4-hydroxybenzaldehyde (4e)-4-aminohex-4-enoic acid 4-hydroxy-3-nitrobenzaldehyde 4-amino hexanoic acid 4-hydroxybenzylamine 1-(4-hydroxyphenyl)prop-2-en-1-one 3-chloro-1-(4-hydroxyphenyl)propan-1-one [1,1':2',1'']-terphenyl-4,3'',5''-triol 6-(3,5-dimethoxy-phenyl)-naphthalen-2-ol 4,3'',5''-trimethoxy-[1,1':2',1'']-terphenyl 6,6-fused nitrogenous heterocyclic compound 1 6,6-fused nitrogenous heterocyclic compound 2 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide 6,6-fused nitrogenous heterocyclic compound 3 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide 4-[(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol 1-[4-(pyridin-4-yloxy)phenyl]-3-[3-(trifluoromethyl)phenyl]urea 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide 2-hexyloxy-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol 4-amino-2-octyloxy-6-hydroxymethyl-tetrahydro-pyran-3,5-diol 4-amino-2-hexyloxy-6-hydroxymethyl-tetrahydro-pyran-3,5-diol 2-hexyloxy-6-hydroxymethyl-tetrahydro-pyran-3,5-diol 2-[4-(2,4-dichlorophenoxy)phenoxy]propanoic acid 3-thiaoctanoyl-coa (z)-2,6-diisopropyl-n-phenyloctadec-9-enamide 9-hydrazino-1,2,3,4-tetrahydroacridine 6-methoxy-1,2-dimethyl-9h-beta-carbolin-2-ium 3-(2-n-piperidyl-propionamino)-rutaecarpine 3-[7-(benzylmethylamino)-heptyloxy]xanthen-9-one 3-[3-(benzylmethylamino)propoxy]xanthen-9-one 9-amino-7h-dibenzo[de,h]quinolin-7-one 9-o-[2-(phenylol-1-yloxy)hexyl]berberine bromide (3-bromo-propyl)-trimethyl-ammonium 6-hydroxy-2-methyl-9h-beta-carbolin-2-ium 2-hex-5-enyl-5-non-8-enyl-3,4-dihydro-2h-pyrrole 9-o-[3-(4-bromo-phenoxyl)butyl]-berberine bromide 9-o-[3-(4-nitro-phenoxyl)butyl]-berberine bromide 9-o-[3-(phenylamino)propyl]-berberine bromide 4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one 6-methyl-4-(4-o-tolylpiperazin-1-yl)coumarin 9-ethyl-2-methyl-beta-carboline-2-ium iodide 9-o-[2-(phenylol-1-yloxy)ethyl]berberine bromide 3-(4-o-tolylpiperazine-1-carbonyl)coumarin (2-chloro-ethyl)-trimethyl-ammonium chloride 1,2-naphthoquinone 3-chloro-9-ethyl-6,7,8,9,10,11-hexahydro-7,11-methanocycloocta[b]quinolin-12-amine (24s)-ethylcholesta-7,9(11),22(e)-triene-3b-ol 3-(2,5-dioxo-pyrrolidin-1-yl)-benzoic acid 4alpha-(hydroxymethyl)-4alpha-demethylterritrem b 9-o-[3-(2-pyridinoxyl)butyl]-berberine bromide 1-deoxy-1-thio-heptaethylene glycol 2-(n-morpholino)-ethanesulfonic acid (2-mercapto-ethyl)-trimethyl-ammonium iodide (-)-huperzine b 2-propyl-beta-carboline-2-ium iodide 3,6,9,12,15-pentaoxaheptadecane 6-methoxy-2-methyl-9h-beta-carbolin-2-ium 3-[6-(benzylmethylamino)hexyloxy]xanthen-9-one 2-(n-morpholino)ethanesulfonic acid 4-pam derivative 1 5-hex-5-enyl-2-nonyl-3,4-dihydro-2h-pyrrole 1,9-bis(pyridinium)-nonane dibromide 1-[3-({[(4-amino-5-fluoro-2-methylquinolin-3-yl)methyl]thio}methyl)phenyl]-2,2,2-trifluoroethane-1,1-diol 3-(2-diethylamino-acetamino)-rutaecarpine 3-(dimethylamino)phenyl phenylcarbamate (rs)-tacrine(10)-hupyridone 4-formylphenyl-o-beta-dglucopyranoside 3-[2-(1-benzyl-piperidin-4-yl)-ethyl]-1h-indazole 24-ethylcholest-6-ene-3,5-diol 1,2-di(berberine-9-o-yl)ethane dibromide (r)-tacrine(10)-hupyridone 9-o-[3-(phenylol-1-yloxy)propyl]berberine bromide 6-chlorotacrine hydrochloride (4as,6r,8as)-11-[8-(1,3-dioxo-1,3-dihydro-2h-isoindol-2-yl)octyl]-6-hydroxy-3-methoxy-5,6,9,10-tetrahydro-4ah-[1]benzofuro[3a,3,2-ef][2]benzazepin-11-ium 9-o-[4-(phenylol-1-yloxy)butyl]berberine bromide (2-ethoxy-ethyl)-trimethyl-ammonium iodide (3,4,8b-trimethyl-3-oxido-2,3a-dihydro-1h-pyrrolo[2,3-b]indol-3-ium-7-yl) n-(2-ethylphenyl)carbamate (s)-tacrine(10)-hupyridone (3r)-9-amino-3-methyl-1,2,3,4-tetrahydroacridine 1,3-di(berberine-9-o-yl)ethane dibromide 9-o-[5-(phenylol-1-yloxy)pentyl]berberine bromide (3-hydroxy-2-methyl-phenyl)-trimethyl-ammonium 2-hex-5-enyl-5-nonyl-pyrrolidine 6-hydroxy-1,2,9-trimethyl-9h-beta-carbolin-2-ium 10-hydroxy-infractopicrin 1,3-bis-(3-imidazolidin-2-yl-phenyl)-urea (-)-tolserine 3-hydroxy-n,n,n-trimethylbenzenaminium iodide (2-butyryloxy-ethyl)-trimethyl-ammonium iodide 6-methoxy-2,9-dimethyl-9h-beta-carbolin-2-ium 24-ethyl-cholest-7-ene-3,5,6-triol 9-amino-1,2,3,4-tetrahydro-acridine-1,7-diol 3-(4-benzoylpiperazine-1-carbonyl)coumarin 6-hydroxy-1,2-dimethyl-9h-beta-carbolin-2-ium 2,3-dihydropyrrolo[2,1-b]quinazolin-9(1h)-imine 2-morpholino-n-phenethylpyrimidin-4-amine 6-hydroxy-2,9-dimethyl-9h-beta-carbolin-2-ium 3-(2-n-piperidyl-acetamino)-rutaecarpine 6-methoxy-1,9-dimethyl-9h-pyrido[3,4-b]indole (5-bromo-pentyl)-trimethyl-ammonium 1,10-bis(pyridinium)-decane dibromide 6,8-dichloro-1,2,3,4-tetrahydro-acridin-9-ylamine 4-[4-(benzhydryloxy)piperidino]butyl benzoate 2-pam derivative 1 1-(3-bromomethyl-phenyl)-2,2,2-trifluoro-ethanone (9s)-9-[(8-ammoniooctyl)amino]-1,2,3,4,9,10-hexahydroacridinium 3-(2-n-pyrrolyl-propionamino)-rutaecarpine 2-(acetylamino)-2-deoxy-a-d-glucopyranose (s,s)-(-)-bis(10)-hupyridone 3-(2-n-pyrrolyl-acetamino)-rutaecarpine 3-[4-(benzylmethylamino)butoxy]xanthen-9-one 5,6-dinitroacenaphthoquinone 3-[(1s)-1-(dimethylamino)ethyl]phenol 1,11-bis(pyridinium)-undecane dibromide (-)-phenserine 3,8-diamino-6-phenyl-5-[6-[1-[2-[(1,2,3,4-tetrahydro-9-acridinyl)amino]ethyl]-1h-1,2,3-triazol-5-yl]hexyl]-phenanthridinium 1,4-di(berberine-9-o-yl)ethane dibromide 3-(3-carboxy-propionylamino)-benzoic acid 1-benzene sulfonyl-cis-2,6-dimethyl piperidine 3,8-diamino-6-phenyl-5-[6-[1-[2-[(1,2,3,4-tetrahydro-9-acridinyl)amino]ethyl]-1h-1,2,3-triazol-4-yl]hexyl]-phenanthridinium 1-ethoxy-2-(2-ethoxyethoxy)ethane 2-[4-(dimethylamino)phenyl]-6-hydroxy-3-methyl-1,3-benzothiazol-3-ium 1-benzyl-4-[(5,6-dimethoxy-1-indanon-2-yl)methyl]piperidine 8-chloro-1,2,3,4-tetrahydro-acridin-9-ylamine 6-methyl-4-(4-benzoylpiperazin-1-yl)coumarin 9-ethyl-beta-carboline 5-chloro-1,2,3,4-tetrahydro-acridin-9-ylamine 3,7-bis(dimethylamino)phenothiazin-5-ium 4-formylphenyl-o-beta-d-ribopyranoside 2-hex-5-enyl-5-non-8-enyl-pyrrolidine 3-(2-diethylamino-propionamino)-rutaecarpine 6-methyl-4-(4-phenylpiperazin-1-yl)coumarin (4-bromo-butyl)-trimethyl-ammonium (s,s)-(-)-bis(12)-hupyridone 3,4,5,6-tetrachloro-[1,2]benzoquinone 4-isopropylphenserine 7-oxo-7h-dibenzo[de,g]quinoline 7-chloro-1,2,3,4-tetrahydro-acridin-9-ylamine 3-[5-(benzylmethylamino)pentyloxy]xanthen-9-one 3-(4-phenylpiperazin-1-carbonyl)coumarin (4-iodo-butyl)-trimethyl-ammonium iodide (1r)-1,2,2-trimethylpropyl (s)-methylphosphinate 3-[8-(benzylmethylamino)octyloxy]xanthen-9-one (-)-hydroxycitrate 4-hydroxy-aconitate ion 2-undecanone (3r)-3-hydroxydodecanoic acid 4-nitrophenyl phosphate (2r,3r)-2,3-dihydroxy-4-oxo-4-(propylamino)butanoic acid 2-(6-hydroxy-1,3-benzothiazol-2-yl)-1,3-thiazol-4(5h)-one 1-methylhistidine (2s)-2-(3-bromophenyl)-3-(5-chloro-2-hydroxyphenyl)-1,3-thiazolidin-4-one 1-((1r)-1-(hydroxymethyl)-3-{6-[(3-phenylpropanoyl)amino]-1h-indol-1-yl}propyl)-1h-imidazole-4-carboxamide 3-(6-amino-purin-9-yl)-non-5-yn-2-ol 3-(6-amino-purin-9-yl)-4-p-tolyl-butan-2-ol 6-hydroxy-1,6-dihydro purine nucleoside 1-((1r,2s)-1-{2-[2-(4-chlorophenyl)-1,3-benzoxazol-7-yl]ethyl}-2-hydroxypropyl)-1h-imidazole-4-carboxamide 3-(6-amino-purin-9-yl)-4-butoxy-butan-2-ol 3-(6-amino-purin-9-yl)-5-m-tolyl-pentan-2-ol 1-{(1r,2s)-2-hydroxy-1-[2-(2-naphthyloxy)ethyl]propyl}-1h-imidazone-4-carboxamide 3-(6-amino-purin-9-yl)-8-phenyl-octan-2-ol (2s,3r)-3-(6-amino-9h-purin-9-yl)nonan-2-ol 6-hydroxy-7,8-dihydro purine nucleoside 3-(6-amino-purin-9-yl)-4-phenethyloxy-butan-2-ol 3-(6-amino-purin-9-yl)-7-phenyl-heptan-2-ol 7,8-dihydroinosine 3-(6-amino-purin-9-yl)-6-phenyl-hexan-2-ol 3-(6-amino-purin-9-yl)-non-5-en-2-ol 1-deaza-adenosine 3-(6-amino-purin-9-yl)-6-o-tolyl-hexan-2-ol 2-(biphenyl-4-ylsulfonamido)-n-hydroxyacetamide 2-(4-bromophenylsulfonamido)-n-hydroxyacetamide (3s)-4-{[4-(but-2-ynyloxy)phenyl]sulfonyl}-n-hydroxy-2,2-dimethylthiomorpholine-3-carboxamide 4-({4-[(4-aminobut-2-ynyl)oxy]phenyl}sulfonyl)-n-hydroxy-2,2-dimethylthiomorpholine-3-carboxamide 3-{[4-(but-2-yn-1-yloxy)phenyl]sulfonyl}propane-1-thiol (3s)-1-{[4-(but-2-yn-1-yloxy)phenyl]sulfonyl}pyrrolidine-3-thiol (1s,3r,6s)-4-oxo-6-{4-[(2-phenylquinolin-4-yl)methoxy]phenyl}-5-azaspiro[2.4]heptane-1-carboxylic acid (2r)-n-hydroxy-2-[(3s)-3-methyl-3-{4-[(2-methylquinolin-4-yl)methoxy]phenyl}-2-oxopyrrolidin-1-yl]propanamide 2-(thiomethylene)-4-methylpentanoic acid (2r,3r)-n^1^-[(1s)-2,2-dimethyl-1-(methylcarbamoyl)propyl]-n^4^-hydroxy-2-(2-methylpropyl)-3-{[(1,3-thiazol-2-ylcarbonyl)amino]methyl}butanediamide 1607004-34-1 (r)-2-(biphenyl-4-sulfonylamino)-propionic acid (2r)-n~4~-hydroxy-2-(3-hydroxybenzyl)-n~1~-[(1s,2r)-2-hydroxy-2,3-dihydro-1h-inden-1-yl]butanediamide 2',5'-dideoxy-adenosine 3'-monophosphate 2,6-diamino-hexanoic acid amide 4-iodopyrazole 2,4-difluorobenzyl alcohol 2,4-difluoro-1-(hydroxymethyl)benzene 2-ethoxyethanol 5-beta-d-ribofuranosylnicotinamide adenine dinucleotide (r)-n-(1-methyl-hexyl)-formamide 3-butylthiolane 1-oxide 2,3-difluorobenzyl alcohol 2,3,4,5,6-pentafluorobenzyl alcohol 12-hydroxydodecanoic acid 7-(5-deoxy-beta-d-ribofuranosyl)-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-4-amine 5-[4-(dimethylamino)phenyl]-6-[(6-morpholin-4-ylpyridin-3-yl)ethynyl]pyrimidin-4-amine 5-iodo,5'-deoxytubercidin 6-benzylthioinosine 5'-iodotubercidin [3h]ccpa 2-(3''-(6''-chloro-indolyl)ethyloxy)adenosine 4-bromo-n-(4-phenyl-thiazol-2-yl)-benzamide 2,6-diphenyl-9h-purine 9-(3-nitrobenzyl)-6-(furan-2-yl)-9h-purin-2-amine 8-bromo-9-(2,3-dihydroxypropyl)-9h-adenine 2-p-tolyl-2h-pyrazolo[3,4-c]quinolin-4-amine 2-chloroadenosine 4-chloro-n-(4-phenyl-thiazol-2-yl)-benzamide 2-ethyl-4-(furan-2-yl)thieno[3,2-d]pyrimidine [3h]neca 4-chloro-7-methyl-2-phenyl-[1,8]naphthyridine 3,4-dichloro-n-(4-phenyl-thiazol-2-yl)-benzamide 2-(3''-(5''-bromo-indolyl)ethyloxy)adenosine 9-allyl-8-bromo-9h-adenine 3-(3-chloro-1h-pyrazol-5-yl)quinoxalin-2(1h)-one 8-bromo-9-cyclohexyl-9h-adenine 3-benzyl-7-methyl-[1,8]naphthyridine-4-thiol 9-isopropyl-9h-adenine 2-(3''-pyrrolylethyloxy)adenosine 2-(4-methyl-1h-benzo[d]imidazol-2-yl)quinoxaline 8-phenyl-1-propyl-3,7-dihydro-purine-2,6-dione 9-(3-aminobenzyl)-6-(furan-2-yl)-9h-purin-2-amine 6-ethylamino-2-(3''-indolyl)ethyloxy)adenosine 2-amino-4,6-diphenyl-pyrimidin-5-carbonitrile 2-(3''-(5''-fluoro-indolyl)ethyloxy)adenosine 5,7-dibromo-9h-pyrido[3,4-b]indol-6-ol 2-(4-chlorophenyl)-6-phenyl-9h-purine 6-guanidino-2-(3''-indolylethyloxy)adenosine (2-chloro-9-methyl-9h-purin-6-yl)-phenyl-amine 8-phenyl-3,7-dihydro-purine-2,6-dione 2,6,8-triphenyl-9h-purine 2-(1h-benzo[d]imidazol-2-yl)quinoxaline 2-cyclopentyl-1h-imidazo[4,5-c]quinolin-4-ylamine 2-(3''-indolylethyloxy)adenosine 8-propyl-2,6-diphenyl-9h-purine 2-p-tolyl-2h-pyrazolo[3,4-c]quinolin-4(5h)-one 7-(3,6,9,12-tetraoxatricos-22-enyl)theophylline 2-(4-chloro-1h-benzo[d]imidazol-2-yl)quinoxaline 1-propyl-3,7-dihydro-purine-2,6-dione 1,3-dipropyl-3,7-dihydro-purine-2,6-dione 2-(hex-1-ynyl)-n6-methoxyadenosine 2,6-diphenyl-8-(1-ethylpropyl)-1-deazapurine 2-m-tolyl-2h-pyrazolo[3,4-c]quinolin-4(5h)-one 8-bromo-9-(2-hydroxypropyl)-9h-adenine 8-bromo-9-cyclobutyl-9h-adenine 2-amino-4-furan-2-yl-6-phenyl-nicotinonitrile 1-methylxanthine 4-methoxy-n-(3-phenyl-isoquinolin-1-yl)-benzamide 2-amino-4,6-diphenyl-nicotinonitrile 9-benzyl-6-(furan-2-yl)-9h-purin-2-amine 9-propyl-9h-adenine 7-dimethylamino-2-phenyl-[1,8]naphthyridin-4-ol 2,5'-dichloro-5'-deoxy-n6-cyclopentyladenosine 2-ethynyl-n6-methoxyadenosine (1-phenyl-propyl)-(9-phenyl-9h-purin-6-yl)-amine 1h-imidazo[4,5-c]quinolin-4-ylamine hcl 9-cyclopentyl-9h-adenine 2-(3''-(5''-hydroxyindolyl)ethyloxy)adenosine 4-(furan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-2-amine (s)-pia 8-phenyl theophylline 2,6-dimethyl-8-ethyl-1-deazapurine 8-bromo-9-(3-hydroxypropyl)-9h-adenine 3-noradamantyl-1,3-dipropylxanthine 2-(6-amino-8-bromo-9h-purin-9-yl)ethanol 8-bromo-9-ethyl-9h-adenine 2-(3''-(5''-methoxy-indolyl)ethyloxy)adenosine 2-amino-4-phenyl-6-thiophen-2-yl-nicotinonitrile 4-tert-butyl-n-(4-phenyl-thiazol-2-yl)-benzamide 2-amino-4,6-di-furan-2-yl-nicotinonitrile 4-methyl-n-(4-phenyl-thiazol-2-yl)-benzamide 2-(3''-(6''-bromo-indolyl)ethyloxy)adenosine 2-amino-4,6-diphenyl-pyrimidine 1-methyl-8-phenyl-3,7-dihydro-purine-2,6-dione 8-bromo-9-propyl-9h-adenine 7-chloro-2-phenyl-[1,8]naphthyridin-4-ol 4-(furan-2-yl)thieno[3,2-d]pyrimidin-2-amine (9-methyl-9h-purin-6-yl)-phenyl-amine 2-(3''-(5''-iodo-indolyl)ethyloxy)adenosine 9-phenyl-9h-purin-6-ylamine 2-(4-methoxyphenyl)-6-phenyl-9h-purine 2-amino-n-benzyl-6-phenyl-9h-purine-9-carboxamide 2-(2-furyl)-6-(1h-pyrazol-1-yl)pyrimidin-4-amine 9-methyl-8-[1,2,3]triazol-2-yl-9h-purin-6-ylamine 2-chloro-4-(thiophen-2-yl)thieno[3,2-d]pyrimidine 8-bromo-9-isobutyl-9h-purin-6-amine 2-(5-cyano-1-pent-1-ynyl)-n6-methoxyadenosine 2-phenyl-1h-imidazo[4,5-c]quinolin-4-ylamine 2,6-bis(4-tolyl)-9h-purine 8-bromo-9-cyclopentyl-9h-adenine 2,6-diphenyl-8-tbutyl-1-deazapurine 2,6-dphenyl-8-propyl-1-deazapurine 2-(2''-indolylethyloxy)adenosine 2'-me-tecadenoson 3-benzyl-7-methyl-[1,8]naphthyridin-4-ol 9-ethyl-9h-adenine 2-(3''-(4''-bromo-indolyl)ethyloxy)adenosine 2-amino-6-phenyl-4-thiophen-2-yl-nicotinonitrile 2-[(4-acetylphenyl)ethynyl]-n6-methoxyadenosine 9-(4-nitrobenzyl)-6-(furan-2-yl)-9h-purin-2-amine 5,7-diphenyl-3h-imidazo[4,5-b]pyridin-2-ol 8-cyclohexyl-6-(4-tolyl)-2-phenyl-9h-purine 4-nitro-n-(4-phenyl-thiazol-2-yl)-benzamide 2-tolyl-6-phenyl-9h-purine 2-phenyl-2h-pyrazolo[3,4-c]quinolin-4-amine 2-(4-hydroxypent-1-yl)-n6-methoxyadenosine [3h]osip339391 (r,s)-phpneca 1,3-diisobutyl-3,7-dihydro-purine-2,6-dione 2-ethyl-4-(thiazol-2-yl)thieno[3,2-d]pyrimidine 1-butyl-8-phenyl-3,7-dihydro-purine-2,6-dione 2-m-tolyl-2h-pyrazolo[3,4-c]quinolin-4-amine [3h]hemado 2,6-diphenyl-1-deazapurine 9-ethyl-8-phenylethynyl-9h-purin-6-ylamine 8-bromo-9-methyl-9h-adenine 2-ethyl-4-(thiophen-2-yl)thieno[3,2-d]pyrimidine 8-bromo-9-(sec-butyl)-9h-adenine 9-benzyl-8-bromo-9h-adenine 8-cyclopentyltheophylline 2-(6-cyclopentylamino-purin-9-yl)-ethanol 2,6-diphenyl-8-ethyl-1-deazapurine 1,3-diethyl-3,7-dihydro-purine-2,6-dione 2-amino-6-furan-2-yl-4-phenyl-nicotinonitrile 2-ethyl-4-(pyridin-2-yl)thieno[3,2-d]pyrimidine [3h]dpcpx 2-azido-n6-methyl-9-(beta-d-ribofuranosyl)adenine 8-bromo-9-phenylethyl-9h-adenine 7-bromo-2-phenyl-[1,8]naphthyridin-4-ol 9-methyl-9h-adenine 4-(ethylthio)-6-phenyl-1,3,5-triazin-2-amine 8-bromo-9-(2-butyl)-9h-adenine 9-cyclobutyl-9h-adenine 2-(4-ethylthiobenzimidazol-2-yl)quinoxaline 2,6-diphenyl-8-methyl-1-deazapurine 2-amino-6-phenyl-4-p-tolylnicotinonitrile 2-(3''(7''-bromo-indolyl)ethyloxy)adenosine 2-chloro-2'-c-methyl-tecadenoson 3-chloro-n-(4-phenyl-thiazol-2-yl)-benzamide 8-bromo-9-isopropyl-9h-adenine 2-ethyl-4-(furan-3-yl)thieno[3,2-d]pyrimidine 7-methyl-2-propyl-[1,8]naphthyridin-4-ol 2-phenyl-2h-pyrazolo[3,4-c]quinolin-4(5h)-one 2-[(4-fluorophenyl)ethynyl]-n6-methoxyadenosine 2-(3''(5''-chloro-indolyl)ethyloxy)adenosine 2,6-diphenyl-pyrimidin-4-ylamine 2-amino-4,6-di-thiophen-2-yl-nicotinonitrile 5-cl-5-deoxy-(+/-)-enba 2-phenylpropoxyadenosine 2,4-dichloro-n-(4-phenyl-thiazol-2-yl)-benzamide 2-chloro-4-(thiazol-2-yl)thieno[3,2-d]pyrimidine 4-ethoxy-7-((e)-styryl)-furo[3,2-g]chromen-5-one 4-amino-2,6-diphenyl-pyrimidine-5-carbonitrile 8-bromo-9-(but-3-enyl)-9h-adenine (e)-8-(3-chlorostyryl)-caffeine (1h-imidazo[4,5-c]quinolin-4-yl)-phenyl-amine hcl 6-(furan-2-yl)-9h-purin-2-amine 1,3-diallyl-3,7-dihydro-purine-2,6-dione 4-(thiazol-2-yl)thieno[3,2-d]pyrimidin-2-amine 9-(sec-butyl)-9h-adenine 1,3,7-tripropyl-3,7-dihydro-purine-2,6-dione 9-(2-hydroxyethyl)-9h-adenine 9-(2-hydroxypropyl)-9h-adenine (s)-dhpa 1-aminoanthracene-9,10-dione 9-butyl-9h-adenine (3-amino-5-bromobenzofuran-2-yl)(phenyl)methanone 7-isopropyl-7h-adenine 9-phenylethyl-9h-adenine 8-br-adenine (e,e)-8-(4-phenylbutadien-1-yl)caffeine 5-azido-6-benzyl-2-methyl-[1,8]naphthyridine 8-chlorotheophylline 1-amino-2,4-bis(phenylthio)anthracene-9,10-dione 9-cycloheptyl-9h-adenine (e,e)-8-[4-(3-bromophenyl)butadien-1-yl]caffeine 4-amino-2-p-tolylisoindoline-1,3-dione 2-amino-3-(m-tolylamino)naphthalene-1,4-dione (e,e)-8-[4-(3-fluorophenyl)butadien-1-yl]caffeine (2r,3s)-3-(6-amino-purin-9-yl)-nonan-2-ol 5-butyl-8-phenyl-3h-[1,2,4]triazolo[5,1-i]purine 1-phenyl-3-(4-pyridin-2-yl-thiazol-2-yl)-urea 2-(3''-(benzoimidazole-1''-yl)ethyloxy)adenosine 1,3-dibenzyl-3,7-dihydro-purine-2,6-dione (z)-8-(3-chlorostyryl)caffeine 1-amino-4-chloroanthracene-9,10-dione 3-isopropyl-1-methyl-3,7-dihydro-purine-2,6-dione 6-furan-2-yl-9-phenethyl-9h-purin-2-ylamine 7-allyl-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 1,3,8-trimethyl-3,7-dihydro-purine-2,6-dione 6-furan-2-yl-9-phenyl-9h-purin-2-ylamine 7-propyl-7h-adenine 9-but-3-enyl-9h-adenine 1,3-diallyl-7-methyl-3,7-dihydro-purine-2,6-dione 9-(3-hydroxypropyl)-9h-adenine (e,e)-8-[4-(3-chlorophenyl)butadien-1-yl]caffeine 1-ethyl-3-methyl-3,7-dihydro-purine-2,6-dione 1-allyl-3,7-dimethyl-3,7-dihydro-purine-2,6-dione 9-benzyl-9h-adenine 1-amino-2-phenoxyanthracene-9,10-dione 1-amino-4-methoxyanthracene-9,10-dione 1,4-diaminoanthracene-9,10-dione 9-cyclopropyl-9h-adenine 4-{2-[(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)amino]ethyl}phenol 7-allyl-1,3-dimethyl-3,7-dihydro-purine-2,6-dione [3h]zm 241385 3-methyl-1-phenethyl-3,7-dihydro-purine-2,6-dione [125i]zm-241385 [125i]abopx 8-(3-fluoro-phenyl)-9-methyl-9h-purin-6-ylamine 1-benzyl-3-methyl-3,7-dihydro-purine-2,6-dione 3-isobutyl-8-pyrrolidinoxanthine 1-butyl-3,7-dihydro-purine-2,6-dione [1,2,4]triazolo[1,5-a]quinoxalin-4(5h)-one 1-cyclopentyl-3,7-dihydro-purine-2,6-dione (+)-butaclamol 2-phenylethylyl-adenosine derivative 4-methoxy-2-phenyl-2h-pyrazolo[4,3-c]quinoline 2-benzoylaminoquinazoline-4-carboxyanilide 2,6-bis(4-methoxyphenyl)-9h-purine 5,6,7-trimethyl-2-p-tolyl-chromen-4-one [125i]ab-meca 2-aminoquinazoline-4-carboxyanilide 1-phenyl-3-(2-(pyridin-2-yl)quinazolin-4-yl)urea 2-(5-chloro-1h-benzo[d]imidazol-2-yl)quinoxaline 2-phenyl-2h-pyrazolo[4,3-d]pyrimidin-7(6h)-one [125i]apnea 2-aminoquinazoline-4-carboxy-(4-bromophenyl)amide [3h]kainate 2,6-bis(4-chlorophenyl)-9h-purine 6-hydroxy-5,7-dimethyl-beta-carboline 2-(1h-imidazo[4,5-c]pyridin-2-yl)quinoxaline 8-hydroxy-5,7,9-trimethyl-delta-carboline 2-(3''-(benzotriazole-1''-yl)ethyloxy)adenosine 1-phenethyl-3,7-dihydro-purine-2,6-dione 9h-purine derivative 1-phenyl-3-(2-(pyridin-3-yl)quinazolin-4-yl)urea 2-acetylaminoquinazoline-4-carboxyanilide 1-phenyl-3-(quinazolin-4-yl)urea 8-hydroxy-7,9-dimethyl-delta-carboline 1-(2-(diethylamino)quinazolin-4-yl)-3-phenylurea 2-(4-nitro-1h-benzo[d]imidazol-2-yl)quinoxaline 1-prop-2-ynyl-3,7-dihydro-purine-2,6-dione 1-allyl-3,7-dihydro-purine-2,6-dione 2-phenyl-2h-pyrazolo[4,3-c]quinoline 1,2-dihydro-2-oxoquinazoline-4-carboxyanilide 1-benzyl-1h-1,3,4b,9-tetraaza-fluorene-2,4-dione 2'-me-ccpa [3h]psb-11 2-benzyl-2h-pyrazolo[3,4-c]quinolin-4(5h)-one 1-phenyl-3-(3-(pyridin-2-yl)isoquinolin-1-yl)urea 1-(pyridin-2-yl)piperazine 1-(3-fluoro-pyridin-2-yl)-4-methyl-piperazine 4-(4-chlorobenzyl)phthalazin-1(2h)-one (2-bromo-phenyl)-(1h-imidazol-2-yl)-amine (2,6-dichloro-phenyl)-(1h-imidazol-2-yl)-amine 4-(1-naphthalen-1-yl-ethyl)-1h-imidazole 5-bromo-8-piperazin-1-yl-imidazo[1,2-a]pyrazine 4-(4-chlorobenzyl)-2-allylphthalazin-1(2h)-one 4-(1-naphthalen-1-yl-vinyl)-1h-imidazole 1-(2-chloro-phenyl)-piperazine 4-(3,4-dihydro-1h-isoquinolin-2-yl)-quinoline 4-benzyl-2-methylphthalazin-1(2h)-one 4-(4-isopropyl-morpholin-2-yl)-benzene-1,2-diol 4-(4-methyl-indan-1-yl)-1h-imidazole 4-morpholin-2-yl-benzene-1,2-diol 2-(4-tert-butyl-phenyl)-4,5-dihydro-1h-imidazole 1',2',3',6'-tetrahydro-[2,4']bipyridinyl [3h]rx821002 [3h]spiperone 4-(3-hydroxy-piperidin-3-yl)-benzene-1,2-diol 4-(4-chlorobenzyl)-2-methylphthalazin-1(2h)-one 4-benzo[b]thiophen-4-yl-1h-imidazole 8-piperazin-1-yl-imidazo[1,2-a]pyrazine 4-(2,3-dihydro-1h-phenalen-1-yl)-1h-imidazole 2-pyridin-4-yl-1,2,3,4-tetrahydro-isoquinoline (+/-)-nantenine 1-(2-methoxy-phenyl)-piperazine 4-methoxyamphetamine 4-((e)-1-naphthalen-1-yl-propenyl)-1h-imidazole 4-(1-naphthalen-1-yl-propyl)-1h-imidazole (-)-snap-5399 4-((z)-1-naphthalen-1-yl-propenyl)-1h-imidazole [125i]be-2254 5-methylurapidil [125i]heat 6-fluoronorepinehprine 6-hydroxy-3-(3',5'-dihydroxyphenyl)coumarin 2,3,4,5-tetrahydro-1h-benzo[c]azepine 8-methoxy-1,2,3,4-tetrahydro-benzo[h]isoquinoline 1,2,3,4-tetrahydro-benzo[h]isoquinolin-8-ol (3-ethyl-indol-1-yl)-propyl-pyridin-4-yl-amine (1h-imidazol-2-yl)-quinoxalin-6-yl-amine (3-methyl-indol-1-yl)-propyl-pyridin-4-yl-amine (1,2,3,4-tetrahydro-isoquinolin-3-yl)-methanol 1,2,3,4-tetrahydroisoquinoline 1,2,3,4,4a,5,10,10a-octahydro-benzo[g]quinoline 2,3,4,5-tetrahydro-benzo[f][1,4]oxazepine 1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 7-methoxy-2,3,4,9-tetrahydro-1h-beta-carboline (1h-benzoimidazol-5-yl)-(1h-imidazol-2-yl)-amine 2,3-dihydro-1h-isoindole 6,7,8,9-tetrahydro-5-thia-8-aza-benzocycloheptene 2-bfi 3-methyl-7-nitro-1,2,3,4-tetrahydro-isoquinoline 3-methoxymethyl-1,2,3,4-tetrahydro-isoquinoline 1-((s)-2-aminopropyl)-1h-indazol-6-ol 5-aminomethyl-naphthalen-2-ol 3-methyl-1,2,3,4-tetrahydro-isoquinoline 2,3,4,5-tetrahydro-1h-benzo[e][1,4]diazepine (s)-3-methyl-1,2,3,4-tetrahydro-isoquinoline (r)-3-methyl-1,2,3,4-tetrahydro-isoquinoline (2-methyl-indol-1-yl)-propyl-pyridin-4-yl-amine 1,2,3,4-tetrahydro-isoquinolin-7-ol 7-nitro-1,2,3,4-tetrahydro-isoquinoline 3-fluoromethyl-1,2,3,4-tetrahydro-isoquinoline 1,2,3,4,5,6-hexahydro-benzo[c]azocine [3h]rauwolscine [3h]mk-912 5-(n,n-hexamethylene)-amiloride 6-fluoro-noradrenaline 2-hydroxymethyl-6-octylsulfanyl-tetrahydro-pyran-3,4,5-triol 4-{[(2s)-3-(tert-butylamino)-2-hydroxypropyl]oxy}-3h-indole-2-carbonitrile [3h]cgp12177 1-(2-isopropylphenoxy)-3-morpholinopropan-2-ol 1-(1h-indol-4-yloxy)-3-phenethylamino-propan-2-ol (r,r)-(-)-fenoterol 1-(2-allylphenoxy)-3-morpholinopropan-2-ol (r,s)-(-)-fenoterol 2-fluoronorepinehprine (s,r)-(+)-fenoterol (s)-carazolol (-)-ro 363 [125i]icyp [3h](-)cgp 12177 6-o-phosphoryl inosine monophosphate 5-butyl-methyl immidazole carboxylate 30 [sar1,bpa2]angii 4-[(diphenylmethyl)amino]-2-phenylquinazoline 4-(2-butyl-benzoimidazol-1-ylmethyl)-phenol [sar1,bpa8]angii [125i]exp985 [bpa1]angii 4-hydroxy-1-methyl-4-(4-methylphenyl)-3-piperidyl 4-methylphenyl ketone [sar1,tdf3]angii [sar1,tdf8]angii (e)-n-(3-iodoprop-2-enyl)-2beta-carbomethoxy-3beta-(4'-methylphenyl)n [3h]gbr12935 [sar1,tdf2]angii [sar1,bpa3]angii 5-oxo-1-2-4-oxadiazol biphenyl [tdf1]angii 1-(biphenyl-4-yl-methyl)-1h-imidazole derivative 1 [125i]cgp42112 4-(2-aminophenyl)-4-oxobutanoic acid 5'-deoxy-5'-ureidoadenosine 5'-s-ethyl-5'-thioadenosine (1'r,2's)-9-(2-hydroxy-3'-keto-cyclopenten-1-yl)adenine 5-methylenearisteromycin 2-propanol, isopropanol 4(z)-(5'-deoxyadenosin-5'-ylidene)butanoic acid 5(e)-(5'-deoxyadenosin-5'-ylidene)pentanoic acid 3'-oxo-adenosine 1-[(4s)-4-amino-5-(1,3-benzothiazol-2-yl)-5-oxopentyl]guanidine 2-(1h-indole-3,-carbonyl)-thiazole-4-carboxylic acid methyl ester 6-formylindolo[3,2-b]carbazole 6-(benzofuran-2-sulfonyl)-2h-pyridazin-3-one 4-(3-benzoyl-1h-pyrrol-1-yl)butanoic acid 7-hydroxy-4-phenylcoumarin 3,5-dichlorosalicylic acid 2-(carboxymethyl)-1-oxo-1,2-dihydronaphtho[1,2-d]isothiazole-4-carboxylic acid 3,3-dioxide 6-(3-chloro-benzenesulfonyl)-2h-pyridazin-3-one 6-phenylmethanesulfonyl-2h-pyridazin-3-one 6-(2-bromo-benzenesulfonyl)-2h-pyridazin-3-one 6-(1h-indole-2-sulfonyl)-2h-pyridazin-3-one 2-benzyl-7-hydroxy-chromen-4-one 6,7-dihydroxy-2-phenyl-chromen-4-one 2-benzhydryl-7-hydroxy-chromen-4-one (4-methyl-2-oxo-2h-quinolin-1-yl)-acetic acid 2-(3,4-dihydroxy-benzyl)-7-hydroxy-chromen-4-one (2-{[(4-bromo-2-fluorobenzyl)amino]carbonyl}-5-chlorophenoxy)acetic acid 6-(4-chloro-benzenesulfonyl)-2h-pyridazin-3-one 2,3-dihydroxypropanal 6-(naphthalene-1-sulfonyl)-2h-pyridazin-3-one 4-(3-methoxy-phenyl)-isoxazolidine-3,5-dione (5-chloro-2-{[(3-nitrobenzyl)amino]carbonyl}phenoxy)acetic acid {4-[(carboxymethoxy)carbonyl]-3,3-dioxido-1-oxonaphtho[1,2-d]isothiazol-2(1h)-yl}acetic acid 6-(naphthalene-2-sulfonyl)-2h-pyridazin-3-one 2-(phenylsulfonamido)acetic acid 4-[3-(3-nitrophenyl)-1,2,4-oxadiazol-5-yl]butanoic acid 6-(4-methoxy-benzenesulfonyl)-2h-pyridazin-3-one (6-methoxy-2-oxo-2h-quinolin-1-yl)-acetic acid 2-(3,4-dihydroxy-phenyl)-7-hydroxy-chromen-4-one 6-(2-chloro-benzenesulfonyl)-2h-pyridazin-3-one 7-hydroxy-6-nitro-2-phenyl-chromen-4-one (8-hydroxy-2-oxo-2h-quinolin-1-yl)-acetic acid 3-(3-benzoyl-1h-pyrrol-1-yl)propanoic acid (r)-minalrestat {3-[(5-chloro-1,3-benzothiazol-2-yl)methyl]-2,4-dioxo-3,4-dihydropyrimidin-1(2h)-yl}acetic acid 7-hydroxy-2-(4-methoxy-benzyl)-chromen-4-one 3-[5-(3-nitrophenyl)thiophen-2-yl]propanoic acid 6-(2-fluoro-benzenesulfonyl)-2h-pyridazin-3-one 7-hydroxy-2-(4-hydroxy-benzyl)-chromen-4-one 6-benzenesulfonyl-2h-pyridazin-3-one {[5-(5-nitro-2-furyl)-1,3,4-oxadiazol-2-yl]thio}acetic acid 6-(toluene-4-sulfonyl)-2h-pyridazin-3-one (6-hydroxy-2-oxo-2h-quinolin-1-yl)-acetic acid 6-methoxykaempferol 3-o-beta-d-robinobioside 6-(4-bromo-benzenesulfonyl)-2h-pyridazin-3-one (s,r)-fidarestat 6-(4-fluoro-benzenesulfonyl)-2h-pyridazin-3-one 2'-monophosphoadenosine 5'-diphosphoribose 6-(benzothiazole-2-sulfonyl)-2h-pyridazin-3-one 6-hydroxy-2-(4-hydroxy-benzyl)-chromen-4-one 6-(biphenyl-2-sulfonyl)-2h-pyridazin-3-one 2-(3-benzoyl-1h-pyrrol-1-yl)acetic acid 2-(4-aminophenylsulfonamido)acetic acid 2-(3-((4,5,7-trifluorobenzo[d]thiazol-2-yl)methyl)-1h-pyrrolo[2,3-b]pyridin-1-yl)acetic acid 2-hydroxy-3,5-diiodobenzoic acid 2-methyl-2,4-pentanediol 2,2-dibenzylcyclopentanol 2-(4-chlorobenzylidene)cyclopentanone 2-(4-chlorobenzylidene)cyclopentylmethyl ether 2-(4-chlorobenzylidene)cyclopentyl ethyl ether 3-phenylcyclopentanecarboxylic acid 4-androstene-3-17-dione 3-carboxamido-1,3,5(10)-estratrien-17(r)-spiro-2'(5',5'-dimethyl-6'oxo)tetrahydropyran 2-[(2,2-diphenylacetyl)amino]benzoic acid 3-bromo-5-phenylsalicylc acid 3,20-pregnanedione 5beta-dihydrotestosterone (z)-3-((1h-pyrrol-2-yl)methylene)indolin-2-one 4,5,6,7-tetrabromo-1h-benzo[d][1,2,3]triazole 4,5,6-trihydroxy-3-methylphthalide 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine (2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amine 4-(4-chlorophenyl)-4-[4-(1h-pyrazol-4-yl)phenyl]piperidine 4-oxosebacic acid 3-(2-aminoethyl)-4-(aminomethyl)heptanedioic acid 5-fluorolevulinic acid 2-sulfhydryl-ethanol 5-hydroxyvaleric acid 4,7-dioxosebacic acid 1,4-dithiothreitol 1,6-di-o-phosphono-d-mannitol 1,6-fructose diphosphate (linear form) 1,2,4-triazolo[1,5a]pyridine derivative 2 3,4,6-tribromo-2-(2,4-dibromo-phenoxy)-phenol (-)-7-n-methyldibromophakellin (+)-(5s,8s,9r,10s)-20-methoxypuupehenone (+)-(5s,8s,10s)-20-methoxy-9,15-ene-puupehenol 2,3,4,5-tetrabromo-6-(2,4-dibromo-phenoxy)-phenol (+)-(5s,8s,10s)-20-methoxypuupehenol 3,6,8-tribromo-dibenzo[1,4]dioxin-1-ol (-)-pinoresinol (2e)-3-(2-oct-1-yn-1-ylphenyl)acrylic acid (-)-3,3'-bisdemethylpinoresinol 3,4-dibromo-2-(5-bromo-2-hydroxy-phenoxy)-phenol (+)-3,3'-bisdemethyltanegool 1-furan-2-yl-3-pyridin-2-yl-propenone (fpp-3) 5-methyl-n-phenylbenzo[d]oxazol-2-amine 2-(4-phenyl-butyl)-1,2-dihydro-indazol-3-one 1,2-dihydroxy-10h-anthracen-9-one 5,3'-dipropyl-biphenyl-2,4'-diol 3-biphenyl-3-yl-n-hydroxy-n-methyl-acrylamide 3-methoxy-n-(4-methylthiazol-2-yl)benzamide 5-chloro-n-(4-ethylphenyl)benzo[d]oxazol-2-amine 10-acetyl-1,8-dihydroxy-10h-anthracen-9-one 2-methyl-1,2-dihydro-indazol-3-one 2,4,5-triarylimidazole analogue 2-pyridin-2-ylmethyl-1,2-dihydro-indazol-3-one 2-(4-methoxy-phenyl)-5-phenyl-thiazol-4-ol (n-(3-phenoxycinnamyl)-acetohydroxamic acid 2-(3-phenyl-propyl)-1,2-dihydro-indazol-3-one 4-methoxy-n-(thiazol-2-yl)benzamide 2-(4-butoxy-phenoxy)-n-hydroxy-acetamide 4-butoxy-n-hydroxy-n-methyl-benzamide 2,4'-diacetoxy-5,3'-di-(2-propenyl)-biphenyl 2-phenyl-n-(1,3,4-thiadiazol-2-yl)acetamide 3,4-dihydroxycinnamic acid 2-phenyl-n-(thiazol-2-yl)acetamide 1-benzyl-1,2-dihydro-indazol-3-one 1-(4-methoxyphenyl)-3-(4-methylthiazol-2-yl)urea 1,2-dihydro-indazol-3-one 1,8-dichloro-10h-anthracen-9-one 2-(4-butoxy-phenyl)-n-hydroxy-n-methyl-acetamide 2-benzyl-1,2-dihydro-indazol-3-one 15-hydroxyeicosatetraenoic acid 4'-methoxy-5,3'-dipropyl-biphenyl-2ol 1-methyl-1,2-dihydro-indazol-3-one 2-thiophen-2-ylmethyl-1,2-dihydro-indazol-3-one 1-(4-methoxyphenyl)-3-(1,3,4-thiadiazol-2-yl)urea 2-(4-butoxy-phenoxy)-n-hydroxy-propionamide 2-(4-butoxy-phenoxy)-n-hydroxy-n-methyl-acetamide 2-naphthalen-2-ylmethyl-1,2-dihydro-indazol-3-one 3-biphenyl-4-yl-n-hydroxy-n-methyl-acrylamide 4-(dimethylamino)-n-(thiazol-2-yl)benzamide 2-phenyl-1,2-dihydro-indazol-3-one 7-tert-butyl-2, 3-dihydro-3, 3-dimethyl substituted dihydrofuran 30 (dhdmbf30) 2-thiazol-5-ylmethyl-1,2-dihydro-indazol-3-one 2-pyridin-4-ylmethyl-1,2-dihydro-indazol-3-one 2-(4-hydroxylphenyl)-3-(3,5-dihydroxylphenyl) propenoic acid (nnu-hdpa) 1,3,8-trihydroxy-6-methyl-10h-anthracen-9-one 3,4,5-trimethoxy-n-(thiazol-2-yl)benzamide 4-bromo-n-hydroxy-benzamide 1-hydroxy-10h-anthracen-9-one 2-pyridin-3-ylmethyl-1,2-dihydro-indazol-3-one 3-benzoyl-n-hydroxy-benzamide 1-hydroxy-8-methoxy-10h-anthracen-9-one 4-hydroxy-5-methoxy-10h-anthracen-9-one 2-phenethyl-1,2-dihydro-indazol-3-one 4,5-dihydroxy-10h-anthracen-9-one 3,4-dihydroxy-10h-anthracen-9-one 5,8-dihydroxy-1,4-naphthoquinone 5-methyl-2-p-tolyl-thiazol-4-ol 4,5-dimethoxy-10h-anthracen-9-one 2'-nitro-biphenyl-4-carboxylic acid hydroxyamide 5s-hete 5-chloro-n-phenylbenzo[d]oxazol-2-amine 5-methoxy-n-phenylbenzo[d]oxazol-2-amine 1,5-dihydroxy-10h-anthracen-9-one 4-(1h-indol-3-yl)-1-morpholinobutan-1-one 1,8,9-trimethoxy-9,10-dihydro-anthracene 3-methoxy-n-(1,3,4-thiadiazol-2-yl)benzamide 2,4'-dimethoxy-5,3'-di-(2-propenyl)-biphenyl 4-pentadeca-1,3,6-trienylsulfanyl-butyric acid 2-(4-methoxyphenyl)-n-(thiazol-2-yl)acetamide 2-biphenyl-4-yl-n-hydroxy-n-methyl-acetamide 1-(4-methoxyphenyl)-3-(5-methylthiazol-2-yl)urea 10-benzoyl-1,8-dihydroxy-10h-anthracen-9-one 3-(4-butoxy-phenyl)-n-hydroxy-n-methyl-acrylamide 2-naphthalen-1-ylmethyl-1,2-dihydro-indazol-3-one 1,8-dihydroxy-2-propionyl-10h-anthracen-9-one 2-furan-2-ylmethyl-1,2-dihydro-indazol-3-one 2-(benzyloxy)naphthalene 2-(1h-indol-3-ylmethyl)-1,2-dihydro-indazol-3-one 5'-([(z)-4-amino-2-butenyl]methylamino)-5'-deoxyadenosine 5'-deoxy-5'-(n,n-dimethylamino)adenosine 5'-deoxy-5'-[(3-hydrazinopropyl)methylamino]adenosine 5'-{[4-(aminooxy)butyl](methyl)amino}-5'-deoxy-8-ethenyladenosine 5'-deoxy-5'-(n,n-dimethylamino)-8-methyladenosine 5'-deoxy-5'-dimethylsulfonioadenosine chloride [(2-aminooxyethyl)methylamino]-5'-deoxyadenosine 5-methyltetrahydrofolic acid 4,6-dideoxy-4-amino-alpha-d-glucose 5-hydroxymethyl-chonduritol 6-deoxy-alpha-d-glucose 4-o-(4,6-dideoxy-4-{[4-[(4-o-hexopyranosylhexopyranosyl)oxy]-5,6-dihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl]amino}hexopyranosyl)hexopyranose 4,6-dideoxy-4-{[4-[(4-o-hexopyranosylhexopyranosyl)oxy]-5,6-dihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl]amino}hexopyranosyl-(1->4)hexopyranosyl-(1->4)hexopyranose 4-o-(4,6-dideoxy-4-{[4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl]amino}-beta-d-lyxo-hexopyranosyl)-alpha-d-erythro-hexopyranose 4,6-dideoxy-4-{[4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl]amino}-alpha-d-lyxo-hexopyranosyl-(1->4)-alpha-d-threo-hexopyranosyl-(1->6)-alpha-l-threo-hexopyranose 1,4-dithio-alpha-d-glucopyranose 4-methylthio-alpha-d-mannose 9-anthroic acid 2-benzyl-n1-hydroxy-n3-phenethylmalonamide (1-amino-2-phenyl-ethyl)-phosphinic acid (1-amino-3-phenyl-propyl)-phosphinic acid 2-amino-n1-benzyl-n3-hydroxymalonamide (s)-2-amino-3-phenyl-propane-1-thiol 2-cinnamamido-n4-hexyl-n1-hydroxysuccinamide (1-amino-3-methyl-butyl)-phosphinic acid 2-cinnamamido-n1-hydroxy-n4-pentylsuccinamide (1-amino-3-methylsulfanyl-propyl)-phosphinic acid 2-benzyl-n1-hydroxy-n3-(3-phenylpropyl)malonamide (amino-phenyl-methyl)-phosphinic acid (s)-2-amino-4-methyl-pentane-1-thiol 1-aminopentylphosphonic acid monophenyl ester (1-amino-ethyl)-phosphinic acid 1-aminobutylphosphonic acid (s)-2-amino-4-methylsulfanyl-butane-1-thiol 2-cinnamamido-n1-hydroxy-n4-octylsuccinamide 1-aminohexylphosphonic acid (s)-2-amino-propane-1-thiol 2-benzyl-n1-hydroxy-n3-(4-phenylbutyl)malonamide (s)-2-amino-4-phenyl-butane-1-thiol [(125)i] rb129 (s)-2-amino-2-phenyl-ethanethiol 1-aminohexylphosphonic acid monophenyl ester 1,4-dideoxy-o2-sulfo-glucuronic acid 1,4-dideoxy-5-dehydro-o2-sulfo-glucuronic acid 6-hydroxydopa quinone 1,3-bis(1,3-benzothiazol-2-ylthio)acetone 3-benzofuran-2-yl-2-benzothiazol-2-yl-3-oxo-propanenitrile 5-fluoro-1h-indole-2-carboxylic acid 1,6-bis(4'-aminophenyl)-hexa-1,3,5-triene 1,6-bis(4'-methylaminophenyl)-hexa-1,3,5-triene 2,5-bis(4-nitrophenyl)thiophene 2,5-bis(2-methoxyphenyl)thiophene 6-iodo-4'-hydroxyflavone 2-(4-(methylamino)phenyl)benzo[d]thiazol-6-ol 6-iodo-4'-dimethyaminoflavone 18f-av-45 dimer 2,5-bis(4-methoxyphenyl)thiophene 5-hydroxy-2-(4-methylaminophenyl)benzofuran 4-(5-(4-aminophenyl)thiophen-2-yl)benzenamine 5-methoxy-2-(4-methylaminophenyl)benzofuran 4-(5-(4-methoxyphenyl)thiophen-2-yl)benzenamine 11c-6-me-bta-1 2,5-bis(4-hydroxyphenyl)thiophene 11c-azd-2184 4-(5-(4-methoxyphenyl)thiophen-2-yl)phenol 6-iodo-4'-methylaminoflavone 5-hydroxy-2-(4-aminophenyl)benzofuran 6-iodo-4'-methoxyflavone 4-(5-(4-aminophenyl)thiophen-2-yl)phenol 4-(5-(4-(methylamino)phenyl)thiophen-2-yl)phenol 5-methoxy-2-(4-dimethylaminophenyl)benzofuran 2-(4-nitrophenyl)-5-(4-methoxyphenyl)thiophene 11a1 5-hydroxy-2-(4-dimethylaminophenyl)benzofuran 1,6-bis(4'-nitrophenyl)-hexa-1,3,5-triene 5-methoxy-2-(4-aminophenyl)benzofuran 123i-drm-106 1,6-bis(4'-dimethylaminophenyl)-hexa-1,3,5-triene 1,6-bis(4'-hydroxyphenyl)-hexa-1,3,5-triene 5-o-phosphono-alpha-d-ribofuranosyl diphosphate 5h-pyrrolo[3,2-d]pyrimidin-4-amine 1-testosterone 2-chloro-4-(o-tolyloxy)benzonitrile 3-methoxy-4-(m-tolyloxy)benzonitrile [3h]methyltrienolone 2'-hydroxy-3-methoxy-biphenyl-4-carbonitrile 4-(cyclobutylmethylthio)-2-methoxybenzonitrile 11-methyl-6,11-dihydro-5h-benzo[a]carbazol-9-ol 3-methoxy-4-(p-tolyloxy)benzonitrile 4-(o-tolyloxy)-2-(trifluoromethyl)benzonitrile 1,2-dibromo-4-(1,2-dibromoethyl)cyclohexane 5-methoxyflavone 6-n-propyl -4-trifluoromethylquinolin-2(1h)-one 6-amino-4-trifluoromethylquinolin-2(1h)-one 4-[(7r,7as)-7-hydroxy-1,3-dioxotetrahydro-1h-pyrrolo[1,2-c]imidazol-2(3h)-yl]-1-naphthonitrile 3-methoxy-4-(o-tolyloxy)benzonitrile 2-methoxy-4-(2-methoxyphenylthio)benzonitrile 4-(butylthio)-2-(trifluoromethyl)benzonitrile [3h]mibolerone 4-(o-tolylthio)-2-(trifluoromethyl)benzonitrile 4-(isopropylthio)-2-methoxybenzonitrile 4-{[(1r,2s)-1,2-dihydroxy-2-methyl-3-(4-nitrophenoxy)propyl]amino}-2-(trifluoromethyl)benzonitrile (3aalpha,4alpha,7alpha,7aalpha)- 3a,4,7,7a-tetrahydro-2-(4-nitro-1-naphthalenyl)-4,7-ethano-1h-isoindole-1,3(2h)-dione 4-(2,6-dimethylphenylthio)-2-methoxybenzonitrile 4-(mesitylthio)-2-(trifluoromethyl)benzonitrile 4-(p-tolyloxy)-2-(trifluoromethyl)benzonitrile 1-tert-butyl-3-(2,5-dimethylbenzyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine 4-(mesitylthio)-2-methoxybenzonitrile (5s,8r,9s,10s,13r,14s,17s)-13-{2-[(3,5-difluorobenzyl)oxy]ethyl}-17-hydroxy-10-methylhexadecahydro-3h-cyclopenta[a]phenanthren-3-one 4-(mesityloxy)-2-(trifluoromethyl)benzonitrile 6,11-dihydrothiochromeno[4,3-b]indol-8-ol (2s)-n-(4-cyano-3-iodophenyl)-3-(4-cyanophenoxy)-2-hydroxy-2-methylpropanamide 4-(cyclopropylmethylthio)-2-methoxybenzonitrile 6-hydroxyflavanone (r)-3-bromo-2-hydroxy-2-methyl-n-[4-nitro-3-(trifluoromethyl)phenyl]propanamide 4-(isopropylthio)-2-(trifluoromethyl)benzonitrile 4-(isopentylthio)-2-(trifluoromethyl)benzonitrile (r)-bicalutamide 2-methoxy-4-(m-tolyloxy)benzonitrile 2-methoxy-4-(propylthio)benzonitrile 2-methoxy-4-(p-tolyloxy)benzonitrile 2-methoxy-4-(o-tolyloxy)benzonitrile 4-(m-tolyloxy)-2-(trifluoromethyl)benzonitrile (2s)-2-hydroxy-2-methyl-n-[4-nitro-3-(trifluoromethyl)phenyl]-3-(pentafluorophenoxy)propanamide 3-[(4-amino-1-tert-butyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)methyl]phenol 4-(butylthio)-2-methoxybenzonitrile 4-(propylthio)-2-(trifluoromethyl)benzonitrile 4-(isopentylthio)-2-methoxybenzonitrile 3-chloro-4-(o-tolyloxy)benzonitrile 3-chloro-4-(o-tolylthio)benzonitrile 2-chloro-4-{[(1r,3z,7s,7as)-7-hydroxy-1-(trifluoromethyl)tetrahydro-1h-pyrrolo[1,2-c][1,3]oxazol-3-ylidene]amino}-3-methylbenzonitrile 3,2'-bis-trifluoromethyl-biphenyl-4-carbonitrile 1,3-propanediol 5'-guanosine-diphosphate-monothiophosphate 2(s)-amino-6-boronohexanoic acid 2-amino-3-hydroxy-3-phosphonooxy-propionic acid 4-nitrocatechol sulfate 5-bromonicotinamide 5-monophosphate-9-beta-d-ribofuranosyl xanthine 2,5-di-tert-butylhydroquinone (6ar,11as,11br)-10-acetyl-9-hydroxy-7,7-dimethyl-2,6,6a,7,11a,11b-hexahydro-11h-pyrrolo[1',2':2,3]isoindolo[4,5,6-cd]indol-11-one 1-acetyl-2-carboxypiperidine 4-(2-aminoethyl)benzenesulfonyl fluoride 1-(5-{2-[(1-methyl-1h-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]urea 7-fluoroindirubin-3-oxime 4-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridine 2-(1h-pyrazol-3-yl)-1h-benzimidazole 6-bromoindirubin-3-oxime 1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]urea 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide 7-bromoindirubin-3-oxime 7-iodoindirubin-3-oxime 7-chloroindirubin-3-oxime 7-fluoroindirubin-3-acetoxime 7-bromoindirubin-3-acetoxime 2np8 [ho1][orn8(5/6c-rhm)]vt [ho1][thr4,orn8(5/6c-flu)]vt [thr4,gly7]ot [lys8(alexa 488) ]pva [phe3]ot [ho1][thr4,lys8(5/6c-flu)]vt [lys8(alexa 546) ]pva [ho1][orn8(5/6c-flu)]vt [val4]avp [ho1][lys8(5/6c-flu)]vt 1'-tosylspiro[indene-1,4'-piperidine] [3h]nelivaptan 3-indolebutyric acid 6-aminohexyl-uridine-c1,5'-diphosphate 4-(4-fluorobenzyl)piperidine 2-amino-6-[2-(1h-indol-6-yl)ethyl]pyrimidin-4(3h)-one (2s)-1-(2,5-dimethylphenoxy)-3-morpholin-4-ylpropan-2-ol 6-[2-(1h-indol-6-yl)ethyl]pyridin-2-amine (2s)-4-(4-fluorobenzyl)-n-(2-sulfanylethyl)piperazine-2-carboxamide 3-(2-amino-6-benzoylquinazolin-3(4h)-yl)-n-cyclohexyl-n-methylpropanamide 6-[2-(3'-methoxybiphenyl-3-yl)ethyl]pyridin-2-amine 4-[(1s)-1-(3-fluoro-4-methoxyphenyl)-2-(2-methoxy-5-nitrophenyl)ethyl]-1h-imidazol-2-amine 4-(2-aminoethyl)-2-ethylphenol 4-(2-aminoethyl)-2-cyclohexylphenol (6s)-2-amino-6-(3'-methoxybiphenyl-3-yl)-3,6-dimethyl-5,6-dihydropyrimidin-4(3h)-one (6r)-2-amino-6-[2-(3'-methoxybiphenyl-3-yl)ethyl]-3,6-dimethyl-5,6-dihydropyrimidin-4(3h)-one (2s)-4-(4-fluorobenzyl)-n-(3-sulfanylpropyl)piperazine-2-carboxamide 2ewy (2r,3r,4s,5r)-2-[6-amino-8-[(3,4-dichlorophenyl)methylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol 1-(10h-phenothiazin-10-yl)-2-phenylethanone (4-nitrophenyl)(10h-phenothiazin-10-yl)methanone 3-[12-(benzylmethylamino)dodecyloxy]xanthen-9-one (-)-phenethylcymserine 1-(3,4-dichlorobenzyl)-1h-indole-2,3-dione 3-isopr-sal-cyclosal-d4tmp (10h-phenothiazin-10-yl)(phenyl)methanone 3-[9-(benzylmethylamino)nonyloxy]xanthen-9-one 1-(10h-phenothiazin-10-yl)-3-phenylpropan-1-one (1'h-phenothiazin-1'-yl)(piperidin-1-yl)methanone 2-methyl-beta-carboline-2-ium iodide 1-(10h-phenothiazin-10-yl)-4-phenylbutan-1-one 1-(10h-phenothiazin-10-yl)-2-phenylbutan-1-one (10h-phenothiazin-10-yl)(p-tolyl)methanone 9-n-phenylmethylamino-tacrine 4-chlorophenyl 10h-phenothiazine-10-carboxylate 2-methoxyphenyl 10h-phenothiazine-10-carboxylate 1,2-di(10h-phenothiazin-10-yl)ethane-1,2-dione 3-methoxyphenyl 10h-phenothiazine-10-carboxylate 3-[11-(benzylmethylamino)undecyloxy]xanthen-9-one 1-(10h-phenothiazin-10-yl)-3-phenylbutan-1-one 4-[4-(benzyloxy)piperidino]butyl-4-nitrobenzoate 9-[5-(beta-carboline-9-yl)pentyl]-beta-carboline 3-[10-(benzylmethylamino)decyloxy]xanthen-9-one 5-methyl-cyclosal-d4tmp 1-methyl-3-(phenylcarbamoyloxy)pyridinium bromide 9-[9-(beta-carboline-9-yl)nonyl]-beta-carboline 4-[4-(benzyloxy)piperidino]butyl-3-fluorobenzoate 1-(10h-phenothiazin-10-yl)-2-phenylpropan-1-one (1s)-menthyl hexyl phosphonate group 1,2-bis(2,3-fluorophenyl)ethane-1,2-dione 2-biphenyl-4-yl-1-phenothiazin-10-yl-ethanone 3-sal-cyclosal-d4tmp 4-[4-(benzyloxy)piperidino]butyl benzoate 4-[4-(benzyloxy)piperidino]butyl-4-fluorobenzoate (3-bromophenyl)(10h-phenothiazin-10-yl)methanone 4-[4-(benzyloxy)piperidino]butyl-4-chlorobenzoate 3-chlorophenyl 10h-phenothiazine-10-carboxylate (1r)-menthyl hexyl phosphonate group (4-bromophenyl)(10h-phenothiazin-10-yl)methanone 9-(3-iodobenzylamino)-1,2,3,4-tetrahydroacridine 4-[4-(benzyloxy)piperidino]butyl-3-chlorobenzoate 3-phenyl-cyclosal-d4tmp (10h-phenothiazin-10-yl)(o-tolyl)methanone 1,2-indanedione (-)-debromoflustramine b 4-methoxyphenyl 10h-phenothiazine-10-carboxylate (10h-phenothiazin-10-yl)(m-tolyl)methanone 5,10-dioxy-2-phenyl-benzo[g]pteridin-4-ylamine 4,5-dibenzylbenzene-1,2-diol 2,3,4-trihydroxy-5-isopropyl-n-phenyl-benzamide 4'-fluoro-1,1'-biphenyl-4-carboxylic acid (d)arg-arg-pro-hyp-gly-thi-cys-(d)phe-phe-cys-arg [des-arg9]bradykinin (d)arg-arg-pro-hyp-gly-thi-ser-(d)tic-aoc-arg [leu8,des-arg9]bradykinin (d)arg-arg-pro-hyp-gly-phe-ser-(d)phe-phe-arg [sar,d-phe8,des-arg9]bradykinin (d)arg-arg-pro-hyp-gly-thi-ser-(d)tic-tic-arg (1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oxime 2-(benzylamino)-6-(3-acetamidophenyl)pyrazine 2-(phenylamino)-6-(3-acetamidophenyl)pyrazine (+)-jq1 [131i]-metuximab 2-(2-hydroxy-1,1-dihydroxymethyl-ethylamino)-ethanesulfonic acid 4-amino-6-chlorobenzene-1,3-disulfonamide 3-(3-phenyl-ureido)-benzenesulfonamide 4-azidobenzenesulfonamide 7-methoxy-2-oxo-2h-chromene-4-carboxylic acid 2-mercapto-n-(4-sulfamoyl-phenyl)-benzamide 5-hydroxy-1-tosyl-1h-pyrrol-2(5h)-one 3-mercapto-n-(4-sulfamoyl-phenyl)-propionamide 3-bromophenyl-difluoromethanesulfonamide 2-oxo-2h-thiochromene-3-carboxylic acid 2-acetamido-5-sulfonamidoindane 4-hydrazino-benzenesulfonamide 4,4'-thiodipyridine-3-sulfonamide 2-morpholin-4-yl-n-(4-sulfamoyl-phenyl)-acetamide 6-methyl-2-oxo-2h-chromene-3-carboxylic acid 4-(2-methyl-8-quinolinoxy)-3-pyridinesulfonamide 6-hydroxy-benzothiazole-2-sulfonic acid amide 4-[2-(2-thienyl)acetamido]benzenesulfonamide 4-(2-phenylacetamido)benzenesulfonamide 4,6-dinitro salicylic acid 4-chloro-n-(5-sulfamoyl-indan-2-yl)-benzamide 1-pentafluorophenylamido-5-sulfonamidoindane 4-bromophenylboronic acid 4-ethynyl benzene sulfonamide 4-(quinolinoxy)-3-pyridinesulfonamide 3-(4-sulfamoylphenyl)propanoic acid 5-chlorosalicylic acid 4-[2-(3-phenyl-ureido)-ethyl]-benzenesulfonamide 6-amino-benzothiazole-2-sulfonic acid amide 3-phenylprop-1-enylboronic acid 4-amino-3-iodo-benzenesulfonamide 5-oxo-1-tosyl-2,5-dihydro-1hpyrrol-2-yl acetate 4-isothiocyanatobenzenesulfonamide (2-bromophenyl)difluoromethanesulfonamide 2-oxo-2h-chromene-3-carboxylic acid 3-chloro-4-hydrazino-benzenesulfonamide 1-acetamido-5-sulfonamidoindane 4-benzenesulfonylamino-benzenesulfonamide (4-bromophenyl)difluoromethanesulfonamide 4-(2-aminoethyl)benzenesulfonamide 4-(2-propynylthio)pyridine-3-sulfonamide 2,3-dihydro-1h-indene-5-sulfonamide 4-nitrophenyl-difluoromethanesulfonamide 4-(2-pyridin-4-ylacetamido)benzenesulfonamide 4-(4-fluorophenoxy)-3-pyridinesulfonamide 4-(n-oxide-2-pyridylthio)pyridine-3-sulfonamide 4-methylthiopyridine-3-sulfonamide [cu(cn)2]- 4-amino-3-chloro-benzenesulfonamide 2,4-disulfamyltrifluoromethylaniline 1-benzyl-1,4-dihydro-4-oxo-3-pyridinesulfonamide 2-butylamido-5-sulfonamidoindane 4-(2-pyridin-2-ylacetamido)benzenesulfonamide 4-methoxyphenylboronic acid [au(cn)2]- 4-[2-(2-thienyl)acetamidoethyl]benzenesulfonamide 4-methanesulfonylamino-benzenesulfonamide 1,4-dihydro-1-methyl-4-oxo-3-pyridinesulfonamide 4-fluoro-n-(4-sulfamoylbenzyl)benzenesulfonamide 4-amino-3-fluoro-benzenesulfonamide 4-phenoxyphenylboronic acid 2-cyclohexylamido-5-sulfonamidoindane 4-methoxy-3-pyridinesulfonamide 2-amino-indan-5-sulfonic acid 4-butylphenylboronic acid 4-(2-phenylacetamido)-3-chlorobenzenesulfonamide 4-amino-3-bromo-benzenesulfonamide 4-(4-cyanophenoxy)-3-pyridinesulfonamide 5-amino-[1,3,4]thiadiazole-2-thiol 4-(methylhydrazino)-3-pyridinesulfonamide 2-acetylamino-indan-5-sulfonic acid hydrate 2-propylamido-5-sulfonamidoindane 4-(carbamolymethylthio)pyridine-3-sulfonamide 4-(hydroxymethyl)benzenesulfonamide 4-ethoxy-3-pyridinesulfonamide 4-hydrazino-3-pyridinesulfonamide 2-ethylamido-5-sulfonamidoindane 1-cyclohexylamido-5-sulfonamidoindane 2-hydroxycinnamic acid 2-pentafluorophenylamido-5-sulfonamidoindane 3-fluoro-4-hydrazino-benzenesulfonamide 2,4-dichloro-5-sulfamoylbenzoic acid 3-phenyl-5-sulfamoyl-1h-indole-2-carboxamide 2-(4-chlorobenzyloxyamino)-n-hydroxypropanamide 2,2,2-trifluoro-n-(4-sulfamoyl-phenyl)-acetamide 1-valproylamido-5-sulfonamidoindane 4-methylstyrylboronic acid 3-[4-(aminosulfonyl)phenyl]propanoic acid 2-nonylamido-5-sulfonamidoindane 4-(2-phenylacetamido)-3-fluorobenzenesulfonamide 4-benzythiopyridine-3-sulfonamide 6-methoxy-2-oxo-2h-chromene-3-carboxylic acid 4-methylphenyl-difluoromethanesulfonamide 2-(4-chlorobenzyloxyamino)-n-hydroxyacetamide 4-hydrazinocarbonyl-benzenesulfonamide 4-(2-aminopyrimidin-4-ylamino)benzenesulfonamide 4-(2-phenylacetamidoethyl)benzenesulfonamide 8-methoxy-2-oxo-2h-chromene-3-carboxylic acid 4-(5-methyl-2-pirazolino)-3-pyridinesulfonamide 4-(cyanomethylthio)pyridine-3-sulfonamide 4-(2-phenylacetamidomethyl)benzenesulfonamide 4-amino-n-(4-sulfamoylbenzyl)benzenesulfonamide 4-(2-phenylacetamido)-3-bromobenzenesulfonamide 2-(biphenyl-4-yl)vinylboronic acid 2-valproylamido-5-sulfonamidoindane 6-(aminomethyl)-2h-chromen-2-one 2-(4-chlorobenzyloxyamino)-n-hydroxyhexanamide 4-(allylamino)-3-pyridinesulfonamide 4-(4'-n-methylphenyl)diazenylbenzenesulfonamide 2-amino-2,3-dihydro-1h-indene-5-sulfonamide 4-(n-methyl-hydrazino)-benzenesulfonamide 4-(2-hydroxy-ethyl)-benzenesulfonamide 6-(hydroxymethyl)-2h-chromen-2-one 7-propoxy-2h-chromen-2-one 3-amino-benzenesulfonamide 3-((4-aminophenyl)diazenyl)benzenesulfonamide 7-(benzyloxy)-2h-chromen-2-one 7-phenethoxy-2h-chromen-2-one 4-methylamino-benzenesulfonamide 3-((4-hydroxyphenyl)diazenyl)benzenesulfonamide 3-(4'-hydroxyphenyl)diazenylbenzenesulfonamide 2-amino-benzenesulfonamide 7-butoxy-2h-chromen-2-one 4-((4-hydroxyphenyl)diazenyl)benzenesulfonamide 4-cyanophenol 2-hydrazinylbenzenesulfonamide 2-acetamido-2,3-dihydro-1h-indene-5-sulfonic acid 2,2-dimethyl-n-(4-sulfamoyl-phenyl)-propionamide 4-aminophenol 2-sulfamoyl-benzoic acid methyl ester 6-chloro-3-(dichloromethyl)-3,4-dihydro-2h-1,2,4-benzothiadiazine-7-sulfonamide 1,1-dioxide 4-(benzylideneamino)benzenesulfonamide 2-methoxyestradiol-17-o-sulfamate 5-(2-chlorophenyl)-1,3,4-thiadiazole-2-sulfonamide 3,5-difluorobenzenesulfonamide 2,6-difluorobenzenesulfonamide 4-sulfonamide-[1-(4-aminobutane)]benzamide (17beta)-17-(cyanomethyl)-2-methoxyestra-1(10),2,4-trien-3-yl sulfamate 4-[(4-o-sulfamoylbenzyl)(4-cyanophenyl)amino]-4h-[1,2,4]-triazole 4-(benzylideneamino)benzoic acid 2,6-di-t-butylphenol 4-(aminosulfonyl)-n-[(4-fluorophenyl)methyl]-benzamide 3-mercuri-4-aminobenzenesulfonamide 6-hydroxy-1,3-benzothiazole-2-sulfonamide 4-methylimidazole 4-methoxyphenylsulfamide 2-(cycloheptylmethyl)-1,1-dioxido-1-benzothiophen-6-yl sulfamate (s)-n-(3-indol-1-yl-2-methyl-propyl)-4-sulfamoyl-benzamide 4-(hydroxymercury)benzoic acid 6-hydroxybenzo[d][1,3]oxathiol-2-one 1-methyl-3-oxo-1,3-dihydro-benzo[c]isothiazole-5-sulfonic acid amide 2-(benzylideneamino)ethanesulfonamide (9beta,13alpha,14beta,17alpha)-2-methoxyestra-1,3,5(10)-triene-3,17-diyl disulfamate 2,6-di-tert-butyl-4-methoxyphenol 1,2,4-triazole (r)-n-(3-indol-1-yl-2-methyl-propyl)-4-sulfamoyl-benzamide 4-(aminosulfonyl)-n-[(3,4,5-trifluorophenyl)methyl]-benzamide 4-({[(4-methylpiperazin-1-yl)amino]carbonothioyl}amino)benzenesulfonamide 4-sulfonamide-[4-(thiomethylaminobutane)]benzamide 5-[(phenylsulfonyl)amino]-1,3,4-thiadiazole-2-sulfonamide 4-(aminosulfonyl)-n-[(2,4-difluorophenyl)methyl]-benzamide 3-nitro-benzenesulfonamide 2-(1,3-thiazol-4-yl)-1h-benzimidazole-5-sulfonamide 1-pentenyl-4-(aminosulfonyl)benzoate 1-n-(4-sulfamoylphenyl-ethyl)-2,4,6-trimethylpyridinium 4-(4-tert-butylbenzylideneamino)benzoic acid 2-(4-tert-butylbenzylideneamino)ethanesulfonamide 4-flourobenzenesulfonamide 4-(aminosulfonyl)-n-[(2,3,4-trifluorophenyl)methyl]-benzamide 1,4-phenylene disulfamate 4-(4-hydroxybenzylideneamino)benzoic acid 2-(n''-acetyl-hydrazino)-benzenesulfonamide 4-[(3-bromo-4-o-sulfamoylbenzyl)(4-cyanophenyl)amino]-4h-[1,2,4]-triazole 1-(3,4-dichlorophenyl)-3-hydroxyurea 2-(benzyloxyamino)-n-hydroxyhexanamide 4-(aminosulfonyl)-n-[(2,5-difluorophenyl)methyl]-benzamide 4-(4-hydroxy-benzylideneamino)-benzenesulfonamide 4-thiocyanato-benzenesulfonamide 2-chloro-5-[(1s)-1-hydroxy-3-oxo-2h-isoindol-1-yl]benzenesulfonamide (2,2-dimethyl-1,3-dioxolan-4-yl)methyl sulfamate 3-hydroxy-2-methoxybenzaldehyde 4-nitro-benzenesulfonamide 2-hydrazinocarbonyl-benzenesulfonamide 5-{[(4-amino-3-chloro-5-fluorophenyl)sulfonyl]amino}-1,3,4-thiadiazole-2-sulfonamide (4s-trans)-4-(methylamino)-5,6-dihydro-6-methyl-4h-thieno(2,3-b)thiopyran-2-sulfonamide-7,7-dioxide (4as,4br,10bs,12as)-12a-methyl-1,3-dioxo-2-(pyridin-3-ylmethyl)-1,2,3,4,4a,4b,5,6,10b,11,12,12a-dodecahydronaphtho[2,1-f]isoquinolin-8-yl sulfamate 4-nitrophenylsulfamide 4-((benzylideneamino)methyl)benzenesulfonamide (s)-indapamide 2-(hydrazinocarbonyl)-3-phenyl-1h-indole-5-sulfonamide 4-(aminosulfonyl)-n-[(2,4,6-trifluorophenyl)methyl]-benzamide 6-nitro-benzothiazole-2-sulfonic acid amide 2-(4-hydroxybenzylideneamino)ethanesulfonamide 2-methoxyestrrone-3-o-sulfamate 3-nitro-4-(2-oxo-pyrrolidin-1-yl)-benzenesulfonamide (4-sulfamoyl-phenyl)-thiocarbamic acid o-(2-thiophen-3-yl-ethyl) ester 2-propyl-pentanoic acid 4-sulfamoyl-benzyl ester 2-propyl-pentanoic acid 4-sulfamoyl-benzylamide [fe(cn)6]4- 8-acetyl-7-hydroxy-2h-chromen-2-one 8-acetyl-7-propoxy-2h-chromen-2-one 6-acetyl-7-propoxy-2h-chromen-2-one 8-acetyl-7-(benzyloxy)-2h-chromen-2-one 2-(benzyloxyamino)-n-hydroxy-3-methylpentanamide 8-acetyl-7-methoxy-2h-chromen-2-one 8-acetyl-7-butoxy-2h-chromen-2-one 6-acetyl-7-hydroxy-2h-chromen-2-one 7-hydroxy-8-propionyl-2h-chromen-2-one 7-ethoxy-8-propionyl-2h-chromen-2-one 6-acetyl-7-ethoxy-2h-chromen-2-one 7-hydroxy-6-propionyl-2h-chromen-2-one 7-methoxy-8-propionyl-2h-chromen-2-one 8-acetyl-7-ethoxy-2h-chromen-2-one 90y-cg250 8-propionyl-7-propoxy-2h-chromen-2-one (4-sulfamoylphenylethylthioureido)fluorescein 2-(benzyloxyamino)-n-hydroxyacetamide 6-acetyl-7-methoxy-2h-chromen-2-one 7-hydroxycoumarin [3h](+)-cis-diltiazem (-)-(r)-efonidipine [3h](+)-isradipine (-)-(s)-bayk8644 [3h](-)devapamil 4-(4-bromobenzylthio)-2-aminobutanoic acid 2-amino-2-(2,3-difluorophenyl)acetic acid 4-(3-fluorobenzylthio)-2-aminobutanoic acid (s)-2-amino-2-cyclohexylacetic acid (s)-2-amino-2-p-tolylacetic acid 2-amino-2-(3-chloro-4-fluorophenyl)acetic acid 2-(1-(aminomethyl)-3-ethylcyclopentyl)acetic acid 3-aminomethyl-5-methyl-hexanoic acid 4-(2-methoxybenzylthio)-2-aminobutanoic acid 4-(2-nitrobenzylthio)-2-aminobutanoic acid 4-(3,5-dichlorobenzylthio)-2-aminobutanoic acid 1-benzhydryl-4-(3,3-diphenylpropyl)piperazine 4-(3-bromobenzylthio)-2-aminobutanoic acid 4-(2,3-dichlorobenzylthio)-2-aminobutanoic acid 3-(aminomethyl)-4-(thiophen-3-yl)butanoic acid 1-benzhydryl-4-(4,4-diphenylbutyl)piperazine 4-(3-chlorobenzylthio)-2-aminobutanoic acid 4-(4-chlorobenzylthio)-2-aminobutanoic acid 3-(aminomethyl)-4-(furan-2-yl)butanoic acid 4-(3-nitrobenzylthio)-2-aminobutanoic acid 4-(4-tert-butylbenzylthio)-2-aminobutanoic acid 2-(1-(aminomethyl)-3-butylcyclopentyl)acetic acid 2-amino-4-(2-methyl-benzylsulfanyl)-butyric acid 2-amino-2-(2,4-difluorophenyl)acetic acid (s)-2-amino-2-o-tolylacetic acid (s)-2-amino-4-(benzylthio)butanoic acid 4-(3,5-dimethylbenzylthio)-2-aminobutanoic acid 4-(2,5-dichlorobenzylthio)-2-aminobutanoic acid 4-(2-cyanobenzylthio)-2-aminobutanoic acid (s)-2-amino-3-(benzylthio)propanoic acid (r)-3-(aminomethyl)-4-(furan-2-yl)butanoic acid 4-(2-bromobenzylthio)-2-aminobutanoic acid 2-amino-2-(3-bromophenyl)acetic acid (s)-2-amino-3-cyclohexylpropanoic acid 4-(3-methoxybenzylthio)-2-aminobutanoic acid 3-(aminomethyl)-4-(thiophen-2-yl)butanoic acid 2-amino-2-(2-fluorophenyl)acetic acid (s)-2-amino-2-phenylpropanoic acid 4-(3-cyanobenzylthio)-2-aminobutanoic acid (s)-phenylglycine 4-(3,4-dimethylbenzylthio)-2-aminobutanoic acid 4-(3,4-dichlorobenzylthio)-2-aminobutanoic acid 3-(aminomethyl)-4-(furan-3-yl)butanoic acid 2-amino-2-(3-chlorophenyl)acetic acid (s)-3-(aminomethyl)-4-(furan-2-yl)butanoic acid 2-amino-2-(thiophen-2-yl)acetic acid (3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamide (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrile 2-[4-[4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl]iminocyclohexa-2,5-dien-1-yl]acetonitrile 1-tert-butyl-3-(3-methylbenzyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine 3-({[(3s)-3,4-dihydroxybutyl]oxy}amino)-1h,2'h-2,3'-biindol-2'-one (2s)-4-methyl-2-(3-phenylthioureido)-n-((3s)-tetrahydro-2-hydroxy-3-furanyl)pentanamide 4-[[(2s)-2-[[(2s)-3-carboxy-2-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]butyl-(diaminomethylidene)azanium (1-benzyl-2-oxo-ethyl)-carbamic acid benzyl ester 3-(1h-pyrrol-3-yl)-propionamide 5-azolone derivative 1 3-{6-[(8-hydroxy-quinoline-2-carbonyl)-amino]-2-thiophen-2-yl-hexanoylamino}-4-oxo-butyri acid 1-methyl-3-trifluoromethyl-1h-thieno[2,3-c]pyrazole-5-carboxylic acid (2-mercapto-ethyl)-amide 2-phenethylisoquinoline-1,3,4-trione [n-(3-dibenzylcarbamoyl-oxiranecarbonyl)-hydrazino]-acetic acid 4-[5-(2-carboxy-1-formyl-ethylcarbamoyl)-pyridin-3-yl]-benzoic acid (1s)-2-oxo-1-phenyl-2-[(1,3,4-trioxo-1,2,3,4-tetrahydroisoquinolin-5-yl)amino]ethyl acetate 5-[4-(1-carboxymethyl-2-oxo-propylcarbamoyl)-benzylsulfamoyl]-2-hydroxy-benzoic acid (1s)-1-(3-chlorophenyl)-2-oxo-2-[(1,3,4-trioxo-1,2,3,4-tetrahydroisoquinolin-5-yl)amino]ethyl acetate 2-allylisoquinoline-1,3,4-trione 2-(4-fluoro-benzyl)isoquinoline-1,3,4-trione 5-(pyrrolidin-1-ylsulfonyl)indoline-2,3-dione 2-(4-methoxy-benzyl)isoquinoline-1,3,4-trione 2-hydroxy-5-(2-mercapto-ethylsulfamoyl)-benzoic acid 2-methylisoquinoline-1,3,4-trione 1-methyl-5-(2-phenoxymethyl-pyrrolidine-1-sulfonyl)-1h-indole-2,3-dione 5-(piperidin-1-ylsulfonyl)indoline-2,3-dione 5-(azepan-1-ylsulfonyl)indoline-2,3-dione 2-benzylisoquinoline-1,3,4-trione 5-(azetidin-1-ylsulfonyl)indoline-2,3-dione 2-furan-2-yl-3-phenethyl-3h-quinazolin-4-one 3-phenethyl-2-phenyl-3h-quinazolin-4-one 2-methyl-3-phenethyl-3h-pyrimidin-4-one 1-arylmethylpyrrolidin-2-yl ethanol amine 2-(2-{2-[2-(2-{2-[2-(2-ethoxy-ethoxy)-ethoxy]-ethoxy}-ethoxy)-ethoxy]-ethoxy}-ethoxy)-ethanol, polyethyleneglycol peg400 3-(4-amino-1-tert-butyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)phenol 1-(3,3-diphenyl-allyl)-3-m-tolyl-urea 1-(4-chloro-phenyl)-3-(3-pentyl-oct-2-enyl)-urea 2-nap 1-(4-chloro-phenyl)-3-(3,3-diphenyl-allyl)-urea 3,4-dichloro-n-(3,3-diphenyl-allyl)-benzamide [3h]devazepide [3h]jb-93182 [3h]pd140376 [3h]pbc-264 [125i]-bdz2 [125i]pd142308 3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-ol 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]-2-pyrimidinamine 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide 1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamide 4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamide 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamide 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide 4-methyl-5-[(2z)-2-{[4-(4-morpholinyl)phenyl]imino}-2,5-dihydro-4-pyrimidinyl]-1,3-thiazol-2-amine (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acid 1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acid 6-o-cyclohexylmethyl guanine 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine (2s)-n-[(3e)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxo-1-imidazolidinyl)phenyl]propanamide 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide 4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-ylamine 1-(3,5-dichlorophenyl)-5-methyl-1h-1,2,4-triazole-3-carboxylic acid 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine 2-anilino-6-cyclohexylmethoxypurine 4-(quinolin-3-yl)-n-p-tolylpyrimidin-2-amine 3,4-diphenyl-1h-pyrrole-2,5-dione 3,4-di-(4-methoxyphenyl)-1h-pyrrole-2,5-dione 3-(4-methoxyphenyl)-4-phenyl-1h-pyrrole-2,5-dione 3-(indole-3-yl)-4-phenyl-1h-pyrrole-2,5-dione 3,4-bis(indol-3-yl)maleimide derivative 4-(quinolin-4-yl)-n-p-tolylpyrimidin-2-amine (s)-3-(2',2'-dimethyl-propionyl)amino-caprolactam (s)-3-(1'-adamantanecarbonyl)amino-caprolactam (r)-3-(1'-adamantanecarbonyl)amino-caprolactam 4-tert-butyl-n-m-tolylthiazol-2-amine 4-tert-butyl-n-(naphthalen-1-yl)thiazol-2-amine 4-tert-butyl-n-phenylthiazol-2-amine 4-isopropyl-n-(naphthalen-1-yl)thiazol-2-amine 4-methyl-n-(naphthalen-1-yl)thiazol-2-amine 4-tert-butyl-n-(2-isopropylphenyl)thiazol-2-amine 4-tert-butyl-n-(naphthalen-1-yl)oxazol-2-amine 4-tert-butyl-n-o-tolylthiazol-2-amine 4-(2-(4-chlorobenzyloxy)-5-bromobenzyl)morpholine (2-(4-chlorobenzyloxy)-5-bromophenyl)methanamine 4scar19 and 4scar20 4scar19 cells 4scar19 and 4scar38 4scar19 and 4scar123 4scar19 and 4scar70 4scar19/22 t cells 19-28z t cells 4scar19 and 4scar30 4scar19 and 4scar22 131 i-omburtamab 124i-8h9 225ac-labelled acd33 212pb-labelled acd37 225ac-labelled acd38 1-beta-ribofuranosyl-1,3-diazepinone (z)-2-(1-decyl-2-oxoindolin-3-ylidene)acetic acid (e)-2-(1-decyl-2-oxoindolin-3-ylidene)acetic acid 3-isopropyl-4-(phenylamino)naphthalene-1,2-dione 3-isopropyl-4-phenylnaphthalene-1,2-dione 3-isopropyl-4-(phenylthio)naphthalene-1,2-dione 4-(p-toluidino)-3-isopropylnaphthalene-1,2-dione 3-isopropylnaphthalene-1,2-dione 1-dodecyl-1h-indole-2,3-dione 2-(1-dodecyl-1h-indol-3-yl)acetic acid 5,6,7,8-tetrahydroanthracene-1,4-dione 6,7-dibromoquinoline-5,8-dione 4-ethoxynaphthalene-1,2-dione 4-phenyl-2-(phenylamino)pyrimidine-5-carbonitrile 9-nitropaullone 2-(p-toluidino)-4-phenylpyrimidine-5-carbonitrile 4-(thiazol-5-yl)-pyrimidine derivative 2 10z-hymenialdisine (2,6-diamino-pyridin-3-yl)-phenyl-methanone [2-amino-6-(2,6-difluoro-benzoyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl-methanone (2'z,3'e)-5-chloro-5'-hydroxy-indirubin-3'-oxime 4-(acetylamino)-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide (5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanol 6-(3,4-dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4(5h)-one 1,5-di-substituted pyridine derivative 1 (2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]-2-pyrimidinyl}amino)phenoxy]-3-(dimethylamino)-2-propanol 5-nitroindirubin-3'-oxime (2'z,3'e)-5-nitro-5'-methoxy-indirubin-3'-oxime 5-fluoro-n-(pyridin-2-yl)pyridin-2-amine derivative 1 4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}-n-(1,3-thiazol-2-yl)benzenesulfonamide 2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurine 4-amino-3,5-di-substituted-thiazole derivative 1 6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamine (2s)-1-{4-[(4-anilino-5-bromo-2-pyrimidinyl)amino]phenoxy}-3-(dimethylamino)-2-propanol 6-(3-methyl-benzyloxy)-9h-purin-2-ylamine 4-{[5-(cyclohexylmethoxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide (2s)-1-[4-({6-[(2,6-difluorophenyl)amino]-4-pyrimidinyl}amino)phenoxy]-3-(dimethylamino)-2-propanol 3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amine 4-{[4-(1-cyclopropyl-2-methyl-1h-imidazol-5-yl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide 3-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]-phenol (2'z,3'e)-5-nitro-5'-hydroxy-indirubin-3'-oxime 4-[(5-isopropyl-1,3-thiazol-2-yl)amino]benzenesulfonamide 4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamide 4-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamide 3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxide (2'z,3'e)-5-fluoro-5'-chloro-indirubin-3'-oxime (2e,3s)-3-hydroxy-5'-[(4-hydroxypiperidin-1-yl)sulfonyl]-3-methyl-1,3-dihydro-2,3'-biindol-2'(1'h)-one (5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonylphenyl)amine (2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]-2-pyrimidinyl}amino)phenoxy]-3-(dimethylamino)-2-propanol 1-(3-(2,4-dimethylthiazol-5-yl)-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)-3-(4-methylpiperazin-1-yl)urea 5-[(4-aminocyclohexyl)amino]-7-(propan-2-ylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile (5e)-2-amino-5-(2-pyridinylmethylene)-1,3-thiazol-4(5h)-one 6-(3-amino-benzyloxy)-9h-purin-2-ylamine 4-{5-[(1z)-1-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)ethyl]-2-furyl}benzenesulfonamide 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amine (2'z,3'e)-5-nitro-5'-methyl-indirubin-3'-oxime 6-cyclohexylmethoxy-pyrimidine-2,4,5-triamine 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline 4-[4-(4-methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenol 2-amino-6-chloropyrazine 4-({5-[(4-aminocyclohexyl)amino][1,2,4]triazolo[1,5-a]pyrimidin-7-yl}amino)benzenesulfonamide 4-(thiazol-5-yl)-pyrimidine derivative 1 (2'z,3'e)-5-chloro-5'-methyl-indirubin-3'-oxime (2r)-1-{4-[(4-anilino-5-bromo-2-pyrimidinyl)amino]phenoxy}-3-(dimethylamino)-2-propanol 1-amino-6-cyclohex-3-enylmethyloxypurine 3-pyridin-4-yl-2,4-dihydro-indeno[1,2-.c.]pyrazole 3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine (3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-one {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide 5-[(2-aminoethyl)amino]-6-fluoro-3-(1h-pyrrol-2-yl)benzo[cd]indol-2(1h)-one 6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxide 6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amine 2-(4-(aminomethyl)piperidin-1-yl)-n-(3_cyclohexyl-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)acetamide 5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine (2r)-1-[4-({6-[(2,6-difluorophenyl)amino]-4-pyrimidinyl}amino)phenoxy]-3-(dimethylamino)-2-propanol 3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amine (5r)-5-{[(2-amino-3h-purin-6-yl)oxy]methyl}-2-pyrrolidinone (2'z,3'e)-5-fluoro-5'-hydroxy-indirubin-3'-oxime (2'z,3'e)-5-nitro-5'-fluoro-indirubin-3'-oxime 4-(2,5-dichloro-thiophen-3-yl)-pyrimidin-2-ylamine 3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine 6-(cyclohex-3-enylmethoxy)-9h-purin-2-ylamine (2s)-1-(dimethylamino)-3-(4-{[4-(2-methylimidazo[1,2-a]pyridin-3-yl)-2-pyrimidinyl]amino}phenoxy)-2-propanol 2-(3,4-dihydroxyphenyl)-8-(1,1-dioxidoisothiazolidin-2-yl)-3-hydroxy-6-methyl-4h-chromen-4-one 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-urea (2'z,3'e)-5-chloro-5'-chloro-indirubin-3'-oxime (4e)-n-(4-fluorophenyl)-4-[(phenylcarbonyl)imino]-4h-pyrazole-3-carboxamide (13r,15s)-13-methyl-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.16,9.1,12,15.0,2,7.0,21,25]heptacosa-1(24),2,4,6,17(25),18,20-heptaene-23,26-dione (2'z,3'e)-5-nitro-5'-chloro-indirubin-3'-oxime (2'z,3'e)-5-fluoro-5'-methoxy-indirubin-3'-oxime 3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amine 5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile 5-hydroxynaphthalene-1-sulfonamide 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine (2'z,3'e)-5-chloro-5'-fluoro-indirubin-3'-oxime 4-{[(2,6-difluorophenyl)carbonyl]amino}-n-[(3s)-piperidin-3-yl]-1h-pyrazole-3-carboxamide 5-bromoindirubin (5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydropyrazolo[1,5-a]pyrimidin-7-amine 3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine 4-{[5-(cyclohexylamino)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide 4-[5-(trans-4-aminocyclohexylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-7-ylamino]-n,n-dimethylbenzenesulfonamide 4-[(6-chloropyrazin-2-yl)amino]benzenesulfonamide 2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanol (2'z,3'e)-5-fluoro-5'-methyl-indirubin-3'-oxime 4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one 4-[(6-amino-4-pyrimidinyl)amino]benzenesulfonamide 4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]benzenesulfonamide 2-((3,5-diamino-1h-pyrazol-4-yl)diazenyl)phenol 1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanol 6-(3-aminophenyl)-n-(tert-butyl)-2-(trifluoromethyl)quinazolin-4-amine 6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amine 3-((3,5-diamino-1h-pyrazol-4-yl)diazenyl)phenol 3-{[(2,2-dioxido-1,3-dihydro-2-benzothien-5-yl)amino]methylene}-5-(1,3-oxazol-5-yl)-1,3-dihydro-2h-indol-2-one (2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-ol 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole (2'z,3'e)-5-fluoro-5'-fluoro-indirubin-3'-oxime 1-(1h-indazol-6-yl)-3-pyridin-2-yl-urea 10-hydroxy-18-methoxybetaenone 1-pyridin-2-yl-3-quinolin-5-yl-urea 1-(9-oxo-9h-fluoren-4-yl)-3-pyridin-2-yl-urea 1-(7-hydroxy-naphthalen-1-yl)-3-pyridin-2-yl-urea 6-phenyl[5h]pyrrolo[2,3-b]pyrazine 3-(2-phenylthiazol-4-yl)quinolin-2(1h)-one 1-phenyl-3-(2-(pyridin-4-yl)thiazol-4-yl)urea (2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methyl-1-butanol 3,7,3',4'-tetrahydroxyflavone 2,5-dichloro-n-p-tolylthiophene-3-sulfonamide 4-(phenyldiazenyl)-1h-pyrazole-3,5-diamine 123-iodine-labeled mfe-23 (2-bromoethyl)(2-'formyl-4'-aminophenyl) acetate (tert-butyloxycarbonyl)-alanyl-amino ethyl-formamide (2s,3s)-3-formyl-2-({[(4-methylphenyl)sulfonyl]amino}methyl)pentanoic acid 2-[5-methanesulfonylamino-2-(4-aminophenyl)-6-oxo-1,6-dihydro-1-pyrimidinyl]-n-(3,3,3-trifluoro-1-isopropyl-2-oxopropyl)acetamide (2r)-3-{[(benzylamino)carbonyl]amino}-2-hydroxypropanoic acid [1-(3-chloro-2-formyl-phenylcarbamoyl)-2-methyl-propyl]-carbamic acid tert-butyl ester (tert-butyloxycarbonyl)-alanyl-alanyl-amine (2s,3s)-3-formyl-2-({[(4-nitrophenyl)sulfonyl]amino}methyl)pentanoic acid 3-[[(methylamino)sulfonyl]amino]-2-oxo-6-phenyl-n-[3,3,3-trifluoro-1-(1-methylethyl)-2-oxophenyl]-1(2h)-pyridine acetamide (3r)-3-ethyl-n-[(4-methylphenyl)sulfonyl]-l-aspartic acid 2-(2-hydroxy-cyclopentyl)-pent-4-enal 1-(4-chloro-phenyl)-2-p-tolyl-ethane-1,2-dione 1,2-bis-(3-methoxy-phenyl)-ethane-1,2-dione 1,2-bis(2,3,5-trifluorophenyl)ethane-1,2-dione 1,2-dicyclohexylethane-1,2-dione 1,2-bis(2,3,5-trifluorophenyl)-2-hydroxyethanone (1r)-1,2,2-trimethylpropyl (r)-methylphosphinate 1,2-bis(2,6-difluorophenyl)-2-hydroxyethanone 1,2-bis(2,6-difluorophenyl)ethane-1,2-dione 1-benzyl-1h-indole-2,3-dione 447c88 4-chloro-1h-indole-2,3-dione (1s,7s,8s,8ar)-1,2,3,7,8,8a-hexahydro-7-methyl-8-[2-[(2r,4r)-tetrahydro-4-hy droxy-6-oxo-2h-pyran-2-yl]ethyl]-1-naphthalenol 1-(3,4-dimethyl-phenyl)-2-phenyl-ethane-1,2-dione 5-(trifluoromethoxy)-1h-indole-2,3-dione 4,5-dichloro-1h-indole-2,3-dione 1-propionyl-1h-indole-2,3-dione 1,1,1-trifluoro-3-(octylsulfinyl)propan-2-one 1-hexadecyl-1h-indole-2,3-dione 4-piperidino-piperidine 1,2-bis(2-fluorophenyl)ethane-1,2-dione 1,2-bis-(4-bromo-phenyl)-ethane-1,2-dione 6,7-dichloro-1h-indole-2,3-dione 7-(trifluoromethyl)-1h-indole-2,3-dione 1,2-bis(3,4,5-trifluorophenyl)ethane-1,2-dione 1-(4-nitro-phenyl)-2-phenyl-ethane-1,2-dione 1-butyryl-1h-indole-2,3-dione 3-(butylthio)-1,1,1-trifluoropropan-2-one 1,2-bis-(2-chloro-phenyl)-ethane-1,2-dione 1,2-bis(4-fluorophenyl)ethane-1,2-dione 1,1,1-trifluoro-3-(hexylsulfonyl)propan-2-one 1,2-bis(2,3-difluorophenyl)-2-hydroxyethanone 3-(decylsulfonyl)-1,1,1-trifluoropropan-2-one 1-(4-chlorobenzyl)-1h-indole-2,3-dione 3-(dodecylsulfonyl)-1,1,1-trifluoropropan-2-one 11,12-dihydro-dibenzo[a,e]cyclooctene-5,6-dione 1,10-phenanthroline-5,6-dione 1-(2-bromoethyl)-1h-indole-2,3-dione 5-chloro-1h-indole-2,3-dione 2,2-dimethyl-3-methyleneheptadecane 1-phenyl-1h-indole-2,3-dione 1,2-bis-(3-nitro-phenyl)-ethane-1,2-dione 1,2-bis(3,4-difluorophenyl)ethane-1,2-dione 1-phenyl-2-p-tolyl-ethane-1,2-dione 1,2-bis(3-fluorophenyl)ethane-1,2-dione (e)-octadec-9-enoic acid phenylamide 1-phenyl-propane-1,2-dione 1,2-bis(2,4-difluorophenyl)-2-hydroxyethanone 1,2-bis(2,5-difluorophenyl)ethane-1,2-dione 1,2-bis(3,4,5-trifluorophenyl)-2-hydroxyethanone 1-(2-iodoethyl)-1h-indole-2,3-dione 1-(4-chloro-phenyl)-2-phenyl-ethane-1,2-dione 3-(decylthio)-1,1,1-trifluoropropan-2-one 7-chloro-1h-indole-2,3-dione 1,2-bis-(4-chloro-phenyl)-ethane-1,2-dione 3-(dodecylsulfinyl)-1,1,1-trifluoropropan-2-one 1,1,1-trifluoro-3-(octylsulfonyl)propan-2-one 1,1,1-trifluoro-3-(hexylthio)propan-2-one 1,2-bis(2,5-difluorophenyl)-2-hydroxyethanone 1-methyl-1h-indole-2,3-dione 4,6-dichloro-1h-indole-2,3-dione 1,2-bis(2-fluorophenyl)-2-hydroxyethanone 1,1,1-trifluoro-3-(octylthio)propan-2-one 1,2-bis(2,3,4-trifluorophenyl)ethane-1,2-dione 6-bromo-5-methyl-1h-indole-2,3-dione 1,2-bis(2,4-difluorophenyl)ethane-1,2-dione 4-chloro-7-methyl-1h-indole-2,3-dione 1,2-di-naphthalen-2-yl-ethane-1,2-dione 1,2-bis(3-fluorophenyl)-2-hydroxyethanon 1,2-bis(2,3,6-trifluorophenyl)ethane-1,2-dione 1,2-bis(3,5-difluorophenyl)ethane-1,2-dione 3,5-di-tert-butyl-[1,2]benzoquinone 1,2-bis(3,4-difluorophenyl)-2-hydroxyethanone 4-(2-oxo-2-phenyl-acetyl)-benzoic acid 3-(decylsulfinyl)-1,1,1-trifluoropropan-2-one 1,2-di-p-tolyl-ethane-1,2-dione 4,7-dichloro-1h-indole-2,3-dione 1,2-bis(2,3,4-trifluorophenyl)-2-hydroxyethanone 1-(4-methoxy-phenyl)-2-phenyl-ethane-1,2-dione 1,1,1-trifluorododecan-2-one 2,2-dimethoxy-1,2-diphenyl-ethanone 3-(butylsulfinyl)-1,1,1-trifluoropropan-2-one 5,7-dichloro-1h-indole-2,3-dione 2-methoxy-3,4-methylenedioxybenzophenone 1,1,1-trifluoro-3-(hexylsulfinyl)propan-2-one 1,2-bis(3,5-difluorophenyl)-2-hydroxyethanone 1,2-bis-(4-methoxy-phenyl)-ethane-1,2-dione 1,1,1-trifluoro-3-(octylthio)acetone 4-guanidinobenzoic acid 3,4-dichloroisocoumarin 2-aminobenzyl alcohol 1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid 9-hydroxypyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione 6-(3-aminopropyl)benzo[h]isoquinolin-1(2h)-one 1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}urea 2-(cyclohexylamino)benzoic acid (5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-acetic (2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-ol 3-(1h-benzimidazol-2-yl)-1h-indazole 5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-one (2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diol 9-chlorobenzo[h]isoquinolin-1(2h)-one 2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acid 6-morpholin-4-yl-9h-purine (5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanol [4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanone 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrile 2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanol (3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylate 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one (2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-ol 1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-one 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol 2-(1h-indazol-3-yl)-1h-benzo[d]imidazole 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one 18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-one 1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine 3-(1h-indol-2-yl)-1h-quinolin-2-one 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenol (3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-one 5-nitro-2-(4-phenoxy-phenyl)-1h-benzoimidazole 2-(4-phenoxy-phenyl)-1h-benzoimidazol-5-ylamine 2-(acetylamino)-2-deoxy-6-o-methyl-alpha-d-allopyranose 2-acetylamino-2-deoxy-b-d-allopyranose (3-exo)-3-(10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-yloxy)-8,8-dimethyl-8-azoniabicyclo[3.2.1]octane 6-dimethylamino-2-methyl-hex-4-ynal oxime 7-dimethylamino-3-methyl-hept-5-yn-2-one 1,1-diphenyl-2-(3-tropanyl)ethanol 7-dimethylamino-hept-5-yn-2-one 1-methyl-1-(4-pyrrolidin-1-yl-but-2-ynyl)-urea 2-methyl-6-pyrrolidin-1-yl-hex-4-ynal oxime 3-(3-benzylamino)-piperidin-2-one 2-(4-diethylamino-but-2-ynyl)-isoindole-1,3-dione 1'-benzyl-3-phenyl-[3,4']bipiperidinyl-2,6-dione 3-tetrazol-2-yl-1-aza-bicyclo[2.2.2]octane 3alpha-(bis-chloro-phenylmethoxy)tropane (s)-oxybutynin 7-pyrrolidin-1-yl-hept-5-yn-2-one 2,8-dimethyl-1-oxa-8-aza-spiro[4.5]decan-3-one 3-methyl-7-pyrrolidin-1-yl-hept-5-yn-2-one (r)-4-[2-[3-(4-methoxy-benzoylamino)-benzyl]-piperidin-1-ylmethyl]piperidine-1-carboxylic acid amide (ro-320-6206) 4-damp 3-(1-carbamoyl-1,1-diphenylmethyl)-1-(4-methoxyphenylethyl)pyrrolidine (app) [3h]oxotremorine-m [3h]qnb [125i]epibatidine [3h]cytisine [3h]methyllycaconitine 1,1-dimethyl-4-phenyl-piperazin-1-ium iodide 1-(piperidin-4-ylmethyl)pyridin-2(1h)-one 2-pyridin-3-yl-7-aza-bicyclo[2.2.1]heptane 5-(1-methyl-pyrrolidin-2-yl)-2-phenethyl-pyridine (s)-3-(azetidin-2-ylmethoxy)-2-fluoropyridine 1-(piperidin-3-ylmethyl)pyridin-2(1h)-one 3-((s)-azetidin-2-yloxy)-5-iodo-pyridine 6'-methylepibatidine (2s,3s)-2-phenyl-3,5,5-trimethylmorpholin-2-ol (2s,3s)-2-(m-tolyl)-3,5,5-trimethylmorpholin-2-ol 3-[2-(n,n,n-trimethylammonium)ethoxy]pyridine [3h]a-585539 3,8-dibromoboldine 4bp-tqs [3h]az11637326 3-bromoboldine [3h]nicotine 18-methylaminocoronaridine 18-methoxycoronaridinate 2-methoxyethylamide 2-methoxyethyl 18-methoxycoronaridinate 2-acetylaminoethyl 18-methoxycoronaridinate 18-dimethylaminocoronaridine 2-hydroxyethyl 18-methoxycoronaridinate 18-methoxycoronaridinate 2-hydroxyethylamide 15-nor-18-methoxycornaridine 5-bromo-6-methoxy-9h-beta-carboline (diaminomethyl-methyl-amino)-acetic acid 2,8-bis[oxido(oxo)vanadio]-1,1,1,3,5,5,7,7,9,9,9-undecaoxopentavanadoxane-2,8-diium (hydroxyethyloxy)tri(ethyloxy)octane 2-[3-({methyl[1-(2-naphthoyl)piperidin-4-yl]amino}carbonyl)-2-naphthyl]-1-(1-naphthyl)-2-oxoethylphosphonic acid [(1s)-1-(5-chloro-1-benzothien-3-yl)-2-(2-naphthylamino)-2-oxoethyl]phosphonic acid [3h]resolvin e1 4-methyl-4,5-dihydro-1h-pyrazole-3-carboxamide derivative 1 (e)-n-(4-methoxyphenethyl)undec-2-enamide 3-benzyl-5-methoxy-7-methylchromen-2-one 5-(1,1-dimethyl-heptyl)-2-pyridin-3-yl-phenol [123i]am251 1-(bis(4-bromophenyl)methyl)-3-phenylurea 3-benzyl-5-isopropyl-8-methylchromen-2-one 1,2,4-triazole derivative 1 3-benzyl-5-methoxychromen-2-one {[(9z)-octadec-9-en-1-yl]sulfamoyl}amine 3'-amino-4-(1,1-dimethyl-heptyl)-biphenyl-2-ol 6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-2,2-dimethyl-3,4-dihydro-2h-pyrano[2,3-b]pyridine-4-carboxamide (enantiomeric mix) 1-(bis(4-chlorophenyl)methyl)-3-phenylurea (4-benzhydrylpiperazin-1-yl)(cyclohexyl)methanone (e)-n-(3,5-dimethoxyphenethyl)undec-2-enamide 1,3,5-triphenylimidazolidine-2,4-dione (e)-n-(4-methoxyphenyl)undec-2-enamide 2-benzylbenzo[f]chromen-3-one 1,2,4-triazole derivative 2 [3h]cp55940 4'-amino-4-(1,1-dimethyl-heptyl)-biphenyl-2-ol 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfinyl)-n-(piperidin-1-yl)-1h-imidazole-4-carboxamide (enantiomeric mix) 2-cycloalkyl resorcinol cannabinoid ligand derivative 2 1-(2-morpholinoethyl)-1h-indol-3-yl acetate (1r,2s)-n-arachidonoylcyclopropanolamide (1r,2r)-n-arachidonoylcyclopropanolamide [3h]hu-243 1,2,4-tri-substituted imidazoline derivative 1 1-[bis(4-bromophenyl)methyl]-3-phenylthiourea (1s,2s)-n-oleoylcyclopropanolamide (2r)-n-(6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-2,2-dimethyl-3,4-dihydro-2h-pyrano[2,3-b]pyridin-4-yl)-2-hydroxypropanamide (enantiomeric mix) 1,2,3-triazole derivative 2 4-benzhydryl-n-butylpiperazine-1-carboxamide 4-cyanophenyl ethyl dodecylphosphonate 6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-n-(1-hydroxy-2-methylpropan-2-yl)-2,2-dimethyl-3,4-dihydro-2h-pyrano[2,3-b]pyridine-4-carboxamide (enantiomeric mix) 2'-amino-4-(1,1-dimethyl-heptyl)-biphenyl-2-ol 1-[bis(4-iodophenyl)methyl]-3-(4-bromophenyl)urea 1,3,5-tris(4-chlorophenyl)imidazolidine-2,4-dione 1,2,4,5-tetra-substituted imidazole derivative 2 1,2,3-triazole derivative 1 [3h]win55212-2 4-(1,1-dimethyl-heptyl)-2'-methoxy-biphenyl-2-ol 5-biphenyl-4-ylmethyl-2-isobutyl-2h-tetrazole 3,4-diarylpyrazoline derivative 1,5-diphenylpyrrolidin-2-one derivative 1 (2s)-n-(7'-(2-chlorophenyl)-6'-(4-chlorophenyl)-3',4'-dihydrospiro[cyclohexane-1,2'-pyrano[2,3-b]pyridine]-4'-yl)-2-hydroxypropanamide (enantiomeric mix) 1-[bis(4-chlorophenyl)methyl]-3-(4-chlorophenyl)- (1r,2s)-n-oleoylcyclopropanolamide 5-methoxy-3-(2-methoxybenzyl)-2h-chromen-2-one 1-[bis(4-chlorophenyl)methyl]-3-phenylthiourea (2r)-n-(7'-(2-chlorophenyl)-6'-(4-chlorophenyl)-3',4'-dihydrospiro[cyclohexane-1,2'-pyrano[2,3-b]pyridine]-4'-yl)-2-hydroxypropanamide (enantiomeric mix) (1s,2s)-n-arachidonoylcyclopropanolamide 4-(1,1-dimethyl-heptyl)-3'-methoxy-biphenyl-2-ol 1,5-diphenylpyrrolidin-2-one derivative 2 6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-n-((r)-1-hydroxyethyl)-1,2,2-trimethyl-1,2,3,4-tetrahydro-1,8-naphthyridine-4-carboxamide (enantiomeric mix) 6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-n-(hydroxymethyl)-1,2,2-trimethyl-1,2,3,4-tetrahydro-1,8-naphthyridine-4-carboxamide (enantiomeric mix) 1,5-bis(4-chlorophenyl)-1h-1,2,3-triazole 4-benzhydryl-n-cyclohexylpiperazine-1-carboxamide 1,4-dihydroindeno[1,2-c]-pyrazole 2-cycloalkyl resorcinol cannabinoid ligand derivative 1 1,2,4,5-tetra-substituted imidazole derivative 1 1,3,5-triazine derivative 1 3-benzoyl-1-pentyl-1,4-dihydroquinolin-4-one 5-biphenyl-4-ylmethyl-1-isobutyl-1h-tetrazole 4'-(1,1-dimethyl-heptyl)-3,5-dimethyl-biphenyl 842166x 2-(2-methoxybenzyl)-3h-benzo[f]chromen-3-one 6,7-dihydroxy-8-nitro-1-tetralone (3,4-dihydroxy-2-nitrophenyl)(phenyl)methanone 1-(3,4-dihydroxy-2-nitrophenyl)-2-phenylethanone 5,6-dihydroxy-7-nitro-2,3-dihydroinden-1-one 3,5-dinitrocatechol 2-methoxyestradiol 7,8-dihydroxy-4-phenyl-2h-chromen-2-one 1-(3,4-dihydroxy-5-nitrophenyl)-2-phenoxyethanone (s)-3-phenyllactic acid 2-benzyl-3-iodopropanoic acid (2r)-2-benzyl-3-nitropropanoic acid 2-thiomethyl-3-phenylpropanoic acid (2r)-4,4-dihydroxy-5-nitro-2-(phenylmethyl)pentanoic acid (2s)-2-[3-(aminomethyl)phenyl]-3-{(s)-hydroxy[(1r)-2-methyl-1-{[(2-phenylethyl)sulfonyl]amino}propyl]phosphoryl}propanoic acid (2s)-2-[3-(aminomethyl)phenyl]-3-[(r)-hydroxy{(1r)-2-methyl-1-[(phenylsulfonyl)amino]propyl}phosphoryl]propanoic acid 2-(3-guanidinophenyl)-3-mercaptopropanoic acid (5r,6s,8s)-8-[3-(aminomethyl)phenyl]-6-hydroxy-5-isopropyl-3-oxo-1-phenyl-2,7-dioxa-4-aza-6-phosphanonan-9-oic acid 6-oxide (2s)-2-[3-(aminomethyl)phenyl]-3-[(r)-[(1r)-1-{[(benzyloxy)carbonyl]amino}-2-methylpropyl](hydroxy)phosphoryl]propanoic acid (2s)-2-(3-carbamimidamidophenyl)-3-[hydroxy(3-phenylpropyl)phosphoryl]propanoic acid 2-(4-benzoylpiperidine-1-carbonyl)benzoic acid (+/-)-5-amino-2-(mercaptomethyl)pentanoic acid 2-(3-aminophenyl)-3-mercaptopropanoic acid 3-mercapto-2-(piperidin-4-yl)propanoic acid 6-amino-2-(1h-imidazol-4-yl)-hexanoic acid 3-mercapto-2-(piperidin-3-yl)propanoic acid (3-carboxy-2-(r)-hydroxy-propyl)-trimethyl-ammonium 9-acetyl-2,3,4,9-tetrahydro-1h-carbazol-1-one 2-aminoisobutyric acid 3-carboxy-n,n,n-trimethyl-2-(octanoyloxy)propan-1-aminium 2-ethoxypropanoic acid 5-cyano-furan-2-carboxylic acid [5-hydroxymethyl-2-(4-methyl-piperidin-1-yl)-phenyl]-amide 6-chloro-3-(3-methylisoxazol-5-yl)-4-phenylquinolin-2(1h)-one 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)ethanol 5-iodotubercidin {4-amino-2-[(4-methoxyphenyl)amino]-1,3-thiazol-5-yl}(4-methoxyphenyl)methanone 4-amino-2-[(3-chlorophenyl)amino]-5-(4-fluorobenzoyl)-1,3-thiazol-3-ium 5,6-dichloro-1-beta-d-ribofuranosylbenzimidazole 1,8-di-hydroxy-4-nitro-anthraquinone 5,6,8-trichloroquinoline-4-one-3-carboxylic acid 19-(cyclopropylamino)-4,6,7,15-tetrahydro-5h-16,1-(azenometheno)-10,14-(metheno)pyrazolo[4,3-o][1,3,9]triazacyclohexadecin-8(9h)-one 5,8-di-amino-1,4-dihydroxy-anthraquinone 7,8-dichloroquinoline-4-one-3-carboxylic acid 2-(cyclohexylmethylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 2-(4-chlorobenzylamino)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 4,5,6,7-tetrabromo-1h-benzimidazole (5-hydroxyindolo[1,2-a]quinazolin-7-yl)acetic acid 3,8-dibromo-7-hydroxy-4-methyl-2h-chromen-2-one 2-(4-ethylpiperazin-1-yl)-4-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile 1,8-di-hydroxy-4-nitro-xanthen-9-one 4-(2-(1h-imidazol-4-yl)ethylamino)-2-(phenylamino)pyrazolo[1,5-a][1,3,5]triazine-8-carbonitrile [1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acid 2-[(3-hydroxy-2-methyl-5-phosphonooxymethyl-pyridin-4-ylmethyl)-imino]-5-phosphono-pent-3-enoic acid 1,1,1-trifluoro-3-acetamido-4-phenyl butan-2-one(n-acetyl-l-phenylalanyl trifluoromethyl ketone) 2,4-dihydroxy-trans cinnamic acid 1,1,1-trifluoro-3-((n-acetyl)-l-leucylamido)-4-phenyl-butan-2-one(n-acetyl-l-leucyl-l-phenylalanyl trifluoromethyl ketone) 2-acetylamino-4-methyl-pentanoic acid (1-formyl-2-phenyl-ethyl)-amide (2s) n-acetyl-l-alanyl-?l-phenylalanyl-chloroethylketone [(3-bromophenyl)-p-tolyl-ketone]thiosemicarbazone (s)-1-benzylcyclopentyl 1-oxohexan-2-ylcarbamate 1-(phenyl(p-tolyl)methylene)thiosemicarbazide 3-amino-4-oxybenzyl-2-butanone 2-aminoethanimidic acid 3-methylphenylalanine 2-pyridinethiol (s)-2-amino-n-(1-cyano-2-phenylethyl)acetamide 1h-benoximidazole-2-carboxylic acid 2-morpholinoethylamine 5-amino-6-cyclohexyl-4-hydroxy-2-isobutyl-hexanoic acid [1-(1-benzyl-3-hydroxy-2-oxo-propylcarbamoyl)-2-phenyl-ethyl]-carbamic acid benzyl ester 4-morpholin-4-yl-piperidine-1-carboxylic acid [1-(3-benzenesulfonyl-1-propyl-allylcarbamoyl)-2-phenylethyl]-amide [1-(1-methyl-4,5-dioxo-pent-2-enylcarbamoyl)-2-phenyl-ethyl]-carbamic acid benzyl ester 1,3-dibenzyl-[1,3]diazetidine-2,4-dione (1r,2r)-n-(2-aminoethyl)-2-{[(4-methoxyphenyl)sulfonyl]methyl}cyclohexanecarboxamide 2-cyclohexylamino-pyrimidine-4-carbonitrile 4-cyclohexylamino-pyrimidine-2-carbonitrile 1-(phenylmethyl)cyclopentyl[(1s)-1-formylpentyl]carbamate 3-amino-5-phenylpentane 4-propyl-6-m-tolylpyrimidine-2-carbonitrile [1-(4-fluorobenzyl)cyclobutyl]methyl (1s)-1-[oxo(1h-pyrazol-5-ylamino)acetyl]pentylcarbamate 4-cycloheptyl-6-propylpyrimidine-2-carbonitrile 4-cyclohexyl-6-propylpyrimidine-2-carbonitrile (s)-tert-butyl 1-oxohexan-2-ylcarbamate 1-{7-cyclohexyl-6-[4-(4-methylpiperazin-1-yl)benzyl]-7h-pyrrolo[2,3-d]pyrimidin-2-yl}methanamine (s)-tert-butyl 4-methyl-1-oxopentan-2-ylcarbamate 4-cyclooctyl-6-propylpyrimidine-2-carbonitrile (2r)-2-(3-biphenylyl)-n-{(2r)-2-hydroxy-3-[(2-pyridinylsulfonyl)amino]propyl}-4-methylpentanamide 2-cyclohexylamino-pyridine-2-carbonitrile 9-cyclopentyl-6-[2-(3-imidazol-1-yl-propoxy)-phenylamino]-9h-purine-2-carbonitrile (2r)-3-methyl-1-phenyl-2-butanyl [(2s)-1-oxo-2-hexanyl]carbamate 6-(cyclohexylamino)-9-[2-(4-methylpiperazin-1-yl)-ethyl]-9h-purine-2-carbonitrile 4-phenyl-6-propylpyrimidine-2-carbonitrile 1-(1,3-diphenylpropylidene)thiosemicarbazide 9-benzyl-6-(benzylamino)-9h-purine-2-carbonitrile (3-bromobenzoylpyridine)thiosemicarbazone [2-phenylacetophenone]thiosemicarbazone [(3-bromophenyl)-m-tolyl-ketone]thiosemicarbazone 6-(benzylamino)-9-butyl-9h-purine-2-carbonitrile 6-(3-(trifluoromethyl)phenyl)picolinonitrile (1r)-2-[(cyanomethyl)amino]-1-({[2-(difluoromethoxy)benzyl]sulfonyl}methyl)-2-oxoethyl morpholine-4-carboxylate 2-[(2',3',4'-trifluorobiphenyl-2-yl)oxy]ethanol 4-methylpiperazin-1-yl carbonyl group 2-(2-(2-fluorophenoxy)phenyl)acetic acid 2-(2-(2,5-dichlorophenylamino)phenyl)acetic acid 2-(2-(2-chlorophenoxy)phenyl)acetic acid 2-(2-(2-fluorophenylamino)phenyl)acetic acid 2-(2-(2-chlorophenylamino)phenyl)acetic acid (r)-n-hydroxy-2-(4-isobutyl-phenyl)-propionamide 1-(2-hydroxy-4-nitrophenyl)-3-phenylurea (r)-2-(4-isobutyl-phenyl)-propionamide 2-[3-(1-hydroxy-propyl)-phenyl]-propionic acid 1-(2-bromo-phenyl)-3-(2,4-dihydroxy-phenyl)-urea 2-[3-(1-phenyl-ethyl)-phenyl]-propionic acid (r)-2-(4-isobutyl-phenyl)-n-methoxy-propionamide 2-(3-isopropyl-phenyl)-propionic acid 2-(3-isobutyl-phenyl)-propionic acid 2-[3-(2-methyl-butyl)-phenyl]-propionic acid (r)-3-(4-isobutyl-phenyl)-butan-2-one 1-(5-chloro-2-hydroxy-4-nitrophenyl)-3-phenylurea 1-(3-cyano-2-hydroxyphenyl)-3-phenylurea 1-(2-hydroxy-3-nitro-phenyl)-3-phenyl-urea 1-(2-hydroxy-5-nitro-phenyl)-3-phenyl-urea 1-(2-bromophenyl)-3-(4-cyano-2-hydroxyphenyl)urea 5-(pentylthio)thiazolo[4,5-d]pyrimidin-7-ol 1-(4-cyano-2-hydroxyphenyl)-3-phenylurea 6-hydroxy-5-undecyl-4,7-benzothiazoledione (s)-famoxadone 5-heptyl-6-hydroxy-1,3-benzothiazole-4,7-dione (5s)-3-anilino-5-(2,4-difluorophenyl)-5-methyl-1,3-oxazolidine-2,4-dione 2-nonyl-4-quinolinol 1-oxide 3-(4-amino-phenyl)-3-pentyl-piperidine-2,6-dione 3-(4-amino-phenyl)-3-butyl-piperidine-2,6-dione 3-[5-methoxy-indan-(1z)-ylidenemethyl]-pyridine 1-phenyl-2-pyridin-3-yl-propan-1-one 6-pyridin-3-yl-3,4-dihydro-1h-quinolin-2-one 3-[4-fluoro-indan-(1e)-ylidenemethyl]-pyridine 4-(4-(thiophen-2-yl)benzyl)pyridine 2-methyl-1,2-di-pyridin-3-yl-propane 3-[(z)-2-phenylvinyl]pyridine 3-[4-methyl-indan-(1e)-ylidenemethyl]-pyridine 3-indan-(1e)-ylidenemethyl-pyridine 3-(naphthalen-2-yl)pyridine 6-(pyridin-3-yl)-2-naphthonitrile 6-isoquinolin-4-yl-3,4-dihydroquinolin-2(1h)-one 1-(4-cyanobenzyl)-5-(2-fluorophenyl)-1h-imidazole 5-[5-bromo-indan-(1z)-ylidenemethyl]-1h-imidazole 3-[5-ethoxy-indan-(1e)-ylidenemethyl]-pyridine 1-(3-methoxy-naphthalen-2-yl)-1h-imidazole 4'-(pyridin-4-ylmethyl)biphenyl-3-amine 1-ethyl-3-imidazol-1-ylmethyl-1h-indole 4-[5-bromo-indan-(1e)-ylidenemethyl]-pyridine 3-indan-(1z)-ylidenemethyl-pyridine 3-[5-ethoxy-indan-(1z)-ylidenemethyl]-pyridine 3-(5,6,7,8-tetrahydronaphthalen-2-yl)pyridine 5-naphthalen-2-yl-oxazole (3-((1h-imidazol-1-yl)methyl)phenyl)methanol (4-((1h-imidazol-1-yl)methyl)phenyl)methanol 1-(4-aminobenzyl)-1h-imidazole 6-pyridin-3-yl-1,2,3,4-tetrahydronaphthalen-2-ol 2-methyl-1,2-di-pyridin-3-yl-propylchloride 3-fluoro-4'-(pyridin-4-ylmethyl)biphenyl-4-ol 4-(4-(thiophen-3-yl)benzyl)pyridine 1-(4-cyanobenzyl)-5-(3-methylphenyl)-1h-imidazole 4-[(3'-hydroxybiphenyl-4-yl)methyl]pyridine 4'-(pyridin-4-ylmethyl)biphenyl-4-amine 4-(6-methoxy-3,4-dihydronaphthalen-2-yl)pyridine 5-[4-(pyridin-4-ylmethyl)phenyl]-1h-indole 1-(4-cyanobenzyl)-5-bromo-1h-imidazole 3-[5-chloro-indan-(1e)-ylidenemethyl]-pyridine 3-(5-methoxy-1h-inden-2-yl)pyridine 3-[3-(4-methoxybenzyl)naphthalen-2-yl]pyridine 3-(4-ethyl-3,4-dihydronaphthalen-2-yl)pyridine 3-[5-chloro-indan-(1z)-ylidenemethyl]-pyridine 5-[5-bromo-indan-(1e)-ylidenemethyl]-1h-imidazole 3-(1-ethyl-3,4-dihydronaphthalen-2-yl)-pyridine 3-[5-fluoro-indan-(1z)-ylidenemethyl]-pyridine 3-(1-chloro-7-methoxy-naphthalen-2-yl)-pyridine 5-pyridin-3-yl-2,3-dihydro-1h-inden-1-one 3-[4-chloro-indan-(1z)-ylidenemethyl]-pyridine 4-[5-fluoro-indan-(1e)-ylidenemethyl]-pyridine 7-pyridin-3-yl-2h-1,4-benzothiazin-3(4h)-one 2-methyl-1,2-di-pyridin-3-yl-propyliodide 1-naphthalen-2-yl-1h-imidazole 3-(6-methoxynaphthalen-2-yl)-5-phenylpyridine 1-(4-cyanobenzyl)-5-formyl-1h-imidazole 3-(3-benzylnaphthalen-2-yl)pyridine 3-(5-chloro-6-methoxy-naphthalen-2-yl)-pyridine 5-[5-fluoro-indan-(1e)-ylidenemethyl]-pyrimidine 1-(6-methoxy-naphthalen-2-yl)-1h-imidazole 1-(4-cyanobenzyl)-5-(4-pyridyl)-1h-imidazole 3-[5-bromo-indan-(1z)-ylidenemethyl]-pyridine 3-(4-methyl-3,4-dihydronaphthalen-2-yl)pyridine 3-[5-methoxy-indan-(1e)-ylidenemethyl]-pyridine 1-(4-bromobenzyl)-5-phenyl-1h-imidazole 4'-(pyridin-4-ylmethyl)biphenyl-3,4-diamine 3-(6-bromo-naphthalen-2-yl)-pyridine 3-(5-bromo-6-methoxy-naphthalen-2-yl)-pyridine 3-(6-methoxy-3-methylnaphthalen-2-yl)pyridine 1-(4-cyanobenzyl)-5-hydroxymethyl-1h-imidazole 5-indan-(1e)-ylidenemethyl-1h-imidazole 2-methyl-1-phenyl-2-pyridin-3-yl-propan-1-ol 4-((3',4'-difluorobiphenyl-4-yl)methyl)pyridine 1-(4-cyanobenzyl)-5-(4-methylphenyl)-1h-imidazole 3-(1h-inden-2-yl)pyridine 1-(3,4-dihydronaphthalen-2-yl)-1h-imidazole 4-(4'-fluoro-biphenyl-4-ylmethyl)pyridine 1-(4-fluorobenzyl)-5-phenyl-1h-imidazole 4-indan-(1z)-ylidenemethyl-pyridine 6-pyridin-3-yl-3,4-dihydronaphthalen-2(1h)-one 3-imidazol-1-ylmethyl-1h-indole 4-[5-chloro-indan-(1e)-ylidenemethyl]-pyridine 1-benzyl-5-phenyl-1h-imidazole 3-[5-bromo-indan-(1e)-ylidenemethyl]-pyridine 1-(4-methoxybenzyl)-5-phenyl-1h-imidazole 3-[4-chloro-indan-(1e)-ylidenemethyl]-pyridine 3-(1,2-dihydroacenaphthylen-3-yl)pyridine 3-imidazol-1-ylmethyl-2-isopropyl-1h-indole 5-(6-methoxynaphthalen-2-yl)pyridin-3-ol 1-(4-cyanobenzyl)-5-(4-fluorophenyl)-1h-imidazole 3-ethoxy-5-(6-methoxynaphthalen-2-yl)pyridine 3-[5-fluoro-indan-(1e)-ylidenemethyl]-pyridine 3-((1h-imidazol-1-yl)methyl)aniline 4-(6-methoxy-3-methylnaphthalen-2-yl)isoquinoline 4-[(4'-hydroxybiphenyl-4-yl)methyl]pyridine 1-(4-bromobenzyl)-1h-imidazole 5-indan-(1z)-ylidenemethyl-1h-imidazole 3-(1-methyl-3,4-dihydronaphthalen-2-yl)-pyridine 1-(4-cyanobenzyl)-5-methyl-1h-imidazole 4'-(pyridin-4-ylmethyl)biphenyl-3,4-diol 3-[1-(4-cyanobenzyl)-1h-imidazol-5-yl]-1-propanol 3-imidazol-1-yl-quinoline 1-(4-fluorobenzyl)-1h-imidazole 3-(3-methyl-3,4-dihydronaphthalen-2-yl)pyridine 1-(4-cyanobenzyl)-5-phenyl-1h-imidazole 3-meso2-dde 2-methyl-1,2-di-pyridin-3-yl-propan-1-one oxime 5-pyridin-3-yl-1,3-dihydro-2h-indol-2-one 5-naphthalen-2-yl-1h-imidazole 7-(1-(1h-imidazol-1-yl)ethyl)-9h-fluoren-2-ol 4-[5-bromo-indan-(1z)-ylidenemethyl]-pyridine 6-[4-(pyridin-4-ylmethyl)phenyl]naphthalen-2-ol 1-(3-chlorobenzyl)-1h-imidazole 3-(6-methoxynaphthalen-2-yl)pyridine 6-(4-methylpyridin-3-yl)-2-naphthonitrile 3-[7-methoxy-indan-(1e)-ylidenemethyl]-pyridine 3-(6-methoxynaphthalen-2-yl)pyridin-4-amine 3-(6-methoxynaphthalen-2-yl)-4-methylpyridine 4-((1h-imidazol-1-yl)methyl)benzonitrile 1-(4-cyanobenzyl)-5-(2-methylphenyl)-1h-imidazole 3-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridine 3-(3-benzyl-6-methoxynaphthalen-2-yl)pyridine 4-(2-imidazol-1-yl-ethoxy)-benzamide 2-methyl-1,2-di-pyridin-3-yl-1-methoxypropane 3-(2-chloro-1,1-dimethyl-2-phenyl-ethyl)-pyridine 1-(4-chlorobenzyl)-5-phenyl-1h-imidazole 1-(2-phenoxy-ethyl)-1h-imidazole 3-(6-ethoxy-naphthalen-2-yl)-pyridine 4-[5-fluoro-indan-(1z)-ylidenemethyl]-pyridine 3-(1,1-dimethyl-2-phenyl-ethyl)-pyridine 3-(1-benzyl-1h-imidazol-5-yl)-1-propanol 6-pyridin-3-yl-naphthalen-2-ol 3-(1,2-dihydroacenaphthylen-5-yl)pyridine 3-[1-(4-bromobenzyl)-1h-imidazol-5-yl]-1-propanol 1-(3-fluorobenzyl)-1h-imidazole 3-(3,4-dihydronaphthalen-2-yl)pyridine 4-(6-methoxynaphthalen-2-yl)isoquinoline 1-(4-cyanobenzyl)-5-(3-fluorophenyl)-1h-imidazole 4-[5-chloro-indan-(1z)-ylidenemethyl]-pyridine 3-phenanthren-9-yl-pyridine 1-(3-bromobenzyl)-1h-imidazole 2-methyl-1-phenyl-2-pyridin-3-yl-propan-1-one 6-pyridin-3-yl-3,4-dihydroquinoline-2(1h)-thione 3-methoxy-5-(6-methoxynaphthalen-2-yl)pyridine 3-(6-methoxy-3,4-dihydronaphthalen-2-yl)pyridine 4'-(2-methyl-1-(pyridin-4-yl)propyl)biphenyl-3-ol 4-[4-(6-methoxynaphthalen-2-yl)benzyl]pyridine 1-(3-(4-fluorophenyl)propyl)-1h-imidazole 4-((1h-imidazol-1-yl)methyl)phenol 1-(4-bromophenethyl)-1h-imidazole 4'-(1-(pyridin-4-yl)propyl)biphenyl-3-ol 2,3,5,6-tetrafluoro-4-pentafluorophenylazo-phenol 1-((9h-fluoren-2-yl)ethyl)-1h-imidazole 1-(3,5-dichlorobenzyl)-1h-imidazole 1-(1-biphenyl-4-yl-ethyl)-1h-imidazole 1-(3,5-bis(trifluoromethyl)benzyl)-1h-imidazole 1-(1-biphenyl-4-yl-2-methyl-propyl)-1h-imidazole 4'-(pyridin-4-ylmethyl)biphenyl-4-carboxamide 2,3,4,5-tetrafluoro-6-pentafluorophenylazo-phenol 1-(3-phenylpropyl)-1h-imidazole 4-[1-(4'-methoxybiphenyl-4-yl)propyl]pyridine 1-(1-(biphenyl-4-yl)allyl)-1h-imidazole 1-(1-biphenyl-4-yl-3-methyl-butyl)-1h-imidazole 1-(1-biphenyl-4-yl-pentyl)-1h-imidazole 1-(3,5-dibromobenzyl)-1h-imidazole 1-(4-iodobenzyl)-1h-imidazole 1-(3-(4-chlorophenyl)propyl)-1h-imidazole 1-(1-(4-thiophen-3-ylphenyl)ethyl)-1h-imidazole 1-(3,4-difluorobenzyl)-1h-imidazole 1-(3,5-difluorobenzyl)-1h-imidazole 3-[4-fluoro-indan-(1z)-ylidenemethyl]-pyridine 3-[(4'-hydroxybiphenyl-4-yl)methyl]pyridine 1-imidazol-1-ylmethylxanthen-9-one 1-(4-methyl-benzyl)-1h-imidazole 1-(1-(4-thiophen-3-yl-phenyl)propyl)-1himidazole 4-bromo-1-imidazol-1-ylmethyl-xanthen-9-one 1-(3,4-dichlorobenzyl)-1h-imidazole 1-(1-biphenyl-4-yl-2-phenyl-ethyl)-1h-imidazole 1-ethyl-5-(imidazol-1-yl-phenyl-methyl)-1h-indole 1-imidazol-1-ylmethyl-4-nitro-xanthen-9-one 1-(1-(4'-ethylbiphenyl-4-yl)propyl)-1h-imidazole 1-(4-nitrobenzyl)-1h-imidazole 1-(bis-biphenyl-4-yl-methyl)-1h-imidazole 3-fluoro-4'-(1-(pyridin-4-yl)propyl)biphenyl-4-ol 6-(3-(pyridin-4-yl)phenyl)naphthalen-2-ol 1-(4-chlorobenzyl)-1h-imidazole 2-(1-imidazol-1-yl-ethyl)-9h-carbazole 1-(1-biphenyl-4-yl-propyl)-1h-imidazole 1-(1-biphenyl-4-yl-butyl)-1h-imidazole 1-(4-chlorophenethyl)-1h-imidazole 1-((9h-fluoren-2-yl)methyl)-1h-imidazole 5-[5-methoxy-indan-(1z)-ylidenemethyl]-thiazole 1-(4-nitro-2-phenoxybenzyl)-1h-imidazole 3-(imidazolylmethyl)-7-methoxy-4'-nitroflavone 5-[5-methoxy-indan-(1e)-ylidenemethyl]-thiazole 4-(1-imidazol-1-yl-vinyl)-benzonitrile 3-(imidazolylmethyl)-4'-nitroflavone 4-((1h-imidazol-1-yl)methyl)-2h-chromen-2-one 2,3,4-trimethoxy-4'-amino-trans-stilbene 4-imidazol-1-yl-2-phenyl-chroman-7-ol 9-hydroxy-7,8-benzoflavone 4-[5-methoxy-indan-(1z)-ylidenemethyl]-pyridine 3-(imidazolylmethyl)flavone 3,5-dihydroxyl-4'-amino-trans-stilbene 5-((1h-imidazol-1-yl)methyl)-7,8-dihydroquinoline 2-imidazol-1-yl-7-methoxy-3-phenyl-chromen-4-one 1-(4-aminophenyl)-2-(1h-imidazol-1-yl)ethanone 4'-cyano-3-(imidazolylmethyl)-7-methoxyflavone 4-[6-methoxy-indan-(1e)-ylidenemethyl]-pyridine 4-[6-methyl-indan-(1e)-ylidenemethyl]-pyridine 3-nitro-4'-nitro-trans-stilbene 3-(4-amino-phenyl)-3-hexyl-piperidine-2,6-dione 1-(9-phenyl-9h-fluoren-9-yl)1h-imidazole 3,5-dimethoxy-4'-amino-trans-stilbene 4'-bromo-3-(imidazolylmethyl)flavone 3,5-diacetoxy-4'-amino-trans-stilbene 1-(2-(benzo[b]thiophen-4-yl)ethyl)-1h-imidazole 4'-bromo-3-(imidazolylmethyl)-7-methoxyflavone 3-[6-methyl-indan-(1e)-ylidenemethyl]-pyridine 3-[6-methoxy-indan-(1e)-ylidenemethyl]-pyridine 4'-cyano-3-(imidazolylmethyl)flavone 4-imidazol-1-ylmethylxanthen-9-one 5-[5-fluoro-indan-(1z)-ylidenemethyl]-pyrimidine 2-(3-hydroxyphenyl)-7-methoxychroman-4-one 1-(1-benzyl-2-biphenyl-4-yl-ethyl)-1h-imidazole 3-(imidazolylmethyl)-4'-methoxyflavone (2s)-5,7,2',4'-tetrahydroxyflavanone 4-[6-methoxy-indan-(1z)-ylidenemethyl]-pyridine 2-phenyl-3-pyridin-4-ylmethylene-chroman-4-one 1-(2-phenoxybenzyl)-1h-imidazole 7,4'-dihydroxyflavone 2,5-dimethoxy-4'-amino-trans-stilbene 4-imidazol-1-ylmethyl-3-nitroxanthen-9-one 3-methoxyl-4'-amino-trans-stilbene 3,4-bis(3,4-dimethoxyphenyl)furan-2(5h)-one 7-[1,2,4]triazol-4-ylmethyl-chromen-4-one 2,3-dimethoxy-4'-amino-trans-stilbene 3-[6-methyl-indan-(1z)-ylidenemethyl]-pyridine 5-(2-(1h-imidazol-1-yl)ethyl)quinoline (2s)-abyssinone ii 4-(3,4,5-trimethoxyphenethyl)aniline 3-[3-methyl-indan-(1z)-ylidenemethyl]-pyridine 3-[3-methyl-indan-(1e)-ylidenemethyl]-pyridine 2-phenyl-4-[1,2,4]triazol-1-yl-chroman-7-ol 8-imidazol-1-ylmethyl-5-nitro-chromen-4-one 3,5-diamino-4'-amino-trans-stilbene 1-[(7-fluoronaphth-2-yl)methyl]-1h-imidazole 3-((1h-imidazol-1-yl)methyl)-9h-xanthen-9-one 2,4-dimethoxy-3'-amino-trans-stilbene 3-(2,2-diphenyl-vinyl)-pyridine 4-imidazol-1-ylmethylthioxanthen-9-one 2,4-dimethoxy-4'-amino-trans-stilbene 1-(9-phenyl-9h-fluoren-9-yl)-1h-1,2,4-triazole 6-((1h-imidazol-1-yl)methyl)-2h-chromene-2-thione 6-imidazol-1-yl-isoquinoline 7-(2-(1h-imidazol-1-yl)ethoxy)-2h-chromen-2-one 3-fluoren-9-ylidenemethyl-pyridine 3-(4-amino-phenyl)-3-heptyl-piperidine-2,6-dione 1-(biphenyl-3-ylmethyl)-1h-1,2,4-triazole 2,3,5-trimethoxy-4'-amino-trans-stilbene 1-bromo-4-imidazol-1-ylmethyl-xanthen-9-one 7-((1h-imidazol-1-yl)methyl)-2h-chromen-2-one 4-(3,4-dimethoxyphenethyl)aniline 7-((1h-imidazol-1-yl)methyl)-4h-chromen-4-one 3-(4-amino-phenyl)-3-ethyl-pyrrolidine-2,5-dione 2-(4-hydroxyphenyl)-7-methoxychroman-4-one 4-imidazol-1-ylmethyl-2-nitroxanthen-9-one (+/-)-7-methoxy-2-(4-methoxyphenyl)chroman-4-one 2-phenyl-2,3-dihydrobenzo[h]chromen-4-one 3-[4-methyl-indan-(1z)-ylidenemethyl]-pyridine 3,4'-(ethane-1,2-diyl)dibenzenamine 1-(9h-fluoren-9-yl)-1h-imidazole 7-((1h-imidazol-1-yl)methyl)isoquinoline 4-indan-(1e)-ylidenemethyl-pyridine 10-epi-8-deoxy-cumambrin b 4-fluoren-9-ylidenemethyl-pyridine 4-[6-methyl-indan-(1z)-ylidenemethyl]-pyridine 2-imidazol-1-ylmethylxanthen-9-one 3-[3-phenyl-indan-(1e)-ylidenemethyl]-pyridine 3,4,5-trimethoxy-4'-amino-trans-stilbene 2-(1h-imidazol-1-yl)-1-(4-nitrophenyl)ethanone 4-(2-(1h-imidazol-1-yl)ethoxy)-2h-chromen-2-one (+/-)-7-methoxy-2-phenylchroman-4-one 3,4-dimethoxy-4'-amino-trans-stilbene (2s)-euchrenone a7 4-(2,2-diphenyl-vinyl)-pyridine 3-amino-4'-amino-trans-stilbene 4-imidazol-1-ylmethyl-1-nitro-xanthen-9-one 11beta,13-dihydro-10-epi-8-deoxycumam-brin b 3-(4-amino-phenyl)-pyrrolidine-2,5-dione 3,4,5-trimethoxy-3'-amino-trans-stilbene 5-bromo-8-imidazol-1-ylmethyl-chromen-4-one 7-hydroxy-2-phenylchroman-4-one 1-(4-nitro-2-phenylsulfanylbenzyl)-1h-imidazole 3-(4-amino-phenyl)-3-methyl-pyrrolidine-2,5-dione 7-hydroxy-2-(3-hydroxyphenyl)chroman-4-one 1-(7-methoxy-2-phenyl-chroman-4-yl)-1h-imidazole 3-(4-amino-phenyl)-1-methyl-pyrrolidine-2,5-dione 4-[5-methoxy-indan-(1e)-ylidenemethyl]-pyridine 3-(4-amino-phenyl)-3-propyl-piperidine-2,6-dione 4-imidazol-1-ylmethyl-1-nitrothioxanthen-9-one 4-(3,5-dimethoxyphenethyl)benzenamine 2-[2-(3,5-dimethoxy-phenyl)-vinyl]-thiophene 3-[2-(3,5-dimethoxy-phenyl)-vinyl]-furan 4-[2-(3,5-dimethoxy-phenyl)-vinyl]-pyridine 4-((+/-)-(1h-imidazol-1-yl)-(e)-retinoic acid 4-((+/-)-(1h-imidazol-1-yl)-(e)-methylretinoate 4,4'-dipyridyl disulfide (5-(pyridin-3-yl)furan-2-yl)methanamine 4-(4-chlorophenyl)imidazole 1-(biphenyl-4-ylmethyl)-1h-imidazole (5r)-5-(4-{[(2r)-6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-2h-chromen-2-yl]methoxy}benzyl)-1,3-thiazolidine-2,4-dione 4-[5-(3-hydroxyphenyl)-2-thienyl)-2-methyl]phenol 4-(3-phenylethynyl-benzyl)-1h-imidazole (2-hydroxy-3-phenoxypropyl)(propan-2-yl)amine 1,5-bis(4-hydroxyphenyl)penta-1,4-dien-3-one 1-(4-butoxy-phenyl)-1h-imidazole 1-(methoxymethyl)-6-(naphthalen-2-yl)-3-azabicyclo[4.1.0]heptane (enantiomeric mix) 2-hexyloxy-5-imidazol-1-yl-pyridine 2-(2-(4-tert-butylphenylthio)ethyl)-1h-imidazole 4-[5-(3-hydroxyphenyl)-3-thienyl]-2-methylphenol 1h-1,2,3-benzotriazol-1-amine 3-[3-(4-imidazol-1-yl-phenoxy)-propyl]-pyridine (5-phenylfuran-2-yl)methanamine 2-[3-(4-imidazol-1-yl-phenoxy)-propyl]-pyridine 1-(3,4-dichlorophenyl)-6-(methoxymethyl)-3-azabicyclo[4.1.0]heptane (enantiomeric mix) 2-(4-imidazol-1-yl-phenoxymethyl)-pyridine 2-fluoro-4-[5-(3-hydroxyphenyl)-2-thienyl]phenol 4-methylaminomethyl-7-methoxycoumarin 4-(spiro[chromene-2,4'-piperidine]-4-yl)benzamide 4-[2-(4-imidazol-1-yl-phenoxy)-ethyl]-morpholine 4-[3-(4-imidazol-1-yl-phenoxy)-propyl]-pyridine 4-(3-pent-1-ynyl-benzyl)-1h-imidazole (5-pyridin-3-yl-furan-2-yl)methanethiol 6-(3,4-dichlorophenyl)-1-[1-(methyloxy)-3-buten-1-yl]-3-azabicyclo[4.1.0]heptane (diastereomeric mix) (-)-dihydroclusin 1-acetoxy-2-tert-butyldimethylsilyl-oxylycorine 1-acetoxylycorine 3-(5-((methylthio)methyl)furan-2-yl)pyridine 3-(5-[1,3]dithiolan-2-yl-furan-2-yl)pyridine 1,1':4',1''-terphenyl-3,3''-diol 3-[5-(4-hydroxyphenyl)-3-thienyl]phenol (-)-clusin 5-(2-phenethylpiperazin-1-yl)-1h-indazole (8r,8'r,9's)-5-methoxyclusin (-)-yatein (8r,8'r)-4-hydroxycubebinone 3,3-(1,3-thiazole-2,5-diyl)diphenol 2-tert-butyldimethylsilyloxylycorine (-)-cubebininolide 3-(pyridin-3-yl)prop-2-yn-1-amine 6-(3-hydroxy-phenyl)-naphthalen-2-ol 5-pyridin-3-yl-thiophene-2-carbaldehyde oxime 2,5-bis(4-hydroxybenzylidene)cyclopentanone (-)-cubebinin (-)-cubebin 3-(3-methylthiophen-2-yl)pyridine (-)-thujaplicatintrimethyl ether 1,2-diacetoxylycorine 2-fluoro-5-(3-methylthiophen-2-yl)pyridine (s)-econazole [3h]ltc4 1d-myo-inositol 1,4,5-trisphosphate (2e)-3-(3,4-dihydroxyphenyl)-2-iminopropanoic acid 3,4-dihydro-2h-pyrrolium-5-carboxylate 6-(3-aminopropyl)-4,9-dimethylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione 5,6-dihydro-benzo[h]cinnolin-3-ylamine 4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acid 2-tert-butyl-9-fluoro-1,6-dihydrobenzo[h]imidazo[4,5-f]isoquinolin-7-one (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile 2'-deoxycytidine 7-methyl-7,8-dihydroguanosine-5'-diphosphate 7-methyl-gpppa 5-{[1-(2,3-dichlorobenzyl)piperidin-4-yl]methoxy}quinazoline-2,4-diamine 7-methyl-5'-guanylic acid 5-{[1-(2-fluorobenzyl)piperidin-4-yl]methoxy}quinazoline-2,4-diamine 7-methyl-guanosine-5'-triphosphate-5'-guanosine 5-[(1s)-1-(3-chlorophenyl)ethoxy]quinazoline-2,4-diamine 3-hydroxybenzylhydrazine 6-methyl-2(propane-1-sulfonyl)-2h-thieno[3,2-d][1,2,3]diazaborinin-1-ol 1954u89 5-[(3r)-3-(5-methoxy-3',5'-dimethylbiphenyl-3-yl)but-1-yn-1-yl]-6-methylpyrimidine-2,4-diamine 2,4-diamino-6-[n-(3',4',5'-trimethoxybenzyl)-n-methylamino]pyrido[2,3-d]pyrimidine 2,4-diamino-6-[n-(3',5'-dimethoxybenzyl)-n-methylamino]pyrido[2,3-d]pyrimidine 5-[(3r)-3-(5-methoxybiphenyl-3-yl)but-1-yn-1-yl]-6-methylpyrimidine-2,4-diamine 5-[(3r)-3-(5-methoxy-2',6'-dimethylbiphenyl-3-yl)but-1-yn-1-yl]-6-methylpyrimidine-2,4-diamine (4as)-5-[(2,4-diaminopteridin-6-yl)methyl]-4a,5-dihydro-2h-dibenzo[b,f]azepin-8-ol 6-(octahydro-1h-indol-1-ylmethyl)decahydroquinazoline-2,4-diamine 5-[(3r)-3-(5-methoxy-4'-methylbiphenyl-3-yl)but-1-yn-1-yl]-6-methylpyrimidine-2,4-diamine 2,4-diamino-5-(3,4,5-trimethoxy-benzyl)-pyrimidin-1-ium [n-(2,4-diaminopteridin-6-yl)-methyl]-dibenz[b,f]azepine 5-[3-(2,5-dimethoxyphenyl)prop-1-yn-1-yl]-6-ethylpyrimidine-2,4-diamine 2,4-diamino-5-methyl-6-[(3,4,5-trimethoxy-n-methylanilino)methyl]pyrido[2,3-d]pyrimidine 2,4-diamino-6-[n-(2',5'-dimethoxybenzyl)-n-methylamino]quinazoline (2r,6s)-6-{[methyl(3,4,5-trimethoxyphenyl)amino]methyl}-1,2,5,6,7,8-hexahydroquinazoline-2,4-diamine 7-[2-methoxy-1-(methoxymethyl)ethyl]-7h-pyrrolo[3,2-f] quinazoline-1,3-diamine 5-(4-morpholin-4-yl-phenylsulfanyl)-2,4-quinazolinediamine 5-(4-methoxyphenoxy)-2,4-quinazolinediamine 5-phenylsulfanyl-2,4-quinazolinediamine 5-[4-tert-butylphenylsulfanyl]-2,4-quinazolinediamine 7-(1-ethyl-propyl)-7h-pyrrolo-[3,2-f]quinazoline-1,3-diamine 5-chloryl-2,4,6-quinazolinetriamine 5-[(4-methylphenyl)sulfanyl]-2,4-quinazolinediamine 3-{[(3-fluoro-3'-methoxybiphenyl-4-yl)amino]carbonyl}thiophene-2-carboxylic acid (2z)-n-biphenyl-4-yl-2-cyano-3-cyclopropyl-3-hydroxyprop-2-enamide 2-({[2,3,5,6-tetrafluoro-3'-(trifluoromethoxy)biphenyl-4-yl]amino}carbonyl)cyclopenta-1,3-diene-1-carboxylic acid 5-methyl-n-[4-(trifluoromethyl)phenyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine 5-carbamoyl-1,1':4',1''-terphenyl-3-carboxylic acid 3,6,9,12,15-pentaoxatricosan-1-ol (2z)-n-(3-chloro-2'-methoxybiphenyl-4-yl)-2-cyano-3-hydroxybut-2-enamide (2z)-n-biphenyl-4-yl-2-cyano-3-hydroxybut-2-enamide 3-({[3,5-difluoro-3'-(trifluoromethoxy)biphenyl-4-yl]amino}carbonyl)thiophene-2-carboxylic acid (2z)-2-cyano-n-(3'-ethoxybiphenyl-4-yl)-3-hydroxybut-2-enamide (2z)-2-cyano-n-(2,2'-dichlorobiphenyl-4-yl)-3-hydroxybut-2-enamide 2-({[3,5-difluoro-3'-(trifluoromethoxy)biphenyl-4-yl]amino}carbonyl)cyclopent-1-ene-1-carboxylic acid 2-[4-(4-chlorophenyl)cyclohexylidene]-3,4-dihydroxy-1(2h)-naphthalenone 1-guanidinium-7-aminoheptane 2,4,6-triaminoquinazoline 10-propargyl-5,8-dideazafolic acid 2-moe phosphorothioate gapmers 1-[6-(triphenylmethoxy)hexyl]thymine 1-[5-(triphenylmethoxy)pentyl]thymine 1-[(z)-4-(triphenylmethoxy)-2-butenyl]thymine (l-)-s-adenosyl-l-homocysteine 2',3'-dideoxyadenosine triphosphate (2-(2-chlorophenyl)pyridin-3-yl)methanamine (7r,8r)-8-(2,4,5-trifluorophenyl)-6,7,8,9-tetrahydroimidazo[1,2-a:4,5-c']dipyridin-7-amine (2r)-4-(2-benzoyl-1,2-diazepan-1-yl)-4-oxo-1-(2,4,5-trifluorophenyl)butan-2-amine 7-(aminomethyl)-6-(2-chlorophenyl)-1-methyl-1h-benzimidazole-5-carbonitrile 1-benzyl-4-(2,4-dichlorophenyl)pyrrolidin-3-amine 4-[(3r)-3-{[2-(4-fluorophenyl)-2-oxoethyl]amino}butyl]benzamide 2-({2-[(3r)-3-aminopiperidin-1-yl]-4-oxoquinazolin-3(4h)-yl}methyl)benzonitrile (2s,3s)-4-cyclopropyl-3-{(3r,5r)-3-[2-fluoro-4-(methylsulfonyl)phenyl]-1,2,4-oxadiazolidin-5-yl}-1-[(3s)-3-fluoropyrrolidin-1-yl]-1-oxobutan-2-amine (2r)-4-[(8r)-8-methyl-2-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[1,5-a]pyrazin-7(8h)-yl]-4-oxo-1-(2,4,5-trifluorophenyl)butan-2-amine (+/-)-6-(2-chlorophenyl)cyclohex-3-enamine (3r)-4-[(3r)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-3-methyl-1,4-diazepan-2-one 5-(aminomethyl)-6-(2,4-dichlorophenyl)-2-(3,5-dimethoxyphenyl)pyrimidin-4-amine (1s)-2-[(2s,5r)-2-(aminomethyl)-5-prop-1-yn-1-ylpyrrolidin-1-yl]-1-cyclopentyl-2-oxoethanamine (1s,2r,5s)-5-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin-7(8h)-yl]-2-(2,4,5-trifluorophenyl)cyclohexanamine 4-(2,4-dichlorophenyl)-1-phenylpyrrolidin-3-amine 2-amino-3-methyl-1-pyrrolidin-1-yl-butan-1-one 1-benzhydryl-3-butylpiperidin-4-amine (s)-2-[(r)-3-amino-4-(2-fluorophenyl)butyryl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 4-iodo-l-phenylalanine (1r,2r)-1,2-diphenylethane-1,2-diamine 3-butyl-1-(naphthalen-1-yl)piperidin-4-amine 6-(4-{(1s,2s)-2-amino-1-[(dimethylamino)carbonyl]-3-[(3s)-3-fluoropyrrolidin-1-yl]-3-oxopropyl}phenyl)-1h-[1,2,4]triazolo[1,5-a]pyridin-4-ium (s)-2-amino-1-thiazolidin-3-yl-propane-1-thione (1s)-2-[(2s,5r)-2-(aminomethyl)-5-ethynylpyrrolidin-1-yl]-1-cyclopentyl-2-oxoethanamine 1-biphenyl-2-ylmethanamine 4-(2,4-dichlorophenyl)-1-tosylpyrrolidin-3-amine (3s,4r)-3-butyl-1-phenylpiperidin-4-amine 2-(2-chlorophenyl)-2-morpholinoethanamine 4'-[(1r)-1-amino-2-(2,5-difluorophenyl)ethyl]biphenyl-3-carboxamide 2-({8-[(3r)-3-aminopiperidin-1-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7h-purin-7-yl}methyl)benzonitrile (2s,3s)-3-amino-4-[(3s)-3-fluoropyrrolidin-1-yl]-n,n-dimethyl-4-oxo-2-(trans-4-[1,2,4]triazolo[1,5-a]pyridin-5-ylcyclohexyl)butanamide (5-phenyl-3h-benzo[d]imidazol-4-yl)methanamine (2r,3r)-7-(methylsulfonyl)-3-(2,4,5-trifluorophenyl)-1,2,3,4-tetrahydropyrido[1,2-a]benzimidazol-2-amine (2s,3s)-3-{3-[4-(methylsulfonyl)phenyl]-1,2,4-oxadiazol-5-yl}-1-oxo-1-pyrrolidin-1-ylbutan-2-amine 1-[2-(s)-amino-3-biphenyl-4-yl-propionyl]-pyrrolidine-2-(s)-carbonitrile (3r,4s)-1-[6-(6-methoxypyridin-3-yl)pyrimidin-4-yl]-4-(2,4,5-trifluorophenyl)pyrrolidin-3-amine (3r,4r)-4-(pyrrolidin-1-ylcarbonyl)-1-(quinoxalin-2-ylcarbonyl)pyrrolidin-3-amine 7-benzyl-1,3-dimethyl-8-piperazin-1-yl-3,7-dihydro-purine-2,6-dione (2r)-n-[(2r)-2-(dihydroxyboryl)-1-l-prolylpyrrolidin-2-yl]-n-[(5r)-5-(dihydroxyboryl)-1-l-prolylpyrrolidin-2-yl]-l-prolinamide 4-iodophenyl-alaninyl-(s)-2-cyano-pyrrolidine 1-(1-phenylcyclopentyl)methylamine (3r,4s)-1-{6-[3-(methylsulfonyl)phenyl]pyrimidin-4-yl}-4-(2,4,5-trifluorophenyl)pyrrolidin-3-amine (s)-2-amino-1-azetidin-1-yl-2-cyclohexyl-ethanone (2s)-pyrrolidin-2-ylmethylamine (s)-pyrrolidin-2-yl(thiazolidin-3-yl)methanone (4r,5r)-5-amino-1-[2-(1,3-benzodioxol-5-yl)ethyl]-4-(2,4,5-trifluorophenyl)piperidin-2-one (1r,2s)-1,2-diphenylethane-1,2-diamine (3r,4s)-1-(3,4-dimethoxyphenyl)-3-(3-methylphenyl)piperidin-4-amine (1-phenylcyclopentyl)methanamine (3r,4r)-1-{6-[3-(methylsulfonyl)phenyl]pyrimidin-4-yl}-4-(2,4,5-trifluorophenyl)piperidin-3-amine (2s,3s)-3-{3-[2-chloro-4-(methylsulfonyl)phenyl]-1,2,4-oxadiazol-5-yl}-1-cyclopentylidene-4-cyclopropyl-1-fluorobutan-2-amine (2-chloro-6-phenoxyphenyl)methanamine (s)-pyrrolidin-1-yl(pyrrolidin-2-yl)methanone 4-[(3r)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-3-(2,2,2-trifluoroethyl)-1,4-diazepan-2-one (1s,3s,5s)-2-{(2s)-2-amino-2-[(1r,3s,5r,7s)-3-hydroxytricyclo[3.3.1.1~3,7~]dec-1-yl]acetyl}-2-azabicyclo[3.1.0]hexane-3-carbonitrile (2s,3s)-3-amino-4-(3,3-difluoropyrrolidin-1-yl)-n,n-dimethyl-4-oxo-2-(trans-4-[1,2,4]triazolo[1,5-a]pyridin-6-ylcyclohexyl)butanamide (r)-1-(2-aminoacetyl)pyrrolidin-2-ylboronic acid 1g244 (5s)-5-iododihydro-2,4(1h,3h)-pyrimidinedione 5-iodouracil 6-carboxymethyluracil 1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1-benzyl-4-(2-iodo-pyrrol-1-yl)-piperidine 3-chloroboldine (r,s)-homoaromaline hydrochloride (r)-(-)-11-hydroxy-n-n-propylnoraporphine (+)-(1r,1's)-berbamunine hydrochloride (r)-(-)-n-ethyl-2-methoxy-11-hydroxynoraporphine 1-[2-(2-benzyl-phenoxy)-ethyl]-pyrrolidine 2-methoxyapomorphine (s)-bulbocapnine (+)-adtn (r)-2,11-diaminoaporphine 4-[2-(2-benzyl-phenoxy)-ethyl]-morpholine 1-(4-(1h-pyrazol-1-yl)benzyl)-4-phenylpiperazine 9-aminomethyl-9h-fluorene-2,5,6-triol 2-{[r-(-)-apomorphine-2'-oxy]ethoxy}-ethanol 1-aminomethyl-3-cyclohexyl-isochroman-5,6-diol (s,s)-oxandrine hydrochloride 11-hexanoyloxy-n-n-propylnoraporphine 1-benzyl-4-(2-ethynyl-pyrrol-1-yl)-piperidine 9-aminomethyl-9h-fluorene-3,4-diol (r)-(+)-coclaurine 1-aminomethyl-3-phenyl-isochroman-5,6-diol 1,2-bis-[r-(-)-apomorphine-2'-oxy]ethane (r)-(-)-10-methyl-11-hydroxyaporphine 1-aminomethyl-isochroman-5,6-diol (r)-11-amino-2-methoxyaporphine 6-(2-dipropylamino-ethyl)-biphenyl-2,3,4'-triol 11-propionyloxy-n-n-propylnoraporphine 1-[2-(2-benzyl-phenoxy)-ethyl]-piperidine (s)apomorphine 1-[3-(2-benzyl-phenoxy)-propyl]-pyrrolidine 1-dibenzo[b,f]oxepin-10-yl-4-methyl-piperazine (-)-(1s,1'r)-o,o-dimethylgrisbine hydrochloride 6-(2-amino-ethyl)-biphenyl-2,3-diol 6-(2-amino-ethyl)-biphenyl-2,3,4'-triol 3-iodoboldine 11-butyryloxy-n-n-propylnoraporphine 11-heptanoyloxy-n-n-propylnoraporphine 1-benzyl-4-(2-oxazol-5-yl-pyrrol-1-yl)-piperidine 2-methyl-8-phenyl-1,2,3,4-tetrahydro-isoquinoline (r)-(-)-2-methoxy-11-hydroxyaporphine 6-(2-dipropylamino-ethyl)-biphenyl-2,3-diol [125i]sch23982 (r)-(-)-n-propyl-2-methoxy-11-hydroxynoraporphine (+)-(1r,1's)-thaligrisine hydrochloride 5-(2-amino-ethyl)-2-chloro-phenol hydrobromide (r)-(-)-2-methoxy-n-npropylnorapomorphine [r-(-)-apomorphine-2-yl]-(2'-hydroxy-ethyl)ether 11-valeryloxynoraporphine 1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 2-{[2-(2-phenylethyl)phenoxy]methyl}pyridine 3-(3,5-dimethyl-phenyl)-piperidine 1-propyl-3-p-tolyl-piperidine hydrochloride 3-naphthalen-1-yl-1-propyl-pyrrolidine 3-(2,3-dimethyl-phenyl)-piperidine (4-ethynyl-cyclohex-3-enyl)-dipropyl-amine 3-butyl-2,3,4,5-tetrahydro-1h-benzo[d]azepin-6-ol [3h]n-methylspiperone 3-(4-phenyl-piperidin-1-ylmethyl)-1h-indole 7-(2-dipropylamino-ethyl)-3h-benzothiazol-2-one 3-(3,4-dimethyl-phenyl)-1-propyl-piperidine (r)-(-)-2-phenyl-apomorphine hydrochloride 3-(4-benzyl-piperazin-1-yl)-phenol 2,3-dihydro-1h-indol-5-ol 1-propyl-3-m-tolyl-piperidine hydrochloride (+)-s-14297 5-oh-dpat (s,r)-pseudoxandrine hydrochloride (5-methoxy-chroman-3-yl)-dipropyl-amine 1-benzyl-4-[3-(methylsulfonyl)phenyl]piperazine 1-benzyl-4-pyrrol-1-yl-piperidine 3-phenyl-1-propyl-pyrrolidine (s,r)-antioquine hydrochloride 3-(3,5-dimethyl-phenyl)-1-propyl-piperidine 1,6-bis(4-m-tolylpiperazin-1-yl)hexane (s,r)-isotetrandrine hydrochloride (s)-secoantioquine hydrochloride 3-(octahydro-quinolizin-3-yl)-phenol 1-(benzyloxy)-2-[2-(3-methoxyphenyl)ethyl]benzene 7-trans-oh-pipat [3h]7-oh-dpat 4-(2-benzylamino-ethoxy)-1,3-dihydro-indol-2-one 4-benzyl-1-chroman-3-ylmethyl-piperidine 2-(4-dipropylamino-cyclohexylidene)-malononitrile 3-(4-phenyl-piperazin-1-ylmethyl)-1h-indole 1,6-bis(4-(3-methoxyphenyl)piperazin-1-yl)hexane 3-(2,6-dimethyl-phenyl)-1-propyl-piperidine 1-[(3-methoxybenzyl)oxy]-2-(2-phenylethyl)benzene 3-(4-methyl-piperidin-1-ylmethyl)-1h-indole 4-(4-benzyl-piperazin-1-yl)-1h-benzoimidazole (r)-(-)-2-methyl-apomorphine hydrochloride 3-phenyl-1-propyl-piperidine hydrochloride 1-propyl-3-(3-trifluoromethyl-phenyl)-pyrrolidine [2-(1h-benzoimidazol-4-yloxy)-ethyl]-benzyl-amine 4-(4-benzyl-piperazin-1-yl)-5-chloro-1h-indole 3-phenyl-pyrrolidine 3-(2,3-dimethyl-phenyl)-1-propyl-piperidine 1-[3-(methylsulfonyl)phenyl]-4-propylpiperazine 1-(3-hydroxyphenyl)-4-propylpiperazine 1-(benzyloxy)-2-(2-phenylethyl)benzene 3-(1-propyl-pyrrolidin-3-yl)-phenol 3-(2,4-dimethyl-phenyl)-1-propyl-piperidine (-)-3-(1-propyl-piperidin-3-yl)-benzonitrile 1-methyl-1,2,3,4-tetrahydro-isoquinoline-6,7-diol 3-(octahydro-indolizin-8-yl)-phenol 1,6-bis(4-(3-chlorophenyl)piperazin-1-yl)hexane 3-ethyl-2,3,4,5-tetrahydro-1h-benzo[d]azepin-6-ol 1,6-bis(4-(pyridin-2-yl)piperazin-1-yl)hexane 3-naphthalen-1-yl-pyrrolidine 4-(4-benzyl-piperazin-1-yl)-7-bromo-1h-indole 1-benzyl-4-[3-(methylsulfonyl)phenyl]piperidine 7-(2-amino-ethyl)-4-hydroxy-3h-benzothiazol-2-one 3-(octahydro-quinolizin-1-yl)-phenol 3-(2-benzylamino-ethoxy)-phenol 1-(4-(4-phenyl-1-piperazinyl)butyl)indolin-2-one (-)-3ppp, maryland 3-(n-propylpiperidin-4-yl)phenol (4-quinolin-2-ylpiperazin-1-yl)acetic acid (s)-amisulpride 4-(4-benzyl-piperazin-1-yl)-1h-indole 3-(3,4-dimethyl-phenyl)-piperidine 3-cyclohexyl-1-propyl-piperidine hydrochloride 3-(2,5-dimethyl-phenyl)-1-propyl-piperidine 3-{[2-(2-phenylethyl)phenoxy]methyl}pyridine 3-(4-benzyl-piperidin-1-ylmethyl)-chroman-4-one 1-propyl-3-o-tolyl-piperidine hydrochloride 4-benzyl-1-indan-2-ylmethyl-piperidine 1,6-bis(4-phenylpiperazin-1-yl)hexane 1-benzyl-4-(3-hydroxyphenyl)piperidine 4-benzyl-1-chroman-2-ylmethyl-piperidine 1192u90 1-benzyl-4-(3-oxazol-5-yl-pyrrol-1-yl)-piperidine (r)-2-(benzylamino-methyl)-chroman-7-ol (+)-aj76 (4-phenylethynyl-cyclohex-3-enyl)-dipropyl-amine (4-dipropylamino-cyclohexylidene)-acetonitrile 4-dipropylamino-cyclohex-1-enecarbonitrile (2-benzyl-phenyl)-(2-pyrrolidin-1-yl-ethyl)-amine [125i]l750667 2',3'-dideoxythymidine-5'-monophosphate 3'-fluoro-3'-deoxythymidine 5'-monophosphate 3'-deoxy-3'-aminothymidine monophosphate 1-{(2s,5s)-4-fluoro-5-[(trityloxy)methyl]tetrahydrofuran-2-yl}pyrimidine-2,4(1h,3h)-dione 5-(2-hydroxyethyl)nonane-1,9-diol 4-(n,n-dimethylamino)cinnamoyl-coa 97-139 [125i]pd151242 [3h]bq123 [3h]s0139 [125i]irl1620 (s)-benzyl 4-chloro-3-oxobutan-2-ylcarbamate (3-bromo-phenyl)-quinazolin-4-yl-amine 5-acrylamido-n-(3-bromophenyl)-2-hydroxybenzamide 4-(3-bromo-phenoxy)-6,7-dimethoxy-quinoline 5,6-bis-p-tolylamino-isoindole-1,3-dione 6-chloro-n-(3-chlorophenyl)quinazolin-4-amine 111in-hegf (e)-5-(4-hydroxybenzylidene)-1-phenethylhydantoin 6,7-dimethoxy-4-(2-phenylethynyl)quinazoline 4-(2-nitroprop-1-enyl)benzene-1,2-diol 4-biphenyl-2-ylethynyl-6,7-dimethoxy-quinazoline 6,7-dimethoxy-4-(4-phenylbut-1-ynyl)quinazoline 4-(2-nitrovinyl)benzene-1,2-diol 4-(3-bromo-phenylamino)-quinazoline-6,7-diol (3-bromo-phenyl)-(5-nitro-quinazolin-4-yl)-amine 4557w 4-(4-(2-nitrovinyl)phenoxysulfonyl)benzoic acid 6,7-dimethoxy-4-(3-phenoxyprop-1-ynyl)quinazoline 2-cyano-3-(3,4-dihydroxyphenyl)acrylamide 4-(3-bromo-phenoxy)-6,7-dimethoxy-quinazoline 4-(5-bromoindole-3-yl)-6,7-dimethoxyquinazoline 6,7-dimethoxy-n-m-tolylquinazolin-4-amine 2-(5,6-dihydroxy-indan-1-ylidene)-malononitrile 6,7-diethoxy-4-(5-phenylpent-1-enyl)quinazoline 4-(2-nitrovinyl)phenol 4-acrylamido-n-(3-bromophenyl)-2-hydroxybenzamide 6,7-diethoxy-4-styrylquinazoline 6,7-diethoxy-4-(4-phenylbut-1-enyl)quinazoline 3-pyridin-4-yl-quinoline-6,7-diol 2-benzoyl-3-(3,4-dihydroxyphenyl)acrylonitrile 2-methoxy-4-(2-nitrovinyl)phenol 3-(3-chloro-phenyl)-5,7-dihydroxy-chromen-4-one 2-(4,5-dihydroxy-indan-1-ylidene)-malononitrile 2-(carboxymethylamino)-2-oxoacetic acid 7n-methyl-8-hydroguanosine-5'-diphosphate 7-methyl-guanosine-5'-triphosphate 6-heptyl-4-hydroxy-3-octanoyl-pyran-2-one (4-nitro-1h-pyrazol-1-yl)(o-tolyl)methanone 3,3-diethyl-1-o-tolylazetidine-2,4-dione 2-pyrazinone derivative 4 4-pyridone derivative 1 2-pyrazinone derivative 3 1-benzyl-3,3-dimethylazetidine-2,4-dione 2-pyrazinone derivative 7 (4-bromo-1h-pyrazol-1-yl)(o-tolyl)methanone 4-pyridone derivative 2 (4-nitro-1h-pyrazol-1-yl)(phenyl)methanone 2-pyrazinone derivative 6 (4-bromo-1h-pyrazol-1-yl)(p-tolyl)methanone 3-butyl-3-ethyl-1-phenylazetidine-2,4-dione (3-nitro-1h-pyrazol-1-yl)(p-tolyl)methanone 2-pyrazinone derivative 5 3,3-diethyl-1-phenylazetidine-2,4-dione 1-benzyl-3,3-diethylazetidine-2,4-dione (3-nitro-1h-pyrazol-1-yl)(phenyl)methanone 2-methylbut-3-yn-2-yl 4-methoxybenzoate 1-(3,3-dimethyl-2-oxo-butyl)-1h-indole-2,3-dione 2-pyrazinone derivative 1 4-hydroxy-3-nonanoyl-6-octyl-pyran-2-one 3-ethyl-3-isobutyl-1-phenylazetidine-2,4-dione 3-benzyl-3-ethyl-1-phenylazetidine-2,4-dione (4-chloro-1h-pyrazol-1-yl)(o-tolyl)methanone 3-decanoyl-4-hydroxy-6-nonyl-pyran-2-one 4-methoxy-n'-(2-phenylacetyl)benzohydrazide 1-benzoyl-n-phenyl-1h-pyrazole-3-carboxamide (4-bromo-1h-pyrazol-1-yl)(m-tolyl)methanone 3,3-diethyl-1-(pyridin-3-yl)azetidine-2,4-dione (3,4-dichlorophenyl)(1h-pyrazol-1-yl)methanone (1h-pyrazol-1-yl)(o-tolyl)methanone 2-pyrazinone derivative 2 3-benzyl-3-methyl-1-phenylazetidine-2,4-dione 2-phosphoglycolic acid 2-phospho-d-glyceric acid 2-oxoheptylphosphonic acid 5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamide 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamide 1-adamantan-1-yl-3-(3-hydroxypropyl)urea 6-{[(cyclohexylamino)carbonyl]amino}hexanoic acid 13-(3-n-pentylureido)tridec-5(z)-enoic acid 1-adamantan-1-yl-3-((r)-1-phenyl-ethyl)-urea 1-adamantan-1-yl-3-(4-pentyloxybutyl)urea 13-(3-n-pentylureido)tridec-8(e)-enoic acid 1-adamantan-1-yl-3-(1-butyl-piperidin-4-yl)-urea 1-adamantan-1-yl-3-piperidin-4-yl-urea 13-(n-isopropylheptanamido)tridec-8(z)-enoic acid 13-(3-n-pentylureido)tridec-8-ynoic acid 1-phenyl-3-(1-propionylpiperidin-4-yl)urea 1-adamantan-1-yl-3-(2-methoxy-phenyl)-urea 9-(3-n-pentylureido)non-4(z)-enoic acid 2-cyclohexyl-n-phenethyl-acetamide 1-adamantan-1-yl-3-(4-methoxy-phenyl)-urea 1-adamantan-1-yl-3-(4-hydroxy-decyl)-urea 2-cyclohexyl-n-(4-methoxy-phenyl)-acetamide 1-cycloheptyl-3-(1-propionylpiperidin-4-yl)urea 1-cyclohexyl-3-(4-methoxy-phenyl)-urea 1-adamantan-1-yl-3-(5-hydroxypentyl)urea 1-adamantan-1-yl-3-(3-hexyloxypropyl)urea 13-(3-n-pentylthioureido)tridec-8(z)-enoic acid 9-(3-n-pentylureido)non-4-ynoic acid 13-(5-n-pentylfuran-2-yl)tridec-8(z)-enoic acid 4-(3-cyclohexylureido)butanoic acid 1-cyclohexyl-3-(1-propionylpiperidin-4-yl)urea 1-adamantan-1-yl-3-phenyl-urea 1-(3-chloro-phenyl)-3-cyclohexyl-urea 1-adamantan-1-yl-3-decyl-urea 1-(3-(3-morpholinopropoxy)phenyl)-3-phenylurea 1-adamantan-1-yl-3-(6-hydroxyhexyl)urea 16-(3-ethylureido)hexadec-11(z)-enoic acid 4-{[(cyclohexylamino)carbonyl]amino}butanoic acid 13-(3-pentyluredo)tridec-8(z)-enoic acid 1-adamantan-1-yl-3-(3-methoxy-phenyl)-urea 1-adamantan-1-yl-3-(2-hydroxy-phenyl)-urea 1-adamantan-1-yl-3-(1-benzyl-piperidin-4-yl)-urea 1-adamantan-1-yl-3-[4-(4-fluorophenoxy)butyl]urea 6-amino-n-(2,4-dichlorobenzyl)nicotinamide 4,4-diphenyl-n-(pyridin-3-yl)-butyramide 13-(n-methyl-n-heptnamido)tridec-8(z)-enoic acid 1-adamantan-1-yl-3-piperidin-4-ylmethyl-urea 1-(1-propionylpiperidin-4-yl)-3-p-tolylurea 1,3-diphenylurea 1-adamantan-1-yl-3-(2-hydroxyethyl)urea 12-(3-adamantan-1-yl-ureido)-dodeca noic acid 1-adamantan-1-yl-3-(4-hydroxybutyl)urea [4-(3-adamantan-1-yl-ureido)-phenyl]-acetic acid 1-(3-chloro-phenyl)-3-(4-hydroxy-decyl)-urea 1-(4-(3-morpholinopropoxy)phenyl)-3-phenylurea 1-(1-propionylpiperidin-4-yl)-3-m-tolylurea 1-adamantan-1-yl-3-(1-propyl-piperidin-4-yl)-urea 14-(n-hexylamino)-14-oxotetradec-8(z)-enoic acid 1-(1-adamantyl)-3-(1-propionylpiperidin-4-yl)urea 3-(3-adamantan-1-yl-ureido)-benzoic acid 1-adamantan-1-yl-3-(5-butoxypentyl)urea 13-(n-pentylcarbamoyloxy)tridec-8(z)-enoic acid 1-cyclohexyl-3-phenyl-urea 2-cyclohexyl-n-phenyl-acetamide 1-adamantan-1-yl-3-(6-propyloxyhexyl)urea 7-{[(cyclohexylamino)carbonyl]amino}heptanoic acid 2-adamantan-1-yl-n-decyl-acetamide 6-amino-n-(3,3-diphenylpropyl)nicotinamide 1-(1-propionylpiperidin-4-yl)-3-o-tolylurea 1-adamantan-1-yl-3-(1-ethyl-piperidin-4-yl)-urea 12-(3-n-pentylureidooxy)dodec-8(z)-enoic acid 1-adamantan-1-yl-3-(4-hydroxy-phenyl)-urea 1-adamantan-1-yl-3-(3-hydroxy-phenyl)-urea 12-(3-n-hexylureido)dodec-8(z)-enoic acid 1-adamantan-1-yl-3-(2-heptyloxyethyl)urea 13-n-heptanamidotridec-8(z)-enoic acid 4-(3-adamantan-1-yl-ureido)-benzoic acid 13-n-heptanamidotridec-5-ynoic acid 1-cyclohexyl-3-phenethyl-urea 1-adamantan-1-yl-3-(4-pentyloxycylclohexyl)urea 1-octyl-3-(1-propionylpiperidin-4-yl)urea 1,4-dioxane 3,5 dibromotyrosine 5'-o-(l-prolylsulfamoyl)adenosine 5'-o-(n-(alanyl)sulfamoyl)adenosine 5'-o-(l-cysteinylsulfamoyl)adenosine 227th-labelled her2-ttc 4-(4-isopropylphenyl)-5-cyano-2h-1,2,3-triazole (1-benzyl-1h-indazol-5-yl)-quinazolin-4-yl-amine 4-(4-chlorophenyl)-5-cyano-2h-1,2,3-triazole 4-(3-phenoxylphenyl)-5-cyano-2h-1,2,3-triazole 4-(4-bromophenyl)-5-cyano-2h-1,2,3-triazole (1-benzyl-1h-indol-5-yl)-quinazolin-4-yl-amine 4-(bis(2-chloroethyl)amino)-n-p-tolylbenzamide 1-ethyl-pyrrolidine-2,5-dione 4-chloro-2-(4-hydroxy-phenyl)-quinolin-6-ol 6-phenyl-naphthalen-2-ol 1-bromo-6-(4-hydroxy-phenyl)-naphthalen-2-ol 2,3-diphenyl-1h-indole 4-(5-hydroxy-benzooxazol-2-yl)-benzene-1,3-diol 1,8-dichloro-6-(4-hydroxy-phenyl)-naphthalen-2-ol 3-[1-ethyl-2-(3-hydroxyphenyl)butyl]phenol 3,8-dihydroxy-4-methyl-6h-benzo[c]chromen-6-one [5-hydroxy-2-(4-hydroxyphenyl)-1-benzofuran-7-yl]acetonitrile 2-(5-hydroxy-naphthalen-1-yl)-benzooxazol-6-ol 4-[(1s,2s,5s)-5-(hydroxymethyl)-6,8,9-trimethyl-3-oxabicyclo[3.3.1]non-7-en-2-yl]phenol 8-(3-methylbutyl)naringenin 2-(4-hydroxyphenyl)-1,2'-spirobi[1h-indene]-5-ol 2-(4-hydroxy-phenyl)-benzooxazol-6-ol 2-(3-fluoro-4-hydroxy-phenyl)-benzooxazol-6-ol 6-(4-hydroxy-2-methyl-phenyl)-naphthalen-2-ol 4-(7-chloro-1-cyclopentyl-1h-indazol-3-yl)phenol 3-(4-hydroxyphenyl)-7-isopropoxychromen-4-one 4-(1-cyclopentyl-7-fluoro-1h-indazol-3-yl)phenol 4-hydroxy-n-isopropyl-n-phenylbenzenesulfonamide 2-(4-hydroxy-phenyl)-quinolin-6-ol 4-hydroxy-n-neopentyl-n-phenylbenzenesulfonamide 6-ethyl-2,4-diisobutylaminopyrimidine 4,7-dimethyl-6h-benzo[c]chromene-3,8-diol 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine 4-[(1s,2s,5s,9r)-5-(hydroxymethyl)-8,9-dimethyl-3-oxabicyclo[3.3.1]non-7-en-2-yl]phenol 17-methyl-17-alpha-dihydroequilenin 5-bromo-2-(4-hydroxy-phenyl)-quinolin-6-ol 4-[1,2-bis(4-hydroxyphenyl)vinyl]phenol 2-(3-hydroxyphenyl)-1,2'-spirobi[1h-indene]-6-ol 1-[4-(octahydro-pyrido[1,2-a]pyrazin-2-yl)-phenyl]-2-phenyl-1,2,3,4-tetrahydro-isoquinolin-6-ol 7-phenyl-naphthalen-2-ol 8-n-nonylnaringenin 2-(4-hydroxy-phenyl)-7-methoxy-benzooxazol-5-ol 3-chloro-4-(4-hydroxyphenyl)salicylaldoxime 8-n-heptylnaringenin (9beta,11alpha,13alpha,14beta,17alpha)-11-(methoxymethyl)estra-1(10),2,4-triene-3,17-diol 7-butyl-2-(4-hydroxy-phenyl)-benzooxazol-5-ol (2r,3r,4s)-3-(4-hydroxyphenyl)-4-methyl-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]chroman-6-ol 6-(4-hydroxy-phenyl)-1-nitro-naphthalen-2-ol 6-(4-hydroxy-phenyl)-1-methoxy-naphthalen-2-ol 5-hydroxy-2-phenylisoindoline-1,3-dione 4,6,7-trimethyl-6h-benzo[c]chromene-3,8-diol 2-(4-hydroxy-phenyl)-benzooxazol-5-ol 4-(6-hydroxy-1h-indazol-3-yl)benzene-1,3-diol 2-phenyl-1-[4-(2-piperidin-1-yl-ethoxy)-phenyl]-1,2,3,4-tetrahydro-isoquinolin-6-ol 2-(4-hydroxy-phenyl)-7-propyl-benzooxazol-5-ol 4',5,7-trihydroxy-6,8-dimethylisoflavone 4-[1,2-bis(4-hydroxyphenyl)hex-1-enyl]phenol 3-hydroxy-8,10-dimethyl-6h-benzo[c]chromen-6-one 7-ethynyl-2-(4-hydroxy-phenyl)-benzooxazol-5-ol 4-(2-amino-1-methyl-1h-imidazo[4,5-b]pyridin-6-yl)phenol (9alpha,13beta,17beta)-2-[(1z)-but-1-en-1-yl]estra-1,3,5(10)-triene-3,17-diol 4-(1-butyl-7-chloro-1h-indazol-3-yl)phenol 4-[(1s,2r,5s)-4,4,8-trimethyl-3-oxabicyclo[3.3.1]non-7-en-2-yl]phenol 3-(4-hydroxyphenyl)-7-isobutoxychromen-4-one 3-(2-hydroxy-phenyl)-benzo[d]isoxazol-6-ol 3-ethyl-2-(4-hydroxyphenyl)-2h-indazol-5-ol 2-(4-hydroxyphenyl)benzo[b]thiophen-6-ol 6-(4-hydroxy-phenyl)-1-methyl-naphthalen-2-ol 4-(2-phenyl-1h-indol-3-yl)phenol 2-(4-hydroxy-phenyl)-7-methyl-benzofuran-5-ol 2-(6-hydroxy-naphthalen-2-yl)-benzooxazol-5-ol 4-naphthalen-2-yl-phenol 4-[1-(4-hydroxyphenyl)-2-phenylvinyl]phenol 4-[(1s,2s,5s)-5-(hydroxymethyl)-8-methyl-3-oxabicyclo[3.3.1]non-7-en-2-yl]phenol 6-(2-chloro-4-hydroxy-phenyl)-naphthalen-2-ol 4-(7-methyl-1-propyl-1h-indazol-3-yl)phenol 4-hydroxy-n-phenyl-n-propylbenzenesulfonamide 2-phenyl-1,2'-spirobi[1h-indene]-5'-ol 6-chloro-2-(4-hydroxy-phenyl)-benzooxazol-5-ol 3-chloro-2-(4-hydroxyphenyl)-2h-indazol-5-ol 4-benzo[d]isoxazol-3-yl-benzene-1,3-diol 2-(3-chloro-4-hydroxy-phenyl)-benzooxazol-5-ol 4-[2,2-bis(4-hydroxyphenyl)-1-methylvinyl]phenol 8-n-undecylnaringenin 7-allyl-2-(4-hydroxy-phenyl)-benzooxazol-5-ol 4-[1-(4-hydroxyphenyl)-2-phenylprop-1-enyl]phenol 3'-methoxy-4'hydroxyclomiphene 2-(3-butoxy-4-hydroxy-phenyl)-benzooxazol-6-ol 4-hydroxy-n,n-diphenylbenzenesulfonamide 3-(5-hydroxy-benzooxazol-2-yl)-benzene-1,2-diol 7-(4-hydroxy-phenyl)-naphthalen-2-ol 6-ethyl-4,7-dimethyl-6h-benzo[c]chromene-3,8-diol 4-[1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenol 3-(4-hydroxy-phenyl)-benzo[d]isoxazol-5-ol 4,10-dimethyl-6h-benzo[c]chromene-3,8-diol 6-(3-hydroxy-phenyl)-naphthalen-1-ol 2-amino-1-methyl-6-phenylimidazo(4,5-b)pyridine 6-(3-fluoro-4-hydroxy-phenyl)-naphthalen-2-ol 8-n-pentylnaringenin 3,8-dihydroxy-7-methyl-6h-benzo[c]chromen-6-one 7-chloro-2-(4-hydroxy-phenyl)-benzofuran-5-ol 2-(3-hydroxyphenyl)-1,2'-spirobi[1h-indene]-5-ol 4-benzyl-2,6-diisobutylamino-pyrimidine 2-(4-hydroxy-phenyl)-7-methoxy-benzofuran-5-ol 6-(3-chloro-4-hydroxy-phenyl)-naphthalen-2-ol 2-(4-hydroxy-naphthalen-1-yl)-benzooxazol-6-ol 4-(7-chloro-1-cyclohexyl-1h-indazol-3-yl)phenol 6-(4-hydroxy-2-methoxy-phenyl)-naphthalen-2-ol 2-(6-hydroxy-naphthalen-2-yl)-benzooxazol-6-ol 2-(4-hydroxy-phenyl)-7-phenyl-benzooxazol-5-ol 8-(2-methylpropyl)naringenin 2-(4-hydroxy-phenyl)-4-methoxy-quinolin-6-ol 3-(6-hydroxy-benzooxazol-2-yl)-benzene-1,2-diol (3as,4r,9br)-2,2-difluoro-4-(4-hydroxyphenyl)-1,2,3,3a,4,9b-hexahydrocyclopenta[c]chromen-8-ol 4-[1-(4-hydroxyphenyl)-2-phenylhex-1-enyl]phenol 4-(7-chloro-1-propyl-1h-indazol-3-yl)phenol 1,2-bis-(4-hydroxy-phenyl)-3h-inden-5-ol 6-(2,6-difluoro-4-hydroxy-phenyl)-naphthalen-2-ol (3as,4r,9br)-4-(4-hydroxyphenyl)-6-(methoxymethyl)-1,2,3,3a,4,9b-hexahydrocyclopenta[c]chromen-8-ol 8-(2,2-dimethylpropyl)naringenin 7-bromo-2-(4-hydroxy-phenyl)-benzofuran-5-ol 1-fluoro-6-(4-hydroxy-phenyl)-naphthalen-2-ol [1,1':2',1'']terphenyl-4'-carbaldehyde oxime 2,4-diisobutylamino-6-isopentylpyrimidine 8-fluoro-6-(4-hydroxy-phenyl)-naphthalen-2-ol 4-[1-allyl-7-(trifluoromethyl)-1h-indazol-3-yl]benzene-1,3-diol 7-ethyl-2-(4-hydroxy-phenyl)-benzooxazol-5-ol 2-(4-hydroxy-phenyl)-4-vinyl-quinolin-6-ol 6-(4-hydroxy-phenyl)-naphthalen-1-ol 6-(4-hydroxy-phenyl)-naphthalen-2-ol 3-(4-hydroxy-phenyl)-benzo[d]isoxazol-6-ol 6-butyl-2,4-dipropylaminopyrimidine 4-(1-benzyl-7-chloro-1h-indazol-3-yl)phenol 4-[1,2-bis(4-hydroxyphenyl)but-1-enyl]phenol 4,6,10-trimethyl-6h-benzo[c]chromene-3,8-diol 4-(3-phenyl-1h-indol-2-yl)phenol 7-(3-hydroxy-phenyl)-naphthalen-2-ol 6-(2,5-difluoro-4-hydroxy-phenyl)-naphthalen-2-ol 4-(2-phenyl-1h-benzo[d]imidazol-1-yl)phenol 8-n-propylnaringenin 2-(3-chloro-4-hydroxy-phenyl)-benzooxazol-6-ol 4-bromo-2-(4-hydroxy-phenyl)-quinolin-6-ol 6-(3,5-difluoro-4-hydroxy-phenyl)-naphthalen-2-ol 5-chloro-2-(4-hydroxy-phenyl)-quinolin-6-ol 2-methoxy-6-{(e)-[(4-methylphenyl)imino]methyl}phenol (3as,4r,9br)-4-(4-hydroxyphenyl)-1,2,3,3a,4,9b-hexahydrocyclopenta[c]chromen-9-ol 2-(4-hydroxy-phenyl)-7-propenyl-benzooxazol-5-ol 4,6,7,10-tetramethyl-6h-benzo[c]chromene-3,8-diol 7-cyclopentyloxy-3-(4-hydroxyphenyl)chromen-4-one 4,6,6,7-tetramethyl-6h-benzo[c]chromene-3,8-diol 8-chloro-6-(4-hydroxy-phenyl)-naphthalen-2-ol 2-naphthalen-1-yl-benzooxazol-6-ol 2-(2-chloro-4-hydroxy-phenyl)-benzooxazol-5-ol 4-ethyl-2-(4-hydroxy-phenyl)-quinolin-6-ol 8-methylnaringenin 1-chloro-6-(4-hydroxyphenyl)-2-naphthol 2-(6-hydroxy-naphthalen-1-yl)-benzooxazol-6-ol 6-(4-hydroxy-phenyl)-1-phenyl-naphthalen-2-ol 2-(3-fluoro-4-hydroxy-phenyl)-benzooxazol-5-ol 2-(6-hydroxy-naphthalen-1-yl)-benzooxazol-5-ol 8-benzylnaringenin 4-(3-(4-hydroxyphenyl)-1h-indol-2-yl)phenol 4-(6-hydroxy-benzooxazol-2-yl)-benzene-1,3-diol 2,4-dibenzylamino-6-isopentylpyrimidine 4-(6-hydroxy-benzooxazol-2-yl)-benzene-1,2-diol 4-ethynyl-2-(4-hydroxy-phenyl)-quinolin-6-ol 2-(4-hydroxy-phenyl)-7-isopropyl-benzooxazol-5-ol 2-(4-hydroxy-phenyl)benzofuran-5-ol 5-chloro-2-(4-hydroxy-phenyl)-benzooxazol-6-ol 4-(1,2-diphenyl-but-1-enyl)-phenol 4-[1-(4-hydroxyphenyl)-2-phenylpent-1-enyl]phenol 2-(4-hydroxy-phenyl)-7-vinyl-benzooxazol-5-ol 4-[1,2-bis(4-hydroxyphenyl)pent-1-enyl]phenol 6-(2-fluoro-4-hydroxy-phenyl)-naphthalen-2-ol 3,4,6-trihydroxy-2-(4-hydroxy-phenyl)-inden-1-one (3as,4r,9br)-2,2-difluoro-4-(4-hydroxyphenyl)-6-(methoxymethyl)-1,2,3,3a,4,9b-hexahydrocyclopenta[c]chromen-8-ol 4-(6-hydroxy-benzo[d]isoxazol-3-yl)benzene-1,3-diol 3-hydroxy-4,7-dimethyl-6h-benzo[c]chromen-6-one 5,7-dihydroxy-3-phenyl-3h-quinazolin-4-one 3,6-dihydroxy-2-(4-hydroxy-phenyl)-inden-1-one 5-alpha-androstane-3-beta,17beta-diol 4-(4-hydroxyphenyl)-1-naphthaldehyde oxime 3-bromo-6-hydroxy-2-(4-hydroxyphenyl)-1h-inden-1-one 2-(5-hydroxy-naphthalen-1-yl)-1,3-benzooxazol-6-ol 3-hydroxy-4,10-dimethyl-6h-benzo[c]chromen-6-one 2-(4-hydroxy-phenyl)-1-p-tolyl-3h-inden-5-ol 3-(4-hydroxy-phenyl)-4h-chromen-7-ol 17alpha-estriol 4-(2-{[4-{[3-(4-chlorophenyl)propyl]sulfanyl}-6-(1-piperazinyl)-1,3,5-triazin-2-yl]amino}ethyl)phenol 5-hydroxy-2-(4-hydroxyphenyl)-1-benzofuran-7-carbonitrile 3-hydroxy-4-methyl-6h-benzo[c]chromen-6-one 3-(6-hydroxy-naphthalen-2-yl)-benzo[d]isooxazol-6-ol 7-hydroxy-3-(4-hydroxyphenyl)-3h-quinazolin-4-one 6-(2-hydroxy-phenyl)-naphthalen-2-ol 7-hydroxy-1,2,9,9a-tetrahydrofluoren-3-one (9as)-4-bromo-9a-butyl-7-hydroxy-1,2,9,9a-tetrahydro-3h-fluoren-3-one 7-ethyl-6h-chromeno[4,3-b]quinoline-3,9-diol 7-ethynyl-6h-chromeno[4,3-b]quinoline-3,9-diol 7-chloro-6h-chromeno[4,3-b]quinoline-3,9-diol 7-vinyl-6h-chromeno[4,3-b]quinoline-3,9-diol 1-cyclohexyl-n-{[1-(4-methylphenyl)-1h-indol-3-yl]methyl}methanamine 7-bromo-6h-chromeno[4,3-b]quinoline-3,9-diol 4-hydroxy-n'-(4-isopropylbenzyl)benzohydrazide 1,2,3,4,6-penta-o-galloyl-beta-d-glucose 3-chlorophenyl 2-oxo-2h-chromene-3-carboxylate 5-chloro-n-(2-(4-(2-oxopyridin-1(2h)-yl)benzamido)ethyl)thiophene-2-carboxamide 5-chloro-n-{(3s)-1-[(2s)-1-(4-morpholinyl)-1-oxo-2-propanyl]-2-oxo-3-pyrrolidinyl}-1h-indole-2-sulfonamide 5-chloro-thiophene-2-carboxylic acid ((3s,4s)-4-fluoro- 1-{[2-fluoro-4-(2-oxo-2h-pyridin-1-yl)-phenylcarbamoyl]-methyl}-pyrrolidin-3-yl)-amide 6-chloro-n-{(3s)-1-[(1s)-1-methyl-2-(4-morpholinyl)-2-oxo ethyl]-2-oxo-3-pyrrolidinyl}-2-naphthalenesulfonamide 4-[(5-chloroindol-2-yl)sulfonyl]-2-(2-methylpropyl)-1-[[5-(pyridin-4-yl)pyrimidin-2-yl]carbonyl]piperazine 1-[[(1e)-2-(4-chlorophenyl)ethenyl]sulfonyl]-4-[[1-(4-pyridinyl)-4-piperidinyl]methyl]piperazine 5-chloro-n-((1r,2s)-2-(4-(2-oxopyridin-1(2h)-yl)benzamido) cyclopentyl)thiophene-2-carboxamide 5-chloro-n-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}-1-benzothiophene-2-sulfonamide 5-chloro-n-[(3r)-1-(2-{[2-fluoro-4-(2-oxopyridin-1(2h)-yl)phenyl]amino}-2-oxoethyl)pyrrolidin-3-yl]thiophene-2-carboxamide 5-desgalloylstachyurin 4-({4-[(6-chloro-1-benzothien-2-yl)sulfonyl]-2-oxopiperazin-1-yl}methyl)benzenecarboximidamide 4-(4-benzyloxy-3-methoxy-benzylamino)-benzamidine (2r)-2-(5-chloro-2-thienyl)-n-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}propene-1-sulfonamide 2-({4-[(5-chloro-1h-indol-2-yl)sulfonyl]piperazin-1-yl}carbonyl)thieno[3,2-b]pyridine 4-oxide 1-{2-[(4-chlorophenyl)amino]-2-oxoethyl}-n-(1-isopropylpiperidin-4-yl)-1h-indole-2-carboxamide 6-chloro-n-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}-1-benzothiophene-2-sulfonamide 2-(5-chloro-2-thienyl)-n-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}ethanesulfonamide 5-(5-chloro-2-thienyl)-n-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}-1h-1,2,4-triazole-3-sulfonamide 5-chloro-thiophene-2-carboxylic acid ((3s,4s)-1-{[2-fluoro-4-(2-oxo-2h-pyridin-1-yl)-phenylcarbamoyl]-methyl}-4-hydroxy-pyrrolidin-3-yl)-amide 4-[[(1e)-2-(4-chlorophenyl)ethenyl]sulfonyl]-1-[[1-(4-pyridinyl)-4-piperidinyl]methyl]piperazinone 4-{[(e)-2-(5-chlorothien-2-yl)vinyl]sulfonyl}-1-(1h-pyrrolo[3,2-c]pyridin-2-ylmethyl)piperazin-2-one 3-({4-[(6-chloro-1-benzothien-2-yl)sulfonyl]-2-oxopiperazin-1-yl}methyl)benzenecarboximidamide 6-carbamimidoyl-4-(3-hydroxy-2-methyl-benzoylamino)-naphthalene-2-carboxylic acid methyl ester (r)-1-(4-(4-(hydroxymethyl)-1,3,2-dioxaborolan-2-yl)benzyl)guanidine (r)-1-(4-(4-(hydroxymethyl)-1,3,2-dioxaborolan-2-yl)phenyl)guanidine 3-hydroxypropyl 3-[(7-carbamimidoyl-1-naphthyl)carbamoyl]benzenesulfonate (1r)-2-[(diaminomethylene)amino]-1-{4-[(4r)-4-(hydroxymethyl)-1,3,2-dioxaborolan-2-yl]phenyl}ethyl nicotinate 4-methyl-pentanoic acid {1-[4-guanidino-1-(thiazole-2-carbonyl)-butylcarbamoyl]-2-methyl-propyl}-amide (r)-1-(4-(4-(hydroxymethyl)-1,3,2-dioxaborolan-2-yl)phenethyl)guanidine 2-(6-chloro-3-{[2,2-difluoro-2-(2-pyridinyl)ethyl]amino}-2-oxo-1(2h)-pyrazinyl)-n-[(2-fluoro-6-pyridinyl)methyl]acetamide 4-iodobenzo[b]thiophene-2-carboxamidine 4-[3-(4-chlorophenyl)-1h-pyrazol-5-yl]piperidine (3z,6s)-6-chloro-1-(2-{[(5-chloro-1-benzothiophen-3-yl)methyl]amino}ethyl)-3-({2-[(2r)-2-piperidinyl]ethyl}imino)-2-piperazinol 2-[n'-(4-amino-butyl)-hydrazinocarbonyl]-pyrrolidine-1-carboxylic acid benzyl ester 1-[2-amino-2-cyclohexyl-acetyl]-pyrrolidine-3-carboxylic acid 5-chloro-2-(2-ethylcarbamoyl-ethoxy)-benzylamide 4-tert-butylbenzenesulfonic acid 4-(2,5-diamino-5-hydroxy-pentyl)-phenol (s)-n-(4-carbamimidoylbenzyl)-1-(2-(cyclopentyloxy)ethanoyl)pyrrolidine-2-carboxamide (s)-n-(4-carbamimidoylbenzyl)-1-(2-(cyclohexyloxy)ethanoyl)pyrrolidine-2-carboxamide 5-(dimethylamino)-1-naphthalenesulfonic acid(dansyl acid) 6-(2-hydroxy-cyclopentyl)-7-oxo-heptanamidine 6-chloro-2-(2-hydroxy-biphenyl-3-yl)-1h-indole-5-carboxamidine 1-(2-{[(6-amino-2-methylpyridin-3-yl)methyl]amino}ethyl)-6-chloro-3-[(2,2-difluoro-2-pyridin-2-ylethyl)amino]-1,4-dihydropyrazin-2-ol 2-(6-chloro-3-{[2,2-difluoro-2-(2-pyridinyl)ethyl]amino}-2-oxo-1(2h)-pyrazinyl)-n-[(2-fluoro-3-methyl-6-pyridinyl)methyl]acetamide 2-[2-(4-chloro-phenylsulfanyl)-acetylamino]-3-(4-guanidino-phenyl)-propionamide 2-(2-hydroxy-phenyl)-3h-benzoimidazole-5-carboxamidine 2-naphthalenesulfonic acid 1-(hydroxymethyleneamino)-8-hydroxy-octane 4-oxo-2-phenylmethanesulfonyl-octahydro-pyrrolo[1,2-a]pyrazine-6-carboxylic acid [1-(n-hydroxycarbamimidoyl)-piperidin-4-ylmethyl]-amide 2-nas-phe(3-am)-4-(2-guanidinoethyl)piperidine 4-(1r,3as,4r,8as,8br)-[1-difluoromethyl-2-(4-fluorobenzyl)-3-oxodecahydropyrrolo[3,4-a]pyrrolizin-4-yl]benzamidine 2-[3-chloro-6-[2,2-difluoro-2-(1-oxidopyridin-1-ium-2-yl)ethyl]imino-1-hydroxypyridin-2-yl]-n-[(1r)-1-(3-chlorophenyl)ethyl]acetamide 6-carbamimidoyl-2-[2-hydroxy-6-(4-hydroxy-phenyl)-indan-1-yl]-hexanoic acid [(2r)-1-[(2s)-2-[[(2s,3s)-1-chloro-6-(diaminomethylideneamino)-2-hydroxyhexan-3-yl]carbamoyl]pyrrolidin-1-yl]-1-oxo-3-phenylpropan-2-yl]azanium 4-hydroxyphenylpyruvic acid 2-{2-hydroxy-[1,1'-biphenyl]-3-yl}-1h-1,3-benzodiazole-5-carboximidamide 1-ethoxycarbonyl-d-phe-pro-2(4-aminobutyl)hydrazine 3-(7-diaminomethyl-naphthalen-2-yl)-propionic acid ethyl ester 1-butanoyl-n-(4-carbamimidoylbenzyl)-l-prolinamide 4-(5-benzenesulfonylamino-1-methyl-1h-benzoimidazol-2-ylmethyl)-benzamidine 1-guanidino-4-(n-phenylmethanesulfonyl-l-leucyl-l-prolylamino)butane 2-(2-hydroxy-phenyl)-1h-indole-5-carboxamidine 1-[(2r)-2-aminobutanoyl]-n-(4-carbamimidoylbenzyl)-l-prolinamide (s)-n-(4-carbamimidoylbenzyl)-1-(3-cyclopentylpropanoyl)pyrrolidine-2-carboxamide (3r)-8-(dioxidosulfanyl)-3-methyl-1,2,3,4-tetrahydroquinoline 3-carbamimidamido-1,1-diphenylurea 4-(3,4-diethoxy-benzylamino)-benzamidine [phenylalaninyl-prolinyl]-[2-(pyridin-4-ylamino)-ethyl]-amine 3-(4-chlorophenyl)-5-(methylthio)-4h-1,2,4-triazole 3-cyclohexyl-d-alanyl-n-(3-chlorobenzyl)-l-prolinamide (s)-n-(4-carbamimidoylbenzyl)-1-(2-(cyclopentylamino)ethanoyl)pyrrolidine-2-carboxamide (s)-n-(4-carbamimidoylbenzyl)-1-(3-cyclohexylpropanoyl)pyrrolidine-2-carboxamide (s)-n-(4-carbamimidoylbenzyl)-1-(2-(cyclohexylamino)ethanoyl)pyrrolidine-2-carboxamide 4-iodobenzo[b]thiophene 2-carboxamidine 4-[(3as,4r,7r,8as,8br)-2-(1,3-benzodioxol-5-ylmethyl)-7-hydroxy-1,3-dioxodecahydropyrrolo[3,4-a]pyrrolizin-4-yl]benzenecarboximidamide 2-(6-chloro-3-{[2,2-difluoro-2-(1-oxido-2-pyridinyl)ethyl]amino}-2-oxo-1(2h)-pyrazinyl)-n-[(2-fluorophenyl)methyl]acetamide 3-amino-3-benzyl-9-carboxamide[4.3.0]bicyclo-1,6-diazanonan-2-one {(2s)-1-[n-(tert-butoxycarbonyl)glycyl]pyrrolidin-2-yl}methyl (3-chlorophenyl)acetate (3asr,4rs,8asr,8brs)-4-(2-(4-fluorobenzyl)-1,3-dioxodeacahydropyrrolo[3,4-a] pyrrolizin-4-yl)benzamidine 6-carbamimidoyl-2-[2-hydroxy-5-(3-methoxy-phenyl)-indan-1-yl]-hexanoic acid [[cyclohexanesulfonyl-glycyl]-3[pyridin-4-yl-aminomethyl]alanyl]piperidine 4-({[4-(3-methylbenzoyl)pyridin-2-yl]amino}methyl)benzenecarboximidamide 1-[(2r)-2-aminobutanoyl]-n-(3-chlorobenzyl)-l-prolinamide 1-guanidino-4-(n-nitro-benzoylamino-l-leucyl-l-prolylamino)butane [5-(5-amino-1h-pyrrolo[3,2-b]pyridin-2-yl)-6-hydroxy-3'-nitro-3-biphenylyl]acetic acid [2'-hydroxy-3'-(1h-pyrrolo[3,2-c]pyridin-2-yl)-biphenyl-3-ylmethyl]-urea 2-(4-hydroxy-5-phenyl-1h-pyrazol-3-yl)-1h-benzoimidazole-5-carboxamidine 3-({1-[3-carbamimidoyl-1-(4-carbamimidoyl-benzylcarbamoyl)-propylcarbamoyl]-2-methyl-butylsulfamoyl}-methyl)-benzoic acid 2-[2-ethanesulfonylamino-3-(5-propoxy-1h-indol-3-yl)-propionylamino]-pentanedioic acid 5-amide 1-(4-carbamimidoyl-benzylamide) 2-[2-ethanesulfonylamino-3-(1h-indol-3-yl)-propionylamino]-pentanedioic acid 5-amide 1-(4-carbamim idoyl-benzylamide) (2r)-({4-[amino(imino)methyl]phenyl}amino){5-ethoxy-2-fluoro-3-[(3r)-tetrahydrofuran-3-yloxy]phenyl}aceticacid 5-benzyloxy-benzo[b]thiophene-2-carboxamidine 4-benzyloxybenzo[b]thiophene-2-carboxamidine 4-phenyl-benzo[b]thiophene-2-carboxamidine 6-benzyloxybenzo[b]thiophene-2-carboxamidine 4-(3-{[5-(trifluoromethyl)pyridin-2-yl]oxy}benzyl)piperidine-1-carboxylic acid 1-dodecanol 4-(quinolin-3-ylmethyl)piperidine-1-carboxylic acid 1-anilinonaphthalene-8-sulfonic acid 5-carbazol-9-yl-pentanoic acid 4-carbazol-9-yl-butyric acid 2-(6-methoxy-indole-1-sulfonyl)-benzoic acid 2-(4-methyl-indole-1-sulfonyl)-benzoic acid 3-carbazol-9-yl-propionic acid 2-(3-methyl-indole-1-sulfonyl)-benzoic acid 2-(5-bromo-indole-1-sulfonyl)-benzoic acid 2-(2,3-bis(2-chlorobenzyloxy)phenyl)acetic acid 1-benzyl-2,3-dimethyl-1h-indole-7-carboxylic acid 2-(4-fluoro-indole-1-sulfonyl)-benzoic acid 2-(carbazole-9-sulfonyl)-benzoic acid 4-[hydroxy-[methyl-phosphinoyl]]-3-oxo-butanoic acid 2-aminophenoxazine-3-one (-)-catechingallate 4-hydroxy-6-nitro-3-phenylquinolin-2(1h)-one 2-hexadecynoic acid 4-hydroxy-8-nitro-3-phenylquinolin-2(1h)-one 4-amino-n-[(2-sulfanylethyl)carbamoyl]benzenesulfonamide 2,5-anhydroglucitol-1,6-biphosphate 2,5-dichloro-n-(5-chloro-1,3-benzoxazol-2-yl)benzenesulfonamide {4-[3-(6,7-diethoxy-quinazolin-4-ylamino)-phenyl]-thiazol-2-yl}-methanol 2,5-dichloro-n-[5-methoxy-7-(6-methoxypyridin-3-yl)-1,3-benzoxazol-2-yl]benzenesulfonamide 3-[7'-(methoxy)-napht-2'-yl]-quinuclidine-2-ene 2-[4-(2-thienyl)phenyl]-4-methylmorpholin-2-ol 1-allyl-2-[3-(isopropylamino)propoxy]-9h-xanthen-9-one 3-[1'-{4'-(benzyloxy)-phenyl}]-quinuclidine-2-ene (z)-3-[2-(9h-fluoren-2-yloxy)ethylidene]-quinuclidine hydrochloride 31 1-allyl-2-[3-(isopropylamino)propoxy]-9h-carbazole 1-[(prop-2-ylamino)ethyl]-1,1-bisphosphonicacid (1-hydroxy-1-phosphono-heptyl)-phosphonic acid [2-(6-chloro-purin-9-yl)ethyl]-bisphosphonic acid 1-[(n-oct-1-ylamino)ethyl]-1,1-bisphosphonic acid 1-(but-2-ylamino)ethyl 1,i-bisphosphonic acid 1-[(n-hex-1-ylamino)ethyl]-1,1-bisphosphonic acid [2-(purin-9-yl)ethyl]-bisphosphonic acid [2-(imidazol-1-yl)ethyl]-bisphosphonic acid [2-(benzoimidazol-1-yl)ethyl]-bisphosphonic acid 1-[(cyclohexylamino)ethyl]-1,1-bisphosphonicacid (biphenyl-3-ylamino)methylenediphosphonic acid (2e, 6e)-farnesylbisphosphonate 1-[(tert-butylamino)ethyl]-1,1-bisphosphonicacid 1-[(prop-1-ylamino)ethyl]-1,1-bisphosphonic acid [2-(imidazol-2-yl-thio)ethyl]-bisphosphonic acid 3-azageranylgeranyl diphosphate 1-[(n-but-1-ylamino)ethyl]-1,1-bisphosphonic acid [2-(pyrazol-1-yl)ethyl]-bisphosphonic acid 1-methylcyclopropanecarboxylic acid (s)-4-cmtb 5-amino-naphtalene-2-monosulfonate 5-aminonaphthalene-2-sulfonic acid 3-benzimidazol-2-ylhydroquinolin-2-one 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone (e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanol 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone 4-[4-(1-amino-1-methylethyl)phenyl]-5-chloro-n-[4-(2-morpholin-4-ylethyl)phenyl]pyrimidin-2-amine 5,11-dimethyl-6h-pyrido[4,3-b]carbazol-9-ol (3r)-4-(p-toluenesulfonyl)-1,4-thiazane-3-carboxylicacid-l-phenylalanine ethyl ester 4-hydroxy-2-butanone (3r)-4-(p-toluenesulfonyl)-1,4-thiazane-3-carboxylicacid-l-leucine (21s)-1aza-4,4-dimethyl-6,19-dioxa-2,3,7,20-tetraoxobicyclo[19.4.0] pentacosane 4-hydroxybutan-2-one {3-[3-(3,4-dimethoxy-phenyl)-1-(1-{1-[2-(3,4,5-trimethoxy-phenyl)-butyryl]-piperidin-2yl}-vinyloxy)-propyl]-phenoxy}-acetic acid 3,6-di-pyridin-4-yl-pyrazolo[1,5-a]pyrimidine 4-chloro-n-(2-chloro-benzoyl)-benzenesulfonamide (2-methoxy-phenyl)-(5-phenyl-oxazol-2-yl)-amine 3-(5-phenyl-oxazol-2-ylamino)-benzonitrile 4-(5-phenyl-oxazol-2-ylamino)-benzenesulfonamide 4-chloro-n-(4-nitro-benzoyl)-benzenesulfonamide 4-chloro-n-(2-methyl-benzoyl)-benzenesulfonamide 4-(isoquinolin-5-yl)-n-m-tolylphthalazin-1-amine 2-(5-phenyl-oxazol-2-ylamino)-benzonitrile 4-chloro-n-(3-chloro-benzoyl)-benzenesulfonamide 4-chloro-n-(4-chloro-benzoyl)-benzenesulfonamide (5-phenyl-oxazol-2-yl)-m-tolyl-amine 4-(isoquinolin-5-yl)-n-o-tolylphthalazin-1-amine [3-(5-phenyl-oxazol-2-ylamino)-phenyl]-methanol (5-fluoro-1h-indol-2-yl)-(1h-indol-2-yl)methanone (1h-indol-2-yl)(5-methoxy-1h-indol-2-yl)methanone (1h-indol-2-yl)(6-methoxy-1h-indol-2-yl)methanone 4-(4-aminophenyl)-1h-indazol-3yl-amine (benzo[b]furan-2-yl)-(1h-indol-2-yl)methanone (5-hydroxy-1h-indol-2-yl)(1h-indol-2-yl)methanone (1h-indol-2-yl)(5-phenoxy-1h-indol-2-yl)methanone 2-(3,4-dimethoxybenzamido)thiophene-3-carboxamide 4sc-203 (20s)-19,20,22,23-tetrahydro-19-oxo-5h,21h-18,20-ethano-12,14-etheno-6,10-methenobenz[d]imidazo[4,3-l][1,6,9,13]oxatriazacyclonoadecosine-9-carbonitrile 2-[methyl-(5-geranyl-4-methyl-pent-3-enyl)-amino]-ethyl-diphosphate 2-chloro-5-(3-chloro-phenyl)-6-[(4-cyano-phenyl)-(3-methyl-3h-imidazol-4-yl)- methoxymethyl]-nicotinonitrile (11s)-8-chloro-11-[1-(methylsulfonyl)piperidin-4-yl]-6-piperazin-1-yl-11h-benzo[5,6]cyclohepta[1,2-b]pyridine (20s)-19,20,21,22-tetrahydro-19-oxo-5h-18,20-ethano-12,14-etheno-6,10-metheno-18h-benz[d]imidazo[4,3-k][1,6,9,12]oxatriaza-cyclooctadecosine-9-carbonitrile [(3,7,11-trimethyl-dodeca-2,6,10-trienyloxycarbamoyl)-methyl]-phosphonic acid (z)-2-methyl-3-tetradecyl-but-2-enedioic acid 4-(2-carboxy-5-mercaptopentyl)benzoic acid 99mtc-mip-1404 227th-labelled psma-ttc 2-mercapto-pentanedioic acid 4scar-psma 5-mercapto-pentanoic acid 2-(3-mercapto-propyl)-pentanedioic acid 177-lu-psma-r2 2-(3-carboxybenzyl)succinic acid 2-(3-hydroxycarbamoyl-propyl)-pentanedioic acid 2-hydroxycarbamoyl-pentanedioic acid 3-(2-carbamoyl-5-mercaptopentyl)benzoic acid 2-benzyl-5-mercaptopentanoic acid 177-lu-psma-617 2-phosphonooxy-pentanedioic acid 2-(2-carboxy-7-mercaptoheptyl)benzoic acid 2-hydroxycarbamoylmethyl-pentanedioic acid (2s)-2-{[hydroxy(4-iodobenzyl)phosphoryl]methyl}pentanedioic acid 2-mercaptomethyl-pentanedioic acid 3-(1-carboxy-4-mercaptobutoxy)benzoic acid 3-(2-carboxy-3-mercaptopropyl)benzoic acid 99mtc-mip-1405 3-(2-carboxy-4-mercaptobutyl)benzoic acid 99mtc-mip-1340 177lu-labelled ctt-1403 177lu-labelled psma-617 3-(2-carboxy-3-phosphonopropyl)benzoic acid 2-(2-hydroxycarbamoyl-ethyl)-pentanedioic acid 2-(2-mercapto-ethyl)-pentanedioic acid 2-(4-mercapto-butyl)-pentanedioic acid 2-(5-mercapto-pentyl)-pentanedioic acid [3h]quisqualate 2-pmpa 3-(2-carboxy-5-mercaptopentyl)benzoic acid 3-(2-carboxy-6-mercaptohexyl)benzoic acid 177lu-labelled psma-r2 2-(3-cyanobenzyl)-5-mercaptopentanoic acid 2-(3-methylsulfanyl-propyl)-pentanedioic acid 99mtc-ec-0652 3-[(1-carboxy-4-mercaptobutyl)thio]benzoic acid 2-(2-carboxy-5-mercaptopentyl)benzoic acid 2-(2-phosphonooxy-ethyl)-pentanedioic acid 2-(3-carbamoylbenzyl)-5-mercaptopentanoic acid 3570-0208 (6r)-folinic acid 99mtc-fanolesomab 1-methoxy-2-[2-(2-methoxy-ethoxy]-ethane 16-bromoepiandrosterone 7-o-b-d-glucopyranosyl-a-homonojirimycin 5-(4-(4-acetylphenyl)piperazin-1-ylsulfonyl)-6-chloroindolin-2-one (-)-uniflorine a (r)-2,6-bis-hydroxymethyl-piperidine-3,4,5-triol 2,5-imino-2,5,6-trideoxy-d-manno-heptitol 4-benzyl-5-(4-piperidyl)isothiazol-3-ol 6-bromo-3-ethoxycarbonyl-4-quinolone (9-benzyl-9h-purin-6-yl)-cyclopropyl-amine 3,3-diethyl-dihydro-furan-2-one 9h-beta-carboline-3-carboxylic acid ethyl ester 3-demethoxy-3-d-mannopyranosylaminothiocolchicine 4-naphthalen-2-yl-5-piperidin-4-yl-isoxazol-3-ol 3-(2,2-dimethyl-propoxy)-9h-beta-carboline 6,6-dimethyl-2-oxa-spiro[4.4]nonan-1-one 2-thiophen-2-yl-3h-imidazo[4,5-c]quinoline 3-methoxycarbonyl-2-methyl-9h-beta-carbolin-2-ium 3-ethoxycarbonyl-6-propyl-4-quinolone 2-(3-bromo-phenyl)-6-nitro-chromen-4-one 3-isothiocyanato-9h-beta-carboline 1,2-benzodiazepine 6,9-dimethyl-2-oxa-spiro[4.4]nonan-1-one 3-ethoxy-9h-beta-carboline (beta-cce)9h-beta-carboline-3-carboxylic acid [3h]ro154513 2-furan-2-yl-6h-pyrazolo[1,5-c]quinazolin-5-one 3-butoxy-9h-beta-carboline 5-[(1r)-1-ammonioethyl]isoxazol-3-olate 3,3-diisopropyl-dihydro-furan-2-one 1-methyl-5-oxa-spiro[2.4]heptan-4-one 2-phenyl-6h-pyrazolo[1,5-c]quinazolin-5-one 6-ethyl-3-(2-methylbutoxycarbonyl)-4-quinolone 7,12-dihydro-5,7,12-triaza-indeno[1,2-a]fluorene 4-methoxymethyl-3,6-dipropoxy-9h-beta-carboline 6-ethyl-3-i-propoxycarbonyl-4-quinolone 4-(biphenyl-3-yl)-5-(piperidin-4-yl)isoxazol-3-ol 3-isopropoxy-9h-beta-carboline 2-(1h-indol-3-yl)-2-oxo-n-phenethyl-acetamide 9h-beta-carbolin-6-ylamine 6-bromo-2-(3-nitro-phenyl)-chromen-4-one 3-butoxycarbonyl-4-quinolone 6-ethyl-3-propylaminocarbonyl-4-quinolone 3-nitro-9h-beta-carboline 1,1-dimethyl-5-oxa-spiro[2.4]heptan-4-one (2-amino-4,5-dihydro-thiazol-4-yl)-acetic acid 3-carboxy-6-ethyl-4-quinolone 3-ethoxycarbonyl-4-quinolone 3-isobutoxy-9h-beta-carboline 3-methyl-2-phenyl-2h-chromeno[4,3-c]pyrazol-4-one 3-methoxy-9h-beta-carboline 6-benzyl-3-propylaminocarbonyl-4-quinolone 4-(4-chlorophenyl)-1-pyrid-2-yl-pyrazole 6-bromo-2-(3-bromo-phenyl)-chromen-4-one 3-amino-3-demethoxythiocolchicine 7,12-dihydro-7,12-diaza-indeno[1,2-a]fluorene 3-methyl-1-phenyl-1h-chromeno[4,3-c]pyrazol-4-one 2-phenyl-5,6-dihydro-pyrazolo[1,5-c]quinazoline 2-pyridin-2-yl-6h-pyrazolo[1,5-c]quinazolin-5-one 2-oxa-spiro[4.4]nonan-1-one 3-chloro-9h-beta-carboline 4-benzyl-5-piperidin-4-yl-isoxazol-3-ol (9h-beta-carbolin-3-yl)-carbamic acid ethyl ester 3-ethyl-3-methyl-dihydro-furan-2-one 2-(3-chloro-phenyl)-chromen-4-one 1,3-diphenyl-1h-chromeno[4,3-c]pyrazol-4-one 6-nitro-2-phenyl-chromen-4-one 6-bromo-2-(4-nitro-phenyl)-chromen-4-one 4-naphthalen-1-yl-5-piperidin-4-yl-isoxazol-3-ol 3-demethoxy-3d-glucopyranosylaminothiocolchicine 3-propoxy-9h-beta-carboline 2-(9-benzyl-9h-purin-6-ylamino)-ethanol 2-phenyl-3h-imidazo[4,5-c]quinoline 1-(9h-beta-carbolin-3-yl)-butan-1-one 2-isoxazol-5-yl-3h-imidazo[4,5-c]quinoline 2-p-tolyl-6h-pyrazolo[1,5-c]quinazolin-5-one 3-tert-butyl-3-ethyl-dihydro-furan-2-one 3-(3-methyl-butoxy)-9h-beta-carboline 1-(9h-beta-carbolin-3-yl)-ethanone 6-benzyl-3-propoxycarbonyl-4-quinolone 3-demethoxy-3-d-lyxopyranosylaminothiocolchicine 6-bromo-2-(2-nitro-phenyl)-chromen-4-one 6-fluoro-2-(3-nitro-phenyl)-chromen-4-one 2-(4-chloro-phenyl)-3h-imidazo[4,5-c]quinoline 4-phenyl-5-piperidin-4-yl-isoxazol-3-ol 4-methyl-5-(4-piperidyl)isothiazol-3-ol 3-sec-butoxy-9h-beta-carboline 5,7,2?-trihydroxy-6,8-dimethoxyflavone 6-nitro-2-(4-nitro-phenyl)-chromen-4-one (9h-beta-carbolin-3-yl)-methanol 2-(4-chlorophenyl)-5-phenyl-4-isoxazolin-3-one 3-isopropyl-3-methyl-dihydro-furan-2-one 6-ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone 3-ethyl-3-isopropyl-dihydro-furan-2-one 1-(4-chlorophenyl)-4-phenyl-1h-imidazole 3-butylaminocarbonyl-6-ethyl-4-quinolone (6-benzylamino-9h-beta-carbolin-3-yl)-methanol 3-(benzyloxy)-9h-pyrido[3,4-b]indole 3-demethoxy-3-d-xylopyranosylaminothiocolchicine 6-ethyl-3-(2-ethylbutoxycarbonyl)-4-quinolone 6-ethyl-3-pentoxycarbonyl-4-quinolone 3-demethoxy-3-l-fucopyranosylaminothiocolchicine (4r)-4-ammoniopentanoate 4-(2-aminoethyl)-1,2,5-oxadiazol-3-ol 2-(3-bromo-phenyl)-chromen-4-one 3-methyl-9h-beta-carboline 6-chloro-2-phenyl-chromen-4-one 5-(piperidin-4-yl)isothiazol-3-ol 2-isoxazol-3-yl-3h-imidazo[4,5-c]quinoline (4s)-4-ammoniopentanoate 5-[(1s)-1-ammonioethyl]isoxazol-3-olate [3h]cgs8216 3-cyclopentoxycarbonyl-6-ethyl-4-quinolone 6-bromo-2-phenyl-chromen-4-one 9h-beta-carboline-3-carboxylic acid propyl ester 5-(piperidin-4-yl)isoxazol-3-ol [3h]cgp27492 6-chloro-2-(3-nitro-phenyl)-chromen-4-one 6-bromo-3-ethoxycarbonyl-2-methyl-4-quinolone 9h-beta-carbolin-3-ol 6-methyl-2-oxa-spiro[4.4]nonan-1-one 6-ethyl-3-(3-pentoxycarbonyl)-4-quinolone 3-(hexa-1,3-dienyloxy)-9h-pyrido[3,4-b]indole 6-ethyl-3-propoxycarbonyl-4-quinolone 6-benzyl-3-ethoxycarbonyl-4-quinolone 6-nitro-2-(3-nitro-phenyl)-chromen-4-one (2e,4s)-4-ammoniopent-2-enoate 5-(4-piperidyl)-4-propylisothiazol-3-ol 3-butoxycarbonyl-6-ethyl-4-quinolone (9h-beta-carbolin-3-yl)-ethyl-amine 3-ethoxycarbonyl-6-ethyl-2-methyl-4-quinolone [35s]tbps [18f]fluoroethylflumazenil [3h]l655708 [3h]ry80 (+/-)-cis-2-camp 5-me-iaa [n-me,des-sar]gal-b2 (sar)wtlnsagyllgpkk(lys-lauroyl)k (sar)wtlnsagyllgpkk(lys-decanoyl)k (sar)wtlnsagyllgpkkkk (sar)wtlnsagyllgpkk(lys-mpeg4)k [sar1gly]gal-b2 (sar)wtlnsagyllgpkk(lys-palmitoyl)k (sar)wtlnsagyllgpkk(lys-myristoyl)k [n-ac,des-sar]gal-b2 (sar)wtlnsagyllgpkk(lys-stearoyl)k [sar1ala]gal-b2 (sar)wtlnsagyllgpkk(lys-octanoyl)k 2'-deoxy-2'-[(3,5-dimethoxybenzoyl)amino]-n-[(1r)-1,2,3,4-tetrahydro-1-naphthalenyl]adenosine (+)-rutamarin alcohol 10-cf3c(oh)2-ddacthf 10-trifluoroacetyl-ddacthf 10-formyl-5,8,10-trideazafolic acid (10r)-10-formyl-5,8,10-trideazafolic acid (2r,3s,4s,5r)-2-hexylpiperidine-3,4,5-triol (2r,3s,4s,5r)-2-nonylpiperidine-3,4,5-triol 1,5-dideoxy-1,5-imino-d-xylitol (2r,3r,4r,5s)-2-(hydroxymethyl)-1-nonylpiperidine-3,4,5-triol (2r,3s,4s,5r)-2-propylpiperidine-3,4,5-triol [des-his1,tyr5,glu9,d-phe10]glucagon-nh2 [des-his1,tyr5,glu9,d-tyr10]glucagon-nh2 [des-his1,tyr5,glu9,d-ala10]glucagon-nh2 [des-his1,tyr5,glu9]glucagon-nh2 3-substituted-2-furancarboxylic acid hydrazide derivative 1 3-substituted-2-furancarboxylic acid hydrazide derivative 5 8-hydroxyguanine 3-[(4-fluorophenyl)sulfanyl]-n-(4-methyl-1,3-thiazol-2-yl)-6-[(4-methyl-4h-1,2,4-triazol-3-yl)sulfanyl]pyridine-2-carboxamide 2-amino-4-fluoro-5-[(1-methyl-1h-imidazol-2-yl)sulfanyl]-n-(1,3-thiazol-2-yl)benzamide 2-amino-n-(4-methyl-1,3-thiazol-2-yl)-5-[(4-methyl-4h-1,2,4-triazol-3-yl)sulfanyl]benzamide 2-(methylamino)-n-(4-methyl-1,3-thiazol-2-yl)-5-[(4-methyl-4h-1,2,4-triazol-3-yl)sulfanyl]benzamide 6-(hydroxyethyldithio)-8-(aminomethylthio)octanoic acid [2-(3-dibenzofuran-4-yl-phenyl)-1-hydroxy-1-phosphono-ethyl]-phosphonic acid (1-hydroxyheptane-1,1-diyl)bis(phosphonic acid) (6e,11e)-heptadeca-6,11-diene-9,9-diylbis(phosphonic acid) (2,2-diphosphonoethyl)(dodecyl)dimethylphosphonium (1-hydroxynonane-1,1-diyl)bis(phosphonic acid) [35s]ibutamoren 4-(3-hexylureido)-n-phenylbenzenesulfonamide 2,5-dideoxy-2,5-imino-d-altritol (+)-5-deoxyadeenophorine [gly8, aib22]glp-1(7-37)-nh2 [gly8,glu22]glp-1(7,37)-nh2 [gly8]glp-1(7-37)-nh2 [123i] iodobenzoyl 12-ex4 [3h]strychnine 10-methoxy-ginkgolide c 3,14-didehydroginkgolide a 3,5-dibromo-2-(2,4-dibromophenoxy)phenol 2,3,4-tribromo-6-(2,4-dibromophenoxy)phenol 3,4,5-tribromo-2-(2', 4'-dibromo-phenoxy)phenol 3-(n-morpholino)propanesulfonic acid 2-deoxy-2-amino glucitol-6-phosphate [d-gln3,d-ncy(so,isopropyl)7]acyline [ncy(2-naphthyl)1]acyline [ncy(isopropyl)7]acyline [d-ncy(2-naphthyl)1]acyline [d-4aph(co-nh-oh)6]degarelix [d-dab(co-nh-och3)3]degarelix [ncy(so,methyl)10]acyline [d-dab(co-nh-oh)3]degarelix [d-gln3,d-ncy(isopropyl)7]acyline [4aph(co-nh-oh)5]degarelix [d-ncy(methyl)10] acyline [d-dap(co-nh-oh)3]degarelix [4aph(co-(c2h4o)3-c2h4-nh-co-nh-och3)5]degarelix [ncy(methyl)4]acyline [d-ncy(so,methyl)10]acyline [d-ncy(methyl)4]acyline [d-ncy(so,isopropyl)7]acyline [4aph(co-nh-och3)5]degarelix [d-4aph(co-nh-(c2h4o)2-c2h5)6]degarelix [125i]cetrorelix [d-gln3,ncy(isopropyl)7]acyline [4aph(co-nh-(c2h4o)2-c2h5)5]degarelix [d-gln3,ncy(so,isopropyl)7]acyline [ncy(so,isopropyl)7]acyline [d-4aph(co-nh-och3)6]degarelix [4aph(co-nh-och3)5,d-4aph(co-nh-och3)6]degarelix [d-gln3,d-ncy(so2,isopropyl)7]acyline [ncy(methyl)10]acyline [d-ncy(isopropyl)7]acyline [d-ncy(so,methyl)4]acyline [d-dap(co-nh-och3)3]degarelix [ncy(so,methyl)4]acyline [d-gln3,ncy(so2,isopropyl)7]acyline 4'-deoxy-4'-acetylyamino-pyridoxal-5'-phosphate 5-phosphoarabinonic acid 6-phospho-d-gluconic acid 5-phospho-d-arabinohydroxamic acid (s)-n-oleoyltyrosinol 1-oleoyl glycerol 2-oleoyl glycerol 1-palmitoyl-lysophosphatidylcholine (r)-n-oleoyltyrosinol 1-stearoyl-lysophosphatidylcholine 9-hydroxyoctadecadienoic acid 27-hydroxycholesterol 7beta-hydroxycholesterol 7alpha-hydroxycholesterol 7alpha,25-dihydroxycholesterol 7alpha,27-dihydroxycholesterol 7beta, 25-dihydroxycholesterol 7beta, 27-dihydroxycholesterol 25-hydroxycholesterol 12s-hete [3h]resolvin d1 2-arachidonoylglycerolphosphoinositol 2-arachidonyl glyceryl ether 2-hydroxylauric acid 6-n-octylaminouracil 3-hydroxy capric acid 2-hydroxy capric acid 3-hydroxylauric acid 4-[(10s,14s,18s)-18-(2-amino-2-oxoethyl)-14-(1-naphthylmethyl)-8,17,20-trioxo-7,16,19-triazaspiro[5.14]icos-11-en-10-yl]benzylphosphonic acid (s)-ampa 7-chloro-3-hydroxyquinazoline-2,4-dione (s)-willardiine [3h]cnqx [3h]ampa (s)-5-fluorowillardiine (s)-des-me-ampa 2,3,6a,7,8,9-hexahydro-11h-[1,4]dioxino[2,3-g]pyrrolo[2,1-b][1,3]benzoxazin-11-one (3r)-3-cyclopentyl-7-[(4-methylpiperazin-1-yl)sulfonyl]-3,4-dihydro-2h-1,2-benzothiazine 1,1-dioxide 2-amino-3-(3-hydroxy-7,8-dihydro-6h-cyclohepta[d]-4-isoxazolyl)propionic acid (2s)-2-ammonio-3-[5-(2-methyl-2-propanyl)-3-oxido-1,2-oxazol-4-yl]propanoate (3s)-3-cyclopentyl-6-methyl-7-[(4-methylpiperazin-1-yl)sulfonyl]-3,4-dihydro-2h-1,2,4-benzothiadiazine 1,1-dioxide (3r)-3-cyclopentyl-6-methyl-7-[(4-methylpiperazin-1-yl)sulfonyl]-3,4-dihydro-2h-1,2-benzothiazine 1,1-dioxide 2-amino-3-(5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl)propionic acid (s)-2-amino-3-(1,3,5,7-pentahydro-2,4-dioxo-cyclopenta[e]pyrimidin-1-yl) proionic acid 2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid 2-(3-bromobenzoylamino)-4-chlorobenzoic acid 8-deoxy-neodysiherbaine (s)-5-iodowillardiine (s)-4-ahcp (2s,4r)-4-(3-methoxy-3-oxopropyl)glutamic acid 2s,4r-4-methylglutamate 2-amino-3-(4-hydroxy-1,2,5-oxadiazol-3-yl)propionic acid (structural mix) 2,4-epi-neodysiherbaine 5,7-dichlorokynurenic acid 4-[2-(4-benzyl-piperidin-1-yl)-ethoxy]-phenol [3h]dizocilpine 2-(4-phenoxy-benzyl)-3h-benzoimidazol-4-ol (+)-ha966 3-hydroxy-8-methyl-1h-benzo[b]azepine-2,5-dione 8-chloro-3-hydroxy-1h-benzo[b]azepine-2,5-dione 3-hydroxy-1h-benzo[b]azepine-2,5-dione 2-(4-phenoxy-benzyl)-1h-benzoimidazole 6,7-dichloro-1,4-dihydro-quinoxaline-2,3-dione 8-fluoro-3-hydroxy-1h-benzo[b]azepine-2,5-dione 1,3-ditolylguanidine 6-chloro-1,4-dihydro-quinoxaline-2,3-dione 3-hydroxy-6-methyl-1h-benzo[b]azepine-2,5-dione 4,6-dichloro-1h-indole-2-carboxylic acid (d)-ala-pro-glu 3-hydroxy-7-nitro-1h-benzo[b]azepine-2,5-dione 2-methylamino-succinic acid(nmda) 5,7-dichloro-3-hydroxy-1h-quinazoline-2,4-dione 4-[2-(4-phenyl-butoxy)-ethyl]-phenol 4-bromo-5,7-dichloro-3-hydroxy-1h-quinolin-2-one 5,7-dichloro-1,4-dihydro-quinoxaline-2,3-dione 3-benzoyl-7-chloro-4-hydroxy-1h-quinolin-2-one 6-nitro-1,4-dihydro-quinoxaline-2,3-dione 4-[2-(5-phenyl-pentylamino)-ethyl]-phenol 6-nitro-2-(4-phenoxy-benzyl)-1h-benzoimidazole 5,7-dibromo-1,4-dihydro-quinoxaline-2,3-dione 4-benzyl-1-phenethyl-piperidine hydrochloride 4-[2-(3-phenyl-propylamino)-ethyl]-phenol 6,7-dichloro-3-hydroxy-1h-quinazoline-2,4-dione 6-methoxy-2-(4-phenoxy-benzyl)-1h-benzoimidazole 4,5,7-trichloro-3-hydroxy-1h-quinolin-2-one 4-{2-[ethyl-(4-phenyl-butyl)-amino]-ethyl}-phenol 4-[2-(4-phenyl-piperidin-1-yl)-ethoxy]-phenol 8-ethyl-3-hydroxy-1h-benzo[b]azepine-2,5-dione 4-[2-(6-phenyl-hexylamino)-ethyl]-phenol (rs)-(tetrazol-5-yl)glycine 4-[3-(4-phenyl-butylamino)-propyl]-phenol 5,6,7-trichloro-1,4-dihydro-quinoxaline-2,3-dione 4-chloro-3-hydroxy-1h-quinolin-2-one 4-[2-(4-phenyl-butylamino)-ethyl]-phenol [3h]cgs19755 4-benzyl-1-(2-phenoxy-ethyl)-piperidine (r)-2-amino-7-phosphono-heptanoic acid 3-carbamoyl-6-chloro-1h-indole-2-carboxylic acid [3h]mdl105519 5,7-dinitro-1,4-dihydro-quinoxaline-2,3-dione 3-phenyl-4-hydroxyquinolin-2(1h)-one 5,7-dichloro-4-hydroxy-3-phenyl-1h-quinolin-2-one [3h]cgp39653 4-bromo-3-hydroxy-1h-quinolin-2-one (r)-2-amino-5-phosphono-pentanoic acid 4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7h)-one 2-(4-phenoxy-benzyl)-3h-benzoimidazol-5-ol 2-(4-phenoxy-benzyl)-3h-benzoimidazol-5-ylamine 8-bromo-3-hydroxy-1h-benzo[b]azepine-2,5-dione [3h]cpp 4-[3-(5-phenyl-pentylamino)-propyl]-phenol 2-(4-benzyl-piperidin-1-ylmethyl)-1h-indol-6-ol (s)-3hpg (1s,3r)-acpd (s)-(+)-cbpg 3,5-dhpg [11c]mmtp 3-matida (e)-1-adamantan-1-yl-3-quinolin-3-yl-propenone 2-methyl-6-(phenylethynyl)pyridine 3,5-dimethyl ppp [3h]em-tbpc [18f]fitm (+)-mcpg 4-(cyclohexyloxy)quinazoline (3,4-dimethylphenyl)(4-phenoxyphenyl)methanone [18f]mk-1312 (s)-4cpg (s)-tbpg (e)-4,4-dimethyl-1-quinolin-3-yl-pent-1-en-3-one 6-bromo-n-(3-chlorophenyl)quinazolin-4-amine (s)-alpha-methyl-4-carboxyphenylglycine (s)-4c3hpg [18f]fpit 4-mppts [3h]jnj-40068782 4-appes [3h]ly341495 3-mppts [3h]2,2,2-temps (2r,4r)-4-aminopyrrolidine-2,4-dicarboxylate 5-mpep 2-m-tolyl-1,8-naphthyridine 2-methyl-6-(4-phenylpent-1-ynyl)pyridine 4-(3-pyridylethynyl)-2-thiazolylamine 6-(4-chlorophenylamino)-n,n-diethylnicotinamide (e)-3-[2-(2-methyl-4-thiazolyl)vinyl]pyridine 2-methyl-4-p-tolylethynyl-thiazole 2-methyl-7-phenyl-1,8-naphthyridine 3-isobutoxy-5-(2-methylquinolin-7-yl)benzonitrile 2-methyl-6-(3-(p-tolyloxy)prop-1-ynyl)pyridine 5-((6-methylpyridin-2-yl)ethynyl)nicotinonitrile 7-(4,6-dimethoxypyrimidin-2-yl)-2-methylquinoline 3-bromo-n-(6-methylpyridin-2-yl)benzamide 2-methyl-4-(m-tolylethynyl)thiazole 3-chloro-n-(4-methylthiazol-2-yl)benzamide 3-methoxy-5-(1,5-naphthyridin-3-yl)benzonitrile 2-(2-methyl-thiazol-4-ylethynyl)-pyridine 3-cyano-n-(3-ethylphenyl)-5-fluorobenzamide 7-(4-methoxypyrimidin-2-yl)-2-methylquinoline 3-hydroxy-5-(2-methylquinolin-7-yl)benzonitrile 2-(3-bromophenyl)-7-methyl-1,8-naphthyridine 2-(3-chlorophenyl)-7-methyl-1,8-naphthyridine 2-methyl-7-m-tolylquinoline 3-(4-pyridin-2-yl-pyrazol-1-yl)-benzonitrile 2-(substituted ethynyl)quinoline derivative 3 2-(3-chlorobenzyloxy)-6-chloroisonicotinonitrile [3h]methoxy-pepy 2-methyl-7-phenylquinoline 2-phenylethynyl-7,8-dihydro-6h-quinolin-5-one [14c]mtep 2-(3-bromophenyl)-7-methylpyrido[2,3-d]pyrimidine 2-methyl-6-(4-phenylbut-1-ynyl)pyridine 2-phenylethynyl-5,6,7,8-tetrahydro-quinoline 4-(3-chlorophenylthio)-2-(pyridin-2-yl)pyrimidine 3-methoxy-5-(2-methylquinolin-7-yl)benzonitrile (3-(2-methylquinolin-7-yl)phenyl)methanol 2-phenyl-5-(2-methylthiazol-4ylethynyl)pyridine 7-methyl-2-m-tolylpyrido[2,3-d]pyrimidine 2-(pyridin-2-yl)-4-(m-tolylthio)pyrimidine 3-chloro-n-(3-isobutyramidophenyl)benzamide 3-fluoro-5-(2-methylquinolin-7-yl)benzonitrile 5-(2-(2,5-dimethylphenyl)ethynyl)pyrimidine 6-aryl-imidazopyridine and 6-aryl-triazolopyridine carboxamide analog 1 2-methyl-6-(3-(phenylthio)prop-1-ynyl)pyridine 3-chloro-5-(2-methylquinolin-7-yl)benzonitrile 3-(3-pyridin-2-yl-pyrrol-1-yl)-benzonitrile 5-[(2-methyl-4-thiazolyl)ethynyl]pyrimidine 5-(phenylethynyl)pyrimidine 5-chloro-2-(2-methylquinolin-7-yl)benzonitrile 2-ethoxy-5-(m-tolylethynyl)pyrimidine 7-(3-methoxyphenyl)-2-methyl-1,6-naphthyridine 6-aryl-imidazopyridine and 6-aryl-triazolopyridine carboxamide analog 3 2-ethynyl-4-(3-fluorophenylethynyl)thiazole 2-benzoxy-5-(2-methylquinolin-7-yl)benzonitrile 6-aryl-imidazopyridine and 6-aryl-triazolopyridine carboxamide analog 2 6-bromo-n-m-tolylquinazolin-4-amine 2-(3-(3-methoxyphenoxy)prop-1-ynyl)pyridine 7-(3-fluoro-5-methylphenyl)-1,6-naphthyridine 3-bromo-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 4-(3-bromophenylthio)-2-(pyridin-2-yl)pyrimidine 7-(4-methoxyphenyl)-2-methylquinoline 2-(substituted ethynyl)quinoline derivative 2 (3-ethoxy-pyridin-2-yl)-pyridin-2-yl-amine 4-(2-methoxyphenylethynyl)-2-methylthiazole 2-methyl-4-(2-thienylethynyl)thiazole 3-cyano-5-fluoro-n-m-tolylbenzamide 2-(substituted ethynyl)quinoline derivative 1 5pam523 4-(3-bromophenoxy)-6-chloroquinazoline 2-(substituted ethynyl)quinoline derivative 4 3-m-tolyl-1,5-naphthyridine 2-(m-tolylethynyl)pyrimidine 4-(3,5-difluorophenylethynyl)-2-methylthiazole 3-cyano-n-(6-ethylpyridin-2-yl)-5-fluorobenzamide 3-iodo-n-(6-methylpyridin-2-yl)benzamide 7-(3-chlorophenyl)-2-methylquinoline 7-(3-fluorophenyl)-2-methylquinoline 6-phenylethynyl-nicotinic acid methyl ester 2-cyclohex-1-enylethynyl-pyridine 2-methyl-7-m-tolyl-1,8-naphthyridine 4-(3-chlorophenylethynyl)-2-methylthiazole 3-methyl-n-(6-methylpyridin-2-yl)benzamide 2-methyl-7-(pyridin-3-yl)quinoline 2-phenylethynyl-5,6,7,8-tetrahydro-quinolin-5-ol 2-cyclopent-1-enylethynyl-pyridine 2-methyl-6-(5-phenylpent-1-ynyl)pyridine 3-cyano-5-fluoro-n-(pyridin-2-yl)benzamide 3-cyano-n-(1,4-diphenyl-1h-pyrazol-5-yl)benzamide 2-methyl-4-phenylethynyl-thiazole 3-(1-pyridin-2-yl-1h-pyrazol-3-yl)-benzonitrile 7-(3-methoxyphenyl)-2-methylquinoline 1-(3-(2-methylquinolin-7-yl)phenyl)ethanone 7-(2-methoxyphenyl)-2-methylquinoline 2-methyl-4-o-tolylethynyl-thiazole 4-(2-(4-fluorophenyl)ethynyl)-2-methylthiazole 6-bromo-n-(3-bromophenyl)quinazolin-4-amine 3-(2-methylquinolin-7-yl)phenol [3h]methoxymethyl-mtep 5-methyl-3-phenylethynyl[1,2,4]triazine 2-bromo-4-(3-fluorophenylethynyl)thiazole 3-(3,4-dimethylphenyl)-1,5-naphthyridine 5-(2-methylquinolin-7-yl)-2-phenylnicotinonitrile 3-cyano-5-fluoro-n-(3-fluorophenyl)benzamide 2-chloro-5-(2-methylquinolin-7-yl)nicotinonitrile 3-(2-methylbenzo[d]thiazol-5-yl)benzonitrile 6-fluoro-n-m-tolylquinazolin-4-amine 2-(3-(2-methylquinolin-7-yl)phenyl)acetonitrile 7-bromo-n-(3-bromophenyl)isoquinolin-1-amine 7-(4,6-dimethylpyrimidin-2-yl)-2-methylquinoline 3-chloro-n-(6-methylpyridin-2-yl)benzamide 3-[(5-ethyl-2-methyl-4-thiazolyl)ethynyl]pyridine 3-methyl-5-(2-methylquinolin-7-yl)benzonitrile 2-cyclohexylethynyl-pyridine 5-(2-(3-chlorophenyl)ethynyl)pyrimidine 7-methyl-2-phenylpyrido[2,3-d]pyrimidine 3-cyano-n-(3-ethynylphenyl)-5-fluorobenzamide 3-(2-pyridin-2-yl-2h-tetrazol-5-yl)-benzonitrile 3-cyano-n-(6-methylpyridin-2-yl)benzamide 5-(2-m-tolylethynyl)pyrimidine 3-[(2-methyl-4-thiazolyl)ethynyl]benzonitrile 4-cyano-n-(1,3-diphenyl-1h-pyrazol-5-yl)benzamide 3-(3-bromophenylethynyl)-5-methyl[1,2,4]triazine 6-bromo-n-(3-fluorophenyl)quinazolin-4-amine 5-(2-methylquinolin-7-yl)isophthalonitrile 7-(3,5-dimethoxyphenyl)-1,6-naphthyridine 4-(2-methyl-thiazol-4-ylethynyl)-pyridine 3-biphenyl-4-ylethynyl-5-methyl-[1,2,4]triazine 5-(2-(3,5-difluorophenyl)ethynyl)pyrimidine 3-ethoxy-5-(2-methylquinolin-7-yl)benzonitrile 3-(1,8-naphthyridin-2-yl)benzonitrile 3-bromo-5-(2-methylquinolin-7-yl)benzonitrile 5-(2-methylquinolin-7-yl)nicotinonitrile 3-cyano-5-fluoro-n-phenylbenzamide 4-(4-chlorophenylthio)-2-(pyridin-2-yl)pyrimidine 2-(3,5-dichlorophenyl)pyrido[2,3-d]pyrimidine 3-fluoro-5-(1,6-naphthyridin-7-yl)benzonitrile 5-(2-(4-fluoro-3-methylphenyl)ethynyl)pyrimidine 7-(3-(methoxymethyl)phenyl)-2-methylquinoline 3-(3-pyridin-2-yl-pyrazol-1-yl)-benzonitrile 2-(3,5-dimethoxyphenyl)-1,8-naphthyridine 4-(3-methoxyphenylethynyl)-2-methylthiazole 2-(3,4-dimethylphenyl)-1,8-naphthyridine 5-(2-methylquinolin-7-yl)-2-phenylbenzonitrile 3-cyano-n-(3-cyanophenyl)-5-fluorobenzamide 3-cyano-n-(1,3-diphenyl-1h-pyrazol-5-yl)benzamide 3-[(2-methyl-4-thiazolyl)ethynyl]benzamide 2-[(2-methyl-4-thiazolyl)ethynyl]pyrazine 3-methoxy-n-(6-methylpyridin-2-yl)benzamide 3-phenyl-1-(2-methylthiazol-4-ylethynyl)benzene 4-(2-fluorophenylethynyl)-2-methylthiazole 4-(3-fluorophenylethynyl)-2-thiazolylamine 5-biphenyl-4-ylethynyl-pyrimidine 3-(4-pyridin-2-yl-imidazol-1-yl)-benzonitrile 2-methyl-4-(3-thienylethynyl)thiazole 2-(phenylethynyl)pyrimidine 2-methyl-7-m-tolyl-1,6-naphthyridine 2-(3,5-difluorophenyl)-7-methyl-1,8-naphthyridine 2-phenyl-1,8-naphthyridine 3-[(2,5-dimethyl-4-thiazolyl)ethynyl]pyridine 2-(3-(benzyloxy)phenyl)isoindoline-1,3-dione 3-[(2-methyl-4-thiazolyl)ethynyl]phenol 3-chloro-n-(6-chloropyridin-2-yl)benzamide 3-(5-pyridin-2-yl-tetrazol-2-yl)-benzonitrile 3-[(2-methyl-4-thiazolyl)ethynyl]-5-vinylpyridine 4-biphenyl-4-ylethynyl-2-methyl-thiazole 4-biphenyl-2-ylethynyl-2-methyl-thiazole 3-(7-methyl-1,8-naphthyridin-2-yl)benzonitrile 5-(3-chlorophenylethynyl)-5-methyl[1,2,4]triazine 2-(3-bromophenyl)pyrido[2,3-d]pyrimidine [3h]fenobam 4-(2-(3-fluorophenyl)ethynyl)-2-methylthiazole 2-benzyloxy-7,8-dihydro-6h-quinolin-5-one 2-(2-methylquinolin-7-yl)benzonitrile 3,3'-difluorobenzaldazine 3-(3-(3-chlorobenzyloxy)-5-methylphenyl)pyridine 7-m-tolyl-1,6-naphthyridine 2-chloro-n-(3-(3-chlorobenzamido)phenyl)benzamide 3-[(6-methylpyridin-2-yl)ethynyl]benzonitrile 2-(4-(3-chlorophenyl)but-1-ynyl)-6-methylpyridine 3-(3-methylphenylethynyl)-5-methyl[1,2,4]triazine 3-(1-pyridin-2-yl-1h-pyrrol-3-yl)-benzonitrile 3-(6-fluoroquinazolin-4-ylamino)benzonitrile 3-(1,5-naphthyridin-3-yl)benzonitrile 3-(2-methylquinolin-7-yl)benzonitrile 3-nitro-n-(1,3-diphenyl-1h-pyrazol-5-yl)benzamide 3-(1-pyridin-2-yl-1h-pyrazol-4-yl)-benzonitrile 3-methoxy-5-(1,6-naphthyridin-7-yl)benzonitrile (s)-3,4-dcpg 2-amino-4-phosphono-butyric acid (r,s)-4-phosphonophenylglycine (ch3)cco-his-trp-ala-val-gly-his-leu-met-nh2 177-lu-neob [tyr4]bombesin (d)phe-gln-trp-ala-val-gly-his-leu-leu-nh2 [(n4-bzdig)0]bb(7-14) [n40,pro1,tyr4,nle 14]bb [(n4-bzdig)0,nle14]bb(7-14) 177lu-labelled neobomb1 [n40,pro1,tyr4]bb 177lu-amba 177lu-labelled rm2 3-(3-aminophenyl)-n-(3-chlorophenyl)pyrazolo[1,5-a]pyrimidin-5-amine (2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol 6-deoxymanzamine x 9-ing-41 (e)-n-(6-(prop-1-enyl)-1h-indazol-3-yl)butyramide (2'z,3'e)-7-azaindirubin-3'-oxime 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione 9-n-ethyl-8-ethoxy-manzamine a 6-bromoindirubin-3'-oxime (7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one 9-n-methyl-8-methoxy-manzamine a 3-(6-(phenylamino)-9h-purin-8-yl)benzonitrile 3-phenyl-4-(phenylamino)-1h-pyrrole-2,5-dione 12,13-dehydro-8-o-acetylmanzamine a 4-(5-bromo-1h-indol-3-yl)pyrimidin-2-amine 8-o-(4-chlorobenzenesulfonyl)manzamine f 8-o-(4-toluenesulfonyl)manzamine a 8-oh-manzamine a 12,13-dehydromanzamine a 8-o-(4-bromobenzenesulfonyl)manzamine f 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione 4-nitrobenzo[c][1,2,5]thiadiazole 3-nitro-l-tyrosine 3-(prop-2-ene-1-sulfinyl)-propene-1-thiol 3-sulfino-l-alanine 6-(3-methyl-1,4-dioxo-1,4-dihydronaphthalen-2-yl)hexanoic acid 1-(2'-chlorophenyl)penta-1,4-dien-3-one 3,6-dihydroxy-xanthene-9-propionic acid 2,4,6 trinitrobenzene sulfonate 1,3-bis (2-chlorethyl)-1-nitrosourea 2-(2-phenyl-3-pyridin-2-yl-4,5,6,7-tetrahydro-2h-isophosphindol-1-yl)pyridine 3-sulfinoalanine 2-hydroxyethyl disulfide 4-s-glutathionyl-5-pentyl-tetrahydro-furan-2-ol (9r,10r)-9-(s-glutathionyl)-10-hydroxy-9,10-dihydrophenanthrene 5-fluorotryptophan (9s,10s)-9-(s-glutathionyl)-10-hydroxy-9,10-dihydrophenanthrene 1-hydroxy-2-s-glutathionyl-3-para-nitrophenoxy-propane 3-hydroxybutyryl-coenzyme a 12b9m 5-(dodecylthio)-1h-1,2,3-triazole-4-carboxylic acid 3-decyl-2,5-dioxo-4-hydroxy-3-pyrroline 4-carboxy-5-(1-pentyl)hexylsulfanyl-1,2,3-triazole (2s)-2-hydroxyoctanoic acid 3-(indol-3-yl) lactate 4-[(5-methoxy-2-methylphenoxy)methyl]pyridine 2-[(2-methoxy-5-methylphenoxy)methyl]pyridine 2,6-dicarboxynaphthalene 4-carboxycinnamic acid 2-[4-({[(3,5-dichlorophenyl)amino]carbonyl}amino)phenoxy]-2-methylpropanoic acid 5-hydroxymethyl-2-furfural 1,3,5-benzenetricarboxylic acid 5-isopropyl-1h-pyrazole-3-carboxylic acid 5-(3-chloro-benzyl)-1h-pyrazole-3-carboxylic acid 5-butyl-1h-pyrazole-3-carboxylic acid 1h-pyrazole-3-carboxylic acid 2-(4-phenylbutyl)pyrido[2,3-d]pyrimidin-4(3h)-one (+)-5-(5-bromothiophen-3-yl)-5-methyl-4-oxo-4,5-dihydro-furan-2-carboxylic acid 2-(3-(naphthalen-2-yl)propanamido)benzoic acid 2-(3-biphenyl-4-yl-propionylamino)-benzoic acid 2-(6-phenylhexyl)pyrido[2,3-d]pyrimidin-4(3h)-one 4,5,6,7-tetrahydro-1h-indazole-3-carboxylic acid 2-(2-(4-tert-butylphenoxy)acetamido)benzoic acid 3-pyridine-acetic acid 5-phenethyl-1h-pyrazole-3-carboxylic acid 5-methyl nicotinic acid 5-benzyl-1h-pyrazole-3-carboxylic acid 2-(cinnamyloxy)pyrido[2,3-d]pyrimidin-4(3h)-one 5-propyl-1h-pyrazole-3-carboxylic acid 5-(4-chloro-benzyl)-1h-pyrazole-3-carboxylic acid 5-(3-phenyl-propyl)-1h-pyrazole-3-carboxylic acid 2-hydroxyoctanoic acid 3-hydroxyoctanoic acid 5-methyl-5-(5-methylthiophen-3-yl)-4-oxo-4,5-dihydrofuran-2-carboxylic acid 4-(n-propyl)amino-3-nitrobenzoic acid 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine 3-(6-allyloxy-2-naphthyl)-1-(4-piperidylmethyl)pyrazolo[3,4-d]pyrimidin-4-amine 1,2-diamino cyclopentane-based derivative 22 1,2-diamino cyclopentane-based derivative 27 1,2-diamino cyclopentane-based derivative 16 1,2-diamino cyclopentane-based derivative 5 1,2-diamino cyclopentane-based derivative 26 1,2-diamino cyclopentane-based derivative 10 1,2-diamino cyclopentane-based derivative 24 1,2-diamino cyclopentane-based derivative 34 1,2-diamino cyclopentane-based derivative 6 1,2-diamino cyclopentane-based derivative 8 1,2-diamino cyclopentane-based derivative 19 1,2-diamino cyclopentane-based derivative 14 1,2-diamino cyclopentane-based derivative 12 1,2-diamino cyclopentane-based derivative 21 1,2-diamino cyclopentane-based derivative 29 1,2-diamino cyclopentane-based derivative 4 1,2-diamino cyclopentane-based derivative 23 1,2-diamino cyclopentane-based derivative 18 1,2-diamino cyclopentane-based derivative 9 1,2-diamino cyclopentane-based derivative 11 1,2-diamino cyclopentane-based derivative 31 1,2-diamino cyclopentane-based derivative 13 1,2-diamino cyclopentane-based derivative 30 1,2-diamino cyclopentane-based derivative 20 1,2-diamino cyclopentane-based derivative 7 1,2-diamino cyclopentane-based derivative 32 [3h]sb-674042 1,2-diamino cyclopentane-based derivative 25 1,2-diamino cyclopentane-based derivative 2 1,2-diamino cyclopentane-based derivative 3 1,2-diamino cyclopentane-based derivative 17 1,2-diamino cyclopentane-based derivative 1 1,2-diamino cyclopentane-based derivative 15 1,2-diamino cyclopentane-based derivative 33 7-(3-benzoyl-ureido)-heptanoic acid hydroxyamide 4-chloro-n-(5-hydroxycarbamoyl-pentyl)-benzamide 9,9,9-trifluoro-8-oxo-nonanoic acid phenylamide 8-(3-benzoyl-ureido)-octanoic acid hydroxyamide 7-mercapto-heptanoic acid quinolin-3-ylamide 8-(biphenyl-4-yloxy)-2-oxo-octanoic acid 8-(biphenyl-4-yl)-n-hydroxy-8-oxooctanamide 8-(biphenyl-3-yloxy)-1,1,1-trifluoro-octan-2-one 4sc-202 6-mercapto-hexanoic acid phenylamide 8-mercapto-octanoic acid phenylamide 7-(biphenyl-4-yloxy)-1,1,1-trifluoro-heptan-2-one 7-(biphenyl-4-yloxy)-heptanoic acid hydroxyamide 4-tert-butyl-n-hydroxybenzamide 7-(biphenyl-4-yloxy)-1-oxazol-2-yl-heptan-1-one 5-mercapto-pentanoic acid phenylamide 6-(2-bromo-acetylamino)-hexanoic acid phenylamide 8-oxo-8-phenyl-octanoic acid hydroxyamide 8-(4-bromophenyl)-n-hydroxy-8-oxooctanamide 7-biphenyl-4-yl-heptanoic acid hydroxyamide 6-phenoxy-hexane-1-thiol 5-(4-hydroxyphenyl)-3h-1,2-dithiole-3-thione 7-(biphenyl-3-yloxy)-1-oxazol-2-yl-heptan-1-one 1,1,1-trifluoro-8-(4-phenoxy-phenoxy)-octan-2-one 4-dimethylamino-n-(6-mercapto-hexyl)-benzamide 7-(4-(dimethylamino)phenoxy)-n-hydroxyheptanamide 6-benzenesulfinylhexanoic acid hydroxamide 6-(9h-carbazol-9-yl)-n-hydroxyhexanamide 4-benzoylamino-n-hydroxy-benzamide 8-phenyl-octanoic acid hydroxyamide 7-mercapto-heptanoic acid biphenyl-3-ylamide 6-phenylsulfanylhexanoic acid hydroxamide 4-benzenesulfonylamino-n-hydroxy-benzamide 7-mercapto-n-(4-phenylthiazol-2-yl)heptanamide 5-(4-chloro-phenyl)-pentanoic acid hydroxyamide 8-oxo-8-phenyl-octanoic acid 7-(1h-indol-5-yloxy)-n-hydroxyheptanamide 1,1,1-trifluoro-8-phenoxy-octan-2-one 4-butyrylamino-n-hydroxy-benzamide 7-mercapto-heptanoic acid pyridin-3-ylamide (e)-8-biphenyl-4-yl-1-oxazol-2-yl-oct-7-en-1-one 7-phenoxy-heptanoic acid hydroxyamide 4-phenylbutyrohydroxamic acid 7-mercapto-heptanoic acid biphenyl-4-ylamide 2-(methylsulfonylthio)ethyl 2-propylpentanoate 4-hydroxy-n-(5-hydroxycarbamoyl-pentyl)-benzamide 6-benzenesulfonylhexanoic acid hydroxamide 8-(biphenyl-4-yloxy)-1,1,1-trifluoro-octan-2-one 6-(3-benzoyl-ureido)-hexanoic acid hydroxyamide 7-(naphthalen-2-yloxy)-1-oxazol-2-yl-heptan-1-one 7-mercapto-heptanoic acid benzothiazol-2-ylamide 7-mercapto-heptanoic acid phenylamide 9-(biphenyl-4-yloxy)-1,1,1-trifluoro-nonan-2-one 2-(benzyloxy)-n7-hydroxy-n1-phenylheptanediamide 2-(allyloxy)-n8-hydroxy-n1-phenyloctanediamide 5-(biphenyl-4-yl)-pentanoic acid n-hydroxyamide 2,2-bis(3-fluorophenyl)-n-hydroxyacetamide 2,2-bis(4-fluorophenyl)-n-hydroxyacetamide 2,2,2-trifluoro-1-{5-[(3-phenyl-5,6-dihydroimidazo[1,2-a]pyrazin-7(8h)-yl)carbonyl]thiophen-2-yl}ethane-1,1-diol 2,2-bis(4-chlorophenyl)-n-hydroxyacetamide (s)-2-amino-n-cyclopentyl-7-mercaptoheptanamide 5-(4-methyl-benzoylamino)-biphenyl-3,4'-dicarboxylic acid 3-dimethylamide-4'-hydroxyamide 4-(dimethylamino)-n-[7-(hydroxyamino)-7-oxoheptyl]benzamide 6-(2-mercaptoacetamido)-n-phenylhexanamide (2e)-n-hydroxy-3-[1-methyl-4-(phenylacetyl)-1h-pyrrol-2-yl]prop-2-enamide 9-mercapto-8-oxo-n-phenylnonanamide (2r,3r,4s,5r)-2-acetamido-3,4-dihydroxy-5-hydroxymethyl-piperidine 2-acetamido-2-deoxy-d-glucono-1,5-lactone (5-(1-benzyl-1h-indazol-3-yl)furan-2-yl)methanol 8-bromo-adenosine-5'-monophosphate 5'-o-(n-ethyl-sulfamoyl)adenosine 1d09c3 3-hydroxyglutaric acid (z)-7-octedecan-9-ynoic acid 3-hydroxy-3-methyl-glutaric acid (r)-mevalonate 7,9-tetradecadiynoic acid 5-ketodihydromevinolin (s)-hmg-coa 9-octadecynoic acid 7,9-octadecadiynoic acid 2-cyclopropyl-4-substituted-phenoxy-quinoline derivative 1 (e)-5-octadecen-7,9-diynoic acid 6-hydroxy-7,9-octadecadiynoic acid (e)-octadecan-9-ynoic acid 3-(1,3 dodecadiynyl)-6-oxiranebutanoic acid (z)-5-octadecen-7,9-diynoic acid (7r,12r,13r)-13-formyl-12,14-dihydroxy-3,5,7-trimethyltetradeca-2,4-dienoic acid 1-(adamantan-1-yl)-2-(1h-imidazol-1-yl)ethanone 12-phenylheme 1-({2-[2-(4-chlorophenyl)ethyl]-1,3-dioxolan-2-yl}methyl)-1h-imidazole 2-phenylheme 4-(dimethylamino)butyl imidothiocarbamate 2-(2-iodo-benzoyl)-cyclohexane-1,3-dione 2-propionyl-cyclohexane-1,3-dione 3-hydroxy-2-propionylcyclohex-2-enone (4-hydroxy-phenoxy)-acetic acid 2-(2-bromo-benzoyl)-cyclohexane-1,3-dione 2-(2-methyl-benzoyl)-cyclohexane-1,3-dione 2-(2-methoxy-benzoyl)-cyclohexane-1,3-dione 3-hydroxy-4-phenyl-5h-furan-2-one 2-acetyl-3-hydroxycyclohex-2-enone 2-acetyl-cyclohexane-1,3-dione 2-cyclopropanecarbonyl-cyclohexane-1,3-dione 2-(2-chloro-benzoyl)-cyclohexane-1,3-dione 2-(2-nitro-benzoyl)-cyclohexane-1,3-dione 3-(4-nitrophenyl)-1h-pyrazole 3-phenyl-5-(1h-pyrazol-3-yl)isoxazole 4-{[4-(4-fluoro-3-methylphenyl)-1,3-thiazol-2-yl]amino}-2-hydroxybenzoic acid 4-(benzhydryloxy)-1-[3-(1h-tetraazol-5-yl)propyl]piperidine 1-phenyl-1h-pyrazole-4-carboxylic acid 2-(2f-benzothiazolyl)-5-styryl-3-(4f-phthalhydrazidyl)tetrazolium chloride 9-deazaguanine 3h-pyrazolo[4,3-d]pyrimidin-7-ol (s)-(+)-dimethindene maleate 2-(2-thiazolyl)ethanamine 2-(9,10-dihydroanthracen-9-yl)-n-methylethanamine (-)-trans-h2-pat 9-(2-aminoethyl)-9,10-dihydroanthracene (+)-cis-h2-pat 4,4-diphenylbutan-1-amine 8r-lisuride 9-phenyl-2,3-dihydro-1h-indeno[2,1-c]pyridine 2-(3-chlorophenyl)histamine (s)-cetirizine 3,3-diphenylpropan-1-amine 9-(2-aminopropyl)-9,10-dihydroanthracene 9-(aminomethyl)-9,10-dihydroanthracene (+)-trans-h2-pat 1-[(furan-2(5h)-one)-4-methyl]-desloratadine 9-oh-risperidone 2-(3-iodophenyl)histamine 1-(4-p-tolyl-butyl)-piperidine (+/-)-cis-h2-pat 2-(3-bromophenyl)histamine 2-pyridylethylamine [125i]iodoaminopotentidine (s)-2-methyl-1-(2-m-tolyl-ethyl)-pyrrolidine (r)-4-(2-(2-methylpyrrolidin-1-yl)ethyl)pyridine (s)-1-(3-methoxyphenethyl)-2-methylpyrrolidine 4-[3-(4-butyl-phenoxy)-propyl]-1h-imidazole [123i]iodoproxyfan 1-(3-methoxyphenethyl)pyrrolidine 4-((2r,3s)-2-methyl-pyrrolidin-3-yl)-1h-imidazole 2-[4-(1-ethyl-propyl)-piperazin-1-yl]-quinoline (s)-1-(4-nitrophenethyl)-2-methylpyrrolidine 4-isopropyl-2-(phenoxymethyl)morpholine 1-(3-(3-phenylpropoxy)propyl)piperidine 3-((1h-imidazol-4-yl)methyl)pyridine (s)-3-(1h-imidazol-4-yl)propyl sec-butylcarbamate 2-(3-methyl-3h-imidazol-4-yl)-ethylamine 5-(2-(pyrrolidin-1-yl)ethyl)isothiazole 1-(3-(2-(3-methoxyphenoxy)ethoxy)propyl)azepane 4-butyl-1-[3-(phenylpropoxy)propyl]piperidine 4-((1h-imidazol-4-yl)methyl)-1-phenylpiperidine 4-[3-(4-ethynyl-phenoxy)-propyl]-1h-imidazole (s)-4-(2-(2-methylpyrrolidin-1-yl)ethyl)pyridine 4-[3-(4-methoxy-phenoxy)-propyl]-1h-imidazole 2-(2-(pyrrolidin-1-yl)ethyl)-1h-indole 4-(2-(3-tert-butylphenylamino)ethyl)-1h-imidazole 2-[2-(1h-imidazol-4-yl)-cyclopropyl]-ethylamine (s)-2-(2-(2-methylpyrrolidin-1-yl)ethyl)pyridine 4-benzyl-1-[3-phenylpropoxy)propyl]piperidine 2-(2-(pyrrolidin-1-yl)ethyl)pyridine 1-(2-p-tolyl-ethyl)-pyrrolidine 4-(7-methyl-oct-3-ynyl)-1h-imidazole (r)-1-(3-methoxyphenethyl)-2-methylpyrrolidine 4-(6-cyclopentyl-hex-3-ynyl)-1h-imidazole 2-(ethoxycarbonyl)-1h-indole-5-carboxylic acid 5-ethyl-2-(2-(pyrrolidin-1-yl)ethyl)pyridine 4-(2-(4-methylphenylamino)ethyl)-1h-imidazole (1r,2r)-2-(1h-imidazol-4-yl)-1-methyl-propylamine 2-(4-cyclopentyl-piperazin-1-yl)-quinoline 2-(4-propyl-piperazin-1-yl)-quinoline (s)-2-(2-(2-methylpyrrolidin-1-yl)ethyl)phenol 4-((1h-imidazol-4-yl)methyl)-1-heptylpiperidine 4-((2s,3r)-2-methyl-pyrrolidin-3-yl)-1h-imidazole 4-(2-(pyrrolidin-1-yl)ethyl)pyridine 1-[2-(2,4,6-trimethyl-phenyl)-ethyl]-pyrrolidine (r)-alpha-methylhistamine (s)-1-(2-methoxyphenethyl)-2-methylpyrrolidine 4-hept-3-ynyl-1h-imidazole 2-((1h-imidazol-4-yl)methyl)pyridine 2-(2-(pyrrolidin-1-yl)ethyl)phenol 2-(4-methyl-piperazin-1-yl)-quinoline 4-(2-(cyclohexylamino)ethyl)-1h-imidazole 1-(2-m-tolyl-ethyl)-pyrrolidine 4-(2-(4-tert-butylphenylamino)ethyl)-1h-imidazole 4-(3-phenoxy-propyl)-1h-imidazole (r)-3-(2-(2-methylpyrrolidin-1-yl)ethyl)pyridine 4-propyl-1-[3-(phenylpropoxy)propyl]piperidine 4-benzylidene-1-(cyclobutylo)piperidine derivative 1 [125i]iodophenpropit 2-(4-cyclopropyl-piperazin-1-yl)-quinoline (1s,2s)-2-(1h-imidazol-4-yl)-cyclopentylamine 2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-b]pyridine 1-(3-(4-(2-fluoroethyl)phenoxy)propyl)piperidine (r)-6-(2-(2-methylpyrrolidin-1-yl)ethyl)quinoline (r)-1-(4-methoxyphenethyl)-2-methylpyrrolidine (r)-1-(4-nitrophenethyl)-2-methylpyrrolidine (r)-2-(2-(2-methylpyrrolidin-1-yl)ethyl)pyridine 5-methoxy-2-(2-(pyrrolidin-1-yl)ethyl)-1h-indole 1-(4-nitrophenethyl)pyrrolidine 4-(6-cyclohexyl-hex-3-ynyl)-1h-imidazole 2-(4-isopropyl-piperazin-1-yl)-quinoline (s)-alpha-methylhistamine 4-(7,7-dimethyl-oct-3-ynyl)-1h-imidazole (r)-2-methyl-1-(2-m-tolyl-ethyl)-pyrrolidine (1r,2s)-2-(1h-imidazol-4-yl)-1-methyl-propylamine 4-(2-(4-cyclohexylphenylamino)ethyl)-1h-imidazole (1h-indol-2-yl)(piperazin-1-yl)methanone 1-(3-(4-(fluoromethyl)phenoxy)propyl)piperidine 4-(2-(3,4-dimethylphenylamino)ethyl)-1h-imidazole (s)-1-(4-methoxyphenethyl)-2-methylpyrrolidine (r)-2-(2-(2-methylpyrrolidin-1-yl)ethyl)phenol (r)-1-(2-methoxyphenethyl)-2-methylpyrrolidine (r)-3-(1h-imidazol-4-yl)propyl sec-butylcarbamate 4-(2-(phenylamino)ethyl)-1h-imidazole (r)-2-methyl-1-(2-p-tolyl-ethyl)-pyrrolidine 4-(2-(4-methoxyphenylamino)ethyl)-1h-imidazole (s)-2-methyl-1-(2-p-tolyl-ethyl)-pyrrolidine 1-(2-(naphthalen-2-yl)ethyl)pyrrolidine 2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-c]pyridine 2-((2-ethoxyphenoxy)methyl)-4-isopropylmorpholine 4-(8-phenyl-oct-3-ynyl)-1h-imidazole 4-hex-3-ynyl-1h-imidazole 5-phenyl-2-(4-(piperidin-1-yl)butyl)oxazole 1-(4-(benzyloxy)phenethyl)pyrrolidine 1-(2-methoxyphenethyl)pyrrolidine 1-(4-methoxyphenethyl)pyrrolidine 4-methylhistamine 6-(4-methylpiperazin-1-yl)pyrimidine-2,4-diamine 2-methylhistamine 6-(4-methylpiperazin-1-yl)-9hpurine 6-(4-methylpiperazin-1-yl)-9h-purin-2-amine [3h]jnj 7777120 9-benzyl-6-(4-methylpiperazin-1-yl)-9h-purine 2-(2-chlorophenylamino)-5-methylthiazol-4(5h)-one 1-(4-tert-butylphenylsulfonyl)-4-methoxyazepane 1-(phenylsulfonyl)butan-2-one 1-(3-methylpyridin-2-yl)-4-tosylpiperazine (5s)-2-(cyclooctylamino)-5-methyl-5-propyl-1,3-thiazol-4(5h)-one 2-(6-{[(3-chloro-2-methylphenyl)sulfonyl]amino}pyridin-2-yl)-n,n-diethylacetamide 1-{[(3r)-3-methyl-4-({4-[(1s)-2,2,2-trifluoro-1-hydroxy-1-methylethyl]phenyl}sulfonyl)piperazin-1-yl]methyl}cyclopropanecarboxamide 2-(adamantan-1-ylamino)-5,5-diethyl-oxazol-4-one 2-(2-chloro-4-fluorophenoxy)-2-methyl-n-[(1r,2s,3s,5s,7s)-5-(methylsulfonyl)-2-adamantyl]propanamide 1-(4-tert-butylphenylsulfonyl)azepan-4-ol 1-(2-adamantyl)-3-benzylpyrrolidin-2-one 3-epicorosolic acid methyl ester 1-(4-chlorophenyl)-2-(phenylsulfonyl)ethanone (5s)-2-{[(1s)-1-(4-fluorophenyl)ethyl]amino}-5-(2-hydroxy-2-propanyl)-5-methyl-1,3-thiazol-4(5h)-one 2-(phenylsulfonyl)-1-(thiophen-3-yl)ethanone 1-(3,4-dichlorophenyl)-2-(phenylsulfonyl)ethanone 2-(o-toluidino)-5-isopropylthiazol-4(5h)-one 2-(benzylamino)-5,5-diethyloxazol-4(5h)-one (5s)-2-{[(1s)-1-(2-fluorophenyl)ethyl]amino}-5-methyl-5-(trifluoromethyl)-1,3-thiazol-4(5h)-one 1-(4-nitrophenyl)-2-(phenylsulfonyl)ethanone (3,3-dimethylpiperidin-1-yl)(6-(3-fluoro-4-methylphenyl)pyridin-2-yl)methanone 1-phenyl-4-(1-phenyl-1h-tetrazol-5-yl)butan-2-one 1-(3-chloropyridin-2-yl)-4-tosylpiperazine 1-(4-ethylphenylsulfonyl)-4-phenylazepan-4-ol 3-acetyl-11-keto-ursolic acid 5,5-diethyl-2-(phenethylamino)oxazol-4(5h)-one 1-(4-fluorophenyl)-3-(phenylsulfonyl)propan-1-one 3-acetyl-11-keto-beta-boswellic acid 1-(4-methoxyphenylsulfonyl)-4-phenylazepan-4-ol 2-(phenylsulfonyl)-1-p-tolylethanone 1-(3,5-dimethylphenyl)-2-(phenylsulfonyl)ethanone (11-beta)-11,21-dihydroxy-pregn-4-ene-3,20-dione 1-phenyl-2-(1-phenyl-1h-tetrazol-5-yloxy)ethanone (2r)-1-[(4-tert-butylphenyl)sulfonyl]-2-methyl-4-(4-nitrophenyl)piperazine (1s,3r,4s,5s,7s)-4-{[2-(4-methoxyphenoxy)-2-methylpropanoyl]amino}adamantane-1-carboxamide 1-(4-fluorophenyl)-2-(phenylsulfonyl)ethanone 2-(cyclooctylamino)-5,5-diethyloxazol-4(5h)-one 11-keto-ursolic acid 1-(4-ethylpiperazin-1-yl)-2-phenylethanone 1-(3-methoxyphenyl)-2-(phenylsulfonyl)ethanone 1-(4-methoxyphenyl)-2-(phenylsulfonyl)ethanone 5-isopropyl-2-(phenylamino)thiazol-4(5h)-one 1-(3-nitropyridin-2-yl)-4-tosylpiperazine (5r)-2-[(2-fluorophenyl)amino]-5-isopropyl-1,3-thiazol-4(5h)-one 2-(o-toluidino)-5-ethylthiazol-4(5h)-one 11-keto-beta-boswellicacid 1-(1-phenyl-1h-tetrazol-5-ylthio)propan-2-one 1-phenyl-3-(phenylsulfonyl)propan-1-one 1-(4-chlorophenylsulfonyl)-4-phenylazepan-4-ol (4-methoxyphenyl)(4-phenylazepan-1-yl)methanone 3-benzyl-1-cyclohexylpyrrolidin-2-one 2-(4-tosylpiperazin-1-yl)nicotinonitrile 1,1-diphenyl-3-(phenylsulfonyl)propan-2-one 1-bromo-6-(3-hydroxyphenyl)-2-naphthol 3,3'-thiene-2,5-diyldiphenol 3-(2-naphthyl)phenol 3'-(5-chloro-2-thienyl)biphenyl-3-ol 3-[5-(4-hydroxyphenyl)-2-thienyl]-5-methylphenol 3-[5-(4-hydroxyphenyl)-2-thienyl]phenol 3-[5-(4-hydroxyphenyl)-1,3-thiazol-2-yl]phenol 16-(2',2'-dimethyl)-propylidene-estrone 3,3'-(3-methylthiene-2,5-diyl]diphenol 6-(3-hydroxyphenyl)-1-phenyl-2-naphthol 2-fluoro-4-[5-(3-hydroxyphenyl)-3-thienyl]phenol 3-[4-(4-hydroxyphenyl)-1,3-oxazol-2-yl]phenol 3-[5-(4-hydroxyphenyl)-1,3-oxazol-2-yl]phenol 6-oxo-16-formyl-estrone 16beta-cyano-estradiol 2-(3-hydroxyphenyl)quinolin-6-ol 3-[5-(3-fluorophenyl)-2-thienyl]phenol 3-hydroxy-7-(3-hydroxyphenyl)-1-naphthonitrile 16-(pyridin-2-yl)methylene-estradiol 1,1':4',1''-terphenyl-3,4''-diol 3-[4-(5-chloro-2-thienyl)pyridin-2-yl]phenol 3,4'-(thiophene-2,4-diyl)diphenol 3-[5-(3,4-difluorophenyl)-2-thienyl]phenol 16-(pyridin-3-yl)methyl-estradiol 16-(4-cyano-benzylidene)-estradiol 3,3',3''-thiene-2,3,5-triyltriphenol 3'-(1-benzothien-2-yl)biphenyl-3-ol 16-isobutylidene-estradiol 3-(6-hydroxy-2-naphthyl)benzoic acid 16-beta-ethoxymethyl-estrone 3-[2-(5-chloro-2-thienyl)pyridin-4-yl]phenol 3-fluoro-5-[5-(4-hydroxyphenyl)-2-thienyl]phenol 16-(pyridin-3-yl)methylene-estradiol 16-(thiophen-2-yl)methylene-estrone 2-fluoro-5-[5-(4-hydroxyphenyl)-2-thienyl]phenol 3,3'-thiene-2,4-diyldiphenol 16-(4-dimethylamino-benzylidene)-estradiol 3,3'-(1,2,4-thiadiazole-3,5-diyl)diphenol 16-(4-dimethylamino-benzylidene)-estrone 4'-(5-chloro-2-thienyl)biphenyl-3-ol 4'-(6-methoxypyridin-3-yl)biphenyl-3-ol 3,3'-(1,2,4-thiadiazol-2,5-diyl)diphenol 5-(6-hydroxy-2-naphthyl)pyridin-3-ol 4-methyl-1,1':4',1''-terphenyl-3,4''-diol 3-[5-(4-fluorophenyl)-2-thienyl]phenol 3-(5-phenyl-2-thienyl)phenol 4-[5-(3-hydroxyphenyl)-2-thienyl]benzene-1,2-diol 3,3'-(1,2,4,5-tetrazine-3,6-diyl)diphenol 3,3'-(1,3-thiazol-2,4-diyl)diphenol 16-(pyridin-4-yl)methyl-estradiol 4-fluoro-1,1':4',1''-terphenyl-3,3''-diol 3,3'-(3-phenylthiene-2,5-diyl)diphenol 3,3'-pyrazine-2,5-diyldiphenol 16-isobutylidene-estrone 5alpha-androstan-3,17-dione 6-oxo-estrone 3-[6-(5-chloro-2-thienyl)pyridin-2-yl]phenol 16-beta-hydroxymethyl-estradiol 3-[3-(4-hydroxyphenyl)isoxazol-5-yl]phenol 3,3'-pyridine-2,5-diyldiphenol 16-(pyridin-2-yl)methyl-estradiol 2-hydroxy-n,6-bis(3-hydroxyphenyl)-1-naphthamide 16-(pyridin-4-yl)methylene-estradiol 16-(2',2'-dimethyl)-propylidene-estradiol 7-hydroxy-3-(3-hydroxyphenyl)-1-naphthonitrile 3-(3-hydroxyphenyl)quinolin-7-ol 1-azepan-1-yl-2-phenyl-2-(4-thioxo-1,4-dihydro-pyrazolo[3,4-d]pyrimidin-5-yl)ethanone adduct (r)-3-hydroxydecanoyl-coa 4-(1h-imidazol-4-yl)-3-(5-ethyl-2,4-dihydroxy-phenyl)-1h-pyrazole 9-butyl-8-(2,5-dimethoxy-benzyl)-2-fluoro-9h-purin-6-ylamine 4-(1,3-benzodioxol-5-yl)-5-(5-ethyl-2,4-dihydroxyphenyl)-2h-pyrazole-3-carboxylic acid 4-(2-methoxyethoxy)-6-methylpyrimidin-2-amine 8-(6-bromo-benzo[1,3]dioxol-5-ylsulfanyl)-9-(3-isopropylamino-propyl)-adenine 6-(3-bromo-2-naphthyl)-1,3,5-triazine-2,4-diamine 9-butyl-8-(4-methoxybenzyl)-9h-purin-6-amine 4-bromo-6-(6-hydroxy-1,2-benzisoxazol-3-yl)benzene-1,3-diol 2-(1h-pyrrol-1-ylcarbonyl)benzene-1,3,5-triol 2-amino-4-(2,4-dichlorophenyl)-n-ethylthieno[2,3-d]pyrimidine-6-carboxamide 4-methyl-7,8-dihydro-5h-thiopyrano[4,3-d]pyrimidin-2-amine (3e)-3-[(phenylamino)methylidene]dihydrofuran-2(3h)-one 3-({2-[(2-amino-6-methylpyrimidin-4-yl)ethynyl]benzyl}amino)-1,3-oxazol-2(3h)-one 2-amino-4-[2,4-dichloro-5-(2-pyrrolidin-1-ylethoxy)phenyl]-n-ethylthieno[2,3-d]pyrimidine-6-carboxamide 9-butyl-8-(3-methoxybenzyl)-9h-purin-6-amine 8-(2,5-dimethoxy-benzyl)-2-fluoro-9-pent-9h-purin-6-ylamine 4-chloro-6-(4-piperazin-1-yl-1h-pyrazol-5-yl)benzene-1,3-diol 9-butyl-8-(2,5-dimethoxy-benzyl)-9h-purin-6-ylamine 9-butyl-8-(3,4,5-trimethoxybenzyl)-9h-purin-6-amine 9-butyl-8-(2-chloro-3,4,5-trimethoxy-benzyl)-9h-purin-6-ylamine 5-(5-chloro-2,4-dihydroxyphenyl)-n-ethyl-4-[4-(morpholin-4-ylmethyl)phenyl]isoxazole-3-carboxamide 2-[(2-methoxyethyl)amino]-4-(4-oxo-1,2,3,4-tetrahydro-9h-carbazol-9-yl)benzamide (5e,7s)-2-amino-7-(4-fluoro-2-pyridin-3-ylphenyl)-4-methyl-7,8-dihydroquinazolin-5(6h)-one oxime 3,6-diamino-5-cyano-4-(4-ethoxyphenyl)thieno[2,3-b]pyridine-2-carboxamide 4-(2,4-dichlorophenyl)-5-phenyldiazenyl-pyrimidin-2-amine 8-(2-chloro-3,4,5-trimethoxy-benzyl)-2-fluoro-9-pent-4-ylnyl-9h-purin-6-ylamine 8-(2,5-dimethoxy-benzyl)-2-fluoro-9h-purin-6-ylamine 4-{[(2r)-2-(2-methylphenyl)pyrrolidin-1-yl]carbonyl}benzene-1,3-diol 8-benzo[1,3]dioxol-,5-ylmethyl-9-butyl-9h- 8-(2-chloro-3,4,5-trimethoxy-benzyl)-9-pent-4-ylnyl-9h-purin-6-ylamine 8-benzo[1,3]dioxol-,5-ylmethyl-9-butyl-2-fluoro-9h-purin-6-ylamine 5-(5-chloro-2,4-dihydroxyphenyl)-n-ethyl-4-(4-methoxyphenyl)isoxazole-3-carboxamide 4-chloro-6-(4-{4-[4-(methylsulfonyl)benzyl]piperazin-1-yl}-1h-pyrazol-5-yl)benzene-1,3-diol 17-desmethoxy-17-aminogeldanamycin 5-(5-chloro-2,4-dihydroxyphenyl)-n-ethyl-4-piperazin-1-yl-1h-pyrazole-3-carboxamide 5-(5-chloro-2,4-dihydroxyphenyl)-n-ethyl-4-(4-methoxyphenyl)-1h-pyrazole-3-carboxamide 4-chloro-6-{5-[(2-morpholin-4-ylethyl)amino]-1,2-benzisoxazol-3-yl}benzene-1,3-diol (5e)-14-chloro-15,17-dihydroxy-4,7,8,9,10,11-hexahydro-2-benzoxacyclopentadecine-1,12(3h,13h)-dione 4-{4-[4-(3-aminopropoxy)phenyl]-1h-pyrazol-5-yl}-6-chlorobenzene-1,3-diol (5e)-12-chloro-13,15-dihydroxy-4,7,8,9-tetrahydro-2-benzoxacyclotridecine-1,10(3h,11h)-dione (5z)-12-chloro-13,15-dihydroxy-4,7,8,9-tetrahydro-2-benzoxacyclotridecine-1,10(3h,11h)-dione (5z)-13-chloro-14,16-dihydroxy-3,4,7,8,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,11(12h)-dione 2-(3-amino-2,5,6-trimethoxyphenyl)ethyl 5-chloro-2,4-dihydroxybenzoate 2-chlorodideoxyadenosine 3-(4-benzyl-piperidin-1-ylmethyl)-chromen-4-one 2-(2-methoxyphenoxy)-3-(piperidin-4-yl)pyridine 4-(2-fluoro-6-(2-fluorophenoxy)phenyl)piperidine 8-methoxy-2-(4-methyl-piperazin-1-yl)-quinoline [3h]8-oh-dpat 1-(3-(pentafluorosulfanyl)phenyl)propan-2-amine 1-(3-nitro-phenyl)-piperazine 2-(2-fluorophenoxy)-3-(piperidin-4-yl)pyridine 3-amino-1-(2-amino-5-methoxy-phenyl)-propan-1-one 1-(2-methoxy-phenyl)-4-propyl-piperazine 4-(3-fluoro-2-phenoxyphenyl)piperidine 8-methoxy-quinolin-2-ylamine 4-(2-(benzyloxy)-3-fluorophenyl)piperidine 4-(2-(benzyloxy)-6-fluorophenyl)piperidine 8-methoxy-1,2,3,4-tetrahydro-naphthalen-2-ylamine 1-(2-(phenoxymethyl)phenyl)piperazine 2-(2-amino-propyl)-5-bromo-4-methoxy-phenol 1-ethyl-4-(2-methoxy-phenyl)-piperazine 4-(2-(benzyloxy)phenyl)piperidine (r)-flurocarazolol 2-piperazin-1-yl-benzonitrile 4-(2-(4-fluorophenoxy)phenyl)piperidine 4-(2-(2-fluorobenzyloxy)phenyl)piperidine 1-(2-(benzyloxy)phenyl)piperazine 1-(4-bromo-2,5-dimethoxy-phenyl)-piperazine 2-(3-bromophenylthio)-n,n-dimethylethanamine 2-(4-methyl-piperazin-1-yl)-4-phenyl-pyrimidine [3h]p-mppf 1-benzyl-4-chroman-2-ylmethyl-piperazine 1-butyl-4-(2-methoxy-phenyl)-piperazine 2-(2-chlorophenoxy)-3-(piperidin-4-yl)pyridine 5-chloro-4-methyl-3,4-dihydroquinazolin-2-amine 4-(2-fluoro-6-(3-fluorophenoxy)phenyl)piperidine [3h]robalzotan 1-naphthalen-2-yl-piperazine 5-chloro-4-ethyl-3,4-dihydroquinazolin-2-amine 4-(2-fluoro-6-phenoxyphenyl)piperidine 1-naphthylpiperazine 1-(2-(2-fluorobenzyloxy)phenyl)piperazine [3h]nlx-112 8-methoxy-2-piperazin-1-yl-quinoline 3-(2-amino-propyl)-1h-indol-5-ol 2-(3-methoxy-phenyl)-1-methyl-ethylamine 1-(2,5-dimethoxy-4-methyl-phenyl)-piperazine 1-(2,5-dimethoxyphenyl)propan-2-amine 1-methyl-1,3-dihydro-indol-2-one 4-(2-phenoxyphenyl)piperidine 1-(2-phenoxyphenyl)piperazine 7-methoxy-1-naphthylpiperazine 1-(2-fluoro-phenyl)-piperazine 1-(2,5-dimethoxy-phenyl)-piperazine 1-(3-fluoro-phenyl)-piperazine 1-(2-butoxy-phenyl)-piperazine 5-chloro-3,4-dihydroquinazolin-2-amine 1-(2-(4-fluorophenoxy)phenyl)piperazine 3-(3-methanesulfonyl-phenyl)-1-propyl-pyrrolidine 3-(piperidin-4-yl)-2-(o-tolyloxy)pyridine 8-methoxy-4-methyl-3,4-dihydroquinazolin-2-amine 1-(2-((3-fluorophenoxy)methyl)phenyl)piperazine [11c]way100635 (s)-flurocarazolol 4-(2-fluoro-6-(4-fluorophenoxy)phenyl)piperidine 5-methoxy-n,n-dimethyltryptamine 4-(2-(2-fluoro-5-methylphenoxy)phenyl)piperidine 1,2,3,4-tetrahydro-naphthalen-2-ylamine 4-(2-(4-fluorobenzyloxy)phenyl)piperidine (3-chloro-phenyl)-piperazin-1-yl-methanone 1-(2-(3-fluorophenoxy)phenyl)piperazine 4-(2-(3-chlorophenoxy)phenyl)piperidine 2-dipropylamino-1,2,3,4-tetrahydro-anthracen-9-ol 2-(2-methoxy-phenyl)-1-methyl-ethylamine 1-(7-methoxy-naphthalen-2-yl)-piperazine 2-phenoxy-3-(piperidin-4-yl)pyridine 1-(2-ethoxy-phenyl)-piperazine 1-(2-(2-chlorophenoxy)pyridin-3-yl)piperazine 2-(biphenyl-3-ylthio)-n,n-dimethylethanamine 2-(4-bromo-phenyl)-1-methyl-ethylamine 2-(4-bromo-2-methoxy-phenyl)-1-methyl-ethylamine 4-(1h-indol-4-yloxy)-1-(isopropylamino)butan-2-ol 2-(5-methoxy-1h-indol-3-yl)-1-methyl-ethylamine 1-(2-isopropoxy-phenyl)-piperazine 2-piperazin-1-yl-phenol 3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1h-indole 5-ct 4-(2-(3-fluorophenoxy)phenyl)piperidine 2-(4-benzyl-piperidin-1-ylmethyl)-chroman-4-one 5,6-dichloro-3,4-dihydroquinazolin-2-amine 2-(2'-methyl-biphenyl-3-yl)-ethylamine 9-methoxy-1,2,3,4-tetrahydro-anthracen-2-ylamine 1-(2-methoxyphenyl)-4-pentylpiperazine 5-isopropyl-3-(2-pyrrolidin-1-yl-ethyl)-1h-indole 2-methyl-5-ht [11c]az10419369 5-ethyl-3-(2-pyrrolidin-1-yl-ethyl)-1h-indole 5-amino-3-(n-methylpiperidin-4-yl)-1h-indole 2-(5-nonyloxy-1h-indol-3-yl)-ethylamine 2-(5-thiophen-2-yl-1h-indol-3-yl)-ethylamine [125i]gti [3h]sumatriptan [3h]gr 125,743 [n-methyl-3h(3)]az-10419369 [2-(5-ethyl-1h-indol-3-yl)-ethyl]-dimethyl-amine [3h]eletriptan 2-(2,6-dimethyl-benzyl)-4,5-dihydro-1h-imidazole [3h]5-ct [3h]5-ht 5-bodmt 2-(5-fluoro-1h-indol-3-yl)ethanamine [125i]lsd 3-dimethylaminomethyl-1-methyl-1h-indol-4-ol 1-(2,6-dimethoxy-4-methylphenyl)propan-2-amine (r,s)-1-(6-fluoro-1h-indol-1-yl)propan-2-amine (2s)-1-(5-fluoro-1h-indazol-1-yl)propan-2-amine [2-(4-fluoro-1h-indol-3-yl)-ethyl]-dimethyl-amine 2-(piperazin-1-yl)-5,6,7,8-tetrahydroquinoline 6-methoxy-2,3,4,9-tetrahydro-1h-beta-carboline 1-((s)-2-aminopropyl)-7-fluoro-1h-indazol-6-ol 1-((r)-2-aminopropyl)-1h-indazol-6-ol 1-(4-bromo-2,5-difluorophenyl)-2-aminopropane 7-chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 5-methoxy-4,9-dihydro-3h-beta-carboline 1-(10-bromoanthracen-9-yl)-2-aminopropane (e)-2-(4-fluorostyryl)-5-(phenylsulfinyl)pyridine 3-(2-dimethylamino-ethyl)-1-methyl-1h-indol-4-ol 4-methoxy-9-aminomethyl-9,10-dihydroanthracene 3-(2-dimethylamino-ethyl)-1h-indol-6-ol 8-bromo-2,3,4,9-tetrahydro-1h-beta-carboline 3-(2-dimethylamino-ethyl)-2-methyl-1h-indol-4-ol 5-methoxytryptamine 2,5-dimethoxy-4-bromophenethylamine 2,2-diphenyl-ethylamine 3-(2-pyrrolidin-1-yl-ethyl)-1h-indol-4-ol 6,7-dichloro-2,3,4,5-tetrahydro-1h-3-benzazepine 5-bromo-2,3,4,9-tetrahydro-1h-beta-carboline 2,5-dimethoxy-4-ethylthioamphetamine 3-methoxy-9-aminomethyl-9,10-dihydroanthracene 2-(3,5-dimethoxy-4-phenethoxyphenyl)ethanamine 3-(2-dimethylamino-propyl)-1h-indol-4-ol (2s)-1-(6-methoxy-1h-indazol-1-yl)propan-2-amine (r,s)-1-(5-bromo-1h-indol-1-yl)propan-2-amine 4-(10h-anthracen-9-ylidene)-1-methyl-piperidine (r,s)-1-(5-fluoro-1h-indol-1-yl)propan-2-amine 2-phenyl-3-(2-piperidin-1-yl-ethyl)-1h-indole (r)-(+)-(4,5,6-trimethoxyindan-1-yl)methanamine 1-((s)-2-aminopropyl)-7-chloro-1h-indazol-6-ol (2-indol-1-yl-ethyl)-dimethyl-amine [2-(6-methoxy-indol-1-yl)-ethyl]-dimethyl-amine 3-dimethylaminomethyl-1h-indol-4-ol (s)-1-(5,6-difluoro-1h-indol-1-yl)propan-2-amine (2s)-1-(1h-furo[2,3-g]indazol-1-yl)propan-2-amine 5-chloro-n-(pyridin-3-yl)indoline-1-carboxamide 1-(4-ethyl-2,5-dimethoxyphenyl)propan-2-amine 1-butyl-3-(2-dimethylamino-ethyl)-1h-indol-4-ol 8-bromo-4,9-dihydro-3h-beta-carboline 2-methoxy-9-aminomethyl-9,10-dihydroanthracene 2-phenyl-3-piperidin-4-yl-1h-indole 3-(1-benzyl-piperidin-4-yl)-2-phenyl-1h-indole 8-chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole (1-phenethyl-piperidin-4-yl)-phenyl-methanone 3-(1-methyl-piperidin-4-yl)-2-phenyl-1h-indole 3-(1-phenethyl-piperidin-4-yl)-2-phenyl-1h-indole 1-methoxy-9-aminomethyl-9,10-dihydroanthracene (r,s)-1-(5-methyl-1h-indol-1-yl)propan-2-amine 4-bromo-2,5-dimethoxyphenethylamine [11c]volinanserin 6-chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole 7,8,9,10-tetrahydro-6h-furo-[3,2-g][3]benzazepine [18f]altanserin 4-benzyl-1-methyl-piperidine hydrochloride 1-((s)-2-aminopropyl)-7-iodo-1h-indazol-6-ol 8-methoxy-4,9-dihydro-3h-beta-carboline 5-methoxy-2,3,4,9-tetrahydro-1h-beta-carboline (2s)-1-(6-fluoro-1h-indazol-1-yl)propan-2-amine 1-(3-(phenylthio)propyl)-4-m-tolylpiperazine 4-(4-fluoro-benzyl)-piperidine hydrochloride 6-chloro-n-(pyridin-3-yl)indoline-1-carboxamide (r)-3-(4-propylmorpholin-2-yl)phenol (r,s)-1-(5-chloro-1h-indol-1-yl)propan-2-amine 3-phenyl pyrazole derivative 1 [125i]doi 1-(2-aminoethyl)-1h-indazol-6-ol 8-methoxy-2,3,4,9-tetrahydro-1h-beta-carboline 1-((s)-2-aminopropyl)-7-methyl-1h-indazol-6-ol 6-bromoaplysinopsin 7,8,9,10-tetrahydro-6h-furo-[2,3-g][3]benzazepine 3-(3-dimethylamino-propyl)-1h-indol-4-ol 5-meo-dmt 2-(1h-indol-3-yl)-n,n-dimethylethanamine (s)-(-)-(4,5,6-trimethoxyindan-1-yl)methanamine (e)-2-(4-fluorostyryl)-5-(phenylsulfonyl)pyridine 9-(n-benzylaminomethyl)-9,10-dihydroanthracene (r)-1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine (5-methoxy-1h-indol-3-yl)methanamine [3h]lsd 6-fluoromelatonin [3h]mesulergine (-)-norfenfluramine (+)-norfenfluramine 1-(piperazin-1-yl)isoquinoline 4-(piperazin-1-yl)-7h-pyrrolo[2,3-d]pyrimidine 6-(piperazin-1-yl)-9-propyl-9h-purine 1-(2-dimethylamino-ethyl)-1h-indol-4-ol 6-methyl-4-(piperazin-1-yl)furo[2,3-d]pyrimidine 4-(piperazin-1-yl)thieno[3,2-c]pyridine 6-bromo-2'-de-n-methylaplysinopsin 6-bromo-8-(piperazin-1-yl)imidazo[1,2-a]pyrazine 4-(piperazin-1-yl)furo[3,2-c]pyridine 4-(piperazin-1-yl)thieno[2,3-d]pyrimidine 4-(piperazin-1-yl)thieno[3,2-d]pyrimidine 10,11-dihydro-5h-dibenzo[b,f]azepine 6-(4-methyl-piperazin-1-yl)-phenanthridine 4-((naphthalen-2-yloxy)methyl)piperidine 7-(piperidin-4-ylmethoxy)-2-naphthonitrile (s)-zacopride 1-(biphenyl-4-yl)-3-(4-(piperidin-1-yl)butyl)urea [3h](s)-zacopride 2-(4-benzyl-piperazin-1-yl)-benzothiazole [3h]gr65630 5-hydroxyindole 2-(1h-imidazol-4-ylmethyl)-4-phenyl-thiazole 3alpha-(2'-indolecarbonyloxy)-nortropane [3h]ramosetron 3alpha-(1'-methyl-2'-indolecarbonyloxy)-tropane 1-phenylbiguanide [3h]granisetron 4-benzoxazo-2-yl-1,4-diazabicyclo[3.2.2]nonane [123i]sb 207710 (r)-zacopride [11c]sb207145 4-methyl-n-propyl-3,4-dihydroquinazolin-2-amine 8-chloro-3,4-dihydroquinazolin-2-amine 3,4-dihydroquinazolin-2-amine hydrobromide 4-propyl-3,4-dihydroquinazolin-2-amine 4-ethyl-3,4-dihydroquinazolin-2-amine 1-benzenesulfonyl-3-piperidin-4-yl-1h-indole 2-(1-(phenylsulfonyl)-1h-indol-3-yl)ethanamine 4-(6-methoxy-1h-indol-1-ylsulfonyl)benzenamine 1-(phenylsulfonyl)-4-(piperazin-1-yl)-1h-indole 4-(3-methyl-indole-1-sulfonyl)-phenylamine 5-(4-methylpiperazin-1-yl)-3-tosyl-1h-indazole 4-(2-benzenesulfonylphenyl)piperazine 4-(indan-1-ylsulfanyl)-phenylamine 4-(4-benzenesulfonamidophenyl)piperazine 4-(piperazin-1-yl)-3-tosyl-1h-indazole 2-(3-benzenesulfonyl)phenyl-1-aminoethane 4-inden-(1e)-ylidenemethyl-phenylamine 4-(4-benzenesulfonylphenyl)piperazine 4-(1h-indol-1-ylsulfonyl)benzenamine 4-(3-benzenesulfonylphenyl)piperazine 4-(4,6-dinitro-1h-indol-1-ylsulfonyl)benzenamine 2-benzyl-4-piperazin-1-yl-1h-benzimidazole 4-(1h-inden-1-ylmethyl)-phenylamine 4-indan-1-ylmethyl-phenylamine 11c-gsk-215083 [2-(3h-indol-1-yl)-ethyl]-dimethyl-amine 2-(3-phenylthio)phenyl)-1-aminoethane 4-(4-methoxy-1h-indol-1-ylsulfonyl)benzenamine 3-(phenylsulfonyl)-1-(pyrrolidin-3-yl)-1h-indole 2-(3-(phenylsulfonyl)-1h-indol-1-yl)ethanamine 1-benzenesulfonyl-3-piperidin-3-yl-1h-indole [2-(3-benzyl-3h-indol-1-yl)-ethyl]-dimethyl-amine 4-(indane-1-sulfonyl)-phenylamine 6-(piperazin-1-yl)-3-tosyl-1h-indazole [2-(3-benzyl-indol-1-yl)-ethyl]-dimethyl-amine [2-(3-benzyl-3h-inden-1-yl)-ethyl]-methyl-amine 4-(naphthalene-1-sulfonyl)-phenylamine 4-(3h-inden-1-ylmethyl)-phenylamine 6-tosyl-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole 4-(piperazin-1-yl)-1h-indole 3-(phenylsulfonyl)-1-(piperidin-4-yl)-1h-indole 4-(3-benzenesulfonamidophenyl)piperazine 2-bromo-lsd 1-phenylthio-n,n-dimethyltryptamine 1-(3-(benzyloxy)-2-methylphenyl)piperazine 2-ethyl-5-methoxy-3-piperidin-4-yl-1h-indole 2-(1-benzyl-1h-indol-3-yl)-n,n-dimethylethanamine [125i]sb-258585 4-(1h-indol-3-ylmethyl)-phenylamine 4-((1h-indol-1-yl)methyl)benzenamine 2-(4-(benzenesulfonyl)phenyl)-1-aminoethane 2-(1-benzyl-1h-inden-3-yl)-n,n-dimethylethanamine 3-(phenylsulfonyl)-1-(piperidin-3-yl)-1h-indole 2-(1-tosyl-1h-indol-3-yl)ethanamine [3h]ro 63-0563 2-[1-(2-chloro-phenyl)-1h-pyrrol-2-yl]-ethylamine 2-(biphenyl-2-yloxy)-n,n-dimethylethanamine 4-oxadiazole derivative 1 2-(2-bromophenoxy)-n,n-dimethylethanamine 2-(biphenyl-2-ylthio)-n,n-dimethylethanamine (r)-8-phenyl-n,n-dipropylchroman-3-amine (2-biphenyl-3-yl-ethyl)-dimethyl-amine 2-(2-bromophenylthio)-n,n-dimethylethanamine 2-(1-o-tolyl-1h-pyrrol-3-yl)ethanamine 2,3-diamino-benzo[b]thiophene derivative 1 2,3-diamino-benzo[b]thiophene derivative 6 4-(benzylamino)-1-naphthol 2,3-diamino-benzo[b]thiophene derivative 8 2,3-dihydrobenzo[d]thiazole-2-thiol 4-(propylamino)naphthalen-1-ol 3-(1h-imidazol-4-yl)benzenethiol 4-(isopropylamino)-1-naphthol 5-phenyl-1h-1,2,3-triazole 1-methyl-l-tryptophan 4-(tert-butylamino)naphthalen-1-ol 2-hydroxygarveatin e 5-aminoquinolin-8-ol 4-amino-1,2,5-oxadiazole-3-carboximidamide 3-(4h-imidazol-4-yl)benzenethiol 4-(methylamino)naphthalen-1-ol 2,3-diamino-benzo[b]thiophene derivative 7 2,3-diamino-benzo[b]thiophene derivative 5 1h-indole-4,7-dione 4-fluorobenzenemethanethiol 1,4-naphthoquinone 2-(1h-imidazol-4-yl)benzene-1,3-diol 2-methoxy-1,4-naphthoquinone 2,3-diamino-benzo[b]thiophene derivative 3 2,2-dimethyl-2h-benzo[g]chromene-5,10-dione 4-phenylthiazole-2-thiol 4-chlorobenzenemethanethiol 4-(2-(diethylamino)ethylamino)-1-naphthol 4-methoxynaphthalen-1-amine 2,3-diamino-benzo[b]thiophene derivative 4 2,4-dichlorobenzenemethanethiol 4-(1h-1,2,3-triazol-5-yl)pyridine 3,4-dichlorobenzenemethanethiol 4-(cyclohexylamino)-1-naphthol 2,3-diamino-benzo[b]thiophene derivative 2 2-(1h-imidazol-4-yl)phenol 2-chlorobenzenemethanethiol 2-hydroxygarvin a 4-(ethylamino)naphthalen-1-ol 4-methoxybenzenemethanethiol 5-(isopropylamino)quinolin-8-ol 4-aminonaphthalen-1-ol 4-methylbenzenemethanethiol 4-phenylimidazole 4-(pent-3-ylamino)-1-naphthol 2,3-dichloro-1,4-naphthoquinone 4-(2-hydroxyethoxy)-1-naphthol 4-((1h-indazol-6-ylamino)methyl)benzene-1,2-diol (4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dione 4-((naphthalen-2-ylamino)methyl)benzene-1,2-diol 3-[5-(1h-imidazol-1-yl)-7-methyl-1h-benzimidazol-2-yl]-4-[(pyridin-2-ylmethyl)amino]pyridin-2(1h)-one 3-{[(9-cyano-9,10-dihydro-10-methylacridin-9-yl)carbonyl]amino}propanoic acid 2-(4-hydroxy-3-nitrophenyl)acetic acid (2-amino-3-phenyl-bicyclo[2.2.1]hept-2-yl)-phenyl-methanone 5-(para-nitrophenyl phosphonate)-pentanoic acid 6-{4-[hydroxy-(4-nitro-phenoxy)-phosphoryl]-butyrylamino}-hexanoic acid 4-nitro-benzylphosphonobutanoyl-glycine 4-(4-styryl-phenylcarbamoyl)-butyric acid (1s,2s,5s)2-(4-glutaridylbenzyl)-5-phenyl-1-cyclohexanol 9-(2-carboxyethyl)-10-methylanthracene endoperoxide 3-(10-methyl-9-anthryl)propanoic acid 3-(hydroxy-phenyl-phosphinoyloxy)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester 3-oxo-n-[(3s)-2-oxopyrrolidin-3-yl]dodecanamide 5-alpha-pregnane-3-beta-ol-hemisuccinate 1-[n-4'-nitrobenzyl-n-4'-carboxybutylamino]methylphosphonic acid 4-hydroxy-5-iodo-3-nitrophenylacetyl-epsilon-aminocaproic acid anion 4-hydroxy-3-nitrophenylacetyl-epsilon-aminocaproic acid anion 4-{[(z)-(5-oxo-2-phenyl-1,3-oxazol-4(5h)-ylidene)methyl]amino}butanoic acid (2s)-2-(butyryloxy)-3-hydroxypropyl nonanoate 4-{4-[2-(1a,7a-dimethyl-4-oxy-octahydro-1-oxa-4-aza-cyclopropa[a]naphthalen-4-yl) -acetylamino]-phenylcarbamoyl}-butyric acid (4z)-2,8:7,12:11,15:14,18:17,22-pentaanhydro-4,5,6,9,10,13,19,20,21-nonadeoxy-d-arabino-d-allo-d-allo-docosa-4,9,20-trienitol [4-(4-acetylamino-phenyl)-3,5-dioxo-4-aza-tricyclo[5.2.2.0 2,6]undec-1-ylcarbamoyloxy]-acetic acid 3-amino-benzo[b]thiophene-2-carboxylic acid amide 3-amino-5-(4-chlorophenyl)thiophene-2-carboxamide 6-phenyl-thieno[3,2-d]pyrimidin-4-ylamine 5-amino-2-p-tolyl-oxazole-4-carboxylic acid amide 2-amino-quinoline-3-carboxylic acid amide 4-amino-biphenyl-3-carboxylic acid amide 5-amino-2-phenyl-oxazole-4-carboxylic acid amide 2-amino-5-phenylthiophene-3-carboxamide 5-mercapto-2-nitro-benzoic acid 3-mercapto-1-(1,3,4,9-tetrahydro-b-carbolin-2-yl)-propan-1-one 2-[2-(2-cyclohexyl-2-guanidino-acetylamino)-acetylamino]-n-(3-mercapto-propyl)-propionamide (1h-indol-3-yl)-(2-mercapto-ethoxyimino)-acetic acid 6-chloropurine riboside, 5'-monophosphate 6-cl-imp 1-methoxy-3-(3-(pyridin-4-yl)-1h-indol-6-yl)urea 3-(pyridin-4-yl)-1h-indol-6-amine 3-(thiophen-3-yl)-1h-indol-6-amine 2-methyl-3-(pyridin-4-yl)-1h-indol-6-amine 1-(3-cyano-1-methyl-1h-indol-6-yl)-3-phenylurea 6-phenyl-3-(pyridin-4-yl)-1h-indole 2-methyl-3-(pyridin-4-yl)-1h-indole 1-methyl-1h-indole-3-carbonitrile 3-(furan-3-yl)-1h-indole 3-(3-cyano-1h-indol-6-yl)-1-methyl-1-phenylurea 6-bromo-1-methyl-3-(pyridin-4-yl)-1h-indole 6-bromo-3-(pyridin-4-yl)-1h-indole 3-(pyridin-4-yl)-1h-indol-7-amine 6-methoxy-5-oxazol-5-yl-2-phenyl-1h-indole 1-methyl-1h-indole-3-carbaldehyde 3-methoxy-4-(oxazol-5-yl)aniline 1-methyl-1h-indole-3-carboxamide 2-benzyl-6-methoxy-5-oxazol-5-yl-1h-indole 3-(furan-3-yl)-1-methyl-1h-indole [4-({5-(aminocarbonyl)-4-[(3-methylphenyl)amino]pyrimidin-2-yl}amino)phenyl]acetic acid 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate 2-deoxy-d-glucitol 6-(e)-vinylhomophosphonate 2-deoxy-glucitol-6-phosphate 3-(3-(carbamoyl)benzamido)-3-phenylpropanoic acid 3-(3-(benzamido)-5-nitrobenzamido)propanoic acid 3-(3-(carbamoyl)benzamido)propanoic acid 3-({4-[(1e)-3-morpholin-4-yl-3-oxoprop-1-en-1-yl]-2,3-bis(trifluoromethyl)phenyl}sulfanyl)aniline 1-acetyl-4-(4-{4-[(2-ethoxyphenyl)thio]-3-nitrophenyl}pyridin-2-yl)piperazine (s)-2-((s)-3-isobutyl-2,5-dioxo-4-quinolin-3-ylmethyl-[1,4]diazepan-1yl)-n-methyl-3-naphtalen-2-yl-propionamide 7a-[(4-cyanophenyl)methyl]-6-(3,5-dichlorophenyl)-5-oxo-2,3,5,7a-tetrahydro-1h-pyrrolo[1,2-a]pyrrole-7-carbonitrile 131i-radretumab 3,5-diiodotyrosine 4-(3-amino-1h-indazol-5-yl)-n-tert-butylbenzenesulfonamide 5-phenyl-1h-indazol-3-amine 4-[(2-{4-[(cyclopropylcarbamoyl)amino]-1h-pyrazol-3-yl}-1h-benzimidazol-6-yl)methyl]morpholin-4-ium 1,2,4-triazolo[1,5a]pyridine derivative 1 1,2,3,4,5,6-hexabromocyclohexane 6-o-tolylquinazolin-2-amine [(r)-(+)-deoxytylophorinidine (3e)-4-(1-methyl-1h-indol-3-yl)but-3-en-2-one [14c]tea 1-benzyl-7-chloro-4-hexyloxy-quinolinium 4-(4-phenoxybutoxy)-7h-furo[3,2-g]chromen-7-one 5-(4-phenylbutoxy)psoralen 2-methoxy-n-(3-methyl-2-phenyl-butyl)-benzamide [1-benzyl-1h-quinolin-(4e)-ylidene]-hexyl-amine 3-(benzyloxy)-2-(4-chlorophenyl)thiazolidin-4-one 2-phenoxy-1-(2-p-tolylthiazolidin-3-yl)ethanone 2-morpholino-2-phenyl-1,1-di(pyridin-3-yl)ethanol 2-phenyl-1,1-di(pyridin-3-yl)ethanol 3-methyl-2-morpholino-1,1-diphenylbutan-1-ol 2-amino-2-phenyl-1,1-di(pyridin-3-yl)ethanol 3-(4-methoxybenzyloxy)-2-phenylthiazolidin-4-one 2-morpholino-1,1-di(pyridin-3-yl)hexan-1-ol 2-morpholino-1,1-di(pyridin-3-yl)octan-1-ol 2-morpholino-1,1,2-triphenylethanol 3-(1-phenethyl-piperidin-3-yl)-2-phenyl-1h-indole 1-(1-phenyl-2-(2-propoxyphenyl)ethyl)piperazine (r)-n-isobutyl-n-(pyrrolidin-3-yl)-2-naphthamide 5-(3-butylpyrrolidin-3-yl)-1h-indole 1-(2-(6-fluoronaphthalen-2-yl)ethyl)piperazine 3-(benzo[b]thiophen-5-yl)-3-benzylpyrrolidine 3 9-dihydro-n-desmethyl-n-isopropylerythromycin a 4-(p-tolyl)spiro[chromene-2,4'-piperidine] 1-(1-(4-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (enantiomeric mix) 5-(3-benzylpyrrolidin-3-yl)-1h-indole (structural mix) 4-(2-thienyl)benzene-1,2-diamine 3-(1-methyl-piperidin-2-yl)-2-phenyl-1h-indole 4-(spiro[chromene-2,4'-piperidine]-4-yl)phenol 3-(1-benzyl-piperidin-3-yl)-2-phenyl-1h-indole 2-[4-(2-piperidin-1-ylethyl)phenoxy]benzothiazole [1-(4-p-tolyl-butyl)-piperidin-4-yl]-methanol (r)-3-(naphthalen-2-ylmethoxy)pyrrolidine 4-(3-thienyl)benzene-1,2-diamine) 1-(2-(2-(difluoromethoxy)phenyl)-1-phenylethyl)piperazine (enantiomeric mix) 4-benzenesulfonyl-1-(3-phenyl-propyl)-piperidine (s)-3-(naphthalen-2-ylmethoxy)pyrrolidine 5-chloro-3-ethyl-1-(4-fluoro-phenyl)-1h-indole 4-phenylspiro[chromene-2,4'-piperidine] 5-(3-benzylpyrrolidin-3-yl)-1-methyl-1h-indole 1-(1-(2-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (enantiomeric mix) 2-phenyl-3-piperidin-3-yl-1h-indole 3-(dimethylamino)-1-(4-heptylphenyl)propan-1-one (1r,5r)-30-oxo-19-oxa-2,6,10,12-tetraazahexacyclo[18.6.2.1^{2,5}.1^{14,18}.0^{8,12}.0^{23,27}]triaconta-8,10,14(29),15,17,20(28),21,23(27)-octaene-17-carbonitrile (structural mix) 4-benzenesulfonyl-1-phenethyl-piperidine 3-(1h-indol-3-yl)-n-methyl-3-phenylpropan-1-amine 5-(3-(4-fluorobenzyl)pyrrolidin-3-yl)-1h-indole 8-azabicyclo[3.2.1]octan-3-yloxy-benzamide (r)-ondansetron 3-(1-methyl-piperidin-3-yl)-2-phenyl-1h-indole 1-((2-chlorophenyl)diphenylmethyl)-1h-pyrazole (3r,4s)-293b 3s,4r-293b (s)-n-[1-(3-morpholin-4-yl-phenyl)-ethyl]-3-phenyl-acrylamide 4-[[2-[[4-chloro-3-(trifluoromethyl)phenyl]amino]-3h-benzimidazol-5-yl]oxy]-n-methyl-pyridine-2-carboxamide 3-(2-aminoquinazolin-6-yl)-1-(3,3-dimethylindolin-6-yl)-4-methylpyridin-2(1h)-one 1-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl]phenyl}-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea 3-methyl-1h-thieno[2,3-c]pyrazole-5-carboxamide 3-(2-aminoquinazolin-6-yl)-4-methyl-1-[3-(trifluoromethyl)phenyl]pyridin-2(1h)-one 3-((3-bromothiophen-2-yl)methylene)indolin-2-one 6-(1h-benzoimidazol-2-yl)-benzocyclohepten-7-one 5-(4-methoxy-phenyl)-1-phenyl-1h-benzoimidazole 4-(4-p-tolylamino-phthalazin-1-yl)-benzamide 2-(pyrimidin-4-ylamino)thiazole-5-carbonitrile (4-phenoxy-phenyl)-quinazolin-4-yl-amine 4-(4-m-tolylamino-phthalazin-1-yl)-benzamide (3-phenoxy-phenyl)-(5-phenyl-oxazol-2-yl)-amine 3-(5-thiophen-3-yl-pyridin-3-yl)-1h-indole 8-methyl-4h,7h-indolo[6,5,4-cd]indol-5-one 3-(4-aminophenyl)thieno[3,2-c]pyridin-4-amine 6-chloro-n-pyrimidin-5-yl-3-{[3-(trifluoromethyl)phenyl]amino}-1,2-benzisoxazole-7-carboxamide 3-phenyl-1,4-dihydroindeno[1,2-c]pyrazole 2-hydroxybenzamide derivative 2 2-hydroxybenzamide derivative 1 4sc-205 11h-benzo[a]carbazole (1s)-1-cyclopropyl-2-[(2s)-4-(2,5-difluorophenyl)-2-phenyl-2,5-dihydro-1h-pyrrol-1-yl]-2-oxoethanamine (2s)-4-(2,5-difluorophenyl)-n-methyl-2-phenyl-n-piperidin-4-yl-2,5-dihydro-1h-pyrrole-1-carboxamide [(4r)-4-(3-hydroxyphenyl)-1,6-dimethyl-2-thioxo-1,2,3,4-tetrahydropyrimidin-5-yl](phenyl)methanone 6-fluoro-2-methyl-9h-carbazole 3-(trifluoromethyl)-9h-carbazole 1-(trifluoromethyl)-9h-carbazole 2-methyl-6-(trifluoromethyl)-9h-carbazole 4'-(trifluoromethyl)-4-biphenylol 2-tert-butyl-7-(trifluoromethyl)-9h-carbazole 9h-carbazole-3-carbaldehyde 1-tert-butyl-9h-carbazole (5s)-5-(3-aminopropyl)-3-(2,5-difluorophenyl)-n-ethyl-5-phenyl-4,5-dihydro-1h-pyrazole-1-carboxamide 4'-trifluoromethyl-biphenyl-4-ylamine (s)-enastron 2,3,4,11-tetrahydro-1h-benzo[a]carbazole 4'-(trifluoromethyl)-4-biphenylsulfonamide 2-methyl-9h-carbazole 2-(trifluoromethoxy)-9h-carbazole 9h-carbazole-2-carbaldehyde 4'-(trifluoromethyl)-4-biphenylyl sulfamate 2-isopropyl-9h-carbazole 7-tert-butyl-9h-carbazole-3-carboxylic acid 4'-(trifluoromethyl)-4-biphenylyl carbamate (s)-dimethylenastron 3-methyl-6-(trifluoromethyl)-9h-carbazole 2-(trifluoromethyl)-9h-carbazole (2s)-4-(2,5-difluorophenyl)-n,n-dimethyl-2-phenyl-2,5-dihydro-1h-pyrrole-1-carboxamide 9-methyl-2-(trifluoromethyl)-9h-carbazole 2-tert-butyl-9h-carbazole 1-(7-methyl-9h-carbazol-3-yl)ethanone 2-tert-butoxy-9h-carbazole 4-(trifluoromethyl)biphenyl 3-tert-butyl-9h-carbazole 2-ethyl-9h-carbazole (4r)-4-(3-hydroxyphenyl)-n,n,7,8-tetramethyl-3,4-dihydroisoquinoline-2(1h)-carboxamide 2-(difluoromethyl)-9h-carbazole (5r)-n,n-diethyl-5-methyl-2-[(thiophen-2-ylcarbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide 3-[(5s)-1-acetyl-3-(2-chlorophenyl)-4,5-dihydro-1h-pyrazol-5-yl]phenol 4-fluorobenzoyl-phe-gly-leu-arg-trp-nh2 9-methoxy-5,11-dimethyl-6h-pyrido[4,3-b]carbazole 9-bromo-5,11-dimethyl-6h-pyrido[4,3-b]carbazole 3-hydroxydesaminokynurenine 3-hydroxyhippuric acid 3-methoxydesaminokynurenine 2-amino-4-[3-hydroxyphenyl]-4-hydroxybutanoic acid (2s)-3-[(r)-[(1s)-1-amino-3-phenylpropyl](hydroxy)phosphoryl]-2-benzylpropanoic acid 3-(2-aminoquinazolin-6-yl)-4-methyl-n-[3-(trifluoromethyl)phenyl]benzamide 1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine 2-(3,4,5-trihydroxy-benzylidene)-malononitrile {4-[(2s)-2-acetamido-3-({(1s)-1-[3-carbamoyl-4-(cyclohexylmethoxy)phenyl]ethyl}amino)-3-oxopropyl]-2-phosphonophenoxy}acetic acid 4-(3-chloro-phenoxy)-6,7-dimethoxy-quinazoline 3-(4-(o-toluidino)pyrimidin-2-ylamino)benzamide 5,6-diphenyl-n-(2-piperazin-1-ylethyl)furo[2,3-d]pyrimidin-4-amine 4-phenylsulfanyl-7h-pyrrolo[2,3-d]pyrimidine 2,3-diphenyl-n-(2-piperazin-1-ylethyl)furo[2,3-b]pyridin-4-amine 2,3,-dihydroxybenzoylserine 2,3-dihydroxy-benzoic acid 6-hydroxy-6-methyl-heptan-3-one 2-methoxy-3-isopropylpyrazine (4r)-limonene 1?,2?-epoxide 2-(sec-butyl)thiazole 2-isobutyl-3-methoxypyrazine 2-deoxy-2-fluoro-?-d-glucose 2-deoxy-2fluoro-glucose 2,5-dideoxy-2,5-imino-dl-glycero-d-manno-heptitol (1s,2s,3r,4s,5s)-2,3,4-trihydroxy-5-(hydroxymethyl)cyclohexyl (1e)-2-phenyl-n-(sulfooxy)ethanimidothioate 2,4-dihydroxy-7-(methyloxy)-2h-1,4-benzoxazin-3(4h)-one (s)-4-hydroxymandelonitrile 4-hydroxy-1,2,5-oxadiazole-3-carboxylic acid 2,3,5,6-tetrafluoro-4-methoxy-benzamide (r)-1-para-nitro-phenyl-2-azido-ethanol 2-(3-methoxybenzylthio)-2-phenylacetic acid (1,1-difluoro-pentadecyl)-phosphonic acid 2-oleoyl-lpa [1-bromo-(3s)-hydrox-4-(palmitoyloxy)butyl]phosphate [3-(biphenyl-4-yloxy)-propyl]-dimethyl-amine 29-methylidene-2,3-oxidosqualene (r)-2-((4-phenoxyphenoxy)methyl)piperidine 2-[4-(2-azepan-1-ylethoxy)phenoxy]benzothiazole 4-(4-propoxyphenoxy)phenol (2s)-2-amino-5-oxo-5-[(4-phenylmethoxyphenyl)amino]pentanoic acid 1-(4-phenoxyphenyl)piperazine 2-(7-(benzyloxy)-1h-indol-3-yl)ethanamine 2-(4-piperidin-1-ylmethylphenoxy)benzothiazole (r)-2-(4-benzylphenoxymethyl)pyrrolidine 1-[4-(4-iodophenoxy)phenyl]piperazine {4-[(2r)-pyrrolidin-2-ylmethoxy]phenyl}(4-thiophen-3-ylphenyl)methanone (r/s)-2-((4-benzylphenoxy)methyl)piperazine 2-(4-phenoxyphenoxy)ethanamine 2-[4-(2-morpholin-4-ylethoxy)phenoxy]benzooxazole 5-[2-(1h-pyrrol-1-yl)ethoxy]-1h-indole (r/s)-2-((4-benzylphenoxy)methyl)piperidine 1-[4-(benzothiazol-2-yloxy)benzyl]piperidin-4-ol 2-[4-(2-azepan-1-ylethoxy)phenoxy]benzooxazole 4-(4-butoxyphenoxy)phenol 3-(benzyloxy)pyridin-2-amine 4s-4,5-diamino-n-(4-phenoxyphenyl)pentanamide 1-(4-thiophen-2-ylphenyl)methanamine (4-(thiophen-2-yl)phenyl)methanamine (r)-2-((4-benzylphenoxy)methyl)piperidine 4-(4-(pentyloxy)phenoxy)phenol (s)-2-((4-phenoxyphenoxy)methyl)piperidine (r)-pyridin-4-yl[4-(2-pyrrolidin-1-ylethoxy)phenyl]methanol 1-(2,2'-bithiophen-5-yl)methanamine 2-(4-benzylphenoxy)ethanamine 4-amino-n-[4-(benzyloxy)phenyl]butanamide (r/s)-2-((4-phenoxyphenoxy)methyl)piperidine 1-(pentyloxy)-4-phenoxybenzene 4-[2-(4-benzylphenoxy)ethyl]pyridine 8(s)-amino-2(r)-methyl-7-oxononanoic acid 5-[2-(4-hydroxyphenyl)ethyl]benzene-1,3-diol 2-amino-n-[4-(phenylmethoxy)phenyl]-acetamide 1-butoxy-4-phenoxybenzene (r)-n-benzyl-4-(pyrrolidin-2-ylmethoxy)aniline (4-fluorophenyl)(pyridin-4-yl)methanone 4-(2-amino-1,3-thiazol-4-yl)phenol (3s,4r)-3-benzyl-7-isopropyl-chroman-4-ol (ltb4-(csa)4)2-glu-h conjugate 20-hydroxy-ltb4 12-epi ltb4 [3h]ltb4 12-hydroxyheptadecatrienoic acid 12r-hete (r)-atenolol 3h-indole-5,6-diol (r)-3-hydroxytetradecanoic acid (s)-aspartimide (r)-propylene glycol 4-methyl-umbelliferyl-n-acetyl-chitobiose 1-3 sugar ring of pentamannosyl 6-phosphate 1,4-butanediol 2-deoxy-2-fluoro-alpha-d-mannosyl fluoride 5-fluoro-beta-l-gulosyl fluoride 1-deoxymannojirimycin (1s,2s,3r,6r)-4-(hydroxymethyl)-6-(octylamino)cyclohex-4-ene-1,2,3-triol 5-thio-a/b-d-mannopyranosylamine (1r,2r,3r,4s,5r)-4-(benzylamino)-5-(methylthio)cyclopentane-1,2,3-triol (+/-)-2-(4'-butoxyphenyl)thiomorpholin-5-one 7-(3-chlorobenzyloxy)-4-carboxaldehyde-coumarin 3-aminoacetamido-4'-methylfuro[3,2-g]coumarin (e)-5-(3-chlorostyryl)isatin (r)-indan-1-yl-methyl-prop-2-ynyl-amine 6-chloro-n-(2-morpholinoethyl)nicotinamide 4-methyl-7-(2-oxocyclopentyloxy)-2h-chromen-2-one 2-phenyl-5h-indeno[1,2-d]pyrimidine 9-methyl-2,3,4,9-tetrahydro-1h-beta-carboline (s)-2-amino-1-(4-methylthiophenyl)-propane 2-bromo-n-(2-morpholinoethyl)nicotinamide 7-acetonyloxy-3-acetylamino-8-methoxycoumarin 4,9-dihydro-3h-beta-carboline 2-furan-2-yl-4,5-dihydro-1h-imidazole 7-bromo-2,3,4,9-tetrahydro-1h-beta-carboline 7-acetonyloxy-3,4-cyclopentene-8-methylcoumarin 1-(1-naphthyl)-2-aminopropane 3,4-benzo-7-acetonyloxy-8-methoxycoumarin (6-butoxy-2-naphthyl)-2-aminopropane (6-benzyloxy-2-naphthyl)-2-aminopropane (7-benzyloxy-2-oxo-2h-chromen-4-yl)acetonitrile (6-methylthio-2-naphthyl)isopropylamine 3,4-benzo-7-(beta-bromoallyloxy)-8-methylcoumarin (+/-)-2-phenylthiomorpholin-5-one 2-phenyl-9h-indeno[2,1-d]pyrimidine 8-(3-methoxybenzyloxy)caffeine 8-(3-fluorobenzyloxy)caffeine 8-[(3-trifluoromethyl)benzyloxy]caffeine (s)-2-amino-1-(4-propylthiophenyl)-propane 2-(4,5-dihydro-1h-imidazol-2-yl)quinoline 1-(2-naphthyl)-2-aminopropane (r/r)befloxatone 6-bromo-2,3,4,9-tetrahydro-1h-beta-carboline 2-chloro-n-(3-morpholinopropyl)nicotinamide 2-[7-(benzyloxy)-2-oxo-2h-chromen-4-yl]acetamide 3-chloro-n-(2-methyl-1h-indol-5-yl)benzamide 6,11-dihydro-5h-benzo[a]carbazole (+/-)-2-(4'-propoxyphenyl)thiomorpholin-5-one 5-bromo-4,9-dihydro-3h-beta-carboline 5-hydroxymethyl-3-pyrrol-1-yl-oxazolidin-2-one 4-chloro-n-(3-morpholinopropyl)nicotinamide 2-amino-1-(4-methylthiophenyl)propane 6-amino-9-methoxy-7h-furo[3,2-g]chromen-7-one 4,8-dimethyl-7-(2'-oxocyclohexyloxy)coumarin (6-propoxy-2-naphthyl)-2-aminopropane (r,s)-n-(r-phenylethyl)-1h-pyrrole-2-carboxamide 2-(naphthalen-2-yl)-4,5-dihydro-1h-imidazole 1-(3-(4-chlorobenzyl)quinoxalin-2-yl)hydrazine 6-methoxy-4,9-dihydro-3h-beta-carboline (+/-)-2-(4'-butoxyphenyl)thiomorpholine 1-(3-benzyl-6,7-dichloroquinoxalin-2-yl)hydrazine 4-chloro-n-(2-morpholinoethyl)nicotinamide 2-oxo-n-phenyl-2h-chromene-3-carboxamide 4-(aminomethyl)-7-(benzyloxy)-2h-chromen-2-one 6-hydroxy-n-(2-morpholinoethyl)nicotinamide (+/-)-2-(4'-methoxyphenyl)thiomorpholine 6-bromo-4,9-dihydro-3h-beta-carboline (e)-5-styrylisatin 3,4-benzo-7-acetonyloxy-8-methylcoumarin (6-methoxy-2-naphthyl)-2-aminopropane 2-phenethyl-4,5-dihydro-1h-imidazole 5,6-dichloro-n-(2-morpholinoethyl)nicotinamide (6-ethoxy-2-naphthyl)-2-aminopropane (+/-)-2-(4'-ethoxyphenyl)thiomorpholin-5-one 2-oxo-n-p-tolyl-2h-chromene-3-carboxamide 2-(2-cyclopentylidenehydrazinyl)-4-phenylthiazole 2-chloro-n-(2-morpholinoethyl)nicotinamide 1-(4-propoxyphenyl)propan-2-amine 1-(3-benzylquinoxalin-2-yl)hydrazine 5,6-dichloro-n-(3-morpholinopropyl)nicotinamide 1-(4-(benzyloxy)phenyl)propan-2-amine 2-phenoxymethyl-4,5-dihydro-1h-imidazole (+/-)-2-(4'-benzyloxyphenyl)thiomorpholine 3-benzyl-n-(2-morpholinoethyl)quinoxalin-2-amine (s)-2-amino-1-(4-butylthiophenyl)-propane (+/-)-2-(4'-ethoxyphenyl)thiomorpholine 3-methyl-2(1h)-thioxo-4(3h)-quinazolinone 2-(4-methoxyphenyl)-4,5-dihydro-1h-imidazole 2-(5-phenyl-furan-2-yl)-4,5-dihydro-1h-imidazole 8-(3-chlorobenzyloxy)caffeine 4-(2-oxo-2h-chromene-3-carboxamido)benzoic acid (+/-)-2-phenylthiomorpholine 8-benzyloxycaffeine 2-oxo-n-m-tolyl-2h-chromene-3-carboxamide 8-(3-methylbenzyloxy)caffeine 2-(3-benzylquinoxalin-2-ylamino)ethanol 7-acetonyloxy-3,4-cyclohexene-8-methylcoumarin 6-chloro-n-(3-morpholinopropyl)nicotinamide 7-methoxy-9h-beta-carboline 5-azidomethyl-3-pyrrol-1-yl-oxazolidin-2-one 2,3,4,5-tetrahydro-1h-pyrido[4,3-b]indole 5-methoxymethyl-3-pyrrol-1-yl-oxazolidin-2-one (s)-2-amino-1-(4-ethylthiophenyl)-propane (+/-)-2-(4'-methoxyphenyl)thiomorpholin-5-one 1-(4-butoxyphenyl)propan-2-amine 7-bromo-4,9-dihydro-3h-beta-carboline 9-(3-aminopropoxy)-7h-furo[3,2-g]chromen-7-one 3,4-dichloro-n-(2-methyl-1h-indol-5-yl)benzamide 6-fluoro-n-(2-morpholinoethyl)nicotinamide 2-(3,4-dimethoxyphenyl)-4,5-dihydro-1h-imidazole (e)-5-(3-fluorostyryl)isatin (+/-)-2-(4'-propoxyphenyl)thiomorpholine 1-(4-ethoxyphenyl)propan-2-amine 4-methyl-2h-benzofuro[3,2-g]chromen-2-one 8-(3-bromobenzyloxy)caffeine 2-(2-cycloheptylidenehydrazinyl)-4-phenylthiazole 7-methoxy-2-p-tolyl-4h-chromene-4-thione (+/-)-2-(4'-benzyloxyphenyl)thiomorpholin-5-one 2-(2-cyclohexylidenehydrazinyl)-4-phenylthiazole (s)(+)-7-methyl-2-p-tolylchroman-4-one (s)-n2-{4-[(3-chlorobenzyl)oxy]benzyl}alaninamide 2-(2,4-dichlorophenyl)-4,5-dihydro-1h-imidazole (s)(+)-7-fluoro-2-phenylchroman-4-one (s)-n2-{4-[(4-chlorobenzyl)oxy]benzyl}alaninamide 3-phenyl-9h-indeno[1,2-e][1,2,4]triazin-9-one 3-(3-methoxyphenyl)-6-methyl-2h-chromen-2-one 2-(4-fluorophenyl)-7-methoxy-4h-chromen-4-one 1,4-diphenyl-(1e,3e)-1,3-butadiene (s)-n2-{4-[(4-nitrobenzyl)oxy]benzyl}serinamide (e)-6-styrylisatin 7-fluoro-2-(4-fluorophenyl)-4h-chromene-4-thione 4-hydroxy-n-propargyl-1(r)-aminoindan 8-bromo-6-methyl-3-(4'-methoxyphenyl)coumarin [(1e)-4-phenylbut-1-enyl]benzene 2-(4-chlorophenyl)-4,5-dihydro-1h-imidazole 7-fluoro-2-(4-methoxyphenyl)-4h-chromen-4-one (s)(+)-2-(4-fluorophenyl)-7-methoxychroman-4-one 1,2,3,4-tetrahydro-naphthalen-1-ylamine 3-(4-hydroxyphenyl)-6-methyl-2h-chromen-2-one 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine 2-(4-methoxyphenyl)-4h-chromene-4-thione 4-phenyl-1,2,3,6-tetrahydropyridine (r)(+)-7-fluoro-2-phenylchroman-4-one (r)-3-prop-2-ynylamino-indan-5-ol 3-(2-bromophenyl)-6-methylcoumarin 8-bromo-6-methyl-3-phenylcoumarin (+/-)-7-fluoro-2-phenylchroman-4-one 3-hydroxy-2-butanone 7-fluoro-2-p-tolyl-4h-chromen-4-one 4-hydroxy-2,5-dimethyl-3(2h)-furanone 7-methyl-2-p-tolyl-4h-chromene-4-thione (r)-n2-{4-[(3-chlorobenzyl)oxy]benzyl}alaninamide (s)(+)-7-methyl-2-phenylchroman-4-one (s)-(+)-2-[4-(fluorobenzyloxy-benzylamino)propionamide] (+/-)-7-fluoro-2-(4-methoxyphenyl)chroman-4-one 7-fluoro-2-p-tolyl-4h-chromene-4-thione 3-(4-methoxyphenyl)-6-methyl-2h-chromen-2-one 4-oxo-4h-chromene-3-carboxylic acid (+/-)-7-fluoro-2-(4-fluorophenyl)chroman-4-one (s)-n2-{4-[(3-chlorobenzyl)oxy]benzyl}serinamide (r)(+)-7-methyl-2-p-tolylchroman-4-one 1h-indole-2,3-dione 2-(2-cyclohexylidenehydrazinyl)-4-p-tolylthiazole (+/-)-7-methyl-2-p-tolylchroman-4-one 7-methoxy-2-p-tolyl-4h-chromen-4-one (r)-n2-{4-[(3-fluorobenzyl)oxy]benzyl}alaninamide (s)-n2-{4-[(4-chlorobenzyl)oxy]benzyl}serinamide (r)-n-methyl-n-2-propynyl-1-indanamine 3,4-dihydroxybenzaldehyde (+/-)-2-(4-fluorophenyl)-7-methylchroman-4-one 7-[(3-chlorobenzyl)oxy]-4-[(methylamino)methyl]-2h-chromen-2-one (r)(+)-7-fluoro-2-(4-fluorophenyl)chroman-4-one 4-fluoroselegiline (r)-n2-{4-[(3-chlorobenzyl)oxy]benzyl}serinamide 2-bromo-n-(3-morpholinopropyl)nicotinamide 2-p-tolyl-4h-chromen-4-one (+/-)-2-(4-fluorophenyl)chroman-4-one (s)-n2-[4-(benzyloxy)benzyl]alaninamide (s)-n2-[4-(benzyloxy)benzyl]serinamide (+/-)-7-methoxy-2-p-tolylchroman-4-one 4-hydroxybenzoicacid 2-p-tolyl-4,5-dihydro-1h-imidazole 4-methoxybenzaldehyde 5-aminomethyl-3-pyrrol-1-yl-oxazolidin-2-one (s)(+)-7-fluoro-2-p-tolylchroman-4-one 7-[(3-chlorobenzyl)oxy]-2-oxo-2h-chromene-4-carbaldehyde 2-(3-nitrophenyl)-4,5-dihydro-1h-imidazole (1z)-4-(4-fluorophenyl)-2-methylidenebutan-1-imine (r)(+)-7-methyl-2-phenylchroman-4-one 2-phenyl-cyclopropylamine hydrochloride (+/-)-2-p-tolylchroman-4-one (+/-)-7-methyl-2-phenylchroman-4-one 4-hydroxybenzylalcohol 2-methyl-9h-indeno[2,1-d]pyrimidin-9-one (s)-n2-{4-[(3-fluorobenzyl)oxy]benzyl}serinamide (s)(+)-7-fluoro-2-(4-fluorophenyl)chroman-4-one (r)(+)-7-fluoro-2-p-tolylchroman-4-one (+/-)-7-fluoro-2-p-tolylchroman-4-one 2-hydrazino-3-methyl-4(3h)-quinazolinone 5-quinoxalin-6-ylmethylene-thiazolidine-2,4-dione (+/-)-2-(4-fluorophenyl)-7-methoxychroman-4-one (r)(+)-2-(4-fluorophenyl)-7-methoxychroman-4-one 3-(phenoxymethyl)-5h-indeno[1,2-c]pyridazin-5-one 2-p-tolyl-4h-chromene-4-thione (+/-)-2-(4-methoxyphenyl)-7-methylchroman-4-one 5-hydroxy-n-propargyl-1(r)-aminoindan 5-phenylamino-4-cyano-3-hydroxy-isothiazole (5s)-4,5-difluoro-6-[(2-fluoro-4-iodophenyl)imino]-n-(2-hydroxyethoxy)cyclohexa-1,3-diene-1-carboxamide 5-bromo-n-[(2s)-2,3-dihydroxypropoxy]-3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]benzamide 2-[(4-ethynyl-2-fluorophenyl)amino]-3,4-difluoro-n-(2-hydroxyethoxy)benzamide 4,5-dibromo-1h-pyrrole-2-carboxylic acid amide 2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamide 8-chloro-quinoline-3-carbonitrile 12-(2-hydroxyethyl)-2-(1-methylethoxy)-13,14-dihydronaphtho[2,1-a]pyrrolo[3,4-c]carbazol-5(12h)-one 6-phenylquinazolin-4-amine 4-[4-(4-fluorophenyl)-2-[4-[(r)-methylsulfinyl]phenyl]-1h-imidazol-5-yl]pyridine (3r,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione (4-fluoro-phenyl)-(9-methyl-9h-purin-6-yl)-amine 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine (s)-n-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamide 2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-n-methylacetamide 7-azaindole derivative 4 9-(4-hydroxyphenyl)-2,7-phenanthroline 1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinoline (3e)-5-fluoro-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-1h-indole-2,3-dione 3-oxime 7-azaindole derivative 7 (3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-[(e)-2-phenylethenyl]-1h-indole-2,3-dione 3-oxime 7-azaindole derivative 5 2,6-dihydroanthra/1,9-cd/pyrazol-6-one 4-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-n-ethylpiperidine-1-carboxamide 5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamide (3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-phenyl-1h-indole-2,3-dione 3-oxime 7-azaindole derivative 1 7-azaindole derivative 3 7-azaindole derivative 6 7-azaindole derivative 2 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde 3-fluoro-5-morpholin-4-yl-n-[1-(2-pyridin-4-ylethyl)-1h-indol-6-yl]benzamide 2-fluoro-4-[4-(4-fluorophenyl)-1h-pyrazol-3-yl]pyridine 6((s)-3-benzylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyrazine 4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridine 9-benzyl-6-phenylsulfanyl-9h-purine 6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amine 2-(2,6-difluorophenoxy)-n-(2-fluorophenyl)-9-isopropyl-9h-purin-8-amine 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one 1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-naphthalen-1-ylurea 6-benzylsulfanyl-9h-purine 3-fluoro-n-1h-indol-5-yl-5-morpholin-4-ylbenzamide 3-(4-fluorophenyl)-1-hydroxy-2-(pyridin-4-yl)-1h-pyrrolo[3,2-b]pyridine 2-chlorophenol [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone 9-benzyl-6-(4-fluoro-phenylsulfanyl)-9h-purine 4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazoline 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-one 4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazole 4-[5-[2-(1-phenyl-ethylamino)-pyrimidin-4-yl]-1-methyl-4-(3-trifluoromethylphenyl)-1h-imidazol-2-yl]-piperidine 8-(2-chlorophenylamino)-2-(2,6-difluorophenylamino)-9-ethyl-9h-purine-1,7-diium 6-phenylsulfanyl-9h-purine 4-phenoxy-n-(pyridin-2-ylmethyl)benzamide 3-fluoro-5-morpholin-4-yl-n-[3-(2-pyridin-4-ylethyl)-1h-indol-5-yl]benzamide 3-(2-chlorophenyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea 4-(2-hydroxybenzylamino)-n-(3-(4-fluorophenoxy)phenyl)piperidine-1-sulfonamide 9-(4-fluoro-benzyl)-6-phenylsulfanyl-9h-purine 4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazole 2-(ethoxymethyl)-4-(4-fluorophenyl)-3-[2-(2-hydroxyphenoxy)pyrimidin-4-yl]isoxazol-5(2h)-one 3-(1-naphthylmethoxy)pyridin-2-amine 6-(4-fluoro-phenylsulfanyl)-9h-purine 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea 4-(2-ethyl-4-m-tolyl-thiazol-5-yl)-pyridine 4-[5-(3-iodo-phenyl)-2-(4-methanesulfinyl-phenyl)-1h-imidazol-4-yl]-pyridine (5-amino-1-phenyl-1h-pyrazol-4-yl)phenylmethanone [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl][3-(piperidin-4-yloxy)phenyl]methanone 6-[(e)-2-(4-fluoro-phenyl)-vinyl]-9h-purine 6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-one 2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamide 5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamide 2-(2-(pentyloxy)pyrimidin-4-ylamino)benzoic acid 2-(2-(butylamino)pyrimidin-4-ylamino)benzoic acid 2-(2-propoxypyrimidin-4-ylamino)benzoic acid 2-(2-butoxypyrimidin-4-ylamino)benzoic acid 2-(2-phenoxypyrimidin-4-ylamino)benzoic acid 2-(2-(phenylamino)pyrimidin-4-ylamino)benzamide 2-(2-sec-butoxypyrimidin-4-ylamino)benzoic acid 2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one (10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one 3-{[(1r)-1-phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dione (4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamide 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one 3-oxiran-2ylalanine 1-methylimidazole 4-(hydrogen sulfate)-beta-d-galactopyranose 1-methyl-4-(1-phenyl-ethyl)-piperazine 1-benzyl-4-methyl-piperazine 3,6,9,12,15-pentaoxaheptadecan-1-ol 8-cyclohexyloxy-quinolin-2-ylamine 8-(3-methyl-cyclopentyloxy)-quinolin-2-ylamine 8-cyclopentylmethoxy-quinolin-2-ylamine 8-(3,3,3-trifluoropropoxy)quinolin-2-amine 8-(1-methyl-butoxy)-quinolin-2-ylamine 8-(2-ethoxy-1-methyl-ethoxy)-quinolin-2-ylamine 8-isopropoxy-quinolin-2-ylamine 8-cycloheptyloxy-quinolin-2-ylamine 8-butoxy-quinolin-2-ylamine 8-(1-ethyl-propoxy)-quinolin-2-ylamine 8-sec-butoxy-quinolin-2-ylamine 8-(2-methoxy-1-methyl-ethoxy)-quinolin-2-ylamine 8-(3-methyl-butoxy)-quinolin-2-ylamine [3h]snap-7941 4-arylphthalazin-1(2h)-3,4-di-f 8-(2-cyclopropyl-ethoxy)-quinolin-2-ylamine 8-propoxy-quinolin-2-ylamine 7-fluorochromone-2-carboxamide 8-(4-methyl-cyclohexyloxy)-quinolin-2-ylamine 8-hexyloxy-quinolin-2-ylamine 8-(1,2-dimethyl-propoxy)-quinolin-2-ylamine 8-pentyloxy-quinolin-2-ylamine 8-(3-methoxy-3-methyl-butoxy)-quinolin-2-ylamine 8-cyclobutylmethoxy-quinolin-2-ylamine 8-(3-methyl-cyclohexyloxy)-quinolin-2-ylamine 8-(2-methyl-cyclohexyloxy)-quinolin-2-ylamine 8-(2-methyl-butoxy)-quinolin-2-ylamine 8-(1,3,3-trimethyl-butoxy)-quinolin-2-ylamine 2-phenyl-n,n-bis(o-tolylthiomethyl)ethanamine 8-(2-ethyl-1-methyl-butoxy)-quinolin-2-ylamine 8-(3,3-dimethyl-butoxy)-quinolin-2-ylamine 1-benzyl-1h-pyrrolo[3,2-b]pyridine 1-[(2-nitrophenyl)sulfonyl]-1h-pyrrolo[3,2-b]pyridine-6-carboxamide 2-(4-fluorophenyl)-n-{[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]carbamoyl}acetamide 1-(phenylsulfonyl)-1h-pyrrolo[3,2-b]pyridine 1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamide 1-(2-nitrophenethyl)-1h-pyrrolo[3,2-b]pyridine 3-(phenylsulfonyl)-1h-pyrrolo[2,3-b]pyridine 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol 3-[(2,2-dimethylpropanoyl)amino]-n-1,3-thiazol-2-ylpyridine-2-carboxamide 5-chloro-6-methyl-n-(2-phenylethyl)-2-pyridin-2-ylpyrimidin-4-amine 5-ethyl-2-(phenylsulfonamido)benzoic acid 5-bromo-2-{[(4-chlorophenyl)sulfonyl]amino}benzoic acid 2-[(phenylsulfonyl)amino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acid 5-chloro-2-(pyridin-2-yl)-1h-benzo[d]imidazole 2-(pyridin-2-yl)-1h-benzo[d]imidazole 5-fluoro-2-(pyridin-2-yl)-1h-benzo[d]imidazole 3-anilino-5-benzylthio-1,2,4-triazole 2-methyl-2-propanol 5-methyl-2-[(phenylsulfonyl)amino]benzoic acid 5-methyl-2-(pyridin-2-yl)-1h-benzo[d]imidazole 2-(pyridin-2-yl)-1h-benzo[d]imidazol-5-amine (2r,3r,4s,5r,6e)-3,4,5-trihydroxy-n-[(3s,6r)-6-hydroxy-2-oxo-3-azepanyl]-2-methoxy-8,8-dimethyl-6-nonenamide 2-(phenylsulfonamido)-1-naphthoic acid 5-butyl-2-(phenylsulfonamido)benzoic acid (2s,3r)-3-amino-2-hydroxy-5-(ethylsulfanyl)pentanoyl-((s)-(-)-(1-naphthyl)ethyl)amide 3,5,6,8-tetramethyl-n-methyl phenanthrolinium 2-(phenylsulfonamido)-5-propylbenzoic acid 5-methyl-2-(phenylsulfonamido)benzoic acid 2-(thiazol-4-yl)-1h-benzo[d]imidazol-5-amine 2-(pyridin-2-yl)-1h-imidazo[4,5-c]pyridine 3-ethyl-6-{[(4-fluorophenyl)sulfonyl]amino}-2-methylbenzoic acid 2-[({2-[(1z)-3-(dimethylamino)prop-1-enyl]-4-fluorophenyl}sulfonyl)amino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acid 2-(4-fluorophenylsulfonamido)-1-naphthoic acid 5-bromo-2-(4-chlorophenylsulfonamido)benzoic acid 3,5-dimethyl-2-(phenylsulfonamido)benzoic acid 5-p-tolyl-1h-[1,2,3]triazole 2-aminomethyl-pyrrolidine-3,4-diol 4'-(p-toluenesulfonamide)-3,4-dihydroxy chalcone 3-(4-(4-hydroxyphenyl)phthalazin-1-ylamino)phenol 1,4-dideoxy-1,4-imino-d-arabinito 2-cyclopentylaminomethyl-pyrrolidine-3,4-diol 2,5-dideoxy-2,5-imino-d-mannitol 6-benzyloxy-9h-purin-2-ylamine 6-benzyloxy-5-nitro-pyrimidine-2,4-diamine 6-allyloxy-9h-purin-2-ylamine 6-benzyloxy-5-nitroso-pyrimidine-2,4-diamine 3-benzyl-6-methylbenzo[d]oxazol-2(3h)-one 2-(4-hydroxystyryl)quinolin-8-ol 7-hydroxy-2-oxo-chromene-3-carboxylic acid ethyl ester 3-benzyl-5-fluorobenzo[d]oxazol-2(3h)-one 4-hydroxybenzaldehyde o-(3,3-dimethylbutanoyl)oxime 4-(4-benzyl-1h-1,2,3-triazol-1-yl)phenol 4-iodo-6-phenylpyrimidine 3-(4-hydroxyphenyl)-4,5-dihydro-5-isoxazole-acetic acid methyl ester 7-hydroxy-3-phenyl-2h-chromen-2-one 3,3,3-tris(4-chlorophenyl)propanoic acid 3-acetyl-7-hydroxy-2h-chromen-2-one 1-phenyl-3-(1,3,4-thiadiazol-2-yl)thiourea 3-fluoro-4-hydroxybenzaldehyde o-(cyclohexylcarbonyl)oxime 3-benzyl-5-methylbenzo[d]oxazol-2(3h)-one 1-(2-chlorophenyl)-3-(pyridin-2-yl)thiourea 4-hydroxybenzaldehyde o-(cyclohexylcarbonyl)oxime 4-((pyridin-4-ylthio)methyl)benzene-1,2-diol 3-(1h-pyrazol-3-yl)benzoic acid 6-phenylpyridazin-3-yl thiophene-2-carboxylate (5r)-2-sulfanyl-5-[4-(trifluoromethyl)benzyl]-1,3-thiazol-4(5h)-one [leu13]motilin (human) [2(r,s)-2-sulfanylheptanoyl]-phe-ala 9-mercaptomethyl-10-oxo-azecane-2-carboxylic acid 2-[(1s)-1-benzyl-2-sulfanylethyl]-1h-imidazo[4,5-c]pyridin-5-ium 3-benzenesulfinyl-heptanoic acid hydroxyamide 3-(4-methoxy-benzenesulfonyl)-cyclohexanethiol 3-(4-phenoxy-benzenesulfonyl)-cyclohexanethiol 4-(4-methoxy-benzenesulfonyl)-butane-2-thiol [[1-[n-hydroxy-acetamidyl]-3-methyl-butyl]-carbonyl-leucinyl]-alanine ethyl ester 3-cyclohexanesulfonyl-heptanoic acid hydroxyamide 3-benzenesulfonyl-heptanoic acid hydroxyamide 3-(4-phenoxy-benzenesulfonyl)-propane-1-thiol 3-(4-methoxy-benzenesulfonyl)-pentane-1-thiol 3-(4-methoxy-benzenesulfonyl)-hexane-1-thiol 4-butoxy-n-hydroxycarbamoylmethyl-benzamide 4-(4-butoxy-phenyl)-n-hydroxy-4-oxo-butyramide 3ts4 2-(2-(biphenyl-4-yl)ethylsulfinyl)acetic acid 4-(4-(dec-1-ynyl)phenyl)-4-oxobutanoic acid 3-(4-phenylethynylbenzoyl)nonanoic acid 2-(biphenyl-4-ylsulfonyl)n-hydroxybenzamide 5-(biphenyl-4-yl)-3-methoxypentanoic acid 3-(4-(2-phenylethynyl)benzoyl)pentanoic acid 5-(4'-cyanobiphenyl-4-yl)-3-hydroxypentanoic acid 5-(3'-cyanobiphenyl-4-yl)-3-hydroxypentanoic acid 2-[(4-fluorophenyl)sulfonylamino]-n-oxo-ethanamide (+/-)5-(biphenyl-4-yl)-3-hydroxypentanoic acid 2-(2-(biphenyl-4-yl)ethylsulfonyl)acetic acid 2-[2-(1,3-dioxo-1,3-dihydro-2h-isoindol-2-yl)ethyl]-4-(4'-ethoxy-1,1'-biphenyl-4-yl)-4-oxobutanoic acid (1s,5s,7r)-n~7~-(biphenyl-4-ylmethyl)-n~3~-hydroxy-6,8-dioxa-3-azabicyclo[3.2.1]octane-3,7-dicarboxamide [2-(biphenyl-4-sulfonyl)phenyl]acetic acid 2-(2-(biphenyl-4-yl)ethylthio)acetic acid 5-(biphenyl-4-yl)-3-oxopentanoic acid 4-{[1-methyl-2,4-dioxo-6-(3-phenylprop-1-yn-1-yl)-1,4-dihydroquinazolin-3(2h)-yl]methyl}benzoic acid 1-(4-methoxy-benzenesulfonyl)-heptane-3-thiol 4-amino-3-(4-(hexyloxy)phenyl)-4-oxobutanoic acid 1-methyloxy-4-sulfone-benzene 4-methoxybenzenesulfinate 3-methylpyridine 4-(methyl(4-phenylthiazol-2-yl)amino)phenol 4-(2,2'-bithiophen-5-ylmethyleneamino)phenol 2-(biphenyl-4-ylsulfonamido)pentanedioic acid 5-(2-ethoxyethyl)-5-[4-(4-fluorophenoxy)phenoxy]pyrimidine-2,4,6(1h,3h,5h)-trione 3-(4-methoxy-benzenesulfonyl)-propane-1-thiol 2-{4-[4-(4-chloro-phenoxy)-benzenesulfonyl]-tetrahydro-pyran-4-yl}-n-hydroxy-acetamide 2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol 3-(4-methoxy-benzenesulfonyl)-cyclopentanethiol 5-hexyl-5-phenyl-pyrimidine-2,4,6-trione 5-(4-phenoxy-phenyl)-pyrimidine-2,4,6-trione 5-biphenyl-4-yl-5-ethyl-pyrimidine-2,4,6-trione 2-(4'-chloro-biphenyl-4-sulfonyl)-pentanoic acid 5-biphenyl-4-yl-5-hexyl-pyrimidine-2,4,6-trione 2-[3-(5-mercapto-[1,3,4]thiadiazol-2yl)-ureido]-n-methyl-3-pentafluorophenyl-propionamide 3-[(4'-cyanobiphenyl-4-yl)oxy]-n-hydroxypropanamide 2-(2-{2-[(biphenyl-4-ylmethyl)-amino]-3-mercapto-pentanoylamino}-acetylamino)-3-methyl-butyric acid methyl ester [4-(4-phenyl-piperidin-1-yl)-benzenesulfonylamino]-acetic acid 3-(1h-indol-3-yl)-2-[4-(4-phenyl-piperidin-1-yl)-benzenesulfonylamino]-propionic acid 1-benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-hexahydro-pyrimidine-4-carboxylic acid hydroxyamide 2-[3-(5-mercapto-[1,3,4]thiadiazol-2-yl)-ureido]-n-methyl-3-phenyl-propionamide (1n)-4-n-butoxyphenylsulfonyl-(2r)-n-hydroxycarboxamido-(4s)-methanesulfonylamino-pyrrolidine [2-(5-mercapto-[1,3,4]thiadiazol-2-ylcarbamoyl)-1-phenyl-ethyl]-carbamic acid benzyl ester 5-methyl-5-(4-phenoxy-phenyl)-pyrimidine-2,4,6-trione (1r)-n,6-dihydroxy-7-methoxy-2-[(4-methoxyphenyl)sulfonyl]-1,2,3,4-tetrahydroisoquinoline-1-carboxamide 5-methyl-3-(9-oxo-1,8-diaza-tricyclo[10.6.1.013,18]nonadeca-12(19),13,15,17-tetraen-10-ylcarbamoyl)-hexanoic acid (1r)-1-{[(4'-methoxy-1,1'-biphenyl-4-yl)sulfonyl]amino}-2-methylpropylphosphonic acid 1-hydroxyamine-2-isobutylmalonic acid 5-[4-(2-hydroxyethyl)-1-piperidinyl]-5-phenyl-2,4,6(1h,3h,5h)-pyrimidinetrione 3-formyl-2-hydroxy-5-methyl-hexanoic acid hydroxyamide (1s)-1-{[(4'-methoxy-1,1'-biphenyl-4-yl)sulfonyl]amino}-2-methylpropylphosphonic acid 3-amino-azacyclotridecan-2-one (5s)-5-(2-amino-2-oxoethyl)-4-oxo-n-[(3-oxo-3,4-dihydro-2h-1,4-benzoxazin-6-yl)methyl]-3,4,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidine-2-carboxamide 2-hydroxycarbamoyl-4-methyl-pentanoic acid 2-(biphenyl-4-sulfonyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (2r)-2-amino-3,3,3-trifluoro-n-hydroxy-2-{[(4-phenoxyphenyl)sulfonyl]methyl}propanamide 5-methyl-5-phenyl-pyrimidine-2,4,6-trione (3r)-4,4-difluoro-3-[(4-methoxyphenyl)sulfonyl]butanoic acid 2-amino-n,3,3-trimethylbutanamide 5-(4-phenoxyphenyl)-5-(4-pyrimidin-2-ylpiperazin-1-yl)pyrimidine-2,4,6(2h,3h)-trione 2-{[formyl(hydroxy)amino]methyl}-4-methylpentanoic acid 4-aminobenzoic acid hydrazide 2lm20-4 227th-rituximab 227th-labelled msln-ttc 6-thiophen-2-yl-imidazo[2,1-b]thiazole 6-thiophen-3-yl-imidazo[2,1-b]thiazole 5'-deoxy-5'-(methylthio)-tubercidin 5'-s-methyl-5'-thioadenosine (2s,3s,4r,5s)-2-(4-amino-4,5-dihydro-1h-pyrrolo[3,2-d]pyrimidin-7-yl)-5-[(methylsulfanyl)methyl]-3,4-pyrrolidinediol 677t 2-iodo-melatonin [125i]div880 [125i]sd6 2-[125i]melatonin 2-(indolin-1yl)-melatonin (hydroxymethylphenyl)agomelatine 6-cl-mlt 5-methoxycarbonylamino-n-acetyltryptamine 2-methoxy-alpha,beta-didehydro-agomelatine 6-hydroxymelatonin 5-methoxy-luzindole [125i]s70254 5-heat 4p-pdot 4-(2-(thiophen-2-yl)-9h-purin-6-yl)morpholine 4-(6-morpholino-9h-purin-2-yl)phenol 2-morpholin-4-yl-pyrimido[2,1-a]isoquinolin-4-one 4-(2-(1h-indol-6-yl)-9h-purin-6-yl)morpholine 4-(2-(thiophen-3-yl)-9h-purin-6-yl)morpholine 3-(6-morpholino-9h-purin-2-yl)phenol 2-(2-methyl-morpholin-4-yl)-benzo[h]chromen-4-one 2-(6-morpholino-9h-purin-2-yl)phenol 2-chloro-n-(6-cyanopyridin-3-yl)propanamide (4-(6-morpholino-9h-purin-2-yl)phenyl)methanol 6-fluoromevalonate pyrophosphate 2-fluoromevalonate 5-diphosphate 6-fluoromevalonate 5-diphosphate 2,2-difluoromevalonate 5-diphosphate (3as)-3a-hydroxy-5-methyl-1-phenyl-1,2,3,3a-tetrahydro-4h-pyrrolo[2,3-b]quinolin-4-one (s)-blebbistatin (3as)-3a-hydroxy-1-phenyl-1,2,3,3a-tetrahydro-4h-pyrrolo[2,3-b]quinolin-4-one (3as)-3a-hydroxy-7-methyl-1-phenyl-1,2,3,3a-tetrahydro-4h-pyrrolo[2,3-b]quinolin-4-one 4-[4-(2,5-dioxo-pyrrolidin-1-yl)-phenylamino]-4-hydroxy-butyric acid (8alpha,10alpha,13alpha,17beta)-17-[(4-hydroxyphenyl)carbonyl]androsta-3,5-diene-3-carboxylic acid (1r,3r)-5-[(2e)-3-{(1s,3r)-2,2,3-trimethyl-3-[6,6,6-trifluoro-5-hydroxy-5-(trifluoromethyl)hex-3-yn-1-yl]cyclopentyl}prop-2-en-1-ylidene]cyclohexane-1,3-diol 1,3-cyclohexanediol, 4-methylene-5-[(2e)-[(1s,3as,7as)-octahydro-1-(5-hydroxy-5-methyl-1,3-hexadiynyl)-7a-methyl-4h-inden-4-ylidene]ethylidene]-, (1r,3s,5z) (2s)-3-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1h-indol-5-yl)-2-ethoxypropanoic acid 2-chloro-5-nitro-n-phenylbenzamide 2-[(2,4-dichlorobenzoyl)amino]-5-(pyrimidin-2-yloxy)benzoic acid (2e,4e)-11-methoxy-3,7,11-trimethyldodeca-2,4-dienoic acid 5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n,2,4-trimethyl-1h-pyrrole-3-carboxamide 2-deoxy-2,3-dehydro-n-acetylneuraminic acid 5-acetamido-5,6-dihydro-4-hydroxy-6-isobutoxy-4h-pyran-2-carboxylic acid 4-(2-cyclohexylethoxy) aniline derivative 1 3-phenyl propanoic derivative 1 1-phenyl-1,3,4-triazole derivative 2 3-phenyl propanoic derivative 2 1-phenyl-1,3,4-triazole derivative 3 1,2,3,4-tetrahydroisoquinoline derivative 1 3-phenyl propanoic derivative 3 4-(2-cyclohexylethoxy) aniline derivative 2 1-phenyl-1,3,4-triazole derivative 1 4-(2-cyclohexylethoxy) aniline derivative 3 4-(2-cyclohexylethoxy) aniline derivative 4 2'-deoxyguanosine-5'-diphosphate 2',3'-dideoxy-3'-fluoro-urididine-5'-diphosphate 2',3'-dehydro-2',3'-deoxy-thymidine 5'-diphosphate 2'-deoxyguanosine-5'-triphosphate 3'-deoxy 3'-amino adenosine-5'-diphosphate 2-(4-chloro-phenylamino)-nicotinic acid (1-methyl-1h-imidazol-2-yl)-(3-methyl-4-{3-[(pyridin-3-ylmethyl)-amino]-propoxy}-benzofuran-2-yl)-methanone 1-(cyclohexylamino)-3-(6-methyl-3,4-dihydro-1h-carbazol-9(2h)-yl)propan-2-ol (z)-3-benzyl-5-(2-hydroxy-3-nitrobenzylidene)-2-thioxothiazolidin-4-one 7-thionicotinamide-adenine-dinucleotide phosphate 4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl]phenol (1s)-1-phenylethyl (4-acetamidobenzyl)phosphonate 4-[(2-methyl-1h-imidazol-1-yl)methyl]pyridine 2-butyl-1-hydroxyguanidine 2-amino-4-methylpyridine 6-bromo-1h-indazole 1-(benzhydrylamino)ethaniminium bromide 4-methyl-pyrrolidin-(2z)-ylideneamine 1-benzyl-2-methyl-1h-imidazole (5-imino-[1,4]thiazepan-3-yl)-methanol 3-(2-nitro-ethyl)-[1,4]oxazepan-(5z)-ylideneamine 5-n-allyl-arginine 4-methyl-oxazolidin-(2z)-ylideneamine 1-hydroxy-2-isopropylguanidine 3-bromo-7-nitroindazole 5-bromomethyl-oxazolidin-(2z)-ylideneamine 1-[(3-methoxybenzyl)amino]ethaniminium chloride 7-bromo-1h-indazole 4-ethyl-pyrrolidin-(2z)-ylideneamine (r)-3-propyl-[1,4]thiazepan-(5e)-ylideneamine [1,4]thiazepan-(5e)-ylideneamine 4-butyl-thiazolidin-(2e)-ylideneamine ((e)-7-but-2-enyl)-azepan-(2z)-ylideneamine 4,5-dimethyl-pyrrolidin-(2z)-ylideneamine 5-ethyl-4-propyl-pyrrolidin-(2z)-ylideneamine (5s,6s)-[octahydro-quinolin-(2e)-ylidene]amine 4-methyl-5-propyl-pyrrolidin-(2z)-ylideneamine 2-aminothiazoline 5-ethyl-4-methyl-pyrrolidin-(2z)-ylideneamine 5-ethyl-oxazolidin-(2z)-ylideneamine 3-propyl-[1,4]thiazepan-(5e)-ylideneamine 5-methyl-oxazolidin-(2z)-ylideneamine 4-methyl-piperidin-(2e)-ylideneamine 5-bromo-1h-indazole [(1s)-4-(1-aminobutylideneamino)-1-carboxybutyl]azanium 4-chloro-1h-indazole 1-(2-amino-benzothiazol-5-yl)-2-ethyl-isothiourea 6-chloro-1h-indazole 7-chloro-1h-indazole 4,5,6,7-tetrafluoro-3-methyl-1h-indazole 5-methyl-pyrrolidin-(2z)-ylideneamine 7-methoxy-1h-indazole 2-methyl-[1,4]thiazepan-(5e)-ylideneamine [1,4]oxazepan-(5e)-ylideneamine 3-methyl-[1,4]thiazepan-(5e)-ylideneamine 7-butyl-azepan-(2z)-ylideneamine 7-methyl-[1,4]thiazepan-(5e)-ylideneamine 3-bromo-7-nitro-1h-indazole 4-ethyl-3-methyl-pyrrolidin-(2z)-ylideneamine 3-(2-amino-ethyl)-5-imino-[1,4]oxazepane 4-isopropyl-pyrrolidin-(2z)-ylideneamine 2-aminopyridine 6-isobutyl-4-methylpyridin-2-amine 3-bromo-1h-indazole-7-carbonitrile 3-ethyl-[1,4]thiazepan-(5e)-ylideneamine [1,4]thiazepan-(3e)-ylideneamine 3-methyl-pyrrolidin-(2z)-ylideneamine [1,3]thiazinan-(2e)-ylideneamine (+/-)-2-methyl-1-(1-phenylethyl)-1h-imidazole 3-isobutyl-[1,4]thiazepan-(5e)-ylideneamine 4-bromo-1h-indazole (6r,1'r,2's)-5,6,7,8 tetrahydrobiopterin 6-(2-fluoropropyl)-4-methylpyridin-2-amine (4s,5r)-4,5-diethyl-oxazolidin-(2z)-ylideneamine 5-iodo-1h-indazole 3,4-dihydro-1h-quinolin-(2e)-ylideneamine 5-chloro-1h-indazole (4s,5s)-4,5-diethyl-oxazolidin-(2z)-ylideneamine [1,4]oxazepan-(3e)-ylideneamine (4s,5r)-4,5-dimethyl-oxazolidin-(2z)-ylideneamine [1,3]oxazinan-(2e)-ylideneamine 2-amino-5-(n-nitro-guanidino)-pentanoic acid 4-iodo-1h-indazole (s)-3-propyl-[1,4]thiazepan-(5e)-ylideneamine 1400w (s)-6-amino-2-(2-imino-ethylamino)-hexanoic acid 5-ethyl-3-methyl-pyrrolidin-(2z)-ylideneamine 2-(2-amino-ethyl)-7-imino-azepane 7-nitro-1h-indazole 4-ethyl-oxazolidin-(2z)-ylideneamine 7-(2-nitro-ethyl)-azepan-(2z)-ylideneamine 3,4-dimethyl-pyrrolidin-(2z)-ylideneamine 3-butyl-[1,4]thiazepan-(5e)-ylideneamine (s)-2-amino-5-(n-methyl-guanidino)-pentanoic acid 4-ethyl-5-methyl-pyrrolidin-(2z)-ylideneamine 1-(2-amino-benzothiazol-6-yl)-2-ethyl-isothiourea 6-(3-fluoropropyl)-4-methylpyridin-2-amine 2-amino-4,6-dimethylpyridine (5s,6r)-[octahydro-quinolin-(2e)-ylidene]amine 4-methyl-6-propylpyridin-2-amine [1,5]thiazocan-(4e)-ylideneamine 6-(4-fluorobutyl)-4-methylpyridin-2-amine 7-nitroindazole 4-(1,3-benzodioxol-5-yloxy)-2-[4-(1h-imidazol-1-yl)phenoxy]-6-methylpyrimidine 6-methyl-5,6-dihydro-4h-1,3-thiazin-2-amine 5-methyl-4-propyl-pyrrolidin-(2z)-ylideneamine 5-nitroindazole (3r)-3-[(1,2,3,4-tetrahydroisoquinolin-7-yloxy)methyl]-2,3-dihydrothieno[2,3-f][1,4]oxazepin-5-amine 4-(1,3-benzodioxol-5-yloxy)-2-[4-(1h-imidazol-1-yl)phenoxy]pyrimidine 1-(6-cyano-3-pyridylcarbonyl)-5',8'-difluorospiro[piperidine-4,2'(1'h)-quinazoline]-4'-amine (4s,5r)-4,5-dipropyl-oxazolidin-(2z)-ylideneamine (s)-n-(1-phenylethyl)acetimidamide hydrobromide 5-(4'-amino-1'-ethyl-5',8'-difluoro-1'h-spiro[piperidine-4,2'-quinazoline]-1-ylcarbonyl)picolinonitrile 4r-fluoro-n6-ethanimidoyl-l-lysine 4-methyl-6-(2-methylprop-1-enyl)pyridin-2-amine 4-(1h-imidazol-1-yl)phenol (2s)-2-methyl-2,3-dihydrothieno[2,3-f][1,4]oxazepin-5-amine 1-[4-(aminomethyl)benzoyl]-5'-fluoro-1'h-spiro[piperidine-4,2'-quinazolin]-4'-amine (e)-4-methyl-6-(prop-1-enyl)pyridin-2-amine (s)-2-amino-6-[(e)-ethylimino]-hexanoic acid 4,5,6,7-tetrafluoro-3-perfluorophenyl-1h-indazole (4s,5s)-4,5-dipropyl-oxazolidin-(2z)-ylideneamine 7,8-dihydrobiopterin 6-nitroindazole 4-({4-[(4-methoxypyridin-2-yl)amino]piperidin-1-yl}carbonyl)benzonitrile (3s)-1-(1,3-benzodioxol-5-ylmethyl)-3-[4-(1h-imidazol-1-yl)phenoxy]piperidine 3-butyl-[1,4]oxazepan-(5z)-ylideneamine 1-(6-amino-4-methylpyridin-2-yl)propan-2-ol 6s-5,6,7,8-tetrahydrobiopterin 7-nitroindazole-2-carboxamidine (3s,5e)-3-propyl-3,4-dihydrothieno[2,3-f][1,4]oxazepin-5(2h)-imine 2,4-diamino-6-phenyl-5,6,7,8,-tetrahydropteridine 1,2,4-triazole-carboxamidine 5,6-cyclic-tetrahydropteridine 4-methyl-5,6-dihydro-1h-pyridin-(2z)-ylideneamine 4-ethyl-5,6-dihydro-1h-pyridin-(2z)-ylideneamine 5-{4-[(3,5-difluorobenzyl)amino]phenyl}-6-ethylpyrimidine-2,4-diamine 4-methyl-3,6-dihydro-1h-pyridin-(2z)-ylideneamine 1dme 4,5,6,7-tetrahydrofuro[3,4-c]pyridine-1(3h)-one derivative 1 4,5,6,7-tetrahydrofuro[3,4-c]pyridine-1(3h)-one derivative 3 4,5,6,7-tetrahydrofuro[3,4-c]pyridine-1(3h)-one derivative 4 4,5,6,7-tetrahydrofuro[3,4-c]pyridine-1(3h)-one derivative 2 [125i]gr231118 [cys-trp-arg-nva-arg-tyr-nh2]2 2,4,4-triphenylimidazoline 5-methoxy-1,2-dimethyl-3-(phenoxymethyl)indole-4,7-dione 2-benzyl-1-hydroxy-3h-benzo[f]chromen-3-one 3-(3,4-dimethylbenzyl)-4-hydroxy-2h-chromen-2-one 4-hydroxy-3-(1-naphthylmethyl)-2h-chromen-2-one 3-(hydroxymethyl)-1-methyl-5-(2-methylaziridin-1-yl)-2-phenyl-1h-indole-4,7-dione 3-benzyl-4-hydroxy-6,7-dimethyl-2h-chromen-2-one 3-benzyl-4-hydroxy-2h-chromen-2-one 3-benzyl-4-hydroxy-2h-benzo[h]chromen-2-one 4-amino-2h-chromen-2-one 4-hydroxy-3-(2-naphthylmethyl)-2h-chromen-2-one 3-hydroxymethyl-5-aziridinyl-1methyl-2-[1h-indole-4,7-dione]-propanol 1,4-dimethylquinolin-2(1h)-one 5,6,8-trimethoxy-1,4-dimethylquinolin-2(1h)-one 5,8-dimethoxy-1,4-dimethylquinolin-2(1h)-one 5,8-dimethoxy-4-methylquinolin-2(1h)-one 6,7,8-trimethoxy-1,4-dimethylquinolin-2(1h)-one 7,8-dimethoxy-1,4-dimethylquinolin-2(1h)-one 5,6,8-trimethoxy-4-methylquinolin-2(1h)-one 6,8-dimethoxy-4-methylquinolin-2(1h)-one (3s)-3-hydroxy-1-methyl-2,3-dihydro-1h-indole-5,6-dione 8-methoxy-1,4-dimethylquinolin-2(1h)-one 6-methyl-[1,3]dioxolo[4,5-h]quinolin-8(9h)-one 6,7,8-trimethoxy-4-methylquinolin-2(1h)-one 6,8-dimethoxy-1,4-dimethylquinolin-2(1h)-one 12,17-dehydroxyriccardin c 24(s)-hydroxycholesterol 4,17-dehydroxyriccardin c 17-dehydroxyriccardin c 24(s), 25-epoxycholesterol 4-dehydroxyriccardin c 12-dehydroxyriccardin c 1,1,1,3,3,3-hexafluoro-2-{4-[(2,2,2-trifluoroethyl)amino]phenyl}propan-2-ol 22r-hydroxycholesterol 2-benzyl-4,5,6,7-tetrachloroisoindoline-1,3-dione 2-benzyl-3-phenyl-7-(trifluoromethyl)-2h-indazole 2-(2-hexylphenyl)isoindoline-1,3-dione 1-benzyl-3-(4-methoxyphenylamino)-4-phenylpyrrole-2,5-dione 67s 4,12,17-dehydroxyriccardin c 2-(2-phenethylphenyl)isoindoline-1,3-dione 5-chloro-2-(4-phenylbutyl)isoindoline-1,3-dione 12-o-deacetyl-12-epi-19-deoxy-21-hydroxyscalarin 1,1-bisphosphonate esters 3-keto-lithocholic acid 16,17-androstene-3-ol (5beta)-pregnane-3,20-dione 1-(2,3-dichlorophenyl)-2,2,2-trifluoro-1-(1-(4-fluorophenyl)-1h-indazol-5-yl)ethanol (enantiomeric mix) 1-(3-chloro-4-fluorophenyl)-2,2,2-trifluoro-1-(1-(4-fluorophenyl)-1h-indazol-5-yl)ethanol (enantiomeric mix) 1-methoxy-6-phenyl-6h-benzo[c]chromene 2,2,2-trifluoro-1-(4-fluorophenyl)-1-(1-(4-fluorophenyl)-1h-indazol-5-yl)ethanol (diastereomeric mix) 1-methoxy-6-phenyl-6h-benzo[c]chromen-8-ylamine (2r)-3-{[{[(2s)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-2-[(9e)-hexadec-9-enoyloxy]propyl (9e)-octadec-9-enoate 3-amino-5-benzyl-substituted indazole derivative 1 [3h]meclinertant 3-(aminooxy)propan-1-amine hydrochloride (2r,5r)-delta-methyl-alpha-acetylenic putrescine 3-methoxy-4-hydroxylonchocarpin 1-amino-3-(aminoxy)-2-propanol dihydrochloride 4-hydroxylonchocarpin 6-(4-(3-(benzylamino)propyl)phenoxy)nicotinamide 1-benzhydryl-4-phenylpiperidin-4-ol 1-benzhydryl-4-(4-methoxyphenyl)piperidin-4-ol 6beta-naltrexol hcl 6-cinnamoylhernandine 1-benzhydryl-4-m-tolylpiperidin-4-ol (-)-eseroline 5-(4-((phenethylamino)methyl)phenoxy)picolinamide 6-(2-phenethylisoindolin-5-yloxy)nicotinamide [dcp1]dyn a(1-11)-nh2 [3h]diprenorphine 4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol 3,6-bis(dmt-tic-nh-butyl)-2(1h)-pyrazinone 1-benzhydryl-4-o-tolylpiperidin-4-ol 4-(4-((phenethylamino)methyl)phenoxy)benzamide 1-benzhydryl-4-(thiophen-2-yl)piperidin-4-ol 3,6-bis(dmt-tic-nh-ethyl)-2(1h)-pyrazinone 1,10-bis-(dmt-tic-amino)decane 3,6-bis(dmt-tic-nh-propyl)-2(1h)-pyrazinone 4-phenyl-1-(1-phenylheptyl)piperidin-4-ol 1-benzhydryl-4-hexylpiperidin-4-ol 3-methylfentanyl 1-(1,2-diphenylethyl)-4-phenylpiperidin-4-ol 6-(allyl-methyl-amino)-4,4-diphenyl-heptan-3-ol 4-phenyl-1-(phenyl(m-tolyl)methyl)piperidin-4-ol 6-(4-((phenethylamino)methyl)phenoxy)nicotinamide 4-phenyl-4-[1h-imidazol-2-yl]-piperidine 1-[3-(3-biphenyl)-(1,2,4-triazol-4-yl) ]-3-phenol [3h]naltrindole 6-(4-((benzylamino)methyl)phenoxy)nicotinamide 1-(2-ethoxy-1-phenylethyl)-4-phenylpiperidin-4-ol 1-benzhydryl-4-benzylpiperidin-4-ol (-)-cyclorphan 1-benzhydryl-4-butylpiperidin-4-ol 2-hydroxymethyl-3-hydroxymorphinan 3,6-bis(dmt-tic-nh-methyl)-2(1h)-pyrazinone 1,6-bis-(dmt-tic-amino)hexane 1,6-bis-(n,n-dimethyl-dmt-tic-nh)hexane (-)-isoelaeocarpiline 1-benzhydryl-4-methoxy-4-phenylpiperidine 1-[3-(4-biphenyl)-(1,2,4-triazol-4-yl) ]-3-phenol 7-benzylidenenaltrexone 1-benzhydryl-4-(2-methoxyphenyl)piperidin-4-ol 1-benzhydryl-4-(4-bromophenyl)piperidin-4-ol 1-benzhydryl-4-(4-fluorophenyl)piperidin-4-ol 1-benzhydryl-4-(benzyloxy)-4-phenylpiperidine 6-desoxonaltrexone 17-methylmorphinan-3-yl 4-iodophenyl carbamate 3-desoxy-3-carboxamidonaltrexone 1-benzhydryl-4-(3-phenylpropyl)piperidin-4-ol 6-(4-(2-(benzylamino)ethyl)phenoxy)nicotinamide 1-benzhydryl-4-p-tolylpiperidin-4-ol 1-benzhydryl-4-cyclohexylpiperidin-4-ol 1-benzhydryl-4-ethoxy-4-phenylpiperidine (h-dmt-tic-glu-nh-(ch(2))(5)-co-dap(6dmn)-nh(2) 8-carboxamidocyclazocine 1-benzhydryl-4-(furan-2-yl)piperidin-4-ol 1-benzhydryl-4-phenyl-4-propoxypiperidine 17-methyl-4'-methyldihydromorphinone 1-benzhydryl-4-(3-methoxyphenyl)piperidin-4-ol 17-(cyclobutylmethyl)-n-phenylmorphinan-3-amine 17-(cyclopropylmethyl)-n-phenylmorphinan-3-amine 4-phenyl-1-(1-phenylpentyl)piperidin-4-ol [leu5]enkephalin 4-phenyl-1-(1-phenylbutyl)piperidin-4-ol 4-phenyl-1-(phenyl(p-tolyl)methyl)piperidin-4-ol 14-o-phenylpropylnaltrexone 1-benzhydryl-4-(3-fluorophenyl)piperidin-4-ol 1,4-bis-(dmt-tic-amino)butane 4-phenyl-1-(1-phenylhexyl)piperidin-4-ol 3-methylthiofentanyl 6-cinnamoyl-n-methylstephasunoline 1-benzhydryl-4-(4-chlorophenyl)piperidin-4-ol 1-(dio-tolylmethyl)-4-phenylpiperidin-4-ol 1-benzhydryl-4-(2-fluorophenyl)piperidin-4-ol [3h]u69593 2-benzylaminomethyl-3-hydroxymorphinan 2-epi-2-thiosalvinorin b 1-benzhydryl-4-tert-butylpiperidin-4-ol [u-13c]ascomycin 3-(1-benzylpiperidin-4-yloxy)benzamide 4-phenyl-1-(1-phenylpropyl)piperidin-4-ol 1-benzhydryl-4-(pyridin-2-yl)piperidin-4-ol 1-benzhydryl-4-isopropylpiperidin-4-ol 1-benzhydryl-4-(4-propylphenyl)piperidin-4-ol 12-epi-salvinorin a 3-(1-benzylpiperidin-4-yl)-5-chloro-1h-indole 1-benzhydryl-4-(4-ethylphenyl)piperidin-4-ol 2-(2-methylquinolin-4-ylamino)-n-phenylacetamide 4-phenyl-1-(1-phenylethyl)piperidin-4-ol 2-epi-2-thiosalvinorin a 2-thiosalvinorin b 2-mepen-ryyrik-nh2 4-(2-(aminomethyl)phenyl)-1-benzylpiperidin-4-ol 2,2-dimebut-ryyrik-nh2 1-benzyl-4-phenylpiperidin-4-ol [asp6,lys10]n/ofq(1-13)nh2 [d-asp7,lys10]n/ofq(1-13)nh2 1-benzhydryl-4-(4-butylphenyl)piperidin-4-ol 1-benzhydryl-4-cyclopropylpiperidin-4-ol [nphe(1)]-nociceptin (1-13)-nh(2) 1-(3,3-diphenylpropyl)-4-phenylpiperidin-4-ol 4-phenyl-1-(3-phenylpropyl)piperidin-4-ol 4-phenyl-1-(1-phenylpropan-2-yl)piperidin-4-ol 6-(4-(2-(benzylamino)ethyl)phenoxy)picolinamide [tyr-pro-phe-nh-ch2-]2 3-(2-methyl-2-aza-bicyclo[3.3.1]non-5-yl)-phenol [tyr-pro-phe-nh-]2 [tyr-pro-phe-phe-nh-ch2-]2 (+/-)-trans-u-50488 methanesulfonate [tyr-pro-phe-phe-nh-]2 6-(2-benzylisoindolin-5-yloxy)nicotinamide [d-ala2]met-enkephalinamide 5-(6-chloro-2-hexyl-1h-indol-1-yl)-5-oxo-valeric acid 5-oxo-ode 5-oxo-15-hete 5-oxo-12-hete [3h]5-oxo-ete 5-oxo-20-hete 5-oxo-c20:3 5s-hpete [mpa1, d-tyr(et)2, d-tic7, d-tic9]ot [mpa1, d-tyr(et)2, aib7, d-tic9]ot [d-tic7]ot [35s]-non-peptide ot antagonist [pip7]ot [mpa1, d-tyr(et)2, d-tic7]ot [mpa1, d-tyr(et)2, l-tic7]ot [mpa1, d-tyr(et)2, pip7]ot [mpa1, d-tic2, aib7]ot [mpa1, l-tic7]ot [mpa1, d-tic7]ot [mpa1, d-tyr(et)2, gly(but)7]ot [aib7]ot [l-tic7]ot [mpa1, d-tyr(et)2, d-tic7, aib9]ot [mpa1, d-tyr(et)2, aib7]ot [mpa1, d-tyr(et)2, gly(but)3, gly(but)7]ot [gly(but)7]ot [3h]a317491 2,2'-pyridylisatogen tosylate 2-cl-adp(alpha-bh3) 1-(3,4-dichlorophenyl)-3-(3,5-dichlorophenyl)urea 2',3'-ddatp 2mesatp [35s]adpbetas 2-chloroadenosine-5-triphosphate [32p]mrs2500 2mesadp [3h]psb-0413 2mesamp [33p]2mesadp 2-thio-udp 4-thio-utp 5brutp 2-thioutp (n)methanocarba-utp 2-amino-uridine-5'-monophosphate 3-phenacyl-udp 12-bromododecanoic acid 6-amino-benzo[de]isoquinoline-1,3-dione 5-fluoro-1-[4-(4-phenyl-3,6-dihydropyridin-1(2h)-yl)butyl]quinazoline-2,4(1h,3h)-dione 3-oxo-2,3-dihydro-1h-indazole-4-carboxamide derivative 2 8-hydroxy-2-(4-nitro-phenyl)-3h-quinazolin-4-one 3-aminobenzo[c][1,5]naphthyridin-6(5h)-one 5-aminoisoquinolin-1(2h)-one 3-phenylquinoline-8-carboxamide 3-ethynylquinoline-8-carboxamide 8-hydroxy-2-phenyl-3h-quinazolin-4-one 3-(4-aminophenyl)quinoxaline-5-carboxamide 2-(3-chlorophenyl)-2h-indazole-7-carboxamide 3-phenyl isoquinolin-1(2h) derivative 1 3-(4-methoxyphenyl)quinoxaline-5-carboxamide 4-benzylphthalazin-1(2h)-one 8-methoxy-2-methyl-3h-quinazolin-4-one 3-methoxybenzamide 2-(3-piperidin-1-yl-propyl)-3h-quinazolin-4-one 5-methylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione 5-amino-3,4-dihydroisoquinolin-1(2h)-one 3-methylquinoline-8-carboxamide 2-(4-amino-phenyl)-8-hydroxy-3h-quinazolin-4-one 8-methoxy-2-phenyl-3h-quinazolin-4-one 2-benzyl-2h-indazole-7-carboxamide 4-carboxamido-isoindolinone derivative 5 4-(4-morpholin-4-yl-butyl)-2h-phthalazin-1-one 3-oxo-2,3-dihydro-1h-indazole-4-carboxamide derivative 4 2-phenyl-2h-benzo[d][1,2,3]triazole-4-carboxamide 3-morpholin-4-ylmethyl-5h-phenanthridin-6-one (e)-n-(4-phenylthiazol-2-yl) cinnamamide 8-methoxy-2-(4-nitro-phenyl)-3h-quinazolin-4-one 3-aminobenzamide 3-ethylquinoline-8-carboxamide 4-carboxamido-isoindolinone derivative 4 8-nitro-6h,11h-indeno[1,2-c]isoquinolin-5-one 9-fluoro-6h,11h-indeno[1,2-c]isoquinolin-5-one 2-(4-methoxyphenyl)quinoline-8-carboxamide 2-(2-chlorophenyl)-2h-indazole-7-carboxamide 2-(4-azido-phenyl)-8-methoxy-3h-quinazolin-4-one 3-oxo-2,3-dihydro-1h-indazole-4-carboxamide derivative 1 2,8-dimethyl-3h-quinazolin-4-one 3-oxo-2,3-dihydro-1h-indazole-4-carboxamide derivative 5 2-phenyl-2h-indazole-7-carboxamide 3-(4-cyanophenyl)quinoxaline-5-carboxamide 4-carboxamido-isoindolinone derivative 1 8-fluoro-6h,11h-indeno[1,2-c]isoquinolin-5-one 4-methylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione 3-phenyl isoquinolin-1(2h) derivative 2 2,3-dihydro-1h-benzo[de]isoquinolin-1-one 2-(4-methoxy-phenyl)-8-methyl-3h-quinazolin-4-one 2-ethylquinoline-8-carboxamide 2-(3'-methoxyphenyl) benzimidazole-4-carboxamide 1,2,3,4,4a,5-hexahydrophenanthridin-6(10bh)-one 2-{3-[4-(4-fluorophenyl)-3,6-dihydro-1(2h)-pyridinyl]propyl}-8-methyl-4(3h)-quinazolinone 2h-isoquinolin-1-one 4-amino-1,8-naphthalimide 1,7,8,9-tetrahydro-1,5-diaza-trindene-4,6-dione 7-azaindole derivative 8 3-prop-1-ynylquinoline-8-carboxamide 2-(4-chlorophenyl)-5-quinoxalinecarboxamide 9-amino-6h,11h-indeno[1,2-c]isoquinolin-5-one 8-methyl-2-phenyl-3h-quinazolin-4-one 2-phenylquinoline-8-carboxamide 8-amino-6h,11h-indeno[1,2-c]isoquinolin-5-one 2-(4-chlorophenyl)-2h-indazole-7-carboxamide 2-(4-hydroxy-phenyl)-8-methyl-3h-quinazolin-4-one 3,4-dihydro-5-methyl-isoquinolinone 4-carboxamido-isoindolinone derivative 3 3-oxo-2,3-dihydro-1h-indazole-4-carboxamide derivative 3 3-ethenylquinoline-8-carboxamide 2-(4-amino-phenyl)-8-methyl-3h-quinazolin-4-one 2-phenylpyrazolo-[1,5-a]pyridine-7-carboxamide 3-hydroxy-benzamide 8-methyl-2-(4-nitro-phenyl)-3h-quinazolin-4-one 4-carboxamido-isoindolinone derivative 2 4-(5-morpholin-4-yl-pentyl)-2h-phthalazin-1-one 2-methylquinoline-8-carboxamide 5-chloro-2-methyl-3h-quinazolin-4-one 2-methyl-3,5,7,8-tetrahydro-4h-thiopyrano[4,3-d]pyrimidin-4-one 4-[3-(1,4-diazepan-1-ylcarbonyl)-4-fluorobenzyl]phthalazin-1(2h)-one 5-(hexahydro-2-oxo-1h-thieno[3,4-d]imidazol-6-yl)pentanal 1-(2-fluorobenzyl)-3-butyl-8-(n-acetyl-4-aminobenzyl)-xanthine 1-allyl-3-butyl-8-(n-acetyl-4-aminobenzyl)-xanthine 5'-guanylylmethylenebisphosphonate 1d05 1,2,4-oxadiazole derivative 1 1,3,4-oxadiazole derivative 2 609a 1,2,4-oxadiazole derivative 2 1,3,4-oxadiazole derivative 1 4,5-bis(4-methoxyphenyl)-2-thiophen-2-yl-1h-imidazole 1,2,4-triazole [4,3-a]quinoxaline derivative 1 6,7-dimethoxy-4-[(3r)-3-(2-naphthyloxy)pyrrolidin-1-yl]quinazoline 1,2,4-triazole [4,3-a]quinoxaline derivative 3 1,2,4-triazole [4,3-a]quinoxaline derivative 2 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 3 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 6 2-({4-[4-(pyridin-4-ylmethyl)-1h-pyrazol-3-yl]phenoxy}methyl)quinoline 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 5 2-{[4-(4-pyridin-4-yl-1h-pyrazol-3-yl)phenoxy]methyl}quinoline 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 4 3-isobutyl-1-methyl-7h-xanthine 2-morpholin-4-yl-8-phenylethynyl-chromen-4-one 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 2 1,2,4-triazole [1,5-a]pyrimidin-7-yl derivative 3 1,2,4-triazole [1,5-a]pyrimidin-7-yl derivative 2 1,2,4-triazole [1,5-a]pyrimidin-7-yl derivative 1 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 1 8-chloro-1,3-dihydro-imidazo[4,5-b]quinolin-2-one 7-iodo-1,5-dihydro-imidazo[2,1-b]quinazolin-2-one 8-methyl-2-morpholino-7-phenyl-4h-chromen-4-one 8-methyl-1,3-dihydro-imidazo[4,5-b]quinolin-2-one 1,5-dihydro-imidazo[2,1-b]quinazolin-2-one 1,3-dihydro-naphtho[2,3-d]imidazol-2-one 6-(2-imidazol-1-yl-vinyl)-1h-quinolin-2-one 7-fluoro-1,3-dihydro-imidazo[4,5-b]quinolin-2-one 2-morpholino-7-(2-phenylethynyl)-4h-chromen-4-one 7-methyl-1,3-dihydro-imidazo[4,5-b]quinolin-2-one 8-methyl-2-morpholino-7-phenoxy-4h-chromen-4-one 1,3-dihydro-imidazo[4,5-b]quinolin-2-one 1,3,9,9a-tetrahydro-imidazo[4,5-b]quinolin-2-one 7-ethoxy-1,3-dihydro-imidazo[4,5-b]quinolin-2-one 5-methyl-1,3-dihydro-imidazo[4,5-b]quinolin-2-one 2-morpholino-7-phenyl-4h-chromen-4-one 6-imidazol-1-yl-3,4-dihydro-1h-quinolin-2-one 7-chloro-1,3-dihydro-imidazo[4,5-b]quinolin-2-one 6-(4-{[2-(3-iodobenzyl)-3-oxocyclohex-1-en-1-yl]amino}phenyl)-5-methyl-4,5-dihydropyridazin-3(2h)-one 6-azido-8-(3-iodo-phenyl)-quinoline (2,5-diphenyl-furan-3-yl)-phenyl-methanone 2,5-bis-(3-cyclopentyloxy-4-methoxy-phenyl)-furan 8-(3-azido-phenyl)-6-pyridin-4-ylmethyl-quinoline 1-methyl-3-propyl-3,7-dihydro-purine-2,6-dione 2,5-bis-(3,4-dimethoxy-phenyl)-furan 8-(3-azido-phenyl)-6-iodo-quinoline (s)-rolipram (4r)-4-(3-butoxy-4-methoxybenzyl)imidazolidin-2-one 6-imidazol-1-ylmethyl-8-phenyl-quinoline 8-(3-nitro-phenyl)-6-phenyl-[1,7]naphthyridine 4-[8-(3-nitrophenyl)-1,7-naphthyridin-6-yl]benzoic acid 8-(3-nitro-phenyl)-6-pyridin-4-ylmethyl-quinoline (r)-rolipram 1-butyl-3-methyl-3,7-dihydro-purine-2,6-dione 4-(2,5-diphenyl-furan-3-yl)-morpholine 1-ethyl-n-(phenylmethyl)-4-(tetrahydro-2h-pyran-4-ylamino)-1h-pyrazolo[3,4-b]pyridine-5-carboxamide 3,5-dimethyl-1-(3-nitrophenyl)-1h-pyrazole-4-carboxylic acid ethyl ester 3-(2-bromophenyl)-2-thioxo-(1h )-quinazolin-4-one 1-(2-chlorophenyl)-3,5-dimethyl-1h-pyrazole-4-carboxylic acid ethyl ester 1-(4-methoxyphenyl)-3,5-dimethyl-1h-pyrazole-4-carboxylic acid ethyl ester 1-(4-aminophenyl)-3,5-dimethyl-1h-pyrazole-4-carboxylic acid ethyl ester 3,5-dimethyl-1h-pyrazole-4-carboxylic acid ethyl ester 2-[3-(2-hydroxy-1,1-dihydroxymethyl-ethylamino)-propylamino]-2-hydroxymethyl-propane-1,3-diol 3,5-dimethyl-1-phenyl-1h-pyrazole-4-carboxylic acid ethyl ester 8-prenylquercetin 7-(2-hydroxyethyl)-3-o-rhamnosylicariin 5-ethoxy-4-(1-methyl-7-oxo-3-propyl-6,7-dihydro-1h-pyrazolo[4,3-d]pyrimidin-5-yl)thiophene-2-sulfonamide 8-prenylapigenin 3,7-bis(2-hydroxyethyl)icaritin 3-(2,6-difluorophenyl)-2-(methylthio)quinazolin-4(3h)-one 8-(2,4-dimethoxyphenyl)-9h-purine-2,6-diamine 8-(2,3,4-trimethoxyphenyl)-9h-purine-2,6-diamine 6-phenylsulfanylmethyl-pteridine-2,4-diamine 5-formyl-6-hydrofolic acid 8-(2,4,6-trimethoxyphenyl)-9h-purine-2,6-diamine 6-(2-phenylsulfanyl-ethyl)-pteridine-2,4-diamine 5-(2-fluorobenzyloxy)quinazoline-2,4-diamine 5-p-tolylsulfanyl-quinazoline-2,4-diamine 8-(3,4,5-trimethoxyphenyl)-9h-purine-2,6-diamine 2'-monophosphoadenosine-5'-diphosphate 2-[(formyl-hydroxy-amino)-methyl]-heptanoic acid [1-(2-hydroxymethyl-pyrrolidine-1-carbonyl)-2-methyl-propyl]-amide 8-pyridin-4-yl-9h-purine-2,6-diamine 3-benzyl-2-mercapto-6-nitroquinazolin-4(3h)-one 5-phenethyl-quinazoline-2,4-diamine 6-m-tolyl-pteridine-2,4,7-triamine 8-(2,6-dichloro-phenyl)-9h-purine-2,6-diamine 8-(3,5-dimethoxyphenyl)-9h-purine-2,6-diamine 5-((e)-styryl)-quinazoline-2,4-diamine 3-phenylsulfanylmethyl-quinoxaline-5,7-diamine 8-(3,4-dimethoxyphenyl)-9h-purine-2,6-diamine 7-methyl-7h-pyrrolo[3,2-f]quinazoline-1,3-diamine 6-phenylaminomethyl-quinazoline-2,4-diamine 6,7-diphenyl-pteridine-2,4-diamine 2-allylthio-6-amino-3-benzyl-quinazolin-4(3h)-one 3-benzyl-2-ethylthio-6-nitro-quinazolin-4(3h)-one 8-(3,4-dichlorophenyl)-9h-purine-2,6-diamine 7h-pyrrolo[3,2-f]quinazoline-1,3-diamine 8-benzyl-9h-purine-2,6-diamine 8-(2,4,5-trimethoxyphenyl)-9h-purine-2,6-diamine 2-allylthio-3-benzyl-6-nitro-quinazolin-4(3h)-one 4-(2,6-diamino-9h-purin-8-yl)-2,6-dimethoxyphenol 8-(2,5-dimethoxyphenyl)-9h-purine-2,6-diamine 3-(3,4-dichloro-phenyl)-6,7-dimethoxy-quinoline 4-(6,7-dimethoxy-quinolin-3-yl)-benzoic acid 5,7-dimethyl-3-thiophen-3-yl-quinoline 5,7-dimethoxy-3-thiophen-3-yl-quinoline 6,7-dimethoxy-3-pyridin-4-yl-quinoline 5-(6,7-dimethoxy-quinolin-3-yl)-1h-pyridin-2-one 6,7-dimethoxy-3-(3-methoxy-phenyl)-quinoline 1-phenyl-1h-benzoimidazole 6-methoxy-3-pyridin-4-yl-quinoline 6,7-dimethoxy-3-phenylethynyl-quinoline 5,6,7-trimethoxy-3-pyridin-4-yl-quinoline 5-methoxy-1-phenyl-1h-benzoimidazole 3-cyclopentyl-6,7-dimethoxy-quinoline 3-benzyloxy-6,7-dimethoxy-quinoline 3-pyridin-4-yl-quinoline 6,7-dimethoxy-3-pyridin-3-yl-quinoline 3-(1h-indol-3-yl)-quinoline 7-methoxy-3-pyridin-4-yl-quinoline 4-(6,7-dimethoxy-quinolin-3-yl)-phenol 3-(4-fluoro-phenyl)-6,7-dimethoxy-quinoline 6,7-dichloro-3-thiophen-3-yl-quinoline 6,7-dimethoxy-3-phenyl-quinoline 6,7-dimethoxy-3-p-tolyl-quinoline 3-(1h-indol-3-yl)-6,7-dimethoxy-quinoline 6,7-dimethoxy-3-(4-nitro-phenyl)-quinoline 5,7-dimethoxy-3-pyridin-4-yl-quinoline 6,7-dimethoxy-3-(2-methoxy-phenyl)-quinoline 6,7-difluoro-3-thiophen-3-yl-quinoline 6,7-dimethoxy-3-thiophen-2-yl-quinoline 3-(3-fluoro-phenyl)-6,7-dimethoxy-quinoline 7-chloro-3-pyridin-4-yl-quinoline 6,7-dimethoxy-3-(4-methoxy-phenyl)-quinoline 7-fluoro-3-thiophen-3-yl-quinoline 4-(5-methoxy-benzoimidazol-1-yl)-phenylamine 3-(3,4-difluoro-phenyl)-6,7-dimethoxy-quinoline 3-(3,4-dimethoxy-phenyl)-6,7-dimethoxy-quinoline 4-(3,4-dimethoxy-phenoxy)-6,7-dimethoxy-quinoline 3-cyclopent-1-enyl-6,7-dimethoxy-quinoline 3-pyridin-4-yl-quinoline-5,7-diol 3-(2-cyclohexyl-ethyl)-6,7-dimethoxy-quinoline 7-thiophen-3-yl-[1,3]dioxolo[4,5-g]quinoline 3-thiophen-3-yl-quinoline 3-pyridin-3-yl-quinoline-6,7-diol 6-methoxy-3-thiophen-3-yl-quinoline 3-pyridin-4-yl-quinolin-7-ol 4-benzoimidazol-1-yl-phenylamine 7-methoxy-3-thiophen-3-yl-quinoline 3-cyclohexylethynyl-6,7-dimethoxy-quinoline 5-fluoro-3-thiophen-3-yl-quinoline 6,7-dimethoxy-3-((e)-styryl)-quinoline 1-phenyl-1h-benzoimidazol-5-ol 3-((e)-styryl)-quinoline 4-(3-ethoxy-phenoxy)-6,7-dimethoxy-quinoline 4-(3-ethyl-phenoxy)-6,7-dimethoxy-quinoline (2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenylamine 6,7-dimethoxy-4-m-tolyloxy-quinoline 6,7-dimethoxy-4-(3-methoxy-phenoxy)-quinoline 6,7-dimethoxy-4-(4-methoxy-phenoxy)-quinoline 6,7-dimethoxy-4-(3-nitro-phenoxy)-quinoline 4-(3,5-dimethoxy-phenoxy)-6,7-dimethoxy-quinoline 3-(4-dimethylamino-benzylidenyl)-2-indolinone 4-(3-fluoro-phenoxy)-6,7-dimethoxy-quinoline 4-(2,3-dimethoxy-phenoxy)-6,7-dimethoxy-quinoline 3-(6,7-dimethoxy-quinolin-4-yloxy)-phenol 3-(6,7-dimethoxy-quinolin-4-yloxy)-phenylamine 6,7-dimethoxy-4-phenoxy-quinoline 6,7-dimethoxy-4-(2-methoxy-phenoxy)-quinoline 4-[(3-chloro-4-{[(2r)-3,3,3-trifluoro-2-hydroxy-2-methylpropanoyl]amino}phenyl)sulfonyl]-n,n-dimethylbenzamide 1,2-dihydroindazolo[4,3-bc][1,5]benzoxazepine derivative 1 4-({(2r,5s)-2,5-dimethyl-4-[(2r)-3,3,3-trifluoro-2-hydroxy-2-methylpropanoyl]piperazin-1-yl}carbonyl)benzonitrile (2r)-n-{4-[ethyl(phenyl)sulfamoyl]-2-methylphenyl}-3,3,3-trifluoro-2-hydroxy-2-methylpropanamide 4-[4-(4-methoxyphenyl)-5-methyl-1h-pyrazol-3-yl]benzene-1,3-diol 5-hydroxy-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-2-one 1-{2-oxo-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-5-yl}urea 2-(1h-imidazol-1-yl)-9-methoxy-8-(2-methoxyethoxy)benzo[c][2,7]naphthyridin-4-amine 3-(1h-indol-3-yl)-4-(1-{2-[(2s)-1-methylpyrrolidinyl]ethyl}-1h-indol-3-yl)-1h-pyrrole-2,5-dione 10,11-dimethoxy-4-methyldibenzo[c,f]-2,7-naphthyridine-3,6-diamine 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione 7-hydroxystaurosporine (2r)-2-({6-[benzyl(methyl)amino]-9-isopropyl-9h-purin-2-yl}amino)butan-1-ol 3po 7-hydroxy-4-methyl-3-(2-hydroxy-ethyl)coumarin 3-phospho-d-glyceric acid (2r)-2-methyl-4,5-dideoxy 6-phosphogluconic acid 4-phospho-d-erythronate 5-deoxy-5-phosphono-d-arabinonate 2-acetamido-2-deoxy-beta-d-glucopyranose(beta1-4)-2-acetamido-1,6-anhydro-3-o-[(r)-1-carboxyethyl]-2-deoxy-beta-d-glucopyranose-l-alanyl-gamma-d-glutamyl-meso-diaminopimelyl-d-alanine 6-(3-nitro-phenyl)-3h-benzothiazol-2-one 1-benzyl-3-phenylquinazoline-2,4(1h,3h)-dione 4-(2,4-diethyl-1h-pyrrol-3-yloxy)benzonitrile 5,n-dihydroxythalidomide 3,3-dimethyl-5-m-tolyl-2,3-dihydro-1h-inden-1-one 2,2,4-trimethyl-6-phenyl-1,2-dihydro-quinoline 3-phenyl-1-propylquinazoline-2,4(1h,3h)-dione 3-(3,3-dimethyl-2-oxoindolin-5-yl)benzonitrile 5-(2-oxoindolin-5-yl)-1h-pyrrole-2-carbonitrile 2-(4-amino-3'-chloro-biphenyl-3-yl)-propan-2-ol 3-(4-morpholinothieno[3,2-d]pyrimidin-2-yl)phenol 2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-one (5e)-5-[(2,2-difluoro-1,3-benzodioxol-5-yl)methylene]-1,3-thiazolidine-2,4-dione 1-methyl-3-naphthalen-2-yl-1h-pyrazolo[3,4-d]pyrimidin-4-amine 5,5-dimethyl-2-morpholin-4-yl-5,6-dihydro-1,3-benzothiazol-7(4h)-one 3-[4-amino-1-(1-methylethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]phenol (4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile 3,4-dihydroxy-1-methylquinolin-2(1h)-one (2s)-1,3-benzothiazol-2-yl{2-[(2-pyridin-3-ylethyl)amino]pyrimidin-4-yl}ethanenitrile 2,3-diphenyl-1h-indole-7-carboxylic acid 6-(5-bromo-2-hydroxyphenyl)-2-oxo-4-phenyl-1,2-dihydropyridine-3-carbonitrile 4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-one 4-[3-(4-chlorophenyl)-2,1-benzisoxazol-5-yl]pyrimidin-2-amine (3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-one (r)-3-(2-naphthamido)-4-m-tolylbutanoic acid 3,6,9,12,15,18-hexaoxaicosane (r)-2-(2-naphthamido)-5-phenylpent-4-ynoic acid (r,)-2-(2-naphthamido)-5-phenylpent-4-enoic acid (r)-2-(2-naphthamido)-3-p-tolylpropanoic acid (r)-2-(2-naphthamido)-3-m-tolylpropanoic acid 1,2-diacyl-sn-glycero-3-phosphoinositol (z,z)-4-hydroxy-n,n,n-trimethyl-10-oxo-7-[(1-oxo-9-octadecenyl)oxy]-3,5,9-trioxa-4-phosphaheptacos-18-en-1-aminium-4-oxide (2s)-2-(4-chlorophenyl)-2-[4-(1h-pyrazol-4-yl)phenyl]ethanamine 4-(4-chlorobenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-aminium 6-{4-[4-(4-chlorophenyl)piperidin-4-yl]phenyl}-9h-purine 3-pyridin-4-yl-2,4-dihydro-indeno[1,2-.c.] pyrazole (1s)-2-(1h-indol-3-yl)-1-[({5-[(e)-2-pyridin-4-ylvinyl]pyridin-3-yl}oxy)methyl]ethylamine 5-(2-methylpiperazine-1-sulfonyl)isoquinoline 5-benzyl-1,3-thiazol-2-amine (2s)-1-(3h-indol-3-yl)-3-{[5-(6-isoquinolinyl)-3-pyridinyl]oxy}-2-propanamine (2r)-2-(4-chlorophenyl)-2-phenylethanamine (1s)-1-(1h-indol-3-ylmethyl)-2-(2-pyridin-4-yl-[1,7]naphtyridin-5-yloxy)-ehylamine 2-[4-(3-methyl-1h-pyrazol-4-yl)phenyl]ethanamine (s)-1-phenyl-1-[4-(9h-purin-6-yl)phenyl]methanamine (s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazine 1-[4-(4-chlorophenyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methanamine 3-pyridin-4-yl-1h-indazole 1-[4-(4-chlorobenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methanamine (2r)-2-(4-chlorophenyl)-2-[4-(1h-pyrazol-4-yl)phenyl]ethanamine (4r,2s)-5'-(4-(4-chlorobenzyloxy)pyrrolidin-2-ylmethanesulfonyl)isoquinoline 6-(2-fluorobenzyl)-2,4-dimethyl-4,6-dihydro-5h-thieno[2',3':4,5]pyrrolo[2,3-d]pyridazin-5-one 1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4-[(4-methoxyphenyl)sulfonyl]piperazine 1-[(2,6-difluorophenyl)sulfonyl]-4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)piperazine 4'-hydroxy-6,3',5'-triprenylisoflavonone 1-o-octyl-2-heptylphosphonyl-sn-glycero-3-phosphoethanolamine 3,9-dihydroxy-2,10-diprenylpterocap-6a-ene 1-decyl-3-trifluoro ethyl-sn-glycero-2-phosphomethanol 1-{2-[2-(2-methoxyethoxy)ethoxy]ethoxy}-4-(1,1,3,3-tetramethylbutyl)benzene 6-phenyl-4(r)-(7-phenyl-heptanoylamino)-hexanoic acid (1-benzyl-5-methoxy-2-methyl-1h-indol-3-yl)acetic acid 4-(1-benzyl-3-carbamoylmethyl-2-methyl-1h-indol-5-yloxy)-butyric acid (2r)-2-acetamido-3-(octadecyloxy)propyl 2-(methylsulfanyl)ethyl hydrogen phosphate [3-(1-benzyl-3-carbamoylmethyl-2-methyl-1h-indol-5-yloxy)-propyl-]-phosphonic acid (2e)-1-[2-hydroxy-4-methoxy-5-(3-methylbut-2-en-1-yl)phenyl]-3-(4-hydroxyphenyl)prop-2-en-1-one (2-carbamoylmethyl-5-propyl-octahydro-indol-7-yl)acetic acid 9-hydroxy-8-methoxy-6-nitro-phenanthrol[3,4-d][1,3]dioxole-5-carboxylic acid 3-{3-[(dimethylamino)methyl]-1h-indol-7-yl}propan-1-ol 1,1,1,2,2-pentafluoro-9-phenyl-nonan-3-one 1,1,1-trifluoro-4-(4-hexyloxy-phenyl)-butan-2-one 1,1,1,2,2-pentafluoro-8-phenyl-octan-3-one (s)-methyl 4-(2-oxohexadecanamido)octanoate [6,4''']biflavone 1,1,1,2,2,3,3,5-octafluoro-8-phenyloctan-4-one (z)-1,1,1,2,2,3,3-heptafluorohenicos-12-en-4-one 1,1,1-trifluoro-5-(4-octylphenoxy)pentan-2-one 1,1,1-trifluoro-7-phenylheptan-2-one [6,3''']biflavone 1,1,1-trifluoro-6-(naphthalen-2-yl)hexan-2-one 1,1,1-trifluoro-8-phenyl-octan-2-one [3,4''']biflavone 4-(4-decyloxy-phenyl)-1,1,1-trifluoro-butan-2-one 4-(2-oxohexadecanamido)butanoic acid 1,1,1,3-tetrafluoro-6-phenylhexan-2-one 1,1,1,2,2,3,3-heptafluoro-8-phenyloctan-4-ol 1,1,1-trifluoro-6-(4-hexyloxy-phenyl)-hexan-2-one 1,1,1-trifluoroheptadecan-2-one [4',4''']-biflavone (s)-tert-butyl 4-(2-oxohexadecanamido)pentanoate 1,1,1,2,2,4-hexafluoro-7-phenylheptan-3-one 1,1,1,3-tetrafluoro-7-phenylheptan-2-one 1,1,1,3-tetrafluoro-heptadecan-2-one (s)-ethyl 6-(2-oxohexadecanamido)decanoate 1-imidazol-1-yl-3-(4-octylphenoxy)propan-2-one 6-(4-decyloxy-phenyl)-1,1,1-trifluoro-hexan-2-one 4-fluorobenzaldehyde o-benzoyloxime 3,4-difluorobenzaldehyde o-benzoyloxime (e)-(thiophen-2-ylmethylidene)amino benzoate 5-(dimethylamino)-2-naphthalenesulfonic acid 1-guanidino-n-phenyl-7-isoquinolinesulphonamide 7-methoxy-8-[1-(methylsulfonyl)-1h-pyrazol-4-yl]naphthalene-2-carboximidamide 4-chloro-1-guanidino-7-isoquinolinesulphonamide 6-fluoro-2-[2-hydroxy-3-(2-methyl-cyclohexyloxy)-phenyl]-1h-indole-5-carboxamidine 4-(2-aminoethoxy)-3,5-dichloro-n-[3-(1-methylethoxy)phenyl]benzamide 2-(2-hydroxy-5-methoxy-phenyl)-1h-benzoimidazole-5-carboxamidine (4-guanidino-benzyl)-carbamic acid benzyl ester 4-(2-aminoethoxy)-n-(3-chloro-2-ethoxy-5-piperidin-1-ylphenyl)-3,5-dimethylbenzamide 6-(n-phenylcarbamyl)-2-naphthalenecarboxamidine 1-[4-(2-oxo-2-phenylethyl)phenyl]guanidine 4-(2-aminoethoxy)-n-(3-chloro-5-piperidin-1-ylphenyl)-3,5-dimethylbenzamide [2,4,6-triisopropyl-phenylsulfonyl-l-[3-amidino-phenylalanine]]-piperazine-n'-beta-alanine 2-amino-1h-benzimidazol-5-ol 6-[(z)-amino(imino)methyl]-n-[4-(aminomethyl)phenyl]-4-(pyrimidin-2-ylamino)-2-naphthamide 6-[n-(1-isopropyl-1,2,3,4-tetrahydro-7-isoquinolinyl)carbamyl]-2-naphthalenecarboxamidine 6-fluoro-2-(2-hydroxy-3-isobutoxy-phenyl)-1h-benzoimidazole-5-carboxamidine 1-guanidino-7-isoquinolinesulphonamide 6-[n-(4-ethyl-1,2,3,4-tetrahydro-6-isoquinolinyl)carbamyl]-2-naphthalenecarboxamidine 6-[(z)-amino(imino)methyl]-n-[3-(cyclopentyloxy)phenyl]-2-naphthamide 2-amino-5-hydroxy-benzimidazole (2r)-1-(2,6-dimethylphenoxy)propan-2-amine 8-(pyrimidin-2-ylamino)naphthalene-2-carboximidamide 6-[n-(4-(aminomethyl)phenyl)carbamyl]-2-naphthalenecarboxamidine 4-(2-aminoethoxy)-n-(2,5-diethoxyphenyl)-3,5-dimethylbenzamide 5-methylsulfanyl-thiophene-2-carboxamidine 6-[n-(1-isopropyl-3,4-dihydro-7-isoquinolinyl)carbamyl]-2-naphthalenecarboxamidine 1-(pyridin-4-yl)piperazine 1-(2-oxo-2-p-tolyl-ethyl)-1h-indole-2,3-dione 1-[5-methyl-2-(trifluoromethyl)furan-3-yl]-3-[5-[2-[[6-(1h-1,2,4-triazol-5-ylamino)pyrimidin-4-yl]amino]ethyl]-1,3-thiazol-2-yl]urea 3-[3-(3-methyl-6-{[(1s)-1-phenylethyl]amino}-1h-pyrazolo[4,3-c]pyridin-1-yl)phenyl]propanamide 3-[3-chloro-5-(5-{[(1s)-1-phenylethyl]amino}isoxazolo[5,4-c]pyridin-3-yl)phenyl]propan-1-ol [(3r)-7-nitro-1,2,3,4-tetrahydroisoquinolin-3-yl]methanol 7-iodo-1,2,3,4-tetrahydro-isoquinoline (1r)-2-amino-1-[3-(trifluoromethyl)phenyl]ethanol (3r)-n-(4-chlorophenyl)-3-(hydroxymethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide (1s,4r,9s)-5-(trifluoromethyl)-1,2,3,4-tetrahydro-1,4-methanonaphthalen-9-amine 1,2,3,4-tetrahydro-isoquinoline-7-sulfonic acid amide (3r)-3-(fluoromethyl)-n-(3,3,3-trifluoropropyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide 8,9-dichloro-2,3,4,5-tetrahydro-1h-benzo[c]azepine (3r)-3-(fluoromethyl)-7-(thiomorpholin-4-ylsulfonyl)-1,2,3,4-tetrahydroisoquinoline 7,8-dichloro-1,2,3,4-tetrahydroisoquinoline 8-iodo-guanine 9-(5,5-difluoro-5-phosphonopentyl)guanine 8-aminoguanine 2-amino-7-[2-(2-hydroxy-1-hydroxymethyl-ethylamino)-ethyl]-1,7-dihydro-purin-6-one 8-aza-dadme-immh 2-hydroxymethyl-pyrrolidine-3,4-diol 9-deazainosine-2',3'-o-ethylidenephosphonate (3r,4r)-3-hydroxy-4-(hydroxymethyl)-1-[(4-oxo-4,4a,5,7a-tetrahydro-3h-pyrrolo[3,2-d]pyrimidin-7-yl)methyl]pyrrolidinium 2'3'-dideoxyinosine 2,6-diamino-(s)-9-[2-(phosphonomethoxy)propyl]purine 3-((2-pyrrolidine-1-yl)-ethyl)uracil 3'-deoxyguanosine 8-amino-9-benzylguanine 5'-methylthio-immucillin-h 5'-deoxy-4'-hydroxy-5'-methylthio-dadme-immh 9-deazahypoxanthine 8-aminoguanosine (+/-)-5'-deoxy-4'-fluoro-5'-methylthio-dadme-immh (2s,3r,4s,5s)-3,4-dihydroxy-2-[(methylsulfanyl)methyl]-5-(4-oxo-4,5-dihydro-1h-pyrrolo[3,2-d]pyrimidin-7-yl)pyrrolidinium 9-deazainosine 5'-phenylthio-immh 8-azaguanine 3-deoxyguanosine 5'-methylthio-immh (1s)-1,2,3,4-tetrahydro-benzo[c]phenanthrene-2,3,4-triol 1,2,3-trihydroxy-1,2,3,4-tetrahydrobenzo[a]pyrene 2'-deoxy-n-(naphthalen-1-ylmethyl)guanosine 5'-(dihydrogen phosphate) 1-[2-deoxyribofuranosyl]-2,4-difluoro-5-methyl-benzene-5'monophosphate (e)-12-nitrooctadec-12-enoic acid (9z,12e)-12-nitrooctadeca-9,12-dienoic acid 8s-hete (e)-13-nitrooctadec-12-enoic acid (e)-4-(3,5-dimethoxystyryl)phenol {4-[3-(4-acetyl-3-hydroxy-2-propylphenoxy)propoxy]phenoxy}acetic acid (2s)-2-{3-[({[2-fluoro-4-(trifluoromethyl)phenyl]carbonyl}amino)methyl]-4-methoxybenzyl}butanoic acid 2-({[3-(3,4-dihydroisoquinolin-2(1h)-ylsulfonyl)phenyl]carbonyl}amino)benzoic acid (11e)-octadec-11-enoic acid (4s,5e,7z,10z,13z,16z,19z)-4-hydroxydocosa-5,7,10,13,16,19-hexaenoic acid 3-fluoro-n-[1-(4-fluorophenyl)-3-(2-thienyl)-1h-pyrazol-5-yl]benzenesulfonamide (e)-6-nitrooctadec-5-enoic acid (e)-9-nitrohexadec-9-enoicacid 2-{5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazol-6-yloxy)propoxy]indol-1-yl}ethanoic acid (9z,11e,13s)-13-hydroxyoctadeca-9,11-dienoic acid (5r,6e,8z,11z,14z,17z)-5-hydroxyicosa-6,8,11,14,17-pentaenoic acid (8r,9z,12z)-8-hydroxy-6-oxooctadeca-9,12-dienoic acid [3h]gw2331 3-[5-(2-nitropent-1-en-1-yl)furan-2-yl]benzoic acid (e)-9-nitrooctadec-9-enoic acid 9(s)-hode (2s)-2-(biphenyl-4-yloxy)-3-phenylpropanoic acid (5e,14e)-11-oxoprosta-5,9,12,14-tetraen-1-oic acid (e)-5-nitrooctadec-5-enoic acid (2s)-2-ethoxy-3-{4-[2-(10h-phenoxazin-10-yl)ethoxy]phenyl}propanoic acid 2-{5-[3-(6-benzoyl-1-propylnaphthalen-2-yloxy)propoxy]indol-1-yl}ethanoic acid 3-phenyl acrylic acid derivative 1 (e)-10-nitrohexadec-9-enoic acid (8e,10s,12z)-10-hydroxy-6-oxooctadeca-8,12-dienoic acid (e)-10-nitrooctadec-9-enoic acid 15-deoxy-delta(12, 14)-prostaglandin j(2) [125i]sb-236636 (2s)-2-(4-ethylphenoxy)-3-phenylpropanoic acid (2s)-2-(4-chlorophenoxy)-3-phenylpropanoic acid 3-(5-methoxy-1h-indol-3-yl)propanoic acid (s)-3-(4-(2-carbazol-9-yl-ethoxy)-phenyl)-2-ethoxy-propionic acid (3r)-1-acetyl-3-methylpiperidine 1-(3-benzyloxy-pyridin-2-yl)-3-phenyl-urea 4-[3-(3-benzyloxy-pyridin-2-yl)-ureido]-benzamide 3-[3-(3-benzyloxy-pyridin-2-yl)-ureido]-benzamide 7-amino-4-methyl-chromen-2-one 2,6,8-trimethyl-3-amino-9-benzyl-9-methoxynonanoic acid 9,10-deepithio-9,10-didehydroacanthifolicin (2s,3s,4e,6e,8s,9s)-3-amino-9-methoxy-2,6,8-trimethyl-10-phenyldeca-4,6-dienoic acid 1-hydroxy-1-thio-glycerol (6s)-1-chloro-3-[(4-fluorobenzyl)oxy]-6-(pyrrolidin-1-ylcarbonyl)pyrrolo[1,2-a]pyrazin-4(6h)-one 1-{3-oxo-3-[(2s)-2-(pyrrolidin-1-ylcarbonyl)pyrrolidin-1-yl]propyl}-3-phenylquinoxalin-2(1h)-one 2-{3-[(2s)-4,4-difluoro-2-(pyrrolidin-1-ylcarbonyl)pyrrolidin-1-yl]-3-oxopropyl}-isoindole-1,3(2h)-dione (2s)-1-(6h-indol-3-yl)-3-{[5-(7h-pyrazolo[3,4-c]pyridin-5-yl)pyridin-3-yl]oxy}propan-2-amine 3-[(3-sec-butyl-4-hydroxybenzoyl)amino]azepan-4-yl 4-(2-hydroxy-5-methoxybenzoyl)benzoate 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione (2s)-1-{[5-(1h-indazol-5-yl)-3-pyridinyl]oxy}-3-(7ah-indol-3-yl)-2-propanamine [3h]camp 5-(2-methylpiperazin-1-ylsulfonyl)isoquinoline (rp)-camps 4-cycloheptyliden(4-hydroxyphenyl)methylphenol 2,3,3-triphenyl-acrylonitrile 3-(1h-indol-3-yl)-4-phenylamino-pyrrole-2,5-dione 4-cyclohexyliden(4-hydroxyphenyl)methylphenol 2-(4-hydroxy-phenyl)-3,3-diphenyl-acrylonitrile (-)-cercosporamide 3,3-bis-(4-methoxy-phenyl)-2-phenyl-acrylonitrile [2,2':5',2'']terthiophene-4-carbaldehyde [2,2':5',2'']terthiophene-4,5''-dicarbaldehyde 3,3-bis-(4-hydroxy-phenyl)-2-phenyl-acrylonitrile 4-cyclopentyliden(4-hydroxyphenyl)methylphenol 4-[1-(4-hydroxyphenyl)-3-methyl-1-butenyl]phenol [2,2':5',2'']terthiophen-4-yl-methanol 3-(4-hydroxy-phenyl)-2,3-diphenyl-acrylonitrile 1,2-dioctanoyl-sn-glycerol 13-acetylphorbol 8-octyl-benzolactam-v9 4-(1h-indol-5-yloxy)-5-styrylnicotinonitrile 4-(3h-indol-4-ylamino)-5-styrylnicotinonitrile 4-(1h-indol-5-ylamino)-5-styrylnicotinonitrile 4-(1h-indol-6-ylamino)-5-styrylnicotinonitrile 2-morpholino-6-(naphthalen-1-yl)-4h-pyran-4-one 2-(piperidin-1-yl)-4h-benzo[h]chromen-4-one 2-(2-fluoro-phenyl)-benzo[h]chromen-4-one 2-morpholino-6-(thiophen-2-yl)-4h-pyran-4-one 7-propoxy-2-(morpholin-4-yl)-chromen-4-one 2-pyridin-3-yl-benzo[h]chromen-4-one 8-phenyl-2-thiomorpholin-4-yl-chromen-4-one 2-(furan-2-yl)-6-morpholino-4h-pyran-4-one 6-(3-hydroxyphenyl)-2-morpholino-4h-chromen-4-one 2-morpholino-6-(naphthalen-2-yl)-4h-pyran-4-one 4-thiomorpholin-4-yl-benzo[g]chromen-2-one 2-morpholino-6-(thianthren-1-yl)-4h-chromen-4-one 1-morpholin-4-yl-benzo[f]chromen-3-one 8-(2-acetylphenyl)-2-morpholin-4-ylchromen-4-one 7-phenylethoxy-2-morpholin-4-yl-chromen-4-one 2-morpholin-4-yl-6-phenyl-4h-thiopyran-4-one 6-(4-hydroxyphenyl)-2-morpholino-4h-chromen-4-one 7-ethyloxyethoxy-2-morpholin-4-yl-chromen-4-one 2-morpholino-6-phenyl-4h-pyran-4-one 4-piperidin-1-yl-chromen-2-one 6-tert-butyl-2-morpholin-4-yl-4h-thiopyran-4-one 4-morpholin-4-yl-benzo[g]chromen-2-one 6-(2-acetylphenyl)-2-morpholin-4-ylchromen-4-one 2-(4-amino-phenyl)-benzo[h]chromen-4-one 2-morpholin-4-yl-8-styrylchromen-4-one 8-(4-hydroxyphenyl)-2-morpholin-4-ylchromen-4-one 3-(6-morpholino-4-oxo-4h-pyran-2-yl)benzonitrile 2-morpholin-4-yl-8-thiophen-3-ylchromen-4-one 2-(2-methoxyphenyl)-6-morpholino-4h-pyran-4-one 7-benzyloxy-2-(morpholin-4-yl)-chromen-4-one 4-morpholin-4-yl-benzo[h]chromen-2-one 2-morpholin-4-yl-6-phenyl-chromen-4-one 7-phenyloxyethoxy-2-morpholin-4-yl-chromen-4-one 3-(6-morpholino-4-oxo-4h-pyran-2-yl)benzaldehyde 2-morpholin-4-yl-benzo[h]chromene-4-thione 2-morpholino-6-styryl-4h-pyran-4-one 8-(4-acetylphenyl)-2-morpholin-4-ylchromen-4-one 2-(4-methoxyphenyl)-6-morpholino-4h-pyran-4-one 8-(3-hydroxyphenyl)-2-morpholin-4-ylchromen-4-one 2-(benzofuran-2-yl)-6-morpholino-4h-pyran-4-one 2-[1,4]oxazepan-4-yl-benzo[h]chromen-4-one 8-dibenzofuran-4-yl-2-morpholin-4-ylchromen-4-one 2-morpholino-6-(thiophen-3-yl)-4h-pyran-4-one 8-methoxy-2-morpholin-4-yl-chromen-4-one 6-(4-fluorostyryl)-2-morpholino-4h-chromen-4-one 6-(4-chlorophenyl)-2-morpholin-4-ylpyridin-4-ol 8-(4-chlorophenyl)-2-morpholin-4-ylchromen-4-one 2-(3-acetylphenyl)-6-morpholino-4h-pyran-4-one 8-methyl-2-morpholin-4-yl-chromen-4-one 7-hydroxy-2-(morpholin-4-yl)chromen-4-one 7-methoxy-4-morpholin-4-yl-chromen-2-one 6-methyl-4-morpholin-4-yl-chromen-2-one 2-dibenzofuran-4-yl-6-morpholin-4-yl-pyran-4-one 7-benzoyloxy-2-(morpholin-4-yl)-chromen-4-one 2-morpholino-4h-benzo[g]chromen-4-one 8-furan-2-yl-2-morpholin-4-ylchromen-4-one 3-morpholino-1h-benzo[f]chromen-1-one 2-(1h-indol-5-yl)-6-morpholino-4h-pyran-4-one 8-(1h-indol-5-yl)-2-morpholin-4-ylchromen-4-one 2-biphenyl-4-yl-6-morpholin-4-yl-pyran-4-one 4-morpholin-4-yl-chromen-2-one 2-morpholin-4-yl-8-naphthalen-2-ylchromen-4-one 2-(4-fluorophenyl)-6-morpholino-4h-pyran-4-one 2-morpholinobenzo[h]quinolin-4(1h)-one 6-(4-chlorophenyl)-4-morpholino-2h-pyran-2-one 2-(3-methoxyphenyl)-6-morpholino-4h-pyran-4-one 8-methyl-4-morpholin-4-yl-chromen-2-one 6-isopropyl-2-morpholin-4-yl-4h-thiopyran-4-one 2-thiomorpholino-4h-benzo[h]chromen-4-one 8-biphenyl-2-yl-2-morpholin-4-ylchromen-4-one 2-(2-aminophenyl)-6-morpholino-4h-pyran-4-one 7-methoxy-2-morpholin-4-yl-chromen-4-one 8-methoxy-4-morpholin-4-yl-chromen-2-one 2-morpholino-6-(quinolin-8-yl)-4h-pyran-4-one 2-pyrrolidin-1-yl-benzo[h]chromen-4-one 4-(6-morpholino-4-oxo-4h-pyran-2-yl)benzonitrile 2-morpholin-4-yl-8-phenoxathiin-4-ylchromen-4-one 6-chloro-4-morpholin-4-yl-chromen-2-one 4-morpholino-6-phenyl-2h-pyran-2-one 2-morpholino-6-(naphthalen-1-yl)-4h-chromen-4-one 2-morpholin-4-yl-pyrido[1,2-a]pyrimidin-4-one 2-thiomorpholin-4-yl-pyrido[1,2-a]pyrimidin-4-one 2-morpholin-4-yl-8-thiophen-2-ylchromen-4-one 2-(4-chlorophenyl)-6-morpholino-4h-pyran-4-one 8-phenyl-2-piperidin-1-yl-chromen-4-one 2-(3-fluoro-phenyl)-benzo[h]chromen-4-one 3-(6-morpholino-4-oxo-4h-pyran-2-yl)benzoic acid 6-(4-methoxyphenyl)-4-morpholino-2h-pyran-2-one 6-biphenyl-2-yl-2-morpholin-4-yl-chromen-4-one 6-methoxy-4-morpholin-4-yl-chromen-2-one 3k3a-apc 4-piperidin-4-ylbutanal (2s,3r)-2-[[4-(tert-butylcarbamoyl)piperazine-1-carbonyl]amino]-6-(diaminomethylideneamino)-3-formylhexanoic acid 2-o-(4'-amidinophenyl)-5-o-(3''-amidinophenyl)-1,4:3,6-dianhydro-d-sorbitol 1-{[1-(2-amino-3-phenyl-propionyl)-pyrrolidine-2-carbonyl]-amino}-2-(3-cyano-phenyl)-ethaneboronic acid 4-phenylbutylamine 2,5-bis-o-{3-[amino(imino)methyl]phenyl}-1,4:3,6-dianhydro-d-glucitol 2-(2-methylphenyl)-1h-indole-5-carboximidamide 2,5-o,o-bis-{4',4''-amidinophenyl}-1,4:3,6-dianhydro-d-sorbitol 3-{5-[amino(iminio)methyl]-1h-indol-2-yl}-5-methoxy-1,1'-biphenyl-2-olate 4-(methylsulfonyl)benzenecarboximidamide 2-(3-methylphenyl)-1h-indole-5-carboximidamide 1-benzyl-1h-indole-5-carboxamidine 3-phenylpropylamine 2-(2-iodo-phenyl)-benzo[d][1,3]oxazin-4-one 4-(5-nitro-indol-1-ylmethyl)-benzamidine 8-furan-3-yl-6-styryl-naphthalene-2-carboxamidine [4-(6-chloro-naphthalene-2-sulfonyl)-piperazin-1-yl]-(3,4,5,6-tetrahydro-2h-[1,4']bipyridinyl-4-yl)-methanone 6-styryl-naphthalene-2-carboxamidine 5-amino-2,4,6-tribromobenzene-1,3-dicarboxylic acid (1r,2s)-2-phenylcyclopropanaminium 2h-benzimidazol-2-amine [n-[n-(4-methoxy-2,3,6-trimethylphenylsulfonyl)-l-aspartyl]-d-(4-amidino-phenylalanyl)]-piperidine [4-({[5-benzyloxy-1-(3-carbamimidoyl-benzyl)-1h-indole-2-carbonyl]-amino}-methyl)-phenyl]-trimethyl-ammonium 1,3-di-p-tolyl-[1,3]diazetidine-2,4-dione 5-amidino-benzimidazole 2-propionyl-1h-indole-6-carboxamidine 1-(3-nitro-benzyl)-1h-indole-5-carboxamidine 2-(2-methylphenyl)-1h-indole-6-carboximidamide [n-(benzyloxycarbonyl)amino](4-amidinophenyl)methane-phosphonate +/-methyl 4-(aminoiminomethyl)-beta-[3- inh (aminoimino)phenyl]benzene pentanoate 1-(4-amidinophenyl)-3-(4-chlorophenyl)urea 4-indol-1-ylmethyl-benzamidine [(1-{2[(4-carbamimidoyl-phenylamino)-methyl]-1-methyl-1h-benzoimidazol-5-yl}-cyclopropyl)-pyridin-2-yl-methyleneaminooxy]-acetic acid ethyl ester 1,4:3,6-dianhydro-2-o-(3-carbamimidoylphenyl)-5-o-(4-carbamimidoylphenyl)-d-glucitol 1-(2-amidinophenyl)-3-(phenoxyphenyl)urea 4-{[1-methyl-5-(2-methyl-benzoimidazol-1-ylmethyl)-1h-benzoimidazol-2-ylmethyl]-amino}-benzamidine 8-bromo-6-styryl-naphthalene-2-carboxamidine 1-(3-amino-benzyl)-1h-indole-5-carboxamidine 4-fluorobenzylamine [4-(1,3,2-dioxaborolan-2-yloxy)methyl]benzamidine 1,3,2-dioxaborolan-2-ol 4-(1,3,2-dioxaborolan-2-yloxy)butan-1-aminium 4-hydroxybutan-1-aminium 4-(hydroxymethyl)benzamidine 1-[4-(hydroxymethyl)phenyl]guanidine 1-benzoyl-2-benzyl-1,2-dihydropyridin-3(6h)-one (2s,3r)-2-(benzyloxy)-3-methoxycyclohexanone (5r,6s)-5,6-bis(benzyloxy)cyclohex-2-enone 1-chloro-4-(1-phenyl-cyclohexanesulfonyl)-benzene (s)-flurbiprofen (5r,6s)-6-(benzyloxy)-5-methoxycyclohex-2-enone (3ar,6r,6as)-6-((s)-((s)-cyclohex-2-enyl)(hydroxy)methyl)-6a-methyl-4-oxo-hexahydro-2h-furo[3,2-c]pyrrole-6-carbaldehyde 3-phosphono-d-alanine 7alpha-nhme-ginkgolide b 7alpha-cl-ginkgolide b 7alpha-nh2-ginkgolide b 10-obn-epi-ginkgolide c 10-obn-7alpha-f-gingkolide b 7-epi-ginkgolide c 7alpha-nhet-ginkgolide b 10-obn-ginkgolide c 60p002 10-obn-ginkgolide b 2-o-ethyl-paf c-16 7alpha-oac-ginkgolide b 2-o-methyl-paf c-18 7alpha-f-ginkgolide b 7alpha-ococh2ph-ginkgolide b 7alpha-n3-ginkgolide b 192c86 15-deoxy-delta12,14-pgj2 15-deoxy-delta12,14-pgd2 2-(2-acetyl-4-bromophenoxy)acetic acid 2-(4-bromo-2-cyclohexylphenoxy)acetic acid 2-(2-formylphenoxy)acetic acid 2-(2-allyl-4-chlorophenoxy)acetic acid 3-(4-chloro-2-cyclohexylphenoxy)propanoic acid 2-(4-chloro-2-cycloheptylphenoxy)acetic acid 2-(2-cyclohexyl-4-methoxyphenoxy)acetic acid 2-(2-cyclohexyl-4-fluorophenoxy)acetic acid 2-(2-benzoyl-4-bromophenoxy)acetic acid 2-(4-bromo-2-(hydroxymethyl)phenoxy)acetic acid 2-(2-cyclohexylphenoxy)acetic acid 2-(2-benzhydryl-4-phenylthiazol-5-yl)acetic acid 2-(4-bromo-2-formylphenoxy)acetic acid 2-(4-bromo-2-tert-butylphenoxy)acetic acid 2-(4-chloro-2-cyclohexylphenoxy)acetic acid 2-(4-chloro-2-cyclopentylphenoxy)acetic acid 4-(4-chloro-2-cyclohexylphenoxy)butanoic acid 13,14-dihydro-15-keto-pgd2 15(s)-15-methyl-pgd2 13,14-dihydro-15-keto-pgf2alpha 2-(2-cyclohexyl-4-methylphenoxy)acetic acid 15(r)-15-methyl-pgd2 2-(2,4-diphenylthiazol-5-yl)acetic acid 2-(4-cyano-2-cyclohexylphenoxy)acetic acid 17-phenyl-omega-trinor-pge2 3-(2-((e)-3-phenylprop-1-enyl)phenyl)acrylic acid 3-(2-(4-methoxycinnamyl)phenyl)acrylic acid 19(r)-oh-pge2 16,16-dimethyl-pge2 11-deoxy-pge1 3-(2-(naphthalen-2-ylmethyl)phenyl)acrylic acid 3-(2-cinnamylphenyl)acrylic acid 11-deoxy-pge2 8-aza-11-deoxyprostaglandin e1 1-oh-pge1 13,14-dihydro-pge1 13,14-dihydro-16-m-chlorophenoxy-w-tetranor-pgf1alpha [3h]pgf2alpha (5z)-7-{(1r,4s,5r,6r)-6-[(1e)-1-octen-1-yl]-2,3-diazabicyclo[2.2.1]hept-2-en-5-yl}-5-heptenoic acid (5e,13e)-11-hydroxy-9,15-dioxoprosta-5,13-dien-1-oic acid (3-chloro-4-propoxy-phenyl)-acetic acid 2-(2-methylpropanoyl)-1,3,5-benzenetriol 1-(4-aminosulfonylphenyl)-2-(2-pyridyl)acetylene 2-(2-(2,6-dimethylphenylamino)phenyl)acetic acid (-)-3-o-acetylspectaline 4,5-bis(4-methoxyphenyl)-3h-1,2-dithiol-3-one 3 beta-o-acetyloleanolic acid 4,5-bis(4-chlorophenyl)isothiazole 2-bromoacetyl group 2-(1,1'-biphenyl-4-yl)propanoic acid 2-(3'-ethylsulfanyl-biphenyl-4-yl)-propionic acid 2-(3'-vinyl-biphenyl-4-yl)-propionic acid 4-amino-n-(4-chlorophenyl)benzenesulfonamide (r)-2-(4-isobutyl-phenyl)-n-phenyl-propionamide 1-(4-aminosulfonylphenyl)-2-(4-pyridyl)acetylene 2-(3'-ethyl-biphenyl-4-yl)-propionic acid 2-(n-(2-fluorophenyl)pyrrol-2-yl) acetic acid 4-(4-chlorophenyl)-5-p-tolyl-3h-1,2-dithiol-3-one 4-amino-n-p-tolylbenzenesulfonamide 1-(4-(methylsulfonyl)phenyl)-3-p-tolylurea (11h-dibenzo[b,e][1,4]dioxepin-7-yl)-acetic acid 2-[1-(4-chlorobenzoyl)-5-methoxy-2-methyl-1h-indol-3-yl]-n-[(1r)-1-(hydroxymethyl)propyl]acetamide 5-(4-chlorophenyl)-4-p-tolyl-1,2-selenazole 2-[4-(1h-indol-5-yl)-phenyl]-propionic acid 2-(2-methoxyphenyl)-1h-indene 2-(3'-allyl-biphenyl-4-yl)-propionic acid 1-(4-(methylsulfonyl)phenyl)-3-phenylurea 2'-epi-guianin 4,5-bis(4-methoxyphenyl)-3h-1,2-dithiole-3-thione (11h-dibenzo[b,e][1,4]dioxepin-8-yl)-acetic acid 5-(4-methoxyphenyl)-4-p-tolylisothiazole 4-(4-chlorophenyl)-5-p-tolylisothiazole 4,5-bis(4-methoxyphenyl)-1,2-selenazole 5-ethyl-3,4-diphenyl-isoxazole 2-[1-(4-chlorobenzoyl)-5-methoxy-2-methyl-1h-indol-3-yl]-n-[(1s)-1-(hydroxymethyl)propyl]acetamide (11h-dibenzo[b,e][1,4]dioxepin-2-yl)-acetic acid 1-(4-iodobenzoyl)-5-methoxy-2-methyl indole-3-acetic acid 5-(2-1h-indenyl)-1,3-benzodioxole 5-(4-chlorophenyl)-4-p-tolylisothiazole 1,2-dihydro-3-(2,3,4-trimethoxyphenyl)naphthalene 5-(2-imidazol-1-yl-ethyl)-7,8-dihydro-quinoline 5-(4-chlorophenyl)-4-p-tolyl-3h-1,2-dithiol-3-one (z)-2'-des-methyl sulindac sulfide 4-(4-chlorophenyl)-5-p-tolyl-1,2-selenazole (+)-2-(4-biphenyl)propionic acid 5-phenyl-pentanoic acid benzyl-hydroxy-amide 4-(5-(4-hydroxyphenyl)isothiazol-4-yl)phenol 4,5-bis(4-methoxyphenyl)isothiazole 2-(2,3,4-trimethoxyphenyl)-1h-indene 2-(p-methylsulfonylbenzoyl)furan 5-(4-methoxyphenyl)-4-p-tolyl-1,2-selenazole 5-(4-chlorophenyl)-4-(4-methoxyphenyl)isothiazole 4,5-bis(4-chlorophenyl)-1,2-selenazole 3-(4-methanesulfonyl-phenyl)-1-phenyl-propynone 2-(n-(2-ffuorophenyl)pyrrol-3-yl) acetic acid 4-(4-chlorophenyl)-5-(4-methoxyphenyl)isothiazole 4-amino-n-(2-chlorophenyl)benzenesulfonamide 5-methyl-3,4-diphenyl-isoxazole 4-((4-methoxyphenyl)diazenyl)benzenesulfonamide 1-phenylsulfonamide-3-trifluoromethyl-5-parabromophenylpyrazole 2,4-dimethoxy-2'-hydroxychalcone 4-fluoro-n-(4-(methylsulfonyl)phenyl)aniline 3-benzyloxy-4-methoxy-2'-hydroxychalcone 3,4-dibenzyloxy-2'-hydroxychalcone 1,3-bis(nitrooxy)propan-2-yl 2-acetoxybenzoate 5-thia-8,11,14,17-eicosatetraenoic acid 4-benzyloxy-2'-hydroxychalcone 1-(4-(methylsulfonyl)phenyl)-1h-pyrrole 4-(4-methyl-benzylideneamino)-benzenesulfonamide 4-(3-nitro-benzylideneamino)-benzenesulfonamide 2,4'-dimethoxy-5,3'-dipropyl-biphenyl 1-(2-hydroxyphenyl)-3-p-tolylprop-2-en-1-one 2'-hydroxychalcone 2-(4-(methylsulfonyl)phenyl)-3-phenylquinoline 2,3-dimethoxy-2'-hydroxychalcone 4-(4-methoxy-benzylideneamino)-benzenesulfonamide (e)-4-(2-(thiophen-2-yl)vinyl)benzenesulfonamide 4-(4-fluoro-phenyliminomethyl)-benzenesulfonamide 6,7'-oxybis(2-phenyl-4h-chromen-4-one) 8alpha,19-dihydroxylabd-13 e-en-15-oic acid 5-methoxy-2-(4-(methylsulfonyl)phenyl)-1h-indole (e)-4-(2-(thiophen-3-yl)vinyl)benzenesulfonamide (e)-4-(2-(furan-2-yl)vinyl)benzenesulfonamide 2,6-dihydroxy-1,7-dimethoxyxanthone 4-amino-n-(4-iodophenyl)benzenesulfonamide 3-bromo-2'-hydroxy-4-methoxychalcone 4-phenyliminomethyl-benzenesulfonamide 2'-hydroxy-3,4,5-trimethoxychalcone (e)-2-(4-(methylsulfonyl)styryl)furan 4-(4-nitro-benzylideneamino)-benzenesulfonamide 4-(4-methyl-phenyliminomethyl)-benzenesulfonamide 2-(4-(methylsulfonyl)phenyl)pyridine 4-(4-fluoro-benzylideneamino)-benzenesulfonamide (e)-3-(4-(methylsulfonyl)styryl)thiophene (e)-2-(4-(methylsulfonyl)styryl)thiophene 4-(3-hydroxy-benzylideneamino)-benzenesulfonamide 4-(3-methoxy-benzylideneamino)-benzenesulfonamide 3,4-dihydroxyxanthone 1-(4-(methylsulfonyl)phenyl)-1h-indole 7-pyridin-2-yl-n-(3,4,5-trimethoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-2-amine 2-({5-chloro-2-[(2-methoxy-4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}amino)-n-methylbenzamide 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide 1,2,5-thiadiazolidin-3-one-1,1-dioxide (4s)-5-[[(2s)-1-[[(2s)-1-amino-3-[4-[difluoro(phosphono)methyl]phenyl]-1-oxopropan-2-yl]amino]-3-[4-[difluoro(phosphono)methyl]phenyl]-1-oxopropan-2-yl]amino]-4-benzamido-5-oxopentanoic acid 4-phosphonooxy-phenyl-methyl-[4-phosphonooxy]benzen 5-(3-hydroxyphenyl)isothiazol-3(2h)-one 1,1-dioxide 3-(carboxymethoxy)thieno[2,3-b]pyridine-2-carboxylic acid 3-(oxalyl-amino)-naphthalene-2-carboxylic acid 2-(oxalyl-amino)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid [{2-bromo-4-[(2r)-3-oxo-2,3-diphenylpropyl]phenyl}(difluoro)methyl]phosphonic acid 3alpha,24-dihydroxyolean-12-en-27-oic acid [(3r)-3-(methylcarbamoyl)-2-{[(2-methyl-2-propanyl)oxy]carbonyl}-1,2,3,4-tetrahydro-7-isoquinolinyl]sulfamic acid 4'-(2-butylbenzofuran-3-yl)biphenyl-4-ol 1-iodyl-4-nitro-benzene 1-methyl-3-phenyl-1h-pyrazol-5-ylsulfamic acid 3-iodyl-benzoic acid 1,2,3,4,6-penta-o-galloyl-d-glucopyranose 3-(4-{2-[2-(2-bromo-acetylamino)-ethyldisulfanyl]-ethylcarbamoyl}-cyclohexylcarbamoyl)-pyrazine-2-carboxylic acid 4-[3-(dibenzylamino)phenyl]-2,4-dioxobutanoic acid [(4-{4-[4-(difluoro-phosphono-methyl)-phenyl]-butyl}-phenyl)-difluoro-methyl]-phosphonic acid 3beta-hydroxyolean-12-en-27-oic acid {[2-(1h-1,2,3-benzotriazol-1-yl)-2-(3,4-difluorophenyl)propane-1,3-diyl]bis[4,1-phenylene(difluoromethylene)]}bis(phosphonic acid) 5-(4-methoxybiphenyl-3-yl)-1,2,5-thiadiazolidin-3-one 1,1-dioxide 5-[3-(benzylamino)phenyl]-4-bromo-3-(carboxymethoxy)thiophene-2-carboxylic acid 6-(oxalyl-amino)-1h-indole-5-carboxylic acid 7-(1,1-dioxo-1h-benzo[d]isothiazol-3-yloxymethyl)-2-(oxalyl-amino)-4,7-dihydro-5h-thieno[2,3-c]pyran-3-carboxylic acid 3-(3,5-dibromo-4-hydroxy-benzoyl)-2-ethyl-benzofuran-6-sulfonic acid [4-(thiazol-2-ylsulfamoyl)-phenyl]-amide 3-(3,5-dibromo-4-hydroxy-benzoyl)-2-ethyl-benzofuran-6-sulfonic acid dimethylamide 4-bromo-3-(carboxymethoxy)-5-[3-(cyclohexylamino)phenyl]thiophene-2-carboxylic acid [(3s)-3-(methylcarbamoyl)-2-{[(2-methyl-2-propanyl)oxy]carbonyl}-1,2,3,4-tetrahydro-7-isoquinolinyl]sulfamic acid 5-(3-{3-[3-hydroxy-2-(methoxycarbonyl)phenoxy]propenyl}phenyl)-4-(hydroxymethyl)isoxazole-3-carboxylic acid 2-(oxalyl-amino)-4,7-dihydro-5h-thieno[2,3-c]pyran-3-carboxylic acid 2-(oxalyl-amino)-benzoic acid 3-epi-masilinic acid 4-[[(2s)-1-[[6-[(1-amino-1-oxo-3-sulfanylpropan-2-yl)amino]-6-oxohexyl]amino]-3-[4-[difluoro(phosphono)methyl]phenyl]-1-oxopropan-2-yl]amino]-3-[[2-[4-[difluoro(phosphono)methyl]phenyl]acetyl]amino]-4-oxobutanoic acid 6-(difluoro-phosphono-methyl)-naphthalene-2-carboxylic acid 3beta-hydroxyurs-12-en-27-oic acid 5-(4-chloro-5-phenyl-3-thienyl)-1,2,5-thiadiazolidin-3-one 1,1-dioxide 4-carbamoyl-4-{[6-(difluoro-phosphono-methyl)-naphthalene-2-carbonyl]-amino}-butyric acid 3-oxoolean-12-en-27-oic acid 3-(3,5-dibromo-4-hydroxy-benzoyl)-2-ethyl-benzofuran-6-sulfonic acid (4-sulfamoyl-phenyl)-amide 2-[{4-[(2s)-2-{[(allyloxy)carbonyl]amino}-3-({4-[3-hydroxy-2-(methoxycarbonyl)phenoxy]butyl}amino)-3-oxopropyl]phenyl}(carboxycarbonyl)amino]benzoic acid 2-{[4-(2-acetylamino-2-pentylcarbamoyl-ethyl)-naphthalen-1-yl]-oxalyl-amino}-benzoic acid [[4-(aminomethyl)phenyl]amino]oxo-acetic acid, 2-(oxalyl-amino)-4,7-dihydro-5h-thieno[2,3-c]thiopyran-3-carboxylic acid (3r)-methylcarbamoyl-7-sulfoamino-3,4-dihydro-1h-isoquinoline-2-carboxylic acid benzyl ester 1-iodyl-3-nitro-benzene {4-[(2s)-2-({[(1s)-1-carboxy-2-phenylethyl]carbamoyl}amino)-3-oxo-3-(pentylamino)propyl]phenoxy}malonic acid {4-[(2s,4e)-2-(1,3-benzothiazol-2-yl)-2-(1h-1,2,3-benzotriazol-1-yl)-5-phenylpent-4-enyl]phenyl}(difluoro)methylphosphonic acid {[7-(difluoro-phosphono-methyl)-naphthalen-2-yl]-difluoro-methyl}-phosphonic acid 3beta,6beta-dihydroxyolean-12-en-27-oic acid 4-iodyl-benzoic acid 5-deoxyabyssinin ii 19alpha,24-dihydroxyurs-12-en-3-on-28-oic acid (4-{(2s)-2-[(tert-butoxycarbonyl)amino]-3-methoxy-3-oxopropyl}phenyl)methaneseleninic acid 3beta-acetoxyolean-12-en-27-oic acid 3-(4,5-bis-biphenyl-4-yl-1h-imidazol-2-yl)-phenol 4-bromo-3-(carboxymethoxy)-5-(4-hydroxyphenyl)thiophene-2-carboxylic acid 4'-((2-butylbenzofuran-3-yl)methyl)biphenyl-4-ol 24-hydroxyursolic acid 3,9-dihydroxy-4-prenyl-[6ar,11ar]pterocarpan 18alpha-glycyrrhetic acid 16-alphah,17-isovaleryloxy-ent-kauran-19-oic acid 2-[(7-hydroxy-naphthalen-1-yl)-oxalyl-amino]-benzoic acid 4-bromo-3-(carboxymethoxy)-5-phenylthiophene-2-carboxylic acid 18beta-glycyrrhetic acid 5-(2-fluoro-5-{(1e)-3-[3-hydroxy-2-(methoxycarbonyl)phenoxy]-1-propen-1-yl}phenyl)-1,2-oxazole-3-carboxylic acid (4-{4-[(tert-butoxycarbonyl)amino]-2,2-bis(ethoxycarbonyl)butyl}phenyl)sulfamic acid {4-[2,2-bis(5-methyl-1,2,4-oxadiazol-3-yl)-3-phenylpropyl]phenyl}sulfamic acid {4-[2-benzyl-3-methoxy-2-(methoxycarbonyl)-3-oxopropyl]phenyl}sulfamic acid (4-ethylphenyl)sulfamic acid 131i-labelled acd45 [131i]-bc8 ({[(3e)-2'-oxo-2',7'-dihydro-2,3'-biindol-3(7h)-ylidene]amino}oxy)acetic acid (2s)-n-[(3s)-1-(2-amino-2-oxoethyl)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]-2-chloro-2h-thieno[2,3-b]pyrrole-5-carboxamide 1-deoxy-1-methoxycarbamido-beta-d-glucopyranose 2-hydroxyiminours-12-en-28-oic acid 1-d-glucopyranosyl cytosine 2alpha-hydroxyurs-12-en-28-oic acid 2alpha-hydroxyolean-12-en-28-oic acid 4-{3-chloro-4-[3-(2,4-dichloro-benzoyl)-ureido]-phenoxy}-butyric acid 2-hydroxyiminoolean-12-en-28-oic acid 1-deoxy-1-acetylamino-beta-d-gluco-2-heptulopyranosonamide (s)-2-chloro-n-(1-(2-(2-hydroxyethylamino)-2-oxoethyl)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)-6h-thieno[2,3-b]pyrrole-5-carboxamide 3,8,9,10-tetrahydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-spiro[4.5]decane-2,4-dione 2beta,3alpha-dihydroxyurs-12-en-28-oic acid (3s,5r,7r,8s,9s,10r)-7-(hydroxymethyl)-3-(4-methylphenyl)-1,6-dioxa-2-azaspiro[4.5]decane-8,9,10-triol 2-(beta-d-glucopyranosyl)-5-methyl-1,3,4-benzothiazole (3r,4r,5r)-5-(hydroxymethyl)-1-(3-phenylpropyl)piperidine-3,4-diol 2-oxoolean-12-en-28-oic acid 2-isooleanolic acid 1-n-acetyl-beta-d-glucosamine (5r,7r,8s,9s,10r)-7-(hydroxymethyl)-3-phenyl-1,6-dioxa-2-azaspiro[4.5]dec-2-ene-8,9,10-triol 2-(beta-d-glucopyranosyl)-5-methyl-1,3,4-oxadiazole 2-isoursolic acid 8,9,10-trihydroxy-7-hydroxymethyl-2-thioxo-6-oxa-1,3-diaza-spiro[4.5]decan-4-one 7-{2,6-dichloro-4-[3-(2-chloro-benzoyl)-ureido]-phenoxy}-heptanoic acid (5s,7r,8s,9s,10r)-3-amino-8,9,10-trihydroxy-7-(hydroxymethyl)-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione 2-chloro-n-[(3r)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]-6h-thieno[2,3-b]pyrrole-5-carboxamide 2-chloro-n-[(1r,2r)-1-hydroxy-2,3-dihydro-1h-inden-2-yl]-6h-thieno[2,3-b]pyrrole-5-carboxamide 4-{2,4-bis[(3-nitrobenzoyl)amino]phenoxy}phthalic acid 2-deoxy-glucose-6-phosphate 2,3-dicarboxy-4-(2-chloro-phenyl)-1-ethyl-5-isopropoxycarbonyl-6-methyl-pyridinium 2-deoxy-3,4-bis-o-[3-(4-hydroxyphenyl)propanoyl]-l-threo-pentaric acid 8,9,10-trihydroxy-7-hydroxymethyl-3-methyl-6-oxa-1,3-diaza-spiro[4.5]decane-2,4-dione (3s,5r,7r,8s,9s,10r)-7-(hydroxymethyl)-3-(2-naphthyl)-1,6-dioxa-2-azaspiro[4.5]decane-8,9,10-triol 2beta,3alpha-dihydroxyolean-12-en-28-oic acid 3alpha-hydroxyurs-12-en-28-oic acid (3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-phosphoramidic acid dimethyl ester 4-{2-[(3-nitrobenzoyl)amino]phenoxy}phthalic acid 2-(beta-d-glucopyranosyl)-5-methyl-1,2,3-benzimidazole 5-{3-[3-(2,4-dichloro-benzoyl)-ureido]-2-methyl-phenoxy}-pentanoic acid 4-{4-[3-(2,4-dichloro-benzoyl)-ureido]-2,3-dimethyl-phenoxy}-butyric acid 23-hydroxybetulinic acid 1-d-glucopyranosyl uracil 1-deoxy-1-methoxycarbamido-beta-d-gluco-2-heptulopyranosonamide 1-benzylimidazole 5-(4-hydroxy-2,6-dimethylstyryl)nicotinic acid 3-fluoro-4-[2-hydroxy-2-(5,5,8,8-tetramethyl-5,6,7,8,-tetrahydro-naphtalen-2-yl)-acetylamino]-benzoic acid 3-fluoro-4-{[(2r)-2-hydroxy-2-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-2-naphthalenyl)acetyl]amino}benzoic acid 1-methyl-2-oxy-5,5-dimethyl pyrrolidine 3-phenyl-1,2-propandiol 2-cyclopropylmethylenepropanal 2-methyl-3-(2-aminothiazolo)propanal 6-(2,4-diamino-6-ethylpyrimidin-5-yl)-4-(3-methoxypropyl)-2,2-dimethyl-2h-1,4-benzoxazin-3(4h)-one (2s)-6-(2,4-diamino-6-ethylpyrimidin-5-yl)-2-(3,5-difluorophenyl)-4-(3-methoxypropyl)-2h-1,4-benzoxazin-3(4h)-one 6-ethyl-5-[9-(3-methoxypropyl)-9h-carbazol-2-yl]pyrimidine-2,4-diamine 6-ethyl-5-[(2s)-1-(3-methoxypropyl)-2-phenyl-1,2,3,4-tetrahydroquinolin-7-yl]pyrimidine-2,4-diamine (h-261)boc-his-pro-phe-his-leu(oh)-val-ile-his-oh 1-hydroxy-2-amino-3-cyclohexylpropane 1-hydroxy-3-methylbutane (z)-5-amino-3-(4-methoxybenzylidene)indolin-2-one (e)-3-(4-hydroxybenzylidene)indolin-2-one [14c]methylamine 1,2-dihexadecanoyl-sn-glycero-3-phosphoethanolamine 2'-deoxycytidine-2'-deoxyadenosine-3',5'-monophosphate 5'-deoxy-5'-piperidin-1-ylthymidine 5-aminouracil 1-(2,5-dideoxy-5-pyrrolidin-1-yl-beta-l-erythro-pentofuranosyl)-5-methylpyrimidine-2,4(1h,3h)-dione 2'-cytidylic acid 3'-phosphate-adenosine-5'-diphosphate 2'-fluoro-2'-deoxyuridine 3'-monophosphate 2'-deoxyuridine 3'-monophosphate 3'-uridinemonophosphate (4-fluoro-phenyl)-(9h-purin-6-yl)-amine 4-phospho-l-threonic acid 1,6-diazanaphthalenes and pyrido[2,3-d] pyrimidine derivative 1 1,6-diazanaphthalenes and pyrido[2,3-d] pyrimidine derivative 2 135pam1 9cuab-30 (o10eq)-beta-alanyl-anhydro-ryanodine (o10eq)-guanidino acetylryanodine (o10eq)-beta-alanylryanodine (o10eq)-beta-guanidinopropionylryanodine (o10eq)-benzyloxycarbonyl-beta-alanylryanodine 8-anilinonaphthalene-1-sulfonic acid 2-[(5-hex-1-yn-1-ylfuran-2-yl)carbonyl]-n-methylhydrazinecarbothioamide (z)-2-[2-(4-methylpiperazin-1-yl)benzyl]diazenecarbothioamide 1-(4-nonylbenzyl)pyrrolidin-3-ylphosphonic acid [3-(4-nonyl-benzylamino)-propyl]-phosphonic acid 3-(n-alkylamino) propylphosphonic acid derivative 1-(4-nonylbenzyl)azetidine-3-carboxylic acid 1-(4-nonylbenzyl)pyrrolidine-3-carboxylic acid 3-amino-5-(4-octylphenyl)pentanoic acid (3-tetradecylamino-cyclohexyl)-phosphonic acid (s)-fty720p 3-(tetradecylamino)propylphosphonic acid 4-amino-6-(4-octylphenyl)hexanoic acid (3-tetradecylamino-cyclopentyl)-phosphonic acid 2-(4-benzoylpiperazin-1-yl)thiazole-5-carboxamide 4,4'-bis([h]methylsulfonyl)-2,2',5,5'-tetrachlorobiphenyl 1-[5-(4-chlorophenyl)-2-furoyl]piperazine 5-(4-chlorophenyl)-n-(2-methylbenzyl)nicotinamide 5-hexyl-5-phenyl-imidazolidine-2,4-dione 4-biphenyl-4-yl-2-hexyl-1h-imidazole 2-hexyl-4-(4-isobutyl-phenyl)-1h-imidazole 5-heptyl-5-phenyl-imidazolidine-2,4-dione 4-biphenyl-4-yl-2-cyclohexylmethyl-1h-imidazole 5-nonyl-5-phenyl-imidazolidine-2,4-dione 5-ethyl-3-methyl-5-phenyl-oxazolidine-2,4-dione 4-biphenyl-4-yl-2-(1-propyl-butyl)-1h-imidazole 2-hydroxy-2-phenyl-nonanoic acid amide 4-biphenyl-4-yl-2-(1-pentyl-hexyl)-1h-imidazole 2-(1-pentyl-hexyl)-4-phenyl-1h-imidazole 4-biphenyl-4-yl-2-methyl-1h-imidazole 3-(4-phenoxy-phenyl)-1h-pyrazole 3-[4-(4-fluoro-phenoxy)-phenyl]-1h-pyrazole 4,9-anhydro-tetrodotoxin 4-(2'-(trifluoromethoxy)biphenyl-3-yl)oxazole 4-(2'-(trifluoromethyl)biphenyl-3-yl)oxazole 4-(2'-(trifluoromethoxy)biphenyl-3-yl)thiazole 1na 2,3,4-trihydroxybenzoic acid 2-[3,4-dihydroxy-2-hydroxymethyl-5-(2-hydroxy-nonyl)-tetrahydro-furan-2-yloxy]-6-hydroxymethyl-tetra hydro-pyran-3,4,5-triol [4-(5-naphthalen-2-yl-1h-pyrrolo[2,3-b]pyridin-3-yl)phenyl]acetic acid 4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid 4'-hydroxyflavanone 5-hydroxymethyl-5,6-dihydrofolic acid (rs)-ppcc (+)-sk&f10047 1,2,4-triazole derivative 3 1,2,4-triazole derivative 4 [3h]pentazocine 2h-chromeno[2,3-d]pyrimidine-2,4(3h)-dione (s)-sirtinol 2,3,4,9-tetrahydro-1h-carbazole-1-carboxamide (r)-sirtinol 2'-o-acetyl adenosine-5-diphosphoribose (2s)-2-(1h-indol-3-yl)hexanoic acid (2s)-8-[(tert-butoxycarbonyl)amino]-2-(1h-indol-3-yl)octanoic acid (2s)-2-(1h-indol-3-yl)pentanoic acid 1-naphthaleneacetic acid 1614235 + 2330672 264w94 [3h]glysar [11c]glysar [14c]glysar [14c]histidine [3h]histidine [11c]dtbz [125i]7-azido-8-iodoketanserine [3h]vesamicol [123i]iodobenzovesamicol [3h]thiamine [3h]etb-tboa 2-ethyl-3-(4-hydroxy) benzoyl benzofuran derivative 1 3-benzyloxyphenyloxoacetic acid derivative 1 3r14s-ochratoxin a 1,2,3-benzenetricarboxylic acid [3-(dodecanoylamino)propyl](hydroxy)dimethylammonium 9-benzyl-6-(4-nitro-benzylsulfanyl)-9h-purine 6-(4-nitro-benzylsulfanyl)-9-phenethyl-9h-purine [3h]nitrobenzylmercaptopurine ribonucleoside [cyclopentyl-(2-nitro-benzoyl)-amino]-acetic acid 5-hydroxy-l-tryptophan [3h]folinic acid [3h]n5-methylfolate 10-methoxy-n(1)-methylburnamine-17-o-veratrate [3h]hemicholinium-3 (r/s) ef-1500 (r)-nipecotic acid (r)-ef-1520 (s)-piperidine-3-carboxylic acid (s)-ef-1520 4-hydroxy-piperidine-3-carboxylic acid 2,4-diamino-butyric acid(gaba) 2-(tert-butylamino)-1-p-tolylpropan-1-one 2-(tert-butylamino)-1-m-tolylpropan-1-one 2-aminomethyl-5-(p-t-butylphenyl)tetrahydrofuran 2-(aminomethyl)-5-(1'-naphthethyl)tetrahydrofuran 1-(3,4-dichloro-phenyl)-3-diethylamino-indan-5-ol 8-methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]octane 2-(2,3-dihydro-1h-indol-5-yl)-1-methyl-ethylamine 2-(n-pyrrolidinyl)-3'-methoxypropiophenone 2-aminomethyl-5-(phenyl)tetrahydrofuran 1-(2-(2-ethylphenyl)-1-phenylethyl)piperazine 2-(aminomethyl)-5-(1'-naphthyl)tetrahydrofuran 3-(3'-furyl)-aniline 1-(2-(2-chlorophenyl)-1-phenylethyl)piperazine 2-((3-iodophenyl)(o-tolyloxy)methyl)morpholine 4-(2-(3-fluorophenoxy)-4-methylphenyl)piperidine 1-(3-bromophenyl)-2-(tert-butylamino)propan-1-one 2-(n-pyrrolidinyl)-3'-bromopropiophenone 1-(2-(2-bromophenyl)-1-phenylethyl)piperazine 3-p-tolyl-8-aza-bicyclo[3.2.1]octane 2-(n-pyrrolidinyl)-3'-nitropropiophenone 2-(n-tert-butylamino)propiophenone (s)-norduloxetine [3-(3,4-dichloro-phenyl)-indan-1-yl]-methyl-amine 2-(n-tert-butylamino)-3'-chloroheptanophenone 2-(n-cyclopentylamino)-3'-chloropropiophenone 1-(3-iodophenyl)-2-pyrrolidin-1-yl-pentan-1-one 2-aminomethyl-5-(p-methoxyphenyl)tetrahydrofuran 2-(n-tert-butylamino)-3'-chloropentanophenone 1-(4-nitrophenyl)-2-pyrrolidin-1-yl-pentan-1-one 3-(1h-indol-1-yl)-n-methyl-3-phenylpropan-1-amine (r)-n-isopropyl-n-(pyrrolidin-3-yl)-2-naphthamide 2-(2'-aminoethyl)-5-benzyltetrahydrofuran 4-(1h-indol-3-yl)-n,n-dimethylcyclohex-3-enamine 2-(tert-butylamino)-1-(3-chlorophenyl)butan-1-one 1-(4-bromophenyl)-2-(tert-butylamino)propan-1-one (s)-n-isobutyl-n-(pyrrolidin-3-yl)-2-naphthamide 2-(n-cyclopentylamino)-3'-methoxypropiophenone [3h]win35428 1-(2-methylphenyl)-2-pyrrolidin-1-yl-pentan-1-one (s)-6-(pyrrolidin-3-ylmethoxy)-2-naphthonitrile 2-((2-iodophenoxy)(phenyl)methyl)morpholine 6-(piperidin-4-ylmethoxy)-2-naphthonitrile 2-(tert-butylamino)-3',4'-dichlorobutyrophenone 4-(3'-furyl)-aniline 2-(aminomethyl)-5-phenethyltetrahydrofuran 2-(n,n-diethylamino)-3'-chloropropiophenone 4-(2-(phenoxymethyl)phenyl)piperidine 1-(2-(3-methoxyphenyl)-1-phenylethyl)piperazine (+/-)-3-((naphthalen-2-yloxy)methyl)pyrrolidine (r)-1-((s)-morpholin-2-yl)-1,2-diphenylethanol 1-(3-chlorophenyl)-2-(dimethylamino)propan-1-one [3h]nisoxetine 1s,2r-milnacipran (r)-duloxetine 2-(n-cyclopentylamino)-3'-bromopropiophenone 2-(2-phenyl-2-(piperazin-1-yl)ethyl)benzonitrile 1-(2,3-dihydro-1h-indol-5-ylmethyl)-propylamine 2-(n-pyrrolidinyl)-3'-fluoropropiophenone 3-(2-phenyl-2-(piperazin-1-yl)ethyl)phenol 1-(4-iodophenyl)-2-pyrrolidin-1-yl-pentan-1-one 1-(4-fluorophenyl)-2-pyrrolidin-1-yl-pentan-1-one 2-(n-cyclopropylamino)-3-chloropropiophenone 2-(n-tert-butylamino)-3'-chlorooctanophenone 2-aminomethyl-5-(p-bromophenyl)tetrahydrofuran 2-(aminomethyl)-5-(2'-naphthyl)tetrahydrofuran 1-(3-methylphenyl)-2-pyrrolidin-1-yl-pentan-1-one 2-(tert-butylamino)-3',4'-dichloropentanophenone 1-(3-chlorophenyl)-2-(piperidin-1-yl)propan-1-one 1-(2-(2-methoxyphenyl)-1-phenylethyl)piperazine (r)-norfluoxetine {2-[3-(phenylsulfonyl)-1h-indol-4-yl]ethyl}amine 2-(n-cyclopentylamino)-3'-fluoropropiophenone 1-(2-(2-ethoxyphenyl)-1-phenylethyl)piperazine 1-(4-bromophenyl)-2-pyrrolidin-1-yl-pentan-1-one 2pyrrolidin-1-yl-1-phenylpentan-1-one 1-(1-phenyl-2-o-tolylethyl)piperazine 18f-lmi-1195 2-(n-pyrrolidinyl)-3'-methylpropiophenone 1-(1,2-diphenylethyl)piperazine 1-(2-(3-chlorophenyl)-1-phenylethyl)piperazine 4-(2-((3-fluorophenoxy)methyl)phenyl)piperidine 2-(n-tert-butylamino)-3',4'-dichloropropiophenone (r)-2-(2-phenyl-2-(piperazin-1-yl)ethyl)phenol (r)-6-(pyrrolidin-3-ylmethoxy)-2-naphthonitrile 1-(3,4-dichloro-phenyl)-3-methylamino-indan-5-ol 3-(2-phenyl-2-(piperazin-1-yl)ethyl)benzonitrile 2-(n-cyclopentylamino)-3'-methylpropiophenone (s)-norfluoxetine ((3r,4r)-4-(o-tolyloxy)chroman-3-yl)methanamine 2-(n-tert-butylamino)-3'-chlorohexanophenone 1-(1,4-diphenylbutan-2-yl)piperazine 2-aminomethyl-5-(p-chlorophenyl)tetrahydrofuran 4-(2-(4-fluorophenoxy)-4-methylphenyl)piperidine 1-naphthalen-2-yl-2-pyrrolidin-1-yl-pentan-1-one (+/-)-threo-n-(5-phenylpentyl)methylphenidate 1-phenyl-3-aza-bicyclo[3.1.0]hexane 2-phenylpiperidine hydrochloride (+/-)-threo-n-methyl-30-methylmethylphenidate (+/-)-threo-n-(4-phenylbutyl)methylphenidate 1-(1-benzo[b]thiophen-2-yl-cycloheptyl)-azepane (+/-)-threo-n-(3-phenylpropyl)ritalinol (+/-)-threo-n-(4-methylpyridine)methylphenidate (+/-)-threo-n-(2-methylthiopene)methylphenidate (+/-)-threo-methylphenidate amide (+/-)-threo-n-(4-methoxybenzyl)methylphenidate (+/-)-threo-n-(3-methylpyridine)methylphenidate 1-biphenyl-4-yl-3-aza-bicyclo[3.1.0]hexane (+/-)-threo-n-benzylmethylphenidate amide (+/-)-threo-n-(2-methylpyridine)methylphenidate 10r-hydroxylobelane 1-(1-(benzo[b]thiophen-2-yl)cyclohexyl)piperidine (+/-)-threo-3-fluororitalinol (+/-)-threo-n-propargylmethylphenidate (+/-)-threo-n-(2-phenylethyl)methylphenidate (rs/sr)-2-[1-(4-chlorophenyl)hexyl]piperidine (+/-)-threo-3',5'-dimethylmethylphenidate (+/-)-threo-n-(6-phenylhexyl)methylphenidate 1-(1-benzo[b]thiophen-2-yl-cyclohexyl)-azepane 1-(4-aminophenyl)-2-pyrrolidin-1-yl-pentan-1-one (+/-)-threo-n-allylmethylphenidate (+/-)-threo-n-benzyl-3',4'-dichlororitalinol 3-phenyl-2-nortropene (rs/sr)-2-[1-(4-chlorophenyl)ethyl]piperidine (+/-)-threo-n-benzyl-3'-chloromethylphenidate (+/-)-threo-n-(4-chlorobenzyl)methylphenidate 4-(2-pyrrolidin-1-yl-pentanoyl)benzonitrile 10s-hydroxylobelane 2-(tert-butylamino)-3'-fluoropropiophenone (+/-)-threo-n-(2-chlorobenzyl)methylphenidate (+/-)-threo-n-(3-chlorobenzyl)methylphenidate (+/-)-threo-n-(2-phenylethyl)ritalinol 1-(thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane (+/-)-threo-n-(4-nitrobenzyl)methylphenidate 2-(n-tert-butylamino)-4'-chloropropiophenone (+/-)-threo-n-(3-methylthiopene)methylphenidate 1-(naphthalen-2-yl)-3-aza-bicyclo[3.1.0]hexane 1-benzo[b]thiophen-2-yl-cycloheptylamine (rs/sr)-2-[1-(4-chlorophenyl)butyl]piperidine 3-(4-trifluoromethylphenyl)-2-nortropene 1-benzo[b]thiophen-2-yl-cyclohexylamine (rs/sr)-2-[1-(3,4-dichlorophenyl)butyl]piperidine (cis)-1,6-diphenyl-3-aza-bicyclo[3.1.0]hexane (+/-)-threo-benzylphenidate (rs/sr)-2-[1-(4-chlorophenyl)pentyl]piperidine (+/-)-threo-3',4'-dichloromethylphenidate amide 3-alpha-phenylmethoxy-3-beta-phenyl-nortropane 2-(tert-butylamino)-3',5'-difluoropropiophenone 3-(4-chlorophenyl)-2-nortropene 1-(1-benzo[b]thiophen-2-yl-cyclopentyl)-azepane (+/-)-threo-4'-ethylmethylphenidate (+/-)-threo-n-(3-phenylpropyl)methylphenidate (rs/sr)-2-[1-(4-chlorophenyl)propyl]piperidine (+/-)-threo-n-(3-methylfuran)methylphenidate 8r-hydroxylobelane 3-(3,4-dichlorophenyl)-2-nortropene (+/-)-threo-n-(2-methylfuran)methylphenidate 1-(benzofuran-2-yl)-3-aza-bicyclo[3.1.0]hexane 8r-hydroxylobel-9-ene 2-(n-isopropylamino)-3'-chloropropiophenone (2r,3s)-2-[(3-iodophenoxy)phenylmethyl]morpholine (2r,3s)-2-[(2-iodophenoxy)phenylmethyl]morpholine (1-phenyl-ethyl)-(2-phenyl-quinazolin-4-yl)-amine 3-(4-fluorophenyl)-2-nortropene 1-benzo[b]thiophen-2-yl-cyclopentylamine 10r-hydroxylobel-7-ene (+/-)-threo-3',4'-dichlororitalinol methyl ether (2s,3s)-iodoreboxetine (2r,3r)-iodoreboxetine [n-[2-[(3'-n'-propyl-3''alpha-(bis(4-fluororphenyl)methoxy)tropane-2''beta-carboxylic acid methyl ester)(2-mercaptoethyl)amino]acetyl]-2-aminoethanethiolato]rhenium(v) oxide (diastereomeric mix) 10s-hydroxylobel-7-ene 8s-hydroxylobelane 1-phenyl-1-(piperidin-2-yl)propan-2-one 1-benzylpiperidine hydrochloride 8s-hydroxylobel-9-ene (+/-)-threo-3',5'-dichloromethylphenidate 6-(3-aza-bicyclo[3.1.0]hexan-1-yl)quinoline (+/-)-threo-n-(4-phenylbutyl)ritalinol (2r,3s)-2-[(4-iodophenoxy)phenylmethyl]morpholine 1-(1,3-diphenylpropyl)piperazine 3-(1h-indol-3-yl)-n,n-dimethylpropan-1-amine 4-benzyl-6-nitro-2-piperazin-1-yl-quinoline 4-bromo-6-nitro-2-piperazin-1-yl-quinoline 3-(3-aminocyclopentyl)-1h-indole-5-carbonitrile 6-nitro-4-phenyl-2-piperazin-1-yl-quinoline 2-n-hydroxyamino-1-(4-methylthiophenyl)propane 2-n-propargylamino-1-(4-methylthiophenyl)propane 4-allyl-6-nitro-2-piperazin-1-yl-quinoline 1-fluoro-5-phenyl-3-aza-bicyclo[3.1.0]hexane 2-n-methylamino-1-(4-methylthiophenyl)propane 2-n,n-dimethylamino-1-(4-methylthiophenyl)propane 6-nitro-2-piperazin-1-yl-4-vinyl-quinoline 2-n-methylamino-1-(4-methylthiophenyl)butane 4-chloro-6-nitro-2-piperazin-1-yl-quinoline 2-n-propargylamino-1-(4-methylthiophenyl)butane 1-methyl-4-p-tolyl-piperidine-4-carbonitrile 6,6-dimethyl-1-phenyl-3-aza-bicyclo[3.1.0]hexane 6-iodo-2-piperazin-1-yl-quinoline 6,8-dinitro-2-piperazin-1-yl-quinoline 6-chloro-2-piperazin-1-yl-quinoline 2-n-hydroxyamino-1-(4-ethylthiophenyl)propane 6-bromo-2-piperazin-1-yl-quinoline 2-n-methylamino-1-(4-ethylthiophenyl)propane 2-n-ethylamino-1-(4-methylthiophenyl)butane 1-(2-(naphthalen-2-yl)ethyl)piperazine 2-n-ethylamino-1-(4-ethylthiophenyl)propane 3-(2-phenyl-2-(piperazin-1-yl)ethyl)benzamide 2-n-(n-propyl)amino-1-(4-methylthiophenyl)butane 2-naphthalen-2-ylmethyl-4,5-dihydro-1h-imidazole 2-n-hydroxyamino-1-(4-methylthiophenyl)butane 4-furan-2-yl-6-nitro-2-piperazin-1-yl-quinoline 2-n-hydroxyamino-1-(4-ethylthiophenyl)butane 4-(2-((dimethylamino)methyl)phenoxy)benzonitrile 1-(1-phenyl-2-(pyridin-4-yl)ethyl)piperazine 1-(2-(naphthalen-1-yl)-1-phenylethyl)piperazine 2-amino-1-(4-ethylthiophenyl)propane 2-n-ethylamino-1-(4-ethylthiophenyl)butane 1-(1-phenyl-2-(pyridin-2-yl)ethyl)piperazine 1-methyl-2-(4-phenylsulfanyl-phenyl)-ethylamine 2-amino-1-(4-ethylthiophenyl)butane 2-n-(isopropyl)amino-1-(4-methylthiophenyl)butane 2-n-methoxyamino-1-(4-methylthiophenyl)propane 2-n-cyclopropylamino-1-(4-methylthiophenyl)butane 4-iodo-6-nitro-2-piperazin-1-yl-quinoline 3-bromo-6-nitro-2-piperazin-1-yl-quinoline 1-(2-(naphthalen-2-yl)-1-phenylethyl)piperazine 2-(3-methyl-piperazin-1-yl)-6-nitro-quinoline 2-n-allylamino-1-(4-methylthiophenyl)propan 2-n-ethylamino-1-(4-methylthiophenyl)propane 2-[1,4]diazepan-1-yl-6-nitro-quinoline 1-(4-benzylsulfanyl-phenyl)-propylamine 2-amino-1-(4-methylthiophenyl)butane [35s]acppb [3h](r)-npts [3h]sb-733993 [3h]gsk931145 [3h]nfps [3h]n-methyl-ssr504734 (+/-)-2-amino-1,2,3,4-tetrahydro-2-naphthoic acid (+/-)-2-aminoindane-2-carboxylic acid 5'-(n-ethyl-n-isopropyl)amiloride [3h]estrone-3-sulphate [3h]estradiol-17beta-glucuronide 4-deoxy-alpha-d-glucose 1-benzyl-4-(4-phenylpiperazin-1-yl)phthalazine 5-fluorouridine 3-fluoro-l-tyrosine (s)-2-amino-6-hydroxy-n-(4-octylphenyl)hexanamide (r)-2-amino-3-(4-octylphenylamino)propan-1-ol (s)-2-amino-4-hydroxy-n-(4-octylphenyl)butanamide (r)-2-amino-4-hydroxy-n-(4-octylphenyl)butanamide 1(beta)-o-galloylpedunculagin 1,2,6-tri-o-galloyl-beta-d-glucose 4-chloro-5,7-diphenyl-7h-pyrrolo[2,3-d]pyrimidine 3-(3-aminobenzo[e][1,2,4]triazin-7-yl)phenol 2-(4-carcoxy-5-isopropylthiazolyl)benzopiperidine 7-(naphthalen-2-yl)benzo[e][1,2,4]triazin-3-amine 4-[(4-methyl-1-piperazinyl)methyl]-n-[3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-benzamide (2e)-n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4-(dimethylamino)but-2-enamide [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrile 5,7-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-ol 1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-phenylurea 1-(1-methylethyl)-3-quinolin-6-yl-1h-pyrazolo[3,4-d]pyrimidin-4-amine 2-[4-[(z)-2-acetamido-3-oxo-3-[[(3s)-2-oxo-1-[(4-phenylphenyl)methyl]azepan-3-yl]amino]prop-1-enyl]-2-formylphenyl]acetic acid 1-cyclobutyl-3-(3,4-dimethoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine 1-methyl-5-phenyl-piperidin-2-one 4,4'-dihydroxyoctafluoroazobenzene 4-methyl-5,6-dihydro-pyrido[1,2-a]quinolin-3-one 5-(4-chloro-phenyl)-1-methyl-piperidin-2-one (e)-3-(4-(4-phenoxybenzoyl)phenyl)acrylic acid {4-[4-(4-bromophenoxy)benzoyl]phenyl}acetic acid 4-[4-(benzhydryloxy)benzoyl]benzoic acid 1-methyl-5-(4-phenylazo-phenyl)-piperidin-2-one (3-fluoro-4-(4-phenoxybenzoyl)phenyl)acetic acid 4-[4-benzyloxy)benzoyl]benzoic acid 1,2,5,6-tetrahydro pyrido[1,2-a]quinolin-3-one 3,4,5,6-tetrahydrobenzo[c]quinolizin-3-(4ah)-one 5-(4-chloro-phenyl)-1-methyl-piperidine-2-thione (3-methyl-4-(4-phenoxybenzoyl)phenyl)acetic acid 4-(4-phenoxybenzoyl)benzoic acid 3-[4-(4-phenoxybenzoyl)phenyl]propanoic acid 4-[3-(benzyloxy)benzoyl]benzoic acid 4-[4-(benzylamino)benzoyl]benzoic acid 4-[4-(benzoylamino)benzoyl]benzoic acid 4-(4-phenoxybenzoyl)phenylacetic acid 99mtc-mip-1407 98mtc-cim-ant 177lu-dotatate 3-tapap 99mtc-14 f7 mab 2-mercapto-n-[1,2,3,10-tetramethoxy-9-oxo-5,6,7,9-tetrahydro-benzo[a]heptalen-7-yl]acetamide 2-adamantan-2-ylidenemethyl-benzooxazol-6-ol 2-(4-cyclohexylthiosemicarbazono)methyl-phenol 2',4'-dicyanobiphenyl-4-yl sulfamate 4-sulfamoyloxy-benzoic acid hexyl ester 4-sulfamoyloxy-benzoic acid nonyl ester 4-sulfamoyloxy-benzoic acid cyclohexyl ester 4-sulfamoyloxy-benzoic acid cycloheptyl ester 4-sulfamoyloxy-benzoic acid cyclopentyl ester 3-{3-[(aminosulfonyl)oxy]benzoyl}phenyl sulfamate 2-methylsulfanylestradiol 3,17-o,o-bis-sulfamate 2-ethylestradiol 3,17-o,o-bis-sulfamate 3-{4-[(aminosulfonyl)oxy]benzoyl}phenyl sulfamate 4-sulfamoyloxy-benzoic acid propyl ester 4-sulfamoyloxy-benzoic acid cyclooctyl ester 2-amino-3-oxo-4-sulfo-butyric acid 3-(4-cyclohexylthiosemicarbazono)methyl-phenol 4-(4-cyclohexylthiosemicarbazono)methyl-phenol 4-sulfamoyloxy-benzoic acid heptyl ester 4-sulfamoyloxy-benzoic acid butyl ester 4-sulfamoyloxy-benzoic acid octyl ester 4-sulfamoyloxy-benzoic acid pentyl ester 3-(4-hexylthiosemicarbazono)methyl-benzoic acid 4-{4-[(aminosulfonyl)oxy]benzoyl}phenyl sulfamate 3,3',5,5'-tetrachlorobiphenyl-4,4'-diol 3'-phospho-5'-adenylyl sulfate {[2-amino-4-oxo-6,7-di(sulfanyl-?s)-3,5,5a,8,9a,10-hexahydro-4h-pyrano[3,2-g]pteridin-8-yl]methyl dihydrogenato(2-) phosphate}(dioxo)sulfanylmolybdenum 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]pyrimidine-5-carboxamide 2-{2-[(3,5-dimethylphenyl)amino]pyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-methylethyl]-4-methyl-1,3-thiazole-5-carboxamide 3-iodothyronamine [125i]l703,606 (d)-phe-(d)-phe-nh2 7-methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide (structural mix) (d)-phe-(l)-phe-nh2 3-benzyloxy-2-phenyl-piperidine [18f]spa-rq 2-phenyl-3-(1-phenyl-ethoxy)-piperidine (l)-phe-(d)-phe-nh2 7-methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (s)-[(s)-1-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide (enantiomeric mix) [sar9,met(o2)11]-sp 3,6-diphenyl-1-oxa-7-aza-spiro[4.5]decane 7-methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (s)-[(r)-1-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide (enantiomeric mix) 3-methoxy-n',2-diphenylquinoline-4-carbohydrazide 2-phenyl-n-(1-phenylethyl)quinoline-4-carboxamide 10,10-difluoro txa2 [125i]sq-29548 [125i]pta-oh [125i]sap [125i]bop 5-imidazol-1-yl-5,6,7,8-tetrahydro-quinoline 2-(8-imidazol-1-yl-octyl)-isoindole-1,3-dione 4-methyl-pyridine 2-(6-imidazol-1-yl-hexyl)-isoindole-1,3-dione 2-(10-imidazol-1-yl-decyl)-isoindole-1,3-dione 4-(4-fluoropyrazol-1-yl)-1,2-oxazol-5-amine 680c91 2-heptyl-1(3)h-anthra[1,2-d]imidazole-6,11-dione 2,7-bis[2-(isobutylamino)acetamido]anthraquinone 2-methyl-1(3)h-anthrasimidazole-6,11-dione 7,8,3',4'-tetrahydroxyflavone 2,3,7-trichloro-5-nitroquinoxaline (tnqx) 2,7-bis(benzoamido)anthraquinone 2,7-bis(acetamido)anthraquinone 2,7-bis(cyclohexanecarbonamido)anthraquinone 2,7-bis[3-(propylamino)propionamido]anthraquinone 2,7-bis(cyclopropanecarbonamido)anthraquinone 2,7-bis[3-(butylamino)propionamido]anthraquinone 1,3-bis(3,4-dihydroxyphenyl)prop-2-en-1-one 2,7-bis[2-(butylamino)acetamido]anthraquinone 2,3-dimethylnaphtho[2,3-f]quinoxaline-7,12-dione 2,7-bis(chloroacetamido)anthraquinone 2,7-bis(cyclopentanecarbonamido)anthraquinone 2-butyl-1(3)h-anthra[1,2-d]imidazole-6,11-dione 2,7-bis[2-(piperidino)acetamido]anthraquinone 2,7-dinitroantraquinone 2,7-bis[3-(piperazino)propionamido]anthraquinone 2,7-bis[2-(dimethylamino)acetamido]anthraquinone 2,7-bis(propionamido)anthraquinone 2,7-bis[2-(ethylamino)acetamido]anthraquinone 2,7-bis(phenylacetamido)anthraquinone 2,7-diaminoanthraquinone 2,7-bis(3-chloropropionamido)anthraquinone 2,7-bis[2-(piperazino)acetamido]anthraquinone 2,7-bis[3-(piperidino)propionamido]anthraquinone 2,7-bis[3-(pyrrolidino)propionamido]anthraquinone 2,7-bis[2-(propylamino)acetamido]anthraquinone 2,7-bis[2-(isopropylamino)acetamido]anthraquinone 2,7-bis(4-chlorobutyramido)anthraquinone 2,7-bis[2-(pyrrolidino)acetamido]anthraquinone 2,7-bis[3-(ethylamino)propionamido]anthraquinone 2,7-bis[2-(diethylamino)acetamido]anthraquinone 2,7-bis(butyramido)anthraquinone 2,7-bis(phenylpropionamido)anthraquinone 4-pyridin-2-yl-5-quinolin-4-yl-thiazol-2-ylamine 5''-quinolin-4-yl-[2,4'']bithiazolyl-2''-ylamine 4-(3-pyridin-2-yl-1h-pyrazol-4-yl)quinoline 2-phenyl-n-(pyridin-4-yl)quinazolin-4-amine 4-pyridin-3-yl-5-quinolin-4-yl-thiazol-2-ylamine 4-pyridin-2-yl-5-quinolin-2-yl-thiazol-2-ylamine 3-(4-fluorophenyl)-2-(6-methylpyridin-2-yl)-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazole 2-(6-methylpyridin-2-yl)-n-pyridin-4-ylquinazolin-4-amine 2-alkyloxy-3-phenylethynyl-4a,5-dihydropyrido[2,3-b]pyrazine derivative 1 3-acylidene-2-oxoindole derivative 1 3-acylidene-2-oxoindole derivative 2 3-chlorotyrosine 3-tyrosine 3-iodotyrosine 3-(dibutylamino)-1-(4-hexylphenyl)propan-1-one 4-hexylphenyl propiolate 3-(4-(benzyloxy)-3,5-dibromophenyl)propanoic acid (e)-1-(4-heptylphenyl)but-2-en-1-one 4-(4-hexylphenyl)-4-oxobut-2-enoic acid 1-(4-hexylphenyl)-3-morpholinopropan-1-one 3-(dimethylamino)-1-(4-hexylphenyl)propan-1-one 3-(3,5-dibromo-4-hexyloxy-phenyl)-propionic acid 3-bromo-1-(4-hexylphenyl)propan-1-one (z)-4-(4-hexylphenylamino)-4-oxobut-2-enoic acid (3,5-dibromo-4-hexyloxy-phenyl)-acetic acid 2-[4-(4-hydroxy-3-isopropyl-phenoxy)-3,5-dimethyl-phenyl]-2h-[1,2,4]triazine-3,5-dione 1-(4-heptylphenyl)prop-2-en-1-one [3,5-dibromo-4-(4-hydroxy-3-phenethylcarbamoyl-phenoxy)-phenyl]-acetic acid (3,5-dibromo-4-butoxy-phenyl)-acetic acid 4-(3-(dimethylamino)propanoyl)-n-hexylbenzamide 1-(4-hexylphenyl)-3-(propylamino)propan-1-one (4-hexylphenyl)(oxiran-2-yl)methanone (3,5-dibromo-4-pentyloxy-phenyl)-acetic acid 1-(4-(hexyloxy)phenyl)-3-morpholinopropan-1-one 1-(4-octylphenyl)prop-2-en-1-one 1-(4-hexylphenyl)prop-2-en-1-one 2-hexylphenyl acrylate 6-hydroxypropylthymine 9-(4-hydroxybutyl)-n2-phenylguanine 9-hydroxypropyladenine, s-isomer (south)-methanocarba-thymidine 3-(2-propyn-1-yl)thymidine 1-[7-(triphenylmethoxy)heptyl]thymine 5-propyl-2'-deoxyuridine 2'-deoxyuridine 9-hydroxypropyladenine, r-isomer 5-iodo-2'-deoxyuridine-5'-monophosphate 3'-(1,2,3-triazol-1-yl)-3'-deoxy-beta-d-thymidine 2-phenylamino-9-(4-hydroxy-butyl)-6-oxopurine 1-[2-(2-triphenylmethoxyethoxy)ethyl]thymine 2'-deoxythymidine triphosphate 5-bromothienyldeoxyuridine 6-(dihydroxy-isobutyl)-thymine 6-(2-aminophenoxy)benzo[d]isothiazol-3-amine 3-hydroxy-myristic acid 8h9 6-[3-(4-morpholinyl)propyl]-2-(3-nitrophenyl)-5-thioxo-5,6,-dihydro-7h-thienol[2',3':4,5]pyrrolo[1,2-c]imidazol-7-one 1,4-diethylene dioxide 5-[1-(3,4-dimethoxy-benzoyl)-1,2,3,4-tetrahydro-quinolin-6-yl]-6-methyl-3,6-dihydro-[1,3,4]thiadiazin-2-one 3-(4-phenyl-2,4'-bipyridin-6-yl)phenol 7-amino-4-hydroxy-2-naphthalenesulfonic acid 2,3-dimethoxy-12h-[1,3]dioxolo[5,6]indeno[1,2-c]isoquinolin-6-ium 5-hydroxy-1h-indole-3-acetic acid 4-(4,6-diphenylpyridin-2-yl)phenol 3-(4-phenyl-6-(thiophen-3-yl)pyridin-2-yl)-phenol (5z,9z)-5,9-heptacosadienoic acid 10-hydroxycamptothecin 3-(4-phenyl-6-(thiophen-2-yl)pyridin-2-yl)-phenol 2,3-dimethoxybenzo[i]phenanthridines 3-(6-phenyl-2,4'-bipyridin-4-yl)phenol 4-hydroxysaprothoquinone 9-aminocamptothecin (s)-drf-1042 4-(6-phenyl-2,4'-bipyridin-4-yl)phenol 7-ethyl-10-hydroxycamptothecin 4-(5,11-dioxo-5h-indeno[1,2-c]isoquinolin-6(11h)-yl)butanoate 3,3'-(4-phenylpyridine-2,6-diyl)diphenol 13-deoxydoxorubicin 3'-thio-thymidine-5'-phosphate 1-(9-ethyl-9h-carbazol-3-yl)-n-methylmethanamine 6-fluorotryptophan 3-(butylsulphonyl)-propanoic acid [2(formyl-hydroxy-amino)-ethyl]-phosphonic acid 3-(2-benzothiazolylthio)-1-propanesulfonic acid 2-carboxyethylphosphonic acid 2-mercaptobenzothiazole (2s)-aminobutyryl-l-proline (r)-sec-butylamide (2s)-aminobutyryl-l-prolinamide (2s)-aminobutyryl-l-proline n-pentylamide (2s)-aminobutyryl-l-proline n-propylamide (2s)-aminobutyryl-(r)-pipecolinic acid amide (2s)-aminobutyryl-l-proline n-butylamide (2s)-aminobutyryl-l-proline-(2s)-methylbutylamide (2s)-aminobutyryl-l-proline isobutylamide 1-[1'-(3-phenylacryloyl)spiro[1-benzofuran-3,4'-piperidin]-5-yl]methanamine 1-(1'-{[3-(methylsulfanyl)-2-benzothiophen-1-yl]carbonyl}spiro[1-benzofuran-3,4'-piperidin]-5-yl)methanamine [4-(3-aminomethyl-phenyl)-piperidin-1-yl]-(5-phenethyl- pyridin-3-yl)-methanone (s)-camphor 2-pentenal 2-methyl-1-(pyridin-4-yl)pent-1-en-3-one oxime 4-oxo-nonenal 1,6-hexamethylene diisocyanate 3-methyl-4-phenylbut-3-en-2-one oxime 2-methyl-1-(thiophen-3-yl)pent-1-en-3-one oxime 1'-acetoxychavicol acetate 2-methyl-1-(pyridin-3-yl)pent-1-en-3-one oxime 2-methyl-1-(thiophen-2-yl)pent-1-en-3-one oxime 2-apb (-)-englerin a 9-phenanthrol 5-benzyloxytryptamine 4-(cyclohexylamino)-n-(quinolin-3-yl)benzamide 6'-iodononivamide [3h]a778317 (e)-octadec-9-enal 4-heptyl-n-(quinolin-3-yl)benzamide 4-(hexyl(methyl)amino)-n-(quinolin-3-yl)benzamide (s)-1-(1h-indazol-4-yl)-3-(1-p-tolylethyl)urea (5e,8e,11e,14e)-icosa-5,8,11,14-tetraenal (e)-3-(4-tert-butyl-phenyl)-n-phenyl-acrylamide 4-decyl-n-(pyridin-3-yl)benzamide (r)-1-(1h-indazol-4-yl)-3-(1-p-tolylethyl)urea 4-(3-methylpyridin-2-yl)-n-p-tolylbenzamide 1,3-dibenzyl urea 4-heptyl-n-(pyridin-3-yl)benzamide 4-butyl-n-(pyridin-3-yl)benzamide 1-(4-bromo-benzyl)-3-quinazolin-8-yl-urea 12s-hpete 1-(isoquinolin-5-yl)-3-(4-morpholinobenzyl)urea 1-(isoquinolin-5-yl)-3-(1-phenylpropyl)urea 4-butyl-n-(7-hydroxynaphthalen-1-yl)benzamide 6-iodo-nordihydrocapsaicin 4-octyl-n-(pyridin-3-yl)benzamide 1-benzhydryl-3-(isoquinolin-5-yl)urea 4-(butyl(methyl)amino)-n-(quinolin-3-yl)benzamide 4-(methyl(octyl)amino)-n-(quinolin-3-yl)benzamide 4-(methyl(nonyl)amino)-n-(quinolin-3-yl)benzamide [125i]resiniferatoxin 4-nonyl-n-(quinolin-3-yl)benzamide 4-butyl-n-phenylbenzamide 2-(4-pentylphenyl)-n-(pyridin-3-yl)acetamide 4-tert-butyl-n-(quinolin-3-yl)benzamide 4-hexyl-n-(quinolin-3-yl)benzamide 4-butyl-n-(quinolin-3-yl)benzamide 15s-hpete 4-butyl-n-(isoquinolin-5-yl)benzamide 4-propyl-n-(quinolin-3-yl)benzamide 4-octyl-n-(quinolin-3-yl)benzamide 4-pyridin-2-yl-piperazine-1-carboxylic acid amide 4-pentyl-n-pyridin-3-yl benzamide 6-tert-butyl-m-cresol 4alpha-pdd 5,6-epoxyeicosatrienoic acid 4alpha-pdh 5'-iodoresiniferatoxin 11c-pbr-28 (r)pk-11195 6-thia-10b-aza-benzo[e]azulen-4-one 18f-fedaa-1106 11c-pbr-170 2-(2-phenyl-1h-indol-3-yl)-n,n-dipropyl-acetamide 5-phenyl-6-thia-10b-aza-benzo[e]azulene 5-phenyl-6-thia-10b-aza-benzo[e]azulen-4-one 4-methoxy-5-phenyl-6-thia-10b-aza-benzo[e]azulene (1r,2r,3s,4r,6s)-3,4,6-trihydroxy-5-{[(s)-hydroxy(3-hydroxy-2-oxopropoxy)phosphoryl]oxy}-1,2-cyclohexanediyl bis[dihydrogen (phosphate)] 3-bromo-4,4',5-trimethoxy-(z)-stilbene 3,4',5-trimethoxy-(z)-stilbene 3,4,4',5-tetramethoxy-(z)-stilbene 6-ile-ustiloxin 2,3'-diamino-3,4,4',5-tetramethoxy-(z)-stillbene 2'-amino-3,4,4',5-tetramethoxy-(z)-stillbene 2-amino-3,4',5-trimethoxy-(z)-stillbene 4-aryl quinol derivative 7 4-aryl quinol derivative 3 4-aryl quinol derivative 4 4,6-dinitrobenzo[c][1,2,5]thiadiazole 4-aryl quinol derivative 2 3-formyl-4-phenyl-1,2,5-oxadiazole 2-oxide 4-aryl quinol derivative 5 4-aryl quinol derivative 1 6-chloro-5-phenylpyrimidine-2,4(1h,3h)-dione 1-benzyl-5'-o-tritylinosine 5-bromo-6-(cyclopropylamino)uracil hydrochloride 6-fluoro-5-phenylpyrimidine-2,4(1h,3h)-dione 5-bromo-6-hydrazinouracil hydrochloride 5-benzyl-6-chloropyrimidine-2,4(1h,3h)-dione 1-(cyclohexyl)methyl-5'-o-tritylinosine 1-(cyclopropyl)methyl-5'-o-tritylinosine 6-amino-5-bromouracil 1-allyl-5'-o-tritylinosine 6-chloro-5-heptylpyrimidine-2,4(1h,3h)-dione 6-bromo-5-phenylpyrimidine-2,4(1h,3h)-dione 6-amino-5-chlorouracil hydrochloride 5-fluoro-6-[(2-aminoimidazol-1-yl)methyl]uracil 1-propyl-5'-o-tritylinosine 5-butyl-6-chloropyrimidine-2,4(1h,3h)-dione 6-chloro-5-pentylpyrimidine-2,4(1h,3h)-dione 5-chloro-6-hydrazinouracil hydrochloride 6-chloro-5-hexylpyrimidine-2,4(1h,3h)-dione 2'-aminoimidazolylmethyluracils 6-chloro-5-propylpyrimidine-2,4(1h,3h)-dione 6-chloro-5-(2-thienyl)pyrimidine-2,4(1h,3h)-dione 2,4-diamino-5-phenyl-6-ethylpyrimidine 6,6-dimethyl-1-[3-(2,4,5-trichlorophenoxy)propoxy]-1,6-dihydro-1,3,5-triazine-2,4-diamine 1-(propan-2-ylidene)thiosemicarbazide 3-(phenoxymethyl) benzylamine derivative 4 1-hydroxy-3-phenylurea 5-{8(z),11(z),14-pentadecatrienyl}resorcinol 2-(butylthiomethyl)-5-hydroxy-4h-pyran-4-one 5-hydroxy-2-(pentylthiomethyl)-4h-pyran-4-one 1-hydroxy-3-(4-nitrophenyl)urea 2,2',4,4'-tetrahydroxychalcone 4'-(4-nitrobenzensulfonamide)-4-hydroxychalcone 5-(6-hydroxynaphthalen-2-yl)benzene-1,3-diol 2,2',4,4',6'-pentahydroxychalcone 1-(1,4-diacetylphenyl)dithiosemicarbazide 3-(phenoxymethyl) benzylamine derivative 1 5-(4-hydroxyphenyl)-1,3,4-oxadiazole-2(3h)-thione 2-hydroxy-3-isopropyl-2,4,6-cycloheptatrien-1-one 1-(butan-2-ylidene)thiosemicarbazide 7-(3,5-dihydroxyphenyl)naphthalene-1,3-diol 3-(2,4-dihydroxyphenyl)propionic acid 1-(2,5-dimethyl-1h-pyrrol-1-yl)thiourea 1-(3-phenoxypropyl)-4-(piperidin-1-yl)piperidine 3,4-dihydroxybenzaldehyde-o-ethyloxime 1-hydroxy-3-(4-(trifluoromethyl)phenyl)urea 2-(cyclohexylthiomethyl)-5-hydroxy-4h-pyran-4-one 5-hydroxy-2-(propylthiomethyl)-4h-pyran-4-one 4'-(4-fluorobenzensulfonamide)-4-hydroxychalcone 4'-amino-4-hydroxychalcone 4,4'-(ethane-1,2-diyl)dibenzene-1,3-diol 1-(1-(4-fluorophenyl)ethylidene)thiosemicarbazide 5-(6-hydroxy-2-naphthyl)-1,2,3-benzenetriol 5-(3-hydroxyphenyl)-1,3,4-oxadiazole-2(3h)-thione 1-(but-2-enylidene)thiosemicarbazide 3-(phenoxymethyl) benzylamine derivative 3 3-(phenoxymethyl) benzylamine derivative 5 3-(phenoxymethyl) benzylamine derivative 2 4-hexyl resorcinol 5-benzhydryl-1,3,4-thiadiazole-2(3h)-thione 5-(pyridin-4-yl)-1,3,4-thiadiazole-2(3h)-thione 5-cyclohexyl-1,3,4-oxadiazole-2(3h)-thione 1-(3-methylbutylidene)thiosemicarbazide 1-(1-p-tolylethylidene)thiosemicarbazide 2-hydroxyphenethyl 3,4,5-trihydroxybenzoate 2-(heptylthiomethyl)-5-hydroxy-4h-pyran-4-one 1-(1-(pyridin-3-yl)ethylidene)thiosemicarbazide 3-hydroxyphenethyl 3,4,5-trihydroxybenzoate 1-(3-phenylallylidene)thiosemicarbazide 2-hydroxy-5-isopropyl-2,4,6-cycloheptatrien-1-one 5-benzhydryl-1,3,4-oxadiazole-2(3h)-thione 5-(pyridin-4-yl)-1,3,4-oxadiazole-2(3h)-thione 5,5'-methylenebis(1,3,4-oxadiazole-2(3h)-thione) 5,5'-methylenebis(1,3,4-thiadiazole-2(3h)-thione) 3hydroxy-1-methyl-1-phenylurea 2-(hexylthiomethyl)-5-hydroxy-4h-pyran-4-one (+/-)-daedalin a 1-(1-(pyrazin-2-yl)ethylidene)thiosemicarbazide 2,2'-bi(1,3,4-thiadiazole)-5,5'(4h,4'h)-dithione 4'-(benzensulfonamide)-4-hydroxychalcone 1-(1-(thiophen-2-yl)ethylidene)thiosemicarbazide 3-(phenoxymethyl) benzylamine derivative 6 1-(4-methylpent-3-en-2-ylidene)thiosemicarbazide 2-(ethylthiomethyl)-5-hydroxy-4h-pyran-4-one 2,2',4,4'-tetrahydroxy-6'-methoxychalcone 5-phenyl-1,3,4-thiadiazole-2(3h)-thione 7,3',4'-trihydroxyisoflavone 5-phenyl-1,3,4-oxadiazole-2(3h)-thione 4-(6-hydroxynaphthalen-2-yl)benzene-1,3-diol 7,8,4'-trihydroxyisoflavone 5-benzyl-1,3,4-oxadiazole-2(3h)-thione 1-(4-bromophenyl)-3-hydroxyurea 2,4,3',5'-tetrahydroxybibenzyl 1-(4-(benzyloxy)phenyl)-3-hydroxyurea 4-hydroxyphenethyl 3,4,5-trihydroxybenzoate 1'-(4-methyl-benzyl)-[1,4']bipiperidinyl 4'-(4-aminobenzensulfonamide)-4-hydroxychalcone 1-ethylidenethiosemicarbazide 1-cyclohexylidenethiosemicarbazide 4',4-dihydroxychalcone 1-(1-(4-bromophenyl)ethylidene)thiosemicarbazide 1-cyclopentylidenethiosemicarbazide 1-propylidenethiosemicarbazide 4'-(p-toluenesulfonamide)-4-hydroxychalcone 4-adamantyl resorcinol 1-(1-phenylethylidene)thiosemicarbazide 5-{8(z),11(z)-pentadecadienyl}resorcinol 1-(3-oxocyclohexylidene)thiosemicarbazide 5-{8(z),-pentadecenyl}resorcinol (4s)-5-fluoro-l-leucine (r,r)-2,3-butanediol 6-hydroxyuridine-5'-phosphate 5-fluoro-6-ethyluridine-5'-o-monophosphate 5-fluoro-6-amino-ump 5-fluoro-6-iodo-ump 5-fluoro-6-azido-ump 1-(2-deoxy-5-o-phosphono-beta-d-erythro-pentofuranosyl)-4-methyl-1h-indole 4-[(1e,7e)-8-(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)-3,6-dioxa-2,7-diazaocta-1,7-dien-1-yl]benzoic acid 3-[(1e,7e)-8-(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)-3,6-dioxa-2,7-diazaocta-1,7-dien-1-yl]benzoic acid 5-benzylacyclouridine 2md 1,6-naphyridine-4-ketone fused heterocyclic derivative 1 3-phenyl-5-ureidoisothiazole-4-carboximide and 3-amino-5-phenylisothiazole derivative 1 (s)-wiskostatin 9-hydroxy-4-phenyl-6h-pyrrolo[3,4-c]carbazole-1,3-dione 8-bromo-4-(2-chlorophenyl)-n-(2-hydroxyethyl)-6-methyl-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-e]indole-7-carboxamide 9-hydroxy-6-(3-hydroxypropyl)-4-(2-methoxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione 3-(9-hydroxy-1,3-dioxo-4-phenyl-2,3-dihydropyrrolo[3,4-c]carbazol-6(1h)-yl)propanoic acid 4-(2-chlorophenyl)-8-(2-hydroxyethyl)-6-methylpyrrolo[3,4-e]indole-1,3(2h,6h)-dione 2-chloro-6(methylamino)purine 3,4'-(1h-1,2,4-triazole-3,5-diyl)dipyridine 3,5-bis(2-methylpyridin-4-yl)-1h-1,2,4-triazole 1-(3-cyano-phenyl)-1h-pyrazole-4-carboxylic acid 3,5-di(pyridin-4-yl)-1h-1,2,4-triazole 3-o-methylquercetin 1-[3,3-dimethyl-2-(2-methylamino-propionylamino)-butyryl]-pyrrolidine-2-carboxylic acid(1,2,3,4-tetrahydro-naphthalen-1-yl)-amide 4-(2,2,2-trifluoroethyl)-l-phenylalanine 3-cyclohexyl-l-alanine 4-o-demethylpenclomedine 4-[3-(2-chloro-4,5-difluoro-benzoyl)ureido]-3-trifluoromethoxybenzoic acid 2-(3,4-dihydroxyphenyl)acetic acid 5-chloro-1h-indole-2-carboxylic acid{[cyclopentyl-(2-hydroxy-ethyl)-carbamoyl]-methyl}-amide 9-amino-n-[3-(dimethylamino)propyl]acridine-4-carboxamide 5-chloro-n-{4-[(1r)-1,2-dihydroxyethyl]phenyl}-1h-indole-2-carboxamide