Gene Information
Gene NameF2RL1
OrganismHomo sapiens (Human)
Gene Length397
Protein NamesProteinase-activated receptor 2 (PAR-2) (Coagulation factor II receptor-like 1) (G-protein coupled receptor 11) (Thrombin receptor-like 1) [Cleaved into: Proteinase-activated receptor 2, alternate cleaved 1; Proteinase-activated receptor 2, alternate cleaved 2]
Target Nameproteinase activated receptor 2
Target TypePatented-recorded target
Gene Age544 ( ENSG00000164251 )
Evolutionary StageEumetazoa
AlphaFoldDBP55085
Gene CardF2RL1
Uniprot IDP55085
PfamPF00001
In ASDyes
Allosteric Predictionyes (1.341816127)
Ortholog in AnimalsAlpaca_ F2RL1 ( ortholog_one2one )
Dog_ F2RL1 ( ortholog_one2one )
GuineaPig_ F2RL1 ( ortholog_one2one )
Macaque_ F2RL1 ( ortholog_one2one )
Mouse_ F2rl1 ( ortholog_one2one )
Pig_ F2RL1 ( ortholog_one2one )
Rat_ F2rl1 ( ortholog_one2one )
Rabbit_ F2RL1 ( ortholog_one2one )
OhnologsNA
ParalogsF2R, F2RL2, F2RL3, P2RY8, GPR20, LPAR4, LPAR6, P2RY10, GPR35, GPR55, GPR18, GPR65, CYSLTR2, GPR17, GPR4, CYSLTR1
TissueNA
Tissue SpecificityWidely expressed in tissues with especially high levels in pancreas, liver, kidney, small intestine, and colon (PubMed:7556175, PubMed:8615752). Moderate expression is detected in many organs, but none in brain or skeletal muscle (PubMed:7556175, PubMed:8615752). Expressed in endothelial cells (PubMed:23202369). {ECO:0000269|PubMed:23202369, ECO:0000269|PubMed:7556175, ECO:0000269|PubMed:8615752}.
Pharmacological Animal ModelsNA
Gene Ontology
(biological process)
Gene Ontology
(cellular component)
Gene Ontology
(molecular function)
PDB 5NDD  (X-ray  2.80A  5NDZ  (X-ray  3.60A  5NJ6  (X-ray  4.00A 
DBSNP rs2243072  rs616235  rs2243062  rs2243083 
Subcellular location [CC]Cell membrane;
Multi-pass membrane protein.
Mouse PG classificationNA
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