| Gene Information | |
|---|---|
| Gene Name | AR |
| Organism | Homo sapiens (Human) |
| Gene Length | 920 |
| Protein Names | Androgen receptor (Dihydrotestosterone receptor) (Nuclear receptor subfamily 3 group C member 4) |
| Target Name | androgen receptor |
| Target Type | Successful target |
| Gene Age | 950 ( ENSG00000169083 ) |
| Evolutionary Stage | Vertebrata |
| AlphaFoldDB | P10275 |
| Gene Card | AR |
| Uniprot ID | P10275 |
| Pfam | PF02166; PF00104; PF00105 |
| In ASD | yes |
| Allosteric Prediction | yes (1.943134088) |
| Ortholog in Animals | Alpaca_ AR ( ortholog_one2one ) Dog_ AR ( ortholog_one2one ) GuineaPig_ AR ( ortholog_one2one ) Macaque_ AR ( ortholog_one2one ) Mouse_ Ar ( ortholog_one2one ) Pig_ AR ( ortholog_one2one ) Rat_ Ar ( ortholog_one2one ) Rabbit_ AR ( ortholog_one2one ) |
| Ohnologs | PGR, NR3C1, NR3C2 |
| Paralogs | ESRRG, ESRRB, NR3C1, ESRRA, ESR1, ESR2, PGR, NR3C2 |
| Tissue | NA |
| Tissue Specificity | [Isoform 2]: Mainly expressed in heart and skeletal muscle. {ECO:0000269|PubMed:15634333}.; [Isoform 3]: Expressed in basal and stromal cells of the prostate (at protein level). {ECO:0000269|PubMed:19244107}. |
| Pharmacological Animal Models | NULL(Chimpanzee);NULL(Mouse);0.006057(Rat);NULL(Rabbit) |
| Gene Ontology (biological process) |
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| Gene Ontology (cellular component) |
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| Gene Ontology (molecular function) |
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| PDB | 1E3G (X-ray 2.40A ) 1GS4 (X-ray 1.95A ) 1T5Z (X-ray 2.30A ) 1T63 (X-ray 2.07A ) 1T65 (X-ray 1.66A ) 1XJ7 (X-ray 2.70A ) 1XOW (X-ray 1.80A ) 1XQ3 (X-ray 2.25A ) 1Z95 (X-ray 1.80A ) 2AM9 (X-ray 1.64A ) 2AMA (X-ray 1.90A ) 2AMB (X-ray 1.75A ) 2AO6 (X-ray 1.89A ) 2AX6 (X-ray 1.50A ) 2AX7 (X-ray 1.90A ) 2AX8 (X-ray 1.70A ) 2AX9 (X-ray 1.65A ) 2AXA (X-ray 1.80A ) 2HVC (X-ray 2.10A ) 2OZ7 (X-ray 1.80A ) 2PIO (X-ray 2.03A ) 2PIP (X-ray 1.80A ) 2PIQ (X-ray 2.40A ) 2PIR (X-ray 2.10A ) 2PIT (X-ray 1.76A ) 2PIU (X-ray 2.12A ) 2PIV (X-ray 1.95A ) 2PIW (X-ray 2.58A ) 2PIX (X-ray 2.40A ) 2PKL (X-ray 2.49A ) 2PNU (X-ray 1.65A ) 2Q7I (X-ray 1.87A ) 2Q7J (X-ray 1.90A ) 2Q7K (X-ray 1.80A ) 2Q7L (X-ray 1.92A ) 2YHD (X-ray 2.20A ) 2YLO (X-ray 2.50A ) 2YLP (X-ray 2.30A ) 2YLQ (X-ray 2.40A ) 2Z4J (X-ray 2.60A ) 3B5R (X-ray 1.80A ) 3B65 (X-ray 1.80A ) 3B66 (X-ray 1.65A ) 3B67 (X-ray 1.90A ) 3B68 (X-ray 1.90A ) 3BTR (X-ray 2.60A ) 3L3X (X-ray 1.55A ) 3L3Z (X-ray 2.00A ) 3RLJ (X-ray 1.90A ) 3RLL (X-ray 1.70A ) 3V49 (X-ray 1.70A ) 3V4A (X-ray 1.95A ) 3ZQT (X-ray 2.29A ) 4HLW (X-ray 2.50A ) 4K7A (X-ray 2.44A ) 4OEA (X-ray 2.12A ) 4OED (X-ray 2.79A ) 4OEY (X-ray 1.83A ) 4OEZ (X-ray 1.80A ) 4OFR (X-ray 2.26A ) 4OFU (X-ray 2.12A ) 4OGH (X-ray 2.98A ) 4OH5 (X-ray 2.00A ) 4OH6 (X-ray 3.56A ) 4OHA (X-ray 1.42A ) 4OIL (X-ray 2.51A ) 4OIU (X-ray 3.01A ) 4OJ9 (X-ray 3.31A ) 4OJB (X-ray 2.00A ) 4OK1 (X-ray 2.09A ) 4OKB (X-ray 2.95A ) 4OKT (X-ray 2.50A ) 4OKW (X-ray 2.00A ) 4OKX (X-ray 2.10A ) 4OLM (X-ray 2.80A ) 4QL8 (X-ray 2.10A ) 5CJ6 (X-ray 2.07A ) 5JJM (X-ray 2.15A ) 5T8E (X-ray 2.71A ) 5T8J (X-ray 2.70A ) 5V8Q (X-ray 1.44A ) 5VO4 (X-ray 2.35A ) |
| DBSNP | rs104894742 rs78686797 rs374549047 rs199554641 rs138454018 rs773996740 rs201934623 rs1355285524 rs139524801 rs137852588 rs1555982864 rs137852586 rs137852586 rs137852587 rs137852569 rs142280455 rs137852573 rs137852576 rs754201976 rs1555990488 rs868669253 rs1800053 rs137852584 rs137852579 rs1555995816 rs1555995822 rs1555995840 rs1555995851 rs864622007 rs925822435 rs137852585 rs137852595 rs1340026226 rs137852583 rs1555996810 rs137852593 rs768869912 rs137852571 rs137852600 rs137852600 rs1085307685 rs1057523747 rs141425171 rs137852567 rs1555996863 rs886041352 rs137852562 rs137852572 rs137852589 rs137852570 rs1254203917 rs1414341563 rs137852591 rs1064793480 rs137852592 rs1555997625 rs1386577803 rs1057521122 rs137852577 rs9332969 rs9332970 rs886041132 rs9332971 rs137852598 rs1555997810 rs137852597 rs137852564 rs137852564 rs137852574 rs143040492 rs137852581 rs137852578 rs137852580 rs755226547 rs886041133 rs1555998105 rs137852582 |
| Subcellular location [CC] | Nucleus {ECO:0000269|PubMed:12958311, ECO:0000269|PubMed:15634333, ECO:0000269|PubMed:17587566, ECO:0000269|PubMed:19244107, ECO:0000269|PubMed:19345326, ECO:0000269|PubMed:25091737}. Cytoplasm {ECO:0000269|PubMed:12958311, ECO:0000269|PubMed:17587566, ECO:0000269|PubMed:19244107}. Note=Detected at the promoter of target genes (PubMed:25091737). Predominantly cytoplasmic in unligated form but translocates to the nucleus upon ligand-binding. Can also translocate to the nucleus in unligated form in the presence of RACK1. {ECO:0000269|PubMed:12958311, ECO:0000269|PubMed:17587566, ECO:0000269|PubMed:25091737}. |
| Mouse PG classification | NA |
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